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Neurociencia

Neurociencia

Los inhibidores en neurociencia son compuestos diseñados para modular la actividad de proteínas, enzimas o receptores específicos dentro del sistema nervioso. Estos inhibidores son cruciales para estudiar los mecanismos moleculares subyacentes a la función neuronal, la transmisión sináptica y las enfermedades neurodegenerativas. Al dirigirse a los receptores de neurotransmisores, canales iónicos y vías de señalización, los inhibidores en neurociencia ayudan en la exploración de la función cerebral y en el desarrollo de estrategias terapéuticas para trastornos neurológicos como el Alzheimer, Parkinson y la epilepsia. En CymitQuimica, ofrecemos una amplia gama de inhibidores de neurociencia de alta calidad para apoyar su investigación en neurobiología, neurofarmacología y ciencias cognitivas.

Subcategorías de "Neurociencia"

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Se han encontrado 5398 productos de "Neurociencia"

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  • Calmodulin-Dependent Protein Kinase II 290-309 acetate


    <p>Calmodulin-Dependent Protein Kinase II 290-309 acetate is an effective antagonist of Ca2+/calmodulin-dependent protein kinase II (IC50 = 52 nM).</p>
    Fórmula:C105H189N31O26S
    Pureza:96.7%
    Forma y color:Solid
    Peso molecular:2333.88
  • (R)-Citalopram oxalate

    CAS:
    <p>(R)-Citalopram oxalate is a weak selective serotonin reuptake inhibitor (SSRI) that antagonises its S-isomer (escitalopram), anticonvulsant and antidepressant</p>
    Fórmula:C22H23FN2O5
    Pureza:99.76%
    Forma y color:White Solid
    Peso molecular:414.43
  • (-)-Coclaurine hydrochloride

    CAS:
    <p>(-)-Coclaurine hydrochloride is an antagonist of nAChRs isolated from Sarcopetalum harveyanum.</p>
    Fórmula:C17H20ClNO3
    Pureza:99.07%
    Forma y color:Soild
    Peso molecular:321.8
  • Dalidnetug

    CAS:
    <p>Dalidnetug is a humanized monoclonal antibody that targets human β-amyloid precursor protein (APP). By specifically binding to APP, Dalidnetug reduces the production of β-amyloid (Aβ), thereby demonstrating activity in clearing β-amyloid. This compound holds potential for research in Alzheimer's disease.</p>
    Forma y color:Liquid
  • Rasagiline 13C3 mesylate racemic

    CAS:
    <p>Rasagiline 13C3 mesylate racemic is the deuterium labeled Rasagiline, which is an irreversible monoamine oxidase inhibitor.</p>
    Fórmula:C13H17NO3S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:270.32
  • Navicixizumab

    CAS:
    <p>Navicixizumab, a bispecific VEGF/DLL4 inhibitor, pairs with Paclitaxel in ovarian and other cancer research.</p>
    Forma y color:Liquid
  • R-(+)-Cotinine

    CAS:
    <p>R-(+)-Cotinine, an inactive nicotine metabolite, boosts Ach-induced current in human α7 nAChRs.</p>
    Fórmula:C10H12N2O
    Forma y color:Solid
    Peso molecular:176.22
  • N-Ethyl-N-(3-pyridylmethyl)amine

    CAS:
    <p>N-Ethyl-N-(3-pyridylmethyl)amine has affinity for nAChR (Ki = 0.97 µM) and can be used in related research in the field of life sciences.</p>
    Fórmula:C8H12N2
    Pureza:99.65%
    Forma y color:Solid
    Peso molecular:136.19
  • BChE-IN-10

    CAS:
    <p>BChE-IN-10, a strong mixed BChE inhibitor (IC50=6.4 μM), comes from Bletilla striata for AD research.</p>
    Fórmula:C23H20O5
    Forma y color:Solid
    Peso molecular:376.4
  • MGS0274

    CAS:
    <p>MGS0274, a lipophilic prodrug of mGlu2/3 agonist MGS0008, enhances oral bioavailability, potentially aiding schizophrenia research.</p>
    Fórmula:C21H32FNO7
    Forma y color:Solid
    Peso molecular:429.485
  • Desfesoterodine

    CAS:
    <p>Desfesoterodine (5-HMT) is a new muscarinic receptor antagonist with Kb of 0.84 nM.</p>
    Fórmula:C22H31NO2
    Pureza:99.77%
    Forma y color:Solid
    Peso molecular:341.49
  • Atracurium

    CAS:
    <p>Atracurium (BW-33A) is a competitive AChR antagonist and non-depolarizing muscle relaxant that may cause bronchoconstriction.</p>
    Fórmula:C53H72N2O122
    Forma y color:Solid
    Peso molecular:929.14
  • AChE/Aβ-IN-6


    <p>BACE1-IN-15 (compound 4j) serves as an effective inhibitor of BACE1 (β-secretase), efficiently mitigating the copper-induced toxicity of Aβ, with an EC50 value of 0.68 μM.</p>
    Forma y color:Odour Solid
  • BTMPS

    CAS:
    <p>BTMPS is a usage-dependent nicotinic antagonist capable of reducing acute withdrawal symptoms associated with morphine use.</p>
    Fórmula:C28H52N2O4
    Pureza:98.1%
    Forma y color:Solid
    Peso molecular:480.72
  • Cisapride hydrate

    CAS:
    <p>Cisapride acts directly as a selective agonist of serotonin 5-HT4 receptor with IC50 value of 0.483 μM. And It also acts indirectly as a parasympathomimetic.</p>
    Fórmula:C23H31ClFN3O5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:483.96
  • OXA(17-33)

    CAS:
    <p>Potent and selective peptide orexin OX1 receptor agonist (EC50 values are 8.29 and 187 nM for OX1 and OX2 receptors respectively). Truncated form of orexin A.</p>
    Fórmula:C79H125N23O22
    Pureza:98%
    Forma y color:Solid
    Peso molecular:1749
  • pCPA methyl ester hydrochloride

    CAS:
    <p>pCPA methyl ester HCl inhibits tryptophan hydroxylase, 5-HT synthesis, crosses blood-brain barrier, lowers central 5-HT.</p>
    Fórmula:C10H13Cl2NO2
    Pureza:99.73% - 99.88%
    Forma y color:Solid
    Peso molecular:250.12
  • COX-2-IN-46


    <p>COX-2-IN-46 (compound 5m) serves as a potent anti-inflammatory and analgesic agent. It demonstrates a significant inhibitory action on COX-2, with an IC 50 value of 87.74 nM.</p>
    Fórmula:C28H19F2N3S
    Forma y color:Solid
    Peso molecular:467.53
  • SB 699551

    CAS:
    <p>SB 699551 is a selective 5-HT5A antagonist (Ki=6.31 nM) that enhances 5-HT neuronal function. It inhibits SERT (Ki=25.12 nM),inhibit breast cancer.</p>
    Fórmula:C34H45N3O
    Pureza:99.83%
    Peso molecular:511.74
  • AChE-IN-46


    <p>AChE-IN-46 (compound 4), a β-cyclocostunolide, functions as an acetylcholinesterase (AChE) inhibitor [1].</p>
    Fórmula:C15H22O2
    Forma y color:Solid
    Peso molecular:234.33