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Neurociencia

Neurociencia

Los inhibidores en neurociencia son compuestos diseñados para modular la actividad de proteínas, enzimas o receptores específicos dentro del sistema nervioso. Estos inhibidores son cruciales para estudiar los mecanismos moleculares subyacentes a la función neuronal, la transmisión sináptica y las enfermedades neurodegenerativas. Al dirigirse a los receptores de neurotransmisores, canales iónicos y vías de señalización, los inhibidores en neurociencia ayudan en la exploración de la función cerebral y en el desarrollo de estrategias terapéuticas para trastornos neurológicos como el Alzheimer, Parkinson y la epilepsia. En CymitQuimica, ofrecemos una amplia gama de inhibidores de neurociencia de alta calidad para apoyar su investigación en neurobiología, neurofarmacología y ciencias cognitivas.

Subcategorías de "Neurociencia"

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Se han encontrado 5389 productos de "Neurociencia"

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  • Telenzepine

    CAS:
    <p>Telenzepine is a potent and selective M1 antimuscarinic.</p>
    Fórmula:C19H22N4O2S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:370.47
  • S 32212 hydrochloride

    CAS:
    <p>S 32212 hydrochloride is a high-affinity inverse agonist at the 5-HT2C receptor and an antagonist at the α2-adrenergic receptor, which is antidepressant .</p>
    Fórmula:C25H29ClN4O2
    Pureza:97.11% - 99.57%
    Forma y color:Solid
    Peso molecular:452.98
  • Dihydro Donepezil

    CAS:
    <p>Dihydro Donepezil (Dihydro E2020), a Donepezil metabolite, is a potent AChE inhibitor (IC50: hAChE 11.6 nM, bAChE 8.12 nM).</p>
    Fórmula:C24H31NO3
    Forma y color:Solid
    Peso molecular:381.51
  • Lesogaberan

    CAS:
    <p>Lesogaberan: selective GABAB agonist, EC50 8.6 nM, Ki 5.1 nM in rats, weak GABAA affinity (Ki 1.4 μM).</p>
    Fórmula:C3H9FNO2P
    Pureza:98%
    Forma y color:Solid
    Peso molecular:141.08
  • SERT-IN-2


    <p>SERT-IN-2, a potent SERT inhibitor (IC 50 = 0.58 nM), exhibits promising efficacy as an anti-depressant.</p>
    Forma y color:Solid
  • NAP-1

    CAS:
    <p>NAP-1 is an anesthetic that enhances CA1 brain inhibition in rats and causes tadpole sedation (EC50 = 0.53 μM).</p>
    Fórmula:C20H18ClNO2
    Forma y color:Solid
    Peso molecular:339.82
  • RU-505

    CAS:
    <p>RU-505 is an interaction inhibitor of Aβ-fibrinogen that acts by rescuing altered thrombosis and cognitive decline in Alzheimer's disease mice.</p>
    Fórmula:C28H32FN5O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:473.58
  • FG-5893

    CAS:
    <p>FG-5893 is a 5-HT1A agonist and 5-HT2 antagonist with potential anxiolytic activity.</p>
    Fórmula:C27H29F2N3O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:465.53
  • BACE2-IN-1

    CAS:
    <p>BACE2-IN-1, a potent BACE2 inhibitor characterized by its exceptional selectivity and a Ki value of 1.6 nM, is utilized in the investigation of Type 2 Diabetes.</p>
    Fórmula:C36H38F3N3O3
    Forma y color:Solid
    Peso molecular:617.7
  • 2-Iodomelatonin

    CAS:
    <p>2-Iodomelatonin, Ki 28 pM, is an MT1 agonist, &gt;5x selective over MT2, used to map melatonin sites in brain/tissues.</p>
    Fórmula:C13H15IN2O2
    Pureza:99.7%
    Forma y color:Solid
    Peso molecular:358.17
  • 8-M-PDOT

    CAS:
    <p>8-M-PDOT (AH-002) is an MT2 receptor agonist that inhibits MT1.8-M-PDOT has anxiolytic activity and may be used in the study of neuropathic pain.</p>
    Fórmula:C14H19NO2
    Pureza:99.54% - 99.54%
    Forma y color:Solid
    Peso molecular:233.31
  • Tracazolate hydrochloride

    CAS:
    <p>Tracazolate hydrochloride (Tracazolate (hydrochloride)) is a modulator of the GABAA receptor with anxiolytic and anticonvulsant activity.</p>
    Fórmula:C16H25ClN4O2
    Pureza:99.52%
    Forma y color:Solid
    Peso molecular:340.85
  • LSP4-2022

    CAS:
    <p>LSP4-2022, a mGlu4 selective agonist, increases behavioral despair in mouse models of antidepressant action.</p>
    Fórmula:C13H18NO8P
    Pureza:100%
    Forma y color:Solid
    Peso molecular:347.26
  • AChE/BuChE-IN-2

    CAS:
    Compound 5f, an oral AChE/BuChE inhibitor, crosses BBB; IC50: 0.72 μM (AChE), 0.16 μM (BuChE), 62.52 μM (Aβ aggregation).
    Fórmula:C20H18N2O2
    Forma y color:Solid
    Peso molecular:318.37
  • Trimedoxime bromide

    CAS:
    <p>Trimedoxime bromide is a cholinesterase reactivator used as an antidote in alkyl phosphate poisoning.</p>
    Fórmula:C15H18Br2N4O2
    Forma y color:Solid
    Peso molecular:446.14
  • Lidanserin

    CAS:
    <p>Lidanserin is an antagonist of the 5-HT2A and α1-adrenergic receptor.</p>
    Fórmula:C26H31FN2O4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:454.53
  • MAO-B-IN-16

    CAS:
    <p>MAO-B-IN-16 selectively inhibits MAO-B with IC50 of 1.55 μM, useful in studying central nervous disorders like Parkinson's.</p>
    Fórmula:C18H19NO3
    Forma y color:Solid
    Peso molecular:297.35
  • UMB68 sodium

    CAS:
    <p>UMB-68 is a GHB receptor ligand with no affinity (IC(50) &gt;100 microM) at GABA(A) or GABA(B) receptors.</p>
    Fórmula:C6H12NaO3
    Forma y color:Solid
    Peso molecular:155.149
  • BChE-IN-14

    CAS:
    <p>BChE-IN-14 reverses cognitive decline, is safe for primary cells, crosses the blood-brain barrier, and selectively inhibits BChE (IC50: 0.011 μM for hBChE).</p>
    Fórmula:C24H29N
    Forma y color:Solid
    Peso molecular:331.49
  • (R)-(+)-8-Hydroxy-DPAT hydrobromide

    CAS:
    <p>5-HT1A serotonin receptor agonist</p>
    Fórmula:C16H26BrNO
    Pureza:98%
    Forma y color:Solid
    Peso molecular:328.29