
Neurociencia
Los inhibidores en neurociencia son compuestos diseñados para modular la actividad de proteínas, enzimas o receptores específicos dentro del sistema nervioso. Estos inhibidores son cruciales para estudiar los mecanismos moleculares subyacentes a la función neuronal, la transmisión sináptica y las enfermedades neurodegenerativas. Al dirigirse a los receptores de neurotransmisores, canales iónicos y vías de señalización, los inhibidores en neurociencia ayudan en la exploración de la función cerebral y en el desarrollo de estrategias terapéuticas para trastornos neurológicos como el Alzheimer, Parkinson y la epilepsia. En CymitQuimica, ofrecemos una amplia gama de inhibidores de neurociencia de alta calidad para apoyar su investigación en neurobiología, neurofarmacología y ciencias cognitivas.
Subcategorías de "Neurociencia"
- Receptor 5-HT(940 productos)
- ACK(1 productos)
- AChR(574 productos)
- ATP Citrato Liasa(16 productos)
- Receptor adrenérgico(2.942 productos)
- BACE(36 productos)
- Beta amiloide(204 productos)
- CAMK(68 productos)
- Inhibidores de ciclooxigenasa (COX)(562 productos)
- Receptor de dopamina(407 productos)
- Receptor GABA(336 productos)
- Gamma-secretasa(59 productos)
- GluR(255 productos)
- GlyT(24 productos)
- Receptor de histamina(358 productos)
- LRRK2(33 productos)
- Receptor de melatonina(24 productos)
- NMDAR(28 productos)
- Receptor de OX(40 productos)
- Receptor de opioides(296 productos)
Mostrar 12 subcategorías más
Se han encontrado 5400 productos de "Neurociencia"
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F-15599
CAS:<p>F-15599 is a highly selective G-protein biased 5-HT1A receptor agonist(Ki : 3.4 nM).</p>Fórmula:C19H21ClF2N4OPureza:98.72%Forma y color:SolidPeso molecular:394.85Lorediplon
CAS:<p>Lorediplon is a novel hypnotic drug acting as a GABAA receptor modulator, differentially active at the α1-subunit, associated with promoting sleep.</p>Fórmula:C20H15FN4O2SPureza:99.12% - 99.19%Forma y color:SolidPeso molecular:394.42Suritozole
CAS:<p>Suritozole (MDL-26479) is a negative modulator at the gamma-aminobutyric acidA (GABAA) receptor</p>Fórmula:C10H10FN3SPureza:99.25%Forma y color:SolidPeso molecular:223.27Succinylcholine Chloride Dihydrate
CAS:<p>Succinylcholine Chloride Dihydrate (Succinyldicholine dichloride) is a nicotinic AChR agonist and also acts as a depolarizing neuromuscular blocker.</p>Fórmula:C14H30N2O4·2Cl·2H2OPureza:99.87%Forma y color:White SolidPeso molecular:397.34PHA 568487 free base
CAS:<p>PHA 568487 free base, an α7 nicotinic receptor agonist, designed to reduce bioactivation and improve in vivo tolerability.</p>Fórmula:C16H20N2O3Pureza:99.74%Forma y color:SolidPeso molecular:288.34Cerlapirdine
CAS:<p>Cerlapirdine (PF-05212365), a 5-HT6 receptor antagonist, is in trials for Alzheimer's and schizophrenia cognition issues.</p>Fórmula:C22H23N3O3SPureza:98.77%Forma y color:SolidPeso molecular:409.5Melatonin
CAS:<p>Melatonin (Melatonine) is a natural hormone that activates melatonin receptors. Melatonin regulates the biological clock. Cost-effective and quality-assured.</p>Fórmula:C13H16N2O2Pureza:98% - 99.89%Forma y color:Pale Yellow Leaflets From Benzene SolidPeso molecular:232.28GNE-7915
CAS:<p>GNE-7915 is a highly potent, selective and brain-penetrable leucine-rich repeat kinase 2 (LRRK2) inhibitor.</p>Fórmula:C19H21F4N5O3Pureza:98% - ≥95%Forma y color:SolidPeso molecular:443.4p-Hydroxybenzaldehyde
CAS:<p>1.</p>Fórmula:C7H6O2Pureza:99.05% - 99.86%Forma y color:SolidPeso molecular:122.12BQCA
CAS:<p>BQCA (benzylquinolone carboxylic acid) a highly selective allosteric M1 mAChR modulator.</p>Fórmula:C18H15NO4Pureza:97.22%Forma y color:SolidPeso molecular:309.32Trazodone
CAS:<p>Trazodone (AF-1161), a 5-HT 2A/2C receptor antagonist, is used as an antidepressant for treating major anxiety disorders and depressive disorder.</p>Fórmula:C19H22ClN5OPureza:99.79% - 99.92%Forma y color:White To Off-White Crystalline PowderPeso molecular:371.86Ramosetron hydrochloride
CAS:<p>Ramosetron hydrochloride (YM-060) is a serotonin 5-HT3 receptor antagonist. It is used to treat diarrhea-predominant irritable bowel syndrome and nausea.</p>Fórmula:C17H18ClN3OPureza:99.95%Forma y color:SolidPeso molecular:315.8E4CPG
