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Neurociencia

Neurociencia

Los inhibidores en neurociencia son compuestos diseñados para modular la actividad de proteínas, enzimas o receptores específicos dentro del sistema nervioso. Estos inhibidores son cruciales para estudiar los mecanismos moleculares subyacentes a la función neuronal, la transmisión sináptica y las enfermedades neurodegenerativas. Al dirigirse a los receptores de neurotransmisores, canales iónicos y vías de señalización, los inhibidores en neurociencia ayudan en la exploración de la función cerebral y en el desarrollo de estrategias terapéuticas para trastornos neurológicos como el Alzheimer, Parkinson y la epilepsia. En CymitQuimica, ofrecemos una amplia gama de inhibidores de neurociencia de alta calidad para apoyar su investigación en neurobiología, neurofarmacología y ciencias cognitivas.

Subcategorías de "Neurociencia"

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Se han encontrado 5398 productos de "Neurociencia"

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  • Triazolomethylindole-3-acetic acid

    CAS:
    <p>Triazolomethylindole-3-acetic acid is a metabolite of Rizatriptan, which acts as an agonist for the serotonin (5-HT) receptor subtypes 5-HT1B and 5-HT1D.</p>
    Fórmula:C13H12N4O2
    Forma y color:Solid
    Peso molecular:256.26
  • MAO-B-IN-38


    <p>MAO-B-IN-38 (Compound 6b) is a reversible, competitive inhibitor of MAO-B, exhibiting IC50 values of 0.03 µM for MAO-B and 21.46 µM for MAO-A. This compound is applicable in research on neurodegenerative diseases, including Alzheimer's disease and Parkinson's disease.</p>
    Fórmula:C14H17FN4O2S3
    Forma y color:Solid
    Peso molecular:388.504
  • DSP-1053

    CAS:
    <p>Dsp-1053 is a powerful SERT (Ki=1.02 nM) inhibitor with partial 5-HT1A receptor (Ki=5.05 nM) agonizing activity.</p>
    Fórmula:C26H32BrNO4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:502.44
  • Cevimeline hydrochloride hemihydrate

    CAS:
    <p>Cevimeline hydrochloride hemihydrate is a novel muscarinic receptor agonist, used as a candidate therapeutic drug for xerostomia in Sjogren's syndrome.</p>
    Fórmula:C20H38Cl2N2O3S2
    Pureza:97.00%
    Forma y color:Solid
    Peso molecular:489.55
  • TAT-CN21


    <p>TatCN21, with an IC 50 of 77 nM, serves as a potent and selective inhibitor peptide of the calcium/calmodulin-dependent protein kinase II (CaMKII), a ubiquitously-expressed multifunctional serine/threonine protein kinase. It is particularly useful in research pertaining to ischemia and neurodegenerative diseases.</p>
    Fórmula:C169H303N69O43
    Forma y color:Solid
    Peso molecular:3989.65
  • PD10


    <p>PD10 is a dual inhibitor of acetylcholinesterase (AChE) and butyrylcholinesterase (BuChE), exhibiting inhibitory potency at human AChE (hAChE IC50: 0.56 μM),</p>
    Fórmula:C23H21BrN2O4
    Forma y color:Solid
    Peso molecular:469.33
  • Asenapine citrate

    CAS:
    <p>Asenapine citrate: atypical antipsychotic for schizophrenia, bipolar disorder; targets serotonin, adrenoceptors, dopamine, histamine (pKi: 8.2-10.5).</p>
    Fórmula:C23H24ClNO8
    Forma y color:Solid
    Peso molecular:477.89
  • α-Conotoxin EI

    CAS:
    <p>Selective antagonist of neuromuscular nicotinic receptors α1β1γδ</p>
    Fórmula:C83H125N27O27S5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:2093.37
  • Nipecotic acid

