
Neurociencia
Los inhibidores en neurociencia son compuestos diseñados para modular la actividad de proteínas, enzimas o receptores específicos dentro del sistema nervioso. Estos inhibidores son cruciales para estudiar los mecanismos moleculares subyacentes a la función neuronal, la transmisión sináptica y las enfermedades neurodegenerativas. Al dirigirse a los receptores de neurotransmisores, canales iónicos y vías de señalización, los inhibidores en neurociencia ayudan en la exploración de la función cerebral y en el desarrollo de estrategias terapéuticas para trastornos neurológicos como el Alzheimer, Parkinson y la epilepsia. En CymitQuimica, ofrecemos una amplia gama de inhibidores de neurociencia de alta calidad para apoyar su investigación en neurobiología, neurofarmacología y ciencias cognitivas.
Subcategorías de "Neurociencia"
- Receptor 5-HT(942 productos)
- ACK(1 productos)
- AChR(576 productos)
- ATP Citrato Liasa(16 productos)
- Receptor adrenérgico(2.949 productos)
- BACE(36 productos)
- Beta amiloide(205 productos)
- CAMK(69 productos)
- Inhibidores de ciclooxigenasa (COX)(565 productos)
- Receptor de dopamina(410 productos)
- Receptor GABA(337 productos)
- Gamma-secretasa(59 productos)
- GluR(255 productos)
- GlyT(24 productos)
- Receptor de histamina(359 productos)
- LRRK2(33 productos)
- Receptor de melatonina(24 productos)
- NMDAR(26 productos)
- Receptor de OX(40 productos)
- Receptor de opioides(298 productos)
Mostrar 12 subcategorías más
Se han encontrado 5389 productos de "Neurociencia"
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Telenzepine
CAS:<p>Telenzepine is a potent and selective M1 antimuscarinic.</p>Fórmula:C19H22N4O2SPureza:98%Forma y color:SolidPeso molecular:370.47S 32212 hydrochloride
CAS:<p>S 32212 hydrochloride is a high-affinity inverse agonist at the 5-HT2C receptor and an antagonist at the α2-adrenergic receptor, which is antidepressant .</p>Fórmula:C25H29ClN4O2Pureza:97.11% - 99.57%Forma y color:SolidPeso molecular:452.98Dihydro Donepezil
CAS:<p>Dihydro Donepezil (Dihydro E2020), a Donepezil metabolite, is a potent AChE inhibitor (IC50: hAChE 11.6 nM, bAChE 8.12 nM).</p>Fórmula:C24H31NO3Forma y color:SolidPeso molecular:381.51Lesogaberan
CAS:<p>Lesogaberan: selective GABAB agonist, EC50 8.6 nM, Ki 5.1 nM in rats, weak GABAA affinity (Ki 1.4 μM).</p>Fórmula:C3H9FNO2PPureza:98%Forma y color:SolidPeso molecular:141.08SERT-IN-2
<p>SERT-IN-2, a potent SERT inhibitor (IC 50 = 0.58 nM), exhibits promising efficacy as an anti-depressant.</p>Forma y color:SolidNAP-1
CAS:<p>NAP-1 is an anesthetic that enhances CA1 brain inhibition in rats and causes tadpole sedation (EC50 = 0.53 μM).</p>Fórmula:C20H18ClNO2Forma y color:SolidPeso molecular:339.82RU-505
CAS:<p>RU-505 is an interaction inhibitor of Aβ-fibrinogen that acts by rescuing altered thrombosis and cognitive decline in Alzheimer's disease mice.</p>Fórmula:C28H32FN5OPureza:98%Forma y color:SolidPeso molecular:473.58FG-5893
CAS:<p>FG-5893 is a 5-HT1A agonist and 5-HT2 antagonist with potential anxiolytic activity.</p>Fórmula:C27H29F2N3O2Pureza:98%Forma y color:SolidPeso molecular:465.53BACE2-IN-1
CAS:<p>BACE2-IN-1, a potent BACE2 inhibitor characterized by its exceptional selectivity and a Ki value of 1.6 nM, is utilized in the investigation of Type 2 Diabetes.</p>Fórmula:C36H38F3N3O3Forma y color:SolidPeso molecular:617.72-Iodomelatonin
CAS:<p>2-Iodomelatonin, Ki 28 pM, is an MT1 agonist, >5x selective over MT2, used to map melatonin sites in brain/tissues.</p>Fórmula:C13H15IN2O2Pureza:99.7%Forma y color:SolidPeso molecular:358.178-M-PDOT
CAS:<p>8-M-PDOT (AH-002) is an MT2 receptor agonist that inhibits MT1.8-M-PDOT has anxiolytic activity and may be used in the study of neuropathic pain.</p>Fórmula:C14H19NO2Pureza:99.54% - 99.54%Forma y color:SolidPeso molecular:233.31Tracazolate hydrochloride
CAS:<p>Tracazolate hydrochloride (Tracazolate (hydrochloride)) is a modulator of the GABAA receptor with anxiolytic and anticonvulsant activity.</p>Fórmula:C16H25ClN4O2Pureza:99.52%Forma y color:SolidPeso molecular:340.85LSP4-2022
CAS:<p>LSP4-2022, a mGlu4 selective agonist, increases behavioral despair in mouse models of antidepressant action.</p>Fórmula:C13H18NO8PPureza:100%Forma y color:SolidPeso molecular:347.26AChE/BuChE-IN-2
CAS:Compound 5f, an oral AChE/BuChE inhibitor, crosses BBB; IC50: 0.72 μM (AChE), 0.16 μM (BuChE), 62.52 μM (Aβ aggregation).Fórmula:C20H18N2O2Forma y color:SolidPeso molecular:318.37Trimedoxime bromide
CAS:<p>Trimedoxime bromide is a cholinesterase reactivator used as an antidote in alkyl phosphate poisoning.</p>Fórmula:C15H18Br2N4O2Forma y color:SolidPeso molecular:446.14Lidanserin
CAS:<p>Lidanserin is an antagonist of the 5-HT2A and α1-adrenergic receptor.</p>Fórmula:C26H31FN2O4Pureza:98%Forma y color:SolidPeso molecular:454.53MAO-B-IN-16
CAS:<p>MAO-B-IN-16 selectively inhibits MAO-B with IC50 of 1.55 μM, useful in studying central nervous disorders like Parkinson's.</p>Fórmula:C18H19NO3Forma y color:SolidPeso molecular:297.35UMB68 sodium
CAS:<p>UMB-68 is a GHB receptor ligand with no affinity (IC(50) >100 microM) at GABA(A) or GABA(B) receptors.</p>Fórmula:C6H12NaO3Forma y color:SolidPeso molecular:155.149BChE-IN-14
CAS:<p>BChE-IN-14 reverses cognitive decline, is safe for primary cells, crosses the blood-brain barrier, and selectively inhibits BChE (IC50: 0.011 μM for hBChE).</p>Fórmula:C24H29NForma y color:SolidPeso molecular:331.49(R)-(+)-8-Hydroxy-DPAT hydrobromide
CAS:<p>5-HT1A serotonin receptor agonist</p>Fórmula:C16H26BrNOPureza:98%Forma y color:SolidPeso molecular:328.29