CAS:<p>E4CPG is a novel group I/II metabotropic glutamate receptor antagonist, more potent than (RS)-MCPG.</p>Fórmula:C11H13NO4Pureza:99.96%Forma y color:SolidPeso molecular:223.23LY900009
CAS:<p>LY900009 is a small molecule inhibitor of Notch signalling via selective inhibition of the γ-secretase protein.</p>Fórmula:C23H27N3O4Pureza:97.07%Forma y color:SolidPeso molecular:409.48Alosetron (Hydrochloride(1:X))
CAS:<p>Alosetron Hydrochloride is a selective 5-HT3 antagonist for treating IBS.</p>Fórmula:C17H18ClN4OForma y color:SolidPeso molecular:329.11691Lurasidone
CAS:<p>Lurasidone (SM-13496) is an antagonist of both dopamine D2 and 5-HT7(IC50=1.68 and 0.495 nM, respectively).It also a partial agonist of 5-HT1A receptor(IC50 : 6</p>Fórmula:C28H36N4O2SPureza:99.78% - 99.91%Forma y color:SolidPeso molecular:492.68SR 57227 hydrochloride
CAS:<p>SR 57227A (SR 57227 hydrochloride) is a potent, orally active and selective 5-HT3 receptor agonist. It with ability to cross the blood brain barrier.</p>Fórmula:C10H14ClN3·HClPureza:99.89%Forma y color:SolidPeso molecular:248.15idalopirdine
CAS:<p>Idalopirdine (Lu AE58054), a selective 5-HT6 receptor antagonist( Ki : 0.83 nM),as a treatment for Alzheimer's disease.</p>Fórmula:C20H19F5N2OPureza:99.73%Forma y color:SolidPeso molecular:398.37IMR-1A
CAS:<p>IMR-1A is the metabolite of IMR-1 which is a novel class of Notch inhibitors targeting the transcriptional activation with IC50 of 6 μMol/L.</p>Fórmula:C13H11NO5S2Pureza:97.1% - 99.76%Forma y color:SolidPeso molecular:325.36Atracurium besylate
CAS:<p>Atracurium besylate (51W89) is a short-acting, non-depolarizing muscle relaxant, not affecting the heart or reliant on kidneys.</p>Fórmula:C65H82N2O18S2Pureza:98.94% - 99.71%Forma y color:SolidPeso molecular:1243.49Naratriptan
CAS:<p>Naratriptan is a selective agonist of 5-HT1 receptor and is is used for the treatment of migraine headaches.</p>Fórmula:C17H25N3O2SPureza:99.08%Forma y color:SolidPeso molecular:335.47Mavacoxib
CAS:<p>Mavacoxib is a selective inhibitor of cyclooxygenase-2 (COX-2) ,with Anti-Tumour activity.</p>Fórmula:C16H11F4N3O2SPureza:99.90%Forma y color:SolidPeso molecular:385.34Eltoprazine
CAS:<p>Eltoprazine(DU28853) is a serenic or antiaggressive agent which as an agonist at the 5-HT1A and 5-HT1B receptors and as an antagonist at the 5-HT2C receptor.</p>Fórmula:C12H16N2O2Forma y color:SolidPeso molecular:220.27Miltirone
CAS:<p>Miltirone is a CYPs inhibitor, it has been characterized as a low-affinity ligand for central benzodiazepine receptors.</p>Fórmula:C19H22O2Pureza:99.22% - 99.66%Forma y color:SolidPeso molecular:282.38Phenylbiguanide
CAS:<p>Phenylbiguanide (N-Phenylbiguanide) is a 5-HT3 receptor selective agonist(EC50 : 3.0±0.1 μM)</p>Fórmula:C8H11N5Pureza:99.54%Forma y color:SolidPeso molecular:177.21TAT-GluA2 3Y acetate(1404188-93-7 free base)
<p>TAT-GluA2 3Y acetate is an inhibitor of AMPA receptor endocytosis.Systemic administration of Tat-GluA2(3Y) during the induction phase of d-amphetamine blocked</p>Fórmula:C115H185N43O29Pureza:99.43%Forma y color:SolidPeso molecular:2634.02Dexketoprofen trometamol
CAS:<p>Dexketoprofen trometamol is a modified non-selective COX inhibitor with a rapid onset of action that is available as both oral and parenteral formulations.</p>Fórmula:C20H25NO6Pureza:99.97% - 99.98%Forma y color:SolidPeso molecular:375.42Isoflurane
CAS:<p>Isoflurane (Forane) is a stable, non-explosive inhalation anesthetic that has been reported to induce caspase-3 activation.</p>Fórmula:C3H2ClF5OPureza:98%Forma y color:Clear Colorless Liquid LiquidPeso molecular:184.49Tebanicline hydrochloride
CAS:<p>Tebanicline hydrochloride (Ebanicline hydrochloride) , is an effective synthetic nicotinic (non-opioid) analgesic drug.</p>Fórmula:C9H12Cl2N2OPureza:91.74% - 98.71%Forma y color:SolidPeso molecular:235.11Syk Inhibitor II dihydrochloride dihydrate
CAS:<p>Potent, selective ATP-competitive Syk Inhibitor II (IC50: 41 nM), with anti-allergic properties, in dihydrochloride dihydrate form.</p>Fórmula:C14H21Cl2F3N6O3Forma y color:SolidPeso molecular:449.26Pergolide mesylate
CAS:<p>Pergolide mesylate (LY127809), a dopamine agonist for Parkinson's and hyperprolactinemia, was withdrawn for heart valve risk.</p>Fórmula:C20H30N2O3S2Pureza:99.70%Forma y color:White To Off-White SolidPeso molecular:410.59PBD-150