    CAS:
    <p>Compound PDK0243, with CAS No. 498-95-3, is a fragment molecule that serves as an important scaffold for molecular linking, expansion, and modification. Compound PDK0243 provides a structural basis and research tool for the design and screening of novel drug candidates, and is commonly used in drug discovery, drug synthesis, and related research.</p>
    Fórmula:C6H11NO2
    Forma y color:Off-White To Pale Yellow-Beige Powder
    Peso molecular:129.16
  • Dipentylone hydrochloride

    CAS:
    <p>Dipentylone hydrochloride (Bk-dmbdp HCl) is a psychoactive synthetic cathinone and sympathomimetic stimulant. Its inhibitory activity towards the dopamine transporter (IC50=0.233µM) is tenfold higher than that towards NET and SERT, inhibiting dopamine uptake and stimulating locomotor activity in mice.</p>
    Fórmula:C14H20ClNO3
    Pureza:99.94%
    Forma y color:Solid
    Peso molecular:285.77
  • AChE-IN-29


    <p>AChE-IN-29, a 3-OH pyrrolidine derivative, acts as a cholinesterase (ChE) inhibitor with potent activity against human acetylcholinesterase (hAChE), electric</p>
    Fórmula:C18H19BrN2O2
    Forma y color:Solid
    Peso molecular:375.26
  • SAHM1

    CAS:
    <p>Notch pathway inhibitor - stabilized hydrocarbon-stapled alpha helical peptide. Targets the protein-protein interface and prevents Notch complex assembly.</p>
    Fórmula:C94H162N36O23S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:2196.58
  • (Rac)-5-Hydroxymethyl Tolterodine hydrochloride

    CAS:
    <p>(Rac)-5-Hydroxymethyl Tolterodine HCl, or (Rac)-Desfesoterodine HCl, is a potent mAChR blocker researched for overactive bladder.</p>
    Fórmula:C22H32ClNO2
    Forma y color:Solid
    Peso molecular:377.95
  • β-Amyloid (29-40)

    CAS:
    <p>β-Amyloid (29-40) is a fragment of Amyloid-β peptide.Alzheimer's beta amyloid peptide (29-40/42) C-terminal fragments have physical and chemical properties</p>
    Fórmula:C49H88N12O13S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:1085.36
  • hAChE/hBuChE-IN-1


    <p>hAChE/hBuChE-IN-1 (compound C2) acts as a dual inhibitor of cholinesterases, exhibiting IC50 values of 514 nM for hAChE and 358 nM for hBuChE. It is orally active and capable of enhancing cognitive function and spatial memory.</p>
    Fórmula:C30H31FN2O3
    Forma y color:Solid
    Peso molecular:486.577
  • AC1-IN-1

    CAS:
    <p>AC1-IN-1 is a selective inhibitor of adenylyl cyclase type 1 (AC1, IC50 = 0.54 µM).</p>
    Fórmula:C18H18FN5O2
    Pureza:99.89%
    Forma y color:Solid
    Peso molecular:355.37
  • AChE-IN-43


    <p>AChE-IN-43 is a potent, selective AChE inhibitor with a K i of 0.41 μM, applicable in the study of neurological diseases [1].</p>
    Forma y color:Odour Solid
  • DCCCyb

    CAS:
    <p>DCCCyb: oral GlyT1 inhibitor with high in vivo occupancy in rhesus monkeys, confirmed by PET tracer displacement.</p>
    Fórmula:C22H29Cl2NO3S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:458.44
  • Isonaringin

    CAS:
    <p>Isonaringin shows anti-Alzheimer’s activity by inhibiting AChE.</p>
    Fórmula:C27H32O14
    Forma y color:Solid
    Peso molecular:580.53
  • (1S,3R)-3-Aminocyclopentane carboxylic acid

    CAS:
    <p>(1S,3R)-3-Aminocyclopentane carboxylic acid exhibits activity on GABAA receptors.</p>
    Fórmula:C6H11NO2
    Forma y color:Solid
    Peso molecular:129.16