
Neurociencia
Los inhibidores en neurociencia son compuestos diseñados para modular la actividad de proteínas, enzimas o receptores específicos dentro del sistema nervioso. Estos inhibidores son cruciales para estudiar los mecanismos moleculares subyacentes a la función neuronal, la transmisión sináptica y las enfermedades neurodegenerativas. Al dirigirse a los receptores de neurotransmisores, canales iónicos y vías de señalización, los inhibidores en neurociencia ayudan en la exploración de la función cerebral y en el desarrollo de estrategias terapéuticas para trastornos neurológicos como el Alzheimer, Parkinson y la epilepsia. En CymitQuimica, ofrecemos una amplia gama de inhibidores de neurociencia de alta calidad para apoyar su investigación en neurobiología, neurofarmacología y ciencias cognitivas.
Subcategorías de "Neurociencia"
- Receptor 5-HT(942 productos)
- ACK(1 productos)
- AChR(576 productos)
- ATP Citrato Liasa(16 productos)
- Receptor adrenérgico(2.949 productos)
- BACE(36 productos)
- Beta amiloide(205 productos)
- CAMK(69 productos)
- Inhibidores de ciclooxigenasa (COX)(565 productos)
- Receptor de dopamina(410 productos)
- Receptor GABA(337 productos)
- Gamma-secretasa(59 productos)
- GluR(255 productos)
- GlyT(24 productos)
- Receptor de histamina(359 productos)
- LRRK2(33 productos)
- Receptor de melatonina(24 productos)
- NMDAR(26 productos)
- Receptor de OX(40 productos)
- Receptor de opioides(298 productos)
Mostrar 12 subcategorías más
Se han encontrado 5389 productos de "Neurociencia"
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α-Conotoxin PIA
CAS:<p>Selective antagonist of α6-containing nicotinic receptors that discriminates between the closely related α6 and α3 subunits (IC50 values are 0.95 and 74.2 nM</p>Fórmula:C79H125N27O25S4Pureza:98%Forma y color:SolidPeso molecular:1981.3IHC3
<p>IHC3 is a competitive and reversible monoamine oxidase B (MAO-B) inhibitor with an IC50 of 1.672 μM, which targets Cys172 within the enzyme's active site.</p>Fórmula:C17H12FN3OPureza:98%Forma y color:SolidPeso molecular:293.3Tetrahydro-β-carboline
CAS:<p>Compound Fr12161, with CAS No. 16502-01-5, is a fragment molecule that serves as an important scaffold for molecular linking, expansion, and modification. Compound Fr12161 provides a structural basis and research tool for the design and screening of novel drug candidates, and is commonly used in drug discovery, drug synthesis, and related research.</p>Fórmula:C11H12N2Pureza:96.31%Forma y color:Tan SolidPeso molecular:172.2264Zicronapine fumarate
CAS:<p>Zicronapine fumarate, an antipsychotic, targets D1/D2 & 5-HT2A receptors; may treat neuropsychiatric conditions.</p>Fórmula:C26H31ClN2O4Forma y color:SolidPeso molecular:470.99Arotinolol hydrochloride
CAS:<p>Arotinolol HCl is a non-selective α/β-blocker, anti-hypertensive, anti-obesity, and improves aortic stiffness.</p>Fórmula:C15H22ClN3O2S3Pureza:99.84%Forma y color:SolidPeso molecular:408NMDA receptor antagonist 6
<p>NMDA Receptor Antagonist 6 (Compound 13b) functions as an antagonist at the glycine-binding site of the NMDA receptor and demonstrates cytoneuroprotective</p>Fórmula:C25H23NO2Pureza:98%Forma y color:SolidPeso molecular:369.46TRV-7019