CAS:<p>PBD-150 is an inhibitor of human glutaminyl cyclase (hQC) Y115E-Y117E variant( ki : 490 nM)</p>Fórmula:C15H20N4O2SPureza:99.68%Forma y color:SolidPeso molecular:320.41Amperozide
CAS:<p>Amperozide (FG 5606), an atypical antipsychotic, antagonizes 5-HT2A and modulates dopamine activity for schizophrenia treatment.</p>Fórmula:C23H29F2N3OPureza:99.68%Forma y color:SolidPeso molecular:401.49N-Desmethylclozapine
CAS:<p>N-Desmethylclozapine: 5-HT2C antagonist (IC50: 7.1 nM), dopamine D4 antagonist, δ-opioid agonist.</p>Fórmula:C17H17ClN4Pureza:97.25% - 99.83%Forma y color:Yellow Crystalline SolidPeso molecular:312.8Dicyclomine
CAS:<p>Dicyclomine: oral muscarinic antagonist, eases GI muscle spasms, high affinity for M1/M2 receptors, Ki of 5.1 nM/54.6 nM.</p>Fórmula:C19H35NO2Forma y color:SolidPeso molecular:309.49β-Amyloid 15-21 acetate
<p>β-Amyloid 15-21 acetate (Beta-Amyloid (15-21) acetate) is a fragment of Amyloid-β peptide, maybe used in the research of neurological disease.</p>Fórmula:C45H69N9O11Pureza:99.62%Forma y color:SolidPeso molecular:912.1Sumatriptan hydrochloride
CAS:<p>Sumatriptan hydrochloride (GR 43175), an oral 5-HT1 receptor agonist, treats migraines; Ki: 5-HT1D - 17 nM, 5-HT1B - 27 nM, 5-HT1A - 100 nM.</p>Fórmula:C14H22ClN3O2SForma y color:SolidPeso molecular:331.86Flutriafol
CAS:<p>Flutriafol is a pesticide, demethylation inhibitor, and NMDA receptor agonist</p>Fórmula:C16H13F2N3OPureza:98.75%Forma y color:SolidPeso molecular:301.29Sarpogrelate
CAS:<p>Sarpogrelate (MCI-9042), an oral 5-HT2 antagonist, boosts platelet aggregation and aids in studying Buerger's disease.</p>Fórmula:C24H31NO6Forma y color:SolidPeso molecular:429.51Acotiamide
CAS:<p>Acotiamide, an oral AChE inhibitor (IC50: 1.79μM), improves gastric motility, targeting functional dyspepsia.</p>Fórmula:C21H30N4O5SForma y color:SolidPeso molecular:450.55PF3274167
CAS:<p>PF3274167 (Cligosiban) is a potent and selective, high-affinity nonpeptide oxytocin receptor antagonist.</p>Fórmula:C19H19ClFN5O3Pureza:99.67% - 99.88%Forma y color:SolidPeso molecular:419.84Flibanserin hydrochloride
CAS:<p>Flibanserin HCl: oral 5-HT1A agonist & 5-HT2A antagonist, Ki values 1 nM & 49 nM, for HSDD, has antidepressant/anxiolytic properties.</p>Fórmula:C20H22ClF3N4OForma y color:SolidPeso molecular:426.87β-amyloid 1-11 acetate(190436-05-6 free base)
<p>β-amyloid 1-11 acetate is a fragment of Amyloid-β peptide, maybe used in the research of neurological disease.</p>Fórmula:C58H80N16O24Pureza:>99.99%Forma y color:SolidPeso molecular:1385.37CI 75300
CAS:<p>CI 75300 targets the P2X purinoceptor 7 (human).</p>Fórmula:C21H20O6Pureza:99.07%Forma y color:SolidPeso molecular:368.38IMR-1
CAS:<p>IMR-1 is a novel class of Notch inhibitors targeting the transcriptional activation with IC50 of 6 μMol/L.</p>Fórmula:C15H15NO5S2Pureza:97.96% - 98.38%Forma y color:SolidPeso molecular:353.41Umeclidinium bromide
CAS:<p>Umeclidinium bromide (GSK573719A) is a novel mAChR antagonist.</p>Fórmula:C29H34BrNO2Pureza:98.4% - 99.89%Forma y color:SolidPeso molecular:508.49Ocinaplon
CAS:<p>Ocinaplon (DOV 273547) is a GABAA receptors modulator.</p>Fórmula:C17H11N5OPureza:99.81%Forma y color:SolidPeso molecular:301.3Ro 67-7476
CAS:<p>Ro 67-7476 is a positive allosteric modulator of mGlu1 receptors.</p>Fórmula:C17H18FNO2SPureza:99.69%Forma y color:SolidPeso molecular:319.39Kavain
CAS:<p>Kavain, a compound extracted from the Kava plant, Piper methysticum, is found to be involved in TNF-α expression in human and mouse cells via regulation of</p>Fórmula:C14H14O3Pureza:99.93% - ≥95%Forma y color:SolidPeso molecular:230.26Piboserod
CAS:<p>Piboserod (SB-207266) (SB 207266) is a selective 5-HT(4) receptor antagonist.</p>Fórmula:C22H31N3O2Pureza:97.21% - 99.49%Forma y color:SolidPeso molecular:369.54i
CAS:<p>4i (CHEMBL1269981) is a 5-HT3 receptor antagonist,It modulates the serotonergic system.</p>Fórmula:C16H12ClN3OPureza:99.49%Forma y color:SolidPeso molecular:297.74AZD-6280
CAS:<p>AZD6280 is a novel, subtype-selective GABAAα2/3 receptor positive modulators, used for treatment of generalized anxiety disorder.</p>Fórmula:C20H22N4O3Pureza:98.99%Forma y color:SolidPeso molecular:366.41PHCCC
CAS:<p>PHCCC is a Group I mGluR antagonist and enhances mGluR4 function; also blocks mGluR2/8.</p>Fórmula:C17H14N2O3Pureza:>99.99%Forma y color:SolidPeso molecular:294.3Ansofaxine hydrochloride
CAS:<p>Ansofaxine hydrochloride (LY03005) is a serotonin-norepinephrine-dopamine reuptake inhibitor (IC50s: 723, 763 and 491 nM, respectively).</p>Fórmula:C24H32ClNO3Pureza:99.57% - 99.77%Forma y color:SolidPeso molecular:417.97Farampator
CAS:<p>Farampator (CX-691) (CX-691;Org24448) is a positive modulator of AMPA receptor.</p>Fórmula:C12H13N3O2Pureza:99.84% - >99.99%Forma y color:SolidPeso molecular:231.25A 582941 HCl (848591-90-2(free base))
<p>A-582941 is a alpha7 neuronal nicotinic receptor agonist with broad spectrum cognition-enhancing properties</p>Fórmula:C17H21ClN4Pureza:99.83%Forma y color:SolidPeso molecular:316.83Firocoxib
CAS:<p>Firocoxib (ML 1785713) is a selective non-steroidal inhibitor of cycooxygenase-2 (COX-2) (IC50 of 0.13 μM), with anti-inflammatory for use in dogs and horses.</p>Fórmula:C17H20O5SPureza:99.84%Forma y color:SolidPeso molecular:336.4Loxapine
CAS:<p>Loxapine, a dibenzoxazepine antipsychotic, treats schizophrenia by blocking D2/D4 and serotonin receptors. Related to clozapine.</p>Fórmula:C18H18ClN3OPureza:99.88%Forma y color:Pale Yellowish Crystals From Petroleum Ether SolidPeso molecular:327.81α-Asarone
CAS:<p>alpha-Asarone (trans-Asarone) is a psychoactive compound with antidepressant-like activity in mice.</p>Fórmula:C12H16O3Pureza:99.64% - 99.64%Forma y color:Monoclinic Needles From Water Monoclinic Needles From WaterPeso molecular:208.25Donitriptan Mesylate
CAS:<p>Donitriptan Mesylate, a 5-HT1B/1D agonist, is used potentially for the treatment of migraines.</p>Fórmula:C24H29N5O5SForma y color:SolidPeso molecular:499.58Thiocolchicoside
CAS:<p>Thiocolchicoside, a muscle relaxant, has anti-inflammatory and analgesic properties; not for seizure-prone people.</p>Fórmula:C27H33NO10SPureza:99.11% - 99.39%Forma y color:SolidPeso molecular:563.62Coluracetam
CAS:<p>Coluracetam (MKC-231)(MKC-231) is a Choline Uptake Enhancer.</p>Fórmula:C19H23N3O3Pureza:99.96%Forma y color:SolidPeso molecular:341.4Dizocilpine Maleate
CAS:<p>Dizocilpine Maleate (MK 801) is a potent noncompetitive antagonist of the NMDA receptor with Kd of 37.2 nM in rat brain membranes.</p>Fórmula:C20H19NO4Pureza:99% - 99.96%Forma y color:White SolidPeso molecular:337.38Acephate
CAS:<p>Acephate (Orthene) is an anticholinesterase insecticide with a weak inhibitory effect on AChE in rats, but it can effectively inhibit AChE in cockroaches.</p>Fórmula:C4H10NO3PSPureza:≥98%Forma y color:Colorless Crystals Acephate Is A White Solid Used As A Contact And Systemic InsecticidePeso molecular:183.17SSD114 HCl
CAS:<p>SSD114 is a novel GABAB receptor positive allosteric modulator.</p>Fórmula:C18H21ClF3N3OPureza:99.03% - 99.95%Forma y color:SolidPeso molecular:387.832'MeO6MF
CAS:<p>2'MeO6MF is a brain-penetrant positive allosteric modulator at α2β1γ2L and all α1-containing GABAA receptors.It offers neuroprotection and improved functional</p>Fórmula:C17H14O3Pureza:99.28% - 99.63%Forma y color:SolidPeso molecular:266.29VU 0357121
CAS:<p>VU0357121, a positive allosteric modulator of mGlu5 (EC50: 33 nM), is inactive or very weakly antagonizing at other mGlu receptor subtypes.</p>Fórmula:C17H17F2NO2Pureza:99% - >99.99%Forma y color:SolidPeso molecular:305.32GSK2578215A
CAS:<p>GSK2578215A is a potent and selective LRRK2 kinase inhibitor.</p>Fórmula:C24H18FN3O2Pureza:99.57% - 99.94%Forma y color:SolidPeso molecular:399.42Pirenperone
CAS:<p>Pirenperone is a putative 5-HT2 receptor antagonist with the central antiserotonergic and antidopaminergic action.</p>Fórmula:C23H24FN3O2Pureza:99.2%Forma y color:SolidPeso molecular:393.45Norfluoxetine Hydrochloride
CAS:<p>Norfluoxetine Hydrochloride (Norfluoxetine HCl) is an active metabolite of fluoxetine. Fluoxetine is an antidepressant drug.</p>Fórmula:C16H17ClF3NOPureza:99.71%Forma y color:SolidPeso molecular:331.76VU10010
CAS:<p>VU10010 (VU 10010) is allosteric potentiator of M4 acetylcholine receptors.</p>Fórmula:C17H16ClN3OSPureza:99.36%Forma y color:SolidPeso molecular:345.85Oxotremorine sesquifumarate