CAS:<p>TRV-7019: BBB-permeable radioligand for brain imaging, used in diagnosing amyloid diseases, MS, and brain tumors.</p>Fórmula:C14H12INO3Forma y color:SolidPeso molecular:369.15Lysyl hydroxylase 2-IN-2
<p>Lysyl Hydroxylase 2-IN-2 (compound 13) is a potent inhibitor of Lysyl Hydroxylase 2 (LH2), exhibiting an IC50 of approximately 500 nM.</p>Fórmula:C19H21N3O2Pureza:98%Forma y color:SolidPeso molecular:323.39Jatrorrhizine hydroxide
CAS:<p>Jatrorrhizine hydroxide: alkaloid from Coptis chinensis; neuroprotective, antimicrobial, antiplasmodial, antioxidant; AChE inhibitor, affects 5-HT/NE uptake.</p>Fórmula:C20H21NO5Forma y color:SolidPeso molecular:355.38MmTx1 toxin
<p>Micrurotoxin 1 (MmTx1 toxin) acts as an allosteric modulator of GABA A receptors, enhancing the receptor's sensitivity to its agonist [1].</p>Fórmula:C295H455N95O97S10Pureza:98%Forma y color:SolidPeso molecular:7205Calmodulin Kinase IINtide, Myristoylated
<p>Myristoylated Calmodulin Kinase IINtide (Myr-CaMKIINtide) serves as a selective and noncompetitive inhibitor of CaMKII [1].</p>Fórmula:C156H275N47O43Pureza:98%Forma y color:SolidPeso molecular:3497.14XL01126
XL01126 degrades LRRK2 (DC50: 14 nM G2019S, 32 nM WT), crosses the blood-brain barrier, aiding Parkinson's studies.Fórmula:C50H64ClFN10O6S2Forma y color:SolidPeso molecular:1019.69Cyclodrine
CAS:<p>Cyclodrine (Cyclopent) is a cholinergic (muscarinic, nicotinic) (mAChR and nAChR) receptor antagonist.</p>Fórmula:C19H29NO3Pureza:97.62%Forma y color:SoildPeso molecular:319.443-Aminopropylphosphinic acid
CAS:<p>3-Aminopropylphosphinic acid (3-APPA) is a phosphonic analog of gamma-aminobutyric acid (GABA).</p>Fórmula:C3H10NO2PForma y color:SolidPeso molecular:123.0922,6-DMA hydrochloride
CAS:<p>2,6-DMA hydrochloride is a phenethylamine and acts as an agonist of the serotonin 5-HT2 receptor, with a pA2 value of 5.09.</p>Fórmula:C11H18ClNO2Forma y color:SolidPeso molecular:231.72Tabernanthalog
CAS:<p>TBG is a 5-HT2A agonist reducing alcohol/heroin cravings and promoting neuroplasticity with antidepressant effects in rodents.</p>Fórmula:C14H18N2OPureza:99.82% - 99.89%Forma y color:SoildPeso molecular:230.31AChE-IN-36
<p>AChE-IN-36 (compound A4) is an acetylcholinesterase inhibitor with an IC50 of 0.04 μM, influencing ROS levels and modulating the gene expression of NRF2 [1].</p>Fórmula:C25H21ClO5SForma y color:SolidPeso molecular:468.95SKF-83566 hydrochloride
CAS:<p>SKF-83566 hydrochloride is a D1-like dopamine receptor antagonist, inhibiting dopamine transporters and mitigating GBP-induced CPP.</p>Fórmula:C17H19BrClNOPureza:99.27%Forma y color:SoildPeso molecular:368.69Feralolide
CAS:<p>Feralolide, a dihydroisocoumarin from the methanolic extract of aloe vera resin, functions as a dual inhibitor of acetylcholinesterase (AChE) and</p>Fórmula:C18H16O7Forma y color:SolidPeso molecular:344.32(R)-(+)-Anatabine
CAS:<p>(R)-(+)-Anatabine is an less active R-enantiomer of Anatabine. Anatabine is a potent agonist of α4β2 nAChR.</p>Fórmula:C10H12N2Pureza:98%Forma y color:SolidPeso molecular:160.22