CAS:<p>Oxotremorine sesquifumarate is a muscarinic agonist.</p>Fórmula:C12H18N2OC4H4O4Pureza:97.94%Forma y color:SolidPeso molecular:380.39MDL 100009
CAS:<p>MDL 100009, the S-enantiomer of MDL 100151 and the opposite enantiomer of MDL 100907, is a selective antagonist of 5-HT2A.</p>Fórmula:C22H28FNO3Pureza:98.96%Forma y color:SolidPeso molecular:373.46IC87201
CAS:<p>IC87201 is a nNOS-PDZ/PSD-95-PDZ inhibitor. IC87201 showed great promise in cellular experiments and animal models of ischemic stroke and pain.</p>Fórmula:C13H10Cl2N4OPureza:97.44%Forma y color:SolidPeso molecular:309.15Dinotefuran
CAS:<p>Dinotefuran (MTI-446), a neonicotinoid insecticide, targets pests by blocking their nervous system.</p>Fórmula:C7H14N4O3Pureza:99.89%Forma y color:White Crystalline PowderPeso molecular:202.21Sofpironium bromide
CAS:<p>Sofpironium bromide (BBI4000) belongs to a class of drugs called anticholinergics, which exert their effect by blocking the action of acetylcholine.</p>Fórmula:C22H32BrNO5Pureza:98.85%Forma y color:SolidPeso molecular:470.4SKF89976A hydrochloride
CAS:<p>SKF89976A hydrochloride (d,l-SKF89976A hydrochloride) is a selective inhibitor GABA transporter such as GAT-1 (IC50s = 0.28 μM), GAT-2 (IC50s = 137.34 μM) and</p>Fórmula:C22H26ClNO2Pureza:98.02%Forma y color:SolidPeso molecular:371.9PNU-282987 S enantiomer free base
CAS:<p>PNU-282987 S enantiomer free base is an agonist of α7 nicotinic acetylcholine receptor (α7 nAChR).</p>Fórmula:C14H17ClN2OPureza:99.74%Forma y color:SolidPeso molecular:264.75Autocamtide 2 TFA(129198-88-5 free base)
<p>Autocamtide 2 TFA, selective CaMKII peptide substrate, used in its activity assay.</p>Fórmula:C67H119F3N22O22Pureza:98%Forma y color:SolidPeso molecular:1641.79SB-200646
CAS:<p>SB-200646 is a selective and potent antagonist of 5-HT2B/5-HT2C receptor</p>Fórmula:C15H14N4OPureza:99.61%Forma y color:SolidPeso molecular:266.35-Benzyloxygramine
CAS:<p>5-Benzyloxygramine blocks the Dopamin receptors and antagonizes the effects of 5-HT on the rat uterus and the rabbit ear.</p>Fórmula:C18H20N2OPureza:99.13%Forma y color:SolidPeso molecular:280.36TBPB
CAS:<p>TBPB is an allosteric M1 mAChR agonist.</p>Fórmula:C25H32N4OPureza:97.87% - 99.9%Forma y color:SolidPeso molecular:404.55BPAM344
CAS:<p>BPAM344 is a potent positive allosteric modulator (PAM) of the KAR subunits GluK1b, GluK2a, and GluK3a.</p>Fórmula:C10H11FN2O2SPureza:99.53%Forma y color:SolidPeso molecular:242.27DNQX disodium salt
CAS:<p>DNQX disodium salt is a water-soluble form of selective antagonist of non-NMDA receptor</p>Fórmula:C8H2N4Na2O6Pureza:98.93%Forma y color:SolidPeso molecular:296.1Almotriptan
CAS:<p>Almotriptan (LAS 31416), a triptan and 5-HT1B/1D agonist, treats migraines by constricting cranial vessels and altering blood flow.</p>Fórmula:C17H25N3O2SPureza:99.85%Forma y color:Light Yellow Or White PowerPeso molecular:335.46Eslicarbazepine Acetate
CAS:<p>Eslicarbazepine Acetate (Zebinix) is an anticonvulsant medication approved for use as an adjunctive therapy for partial-onset seizures.</p>Fórmula:C17H16N2O3Pureza:99.58% - >99.99%Forma y color:White To Off-White SolidPeso molecular:296.32Metoclopramide
CAS:<p>Metoclopramide: dopamine D2 antagonist, treats nausea, vomiting, gastroparesis, GERD; safe for pregnancy.</p>Fórmula:C14H22ClN3O2Pureza:99.75%Forma y color:SolidPeso molecular:299.80Idalopirdine Hydrochloride
CAS:<p>Idalopirdine Hydrochloride (Lu AE58054 Hydrochloride) is an in-vivo binding affinity and effect, in-vitro selectivity and potency of 5-HT(6)R antagonist (Ki: 0.</p>Fórmula:C20H20ClF5N2OPureza:99.77%Forma y color:SolidPeso molecular:434.83TG6-10-1
CAS:<p>TG6-10-1 is an EP2 antagonist.</p>Fórmula:C23H23F3N2O4Pureza:99.66% - ≥95%Forma y color:SolidPeso molecular:448.43MCI-225
CAS:<p>MCI-225 is a selective inhibitor of NA reuptake with 5-HT3 receptor antagonism.</p>Fórmula:C17H17FN4SPureza:99.32%Forma y color:SolidPeso molecular:328.4Tasimelteon
CAS:<p>Tasimelteon (BMS-214778) is a melatonin receptor agonist that is used for the treatment of non-24 hour sleep-wake disorder in blind individuals.</p>Fórmula:C15H19NO2Pureza:98.93% - 99.93%Forma y color:SolidPeso molecular:245.32L-701324
CAS:<p>L-701324 is an NMDA receptor with high affinity and selectivity for the glycine site, used as an orally active and long-acting anticonvulsant.</p>Fórmula:C21H14ClNO3Pureza:98.63% - >99.99%Forma y color:SolidPeso molecular:363.79IPSU
CAS:<p>IPSU is an antagonist of OX2 receptor. IPSU Exhibits approximately six-fold selectivity for OX2 versus OX1 receptors.</p>Fórmula:C23H27N5O2Pureza:97.05%Forma y color:SolidPeso molecular:405.49Bromfenac Sodium
CAS:<p>Bromfenac Sodium (AHR 10282R) is a nonsteroidal anti-inflammatory drug (NSAID) and an orally available COX inhibitor, which has anti-inflammatory activity.</p>Fórmula:C15H11BrNO3·NaPureza:99.93%Forma y color:SolidPeso molecular:356.15NAN-190 hydrobromide
CAS:<p>NAN-190 hydrobromide is an antagonist of serotonin receptor 5-HT.</p>Fórmula:C23H28BrN3O3Pureza:95.20%Forma y color:SolidPeso molecular:474.39Medetomidine hydrochloride
CAS:<p>Medetomidine hydrochloride (MPV785) is a selective α2-adrenoceptor agonist, with Ki of 1.08 nM, exhibts 1620-fold selectivity over α1-adrenoceptor.</p>Fórmula:C13H16N2·HClPureza:99.96%Forma y color:White Or Off White Crystalline PowderPeso molecular:236.74JH-II-127
CAS:<p>JH-II-127 is an oral LRRK2 inhibitor with IC50s: 6.6 nM (WT), 2.2 nM (G2019S), 47.7 nM (A2016T).</p>Fórmula:C19H21ClN6O3Pureza:98.32%Forma y color:SolidPeso molecular:416.86KN-62
CAS:<p>KN-62 is a potent and specific Ca2+/calmodulin-dependent protein kinase II (CaMKII) inhibitor with Ki of 0.9 μM.</p>Fórmula:C38H35N5O6S2Pureza:99.80% - >99.99%Forma y color:White SolidPeso molecular:721.84Homocarnosine acetate
<p>Homocarnosine acetate is a dipeptide unique to brain consisting of γ-aminobutyric acid (GABA) and histidine.</p>Fórmula:C12H20N4O5Pureza:99.52%Forma y color:SolidPeso molecular:300.31GNE-9605
CAS:<p>GNE-9605 is a highly effective, specifical, and brain-penetrant LRRK2 inhibitor (IC50: 19 nM).</p>Fórmula:C17H20ClF4N7OPureza:98.55% - 98.75%Forma y color:SolidPeso molecular:449.83Vilazodone Hydrochloride
CAS:<p>Vilazodone Hydrochloride (EMD 68843) , a partial agonist of 5-HT1A receptors and specific serotonin reuptake inhibitor (SSRI), is utilized in treating of the</p>Fórmula:C26H27N5O2·HClPureza:99.56% - >99.99%Forma y color:SolidPeso molecular:477.99CZC-25146
CAS:<p>CZC-25146, a stable LRRK2 inhibitor, IC50: 4.76 nM (wild-type), 6.87 nM (G2019S).</p>Fórmula:C22H25FN6O4SPureza:97.68%Forma y color:SolidPeso molecular:488.54Tinoridine hydrochloride
CAS:<p>Tinoridine HCl is an NSAID that inhibits lipid peroxides and renin release, unlike indomethacin and corticosteroids.</p>Fórmula:C17H21ClN2O2SPureza:97.49%Forma y color:SolidPeso molecular:352.88A-484954
CAS:<p>A-484954 (A 484954) is a highly specific eukaryotic elongation factor-2 (eEF2, IC50: 280 nM) inhibitor.</p>Fórmula:C13H15N5O3Pureza:97.47% - 99.86%Forma y color:SolidPeso molecular:289.29Bicuculline
CAS:<p>Bicuculline, a plant-derived GABAA receptor antagonist, identified in 1932, reacts to light.</p>Fórmula:C20H17NO6Pureza:98% - 99.99%Forma y color:Light Yellow PowderPeso molecular:367.35RS-67333
CAS:<p>RS-67333 is a partial agonist of 5-HT4R with neuroprotective effects.</p>Fórmula:C19H29ClN2O2Pureza:99.24%Forma y color:SolidPeso molecular:352.9CL 218872
CAS:<p>CL 218872: selective α1 GABAA receptor agonist, anxiolytic, and anticonvulsant; Ki=130 nM for α1, less potent for α2-α6.</p>Fórmula:C13H9F3N4Pureza:99.92%Forma y color:SolidPeso molecular:278.231,1'-Methylenedi-2-naphthol
CAS:<p>1,1'-Methylenedi-2-naphthol target CYP2C19 - cytochrome P450 family 2 subfamily C member 19 (human).</p>Fórmula:C21H16O2Pureza:98.91%Forma y color:Light Pink To Light Brown Crystalline PowderPeso molecular:300.35(S)-UFR2709
CAS:<p>(S)-UFR2709, a nAChR competitive antagonist, favors α4β2 over α7, reduces anxiety and alcohol use in rats.</p>Fórmula:C13H17NO2Forma y color:SolidPeso molecular:219.284GSK163090
CAS:<p>GSK163090 is a specific and orally active 5-HT1A/B/D receptor antagonist (pKis: 9.4/8.5/9.7, and 6.3/6.7 for 5-HT1A/B/D, and dopamine D2/D3).</p>Fórmula:C25H29N5OPureza:99.2%Forma y color:SolidPeso molecular:415.53Solifenacin hydrochloride
CAS:<p>Solifenacin Hcl is a muscarinic receptor antagonist.</p>Fórmula:C23H27ClN2O2Pureza:98%Forma y color:SolidPeso molecular:398.93Rapastinel Trifluoroacetate
CAS:<p>Rapastinel Trifluoroacetate (GLYX-13 Trifluoroacetate) is an NMDA receptor modulator with glycine-site partial agonist properties.</p>Fórmula:C20H32F3N5O8Pureza:99.01% - 99.77%Forma y color:SolidPeso molecular:527.49Bestim
CAS:<p>Bestim is an immunomodulatory dipeptide that is synthetic.</p>Fórmula:C16H19N3O5Pureza:99.76%Forma y color:SolidPeso molecular:333.34Oxyphenonium bromide
CAS:<p>Oxyphenonium bromide is an anticholinergic used to study and treat ulcers and relieve visceral spasms.</p>Fórmula:C21H34BrNO3Pureza:98.96%Forma y color:SolidPeso molecular:428.404SB-203186 hydrochloride
CAS:<p>SB 203186 hydrochloride is a potent 5-HT4 receptor antagonist</p>Fórmula:C16H20N2O2·HClPureza:99.64%Forma y color:SolidPeso molecular:308.81Aripiprazole monohydrate
CAS:<p>Aripiprazole (OPC-14597) is a potent D2 partial agonist and inverse agonist of 5-HT2 receptors, used for schizophrenia and COVID-19 studies.</p>Fórmula:C23H29Cl2N3O3Forma y color:SolidPeso molecular:466.4Tandospirone hydrochloride
CAS:<p>Tandospirone (SM-3997) HCl: potent 5-HT1A partial agonist; Ki: 27 nM; anxiolytic, antidepressant, for CNS disorder research.</p>Fórmula:C21H30ClN5O2Forma y color:SolidPeso molecular:419.95Propiverine
CAS:<p>Propiverine reduces muscle spasms by limiting calcium influx, targeting bladder smooth muscles, aiding OAB research.</p>Fórmula:C23H29NO3Forma y color:SolidPeso molecular:367.48Tiprenolol
CAS:<p>Tiprenolol is a beta adrenergic receptor antagonist.[1]</p>Fórmula:C13H21NO2SPureza:99.43%Forma y color:SolidPeso molecular:255.38Clozapine HCl
CAS:<p>Clozapine HCl, an atypical antipsychotic, binds CNS receptors, targets 5-HT2A/2C, has weaker D2 antagonism. Risk: Agranulocytosis.</p>Fórmula:C18H20Cl2N4Forma y color:SolidPeso molecular:363.29VU0357017 hydrochloride
CAS:<p>VU0357017 hydrochloride (ML071 hydrochloride) is highly selective M1 agonists act at an allosteric site to activate the receptor (EC50: 477 ± 172 nM; Pec50: 6.</p>Fórmula:C18H28ClN3O3Pureza:99% - 99.97%Forma y color:SolidPeso molecular:369.89ADX-47273
CAS:<p>ADX-47273 (BA 94673139) is a positive and selective allosteric modulator for the metabotropic glutamate receptor subtype mGluR5(EC50=170 nM).</p>Fórmula:C20H17F2N3O2Pureza:97% - 99.18%Forma y color:SolidPeso molecular:369.36PHA 543613 hydrochloride
CAS:<p>PHA-543613 hydrochloride, a potent α7 nicotinic receptor agonist, may treat schizophrenia-related cognitive deficits.</p>Fórmula:C15H18ClN3O2Forma y color:SolidPeso molecular:307.78Quipazine
CAS:<p>Quipazine: 5-HT agonist, Ki 1.4 nM at 5-HT3R, anti-SARS-CoV-2 (EC50 31.64 μM), for neurological research.</p>Fórmula:C13H15N3Forma y color:SolidPeso molecular:213.28γ-secretase modulator 1 hydrochloride
CAS:<p>gamma-secretase inhibitior-1 is a gamma-secretase modulator that is useful to Alzheimer's disease [1].</p>Fórmula:C24H25ClN4OSPureza:98%Forma y color:SolidPeso molecular:453Vortioxetine
CAS:<p>Vortioxetine (Lu AA 21004) is a serotonergic antidepressant used for major depression disorders.</p>Fórmula:C18H22N2SPureza:99.34% - 99.34%Forma y color:SolidPeso molecular:298.45SAX-187 hydrochloride
CAS:<p>WAY-181187 is a potent, selective 5-HT6 agonist with high affinity (2.2-4.8 nM), and increases GABA in rat cortex at 3-30 mg/kg s.c.</p>Fórmula:C15H14Cl2N4O2S2Forma y color:SolidPeso molecular:417.33RU 24969 succinate
CAS:<p>RU 24969 succinate, a 5-HT receptor agonist, exhibits K i values of 0.38 nM for 5-HT 1B and 2.5 nM for 5-HT 1A, indicating its affinity towards these receptors. It reduces fluid consumption and enhances forward locomotion. This compound is utilized in neurological disease research.</p>Fórmula:C18H22N2O5Forma y color:SolidPeso molecular:346.38Acotiamide hydrochloride
CAS:<p>Acotiamide hydrochloride, an oral AChE inhibitor (IC50: 1.79 μM), boosts gastric movement and treats functional dyspepsia.</p>Fórmula:C21H31ClN4O5SForma y color:SolidPeso molecular:487.01Eltoprazine dihydrochloride
CAS:<p>Eltoprazine dihydrochloride, a drug developed for aggression, is now studied for L-DOPA-induced dyskinesia in Parkinson's.</p>Fórmula:C12H18Cl2N2O2Pureza:99.64%Forma y color:SolidPeso molecular:293.19Ginkgolide A
CAS:<p>Ginkgolide A (BN-52020), from Ginkgo biloba leaves, is an active PAF antagonist with potential in treating inflammation and immune disorders.</p>Fórmula:C20H24O9Pureza:98.76% - 99.81%Forma y color:White PowderPeso molecular:408.4Loxapine hydrochloride
CAS:<p>Loxapine hydrochloride, an oral anti-psychotic, inhibits dopamine and blocks 5-HT receptors.</p>Fórmula:C18H19Cl2N3OForma y color:SolidPeso molecular:364.27Propantheline
CAS:<p>Propantheline: oral muscarinic receptor blocker for smooth muscle issues, hyperhidrosis, and bladder control.</p>Fórmula:C23H30NO3Forma y color:SolidPeso molecular:368.49LY 2886721 Hydrochloride
CAS:<p>Potent, selective BACE inhibitor; IC50 of 10.2 nM (BACE2) & 20.3 nM (BACE1). >5000x selectivity vs. other proteases. Lowers Aβ & sAPPβ in Alzheimer's mice.</p>Fórmula:C18H17ClF2N4O2SForma y color:SolidPeso molecular:426.876-fluoro-DL-Tryptophan
CAS:<p>6-fluoro-DL-Tryptophan is an inhibitor of serotonin (5-HT) synthesis.</p>Fórmula:C11H11FN2O2Pureza:99.25%Forma y color:Off-White PowderPeso molecular:222.22SSR504734
CAS:<p>SSR504734 is a novel potent glycine transporter 1 (GlyT1) inhibitor.</p>Fórmula:C20H20ClF3N2OForma y color:SolidPeso molecular:396.83Cyclopiazonic acid
CAS:<p>Cyclopiazonic acid (CPA) is a neurotoxic secondary metabolite (SM) made by A.</p>Fórmula:C20H20N2O3Pureza:99.27% - 99.80%Forma y color:SolidPeso molecular:336.38Piboserod hydrochloride
CAS:<p>Piboserod HCl is a selective antagonist of 5-HT4 and muscarinic receptor.</p>Fórmula:C22H32ClN3O2Forma y color:SolidPeso molecular:405.96Niaprazine
CAS:<p>Niaprazine is a histamine H1-receptor antagonist with marked sedative properties.</p>Fórmula:C20H25FN4OPureza:99.56%Forma y color:SolidPeso molecular:356.44MPEP hydrochloride
CAS:<p>MPEP hydrochloride is an effective and highly specific non-competitive antagonist at the mGlu5 receptor subtype (IC50: 36 nM).</p>Fórmula:C14H12ClNPureza:99.87% - >99.99%Forma y color:SolidPeso molecular:229.7CRANAD 2
CAS:<p>CRANAD-2, a near-infrared probe, detects amyloid-beta in vivo, increasing fluorescence 70x and shifting blue 90 nm upon binding.</p>Fórmula:C23H25BF2N2O2Pureza:99.44%Forma y color:Dark Blue To Black PowderPeso molecular:410.27JI130
CAS:<p>JI130 hinders Hes1 transcription repression; notably shrinks pancreatic tumor volume in mice.</p>Fórmula:C23H24N2O3Pureza:99.61%Forma y color:SolidPeso molecular:376.45Alprenolol hydrochloride
CAS:<p>Alprenolol hydrochloride is a non-selective blocker of beta, and also is a antagonist of5-HT1A receptor.</p>Fórmula:C15H24ClNO2Pureza:99.79%Forma y color:SolidPeso molecular:285.81Paroxetine maleate
CAS:<p>Paroxetine maleate is a selective inhibitor of serotonin reuptake and an antidepressant.</p>Fórmula:C23H24FNO7Forma y color:SolidPeso molecular:445.443Spiperone hydrochloride
CAS:<p>5-HT2A serotonin and selective D2-like dopamine receptor antagonist</p>Fórmula:C23H27ClFN3O2Pureza:98%Forma y color:SolidPeso molecular:431.93PHA 568487
CAS:<p>PHA 568487: α-7 nAChR agonist, rapid brain uptake, lessens oxidative stress & neuroinflammation.</p>Fórmula:C20H24N2O7Forma y color:SolidPeso molecular:404.419Verubecestat TFA
CAS:<p>Verubecestat (MK-8931/SCH 900931), a potent BACE1 inhibitor, shows promise for Alzheimer's, cuts Aβ CSF levels by 92%.</p>Fórmula:C19H18F5N5O5SForma y color:SolidPeso molecular:523.435Ladostigil hydrochloride
CAS:<p>Ladostigil hydrochloride: oral dual cholinesterase and MAO-B/AChE inhibitor; IC50s: 37.1 & 31.8 μM; potential for depression and Alzheimer's research.</p>Fórmula:C16H21ClN2O2Forma y color:SolidPeso molecular:308.8LOX-IN-3 dihydrochloride monohydrate
CAS:<p>LOX-IN-3 dihydrochloride monohydrate is an oral lysyl oxidase inhibitor for research in fibrosis, cancer, and angiogenesis.</p>Fórmula:C13H17Cl2FN2O3SForma y color:SolidPeso molecular:371.25Sivopixant
CAS:<p>Sivopixant (S-600918), a potent P2X3 receptor antagonist, has a high analgesic effect (P2X3 IC50=4.2 nM, P2X2/3 IC50=1100 nM).</p>Fórmula:C25H22ClN5O5Pureza:99.34%Forma y color:SolidPeso molecular:507.93Rivanicline hemioxalate
<p>Rivanicline hemioxalate is a selective α4β2 nicotinic receptor agonist (K i =26 nM), over 1,000x preference to α7 (K i =3.6 μM), with limited side effects.</p>Fórmula:C12H16N2O4Pureza:98%Forma y color:SolidPeso molecular:207.23BRL-15572 hydrochloride
CAS:<p>BRL-15572 hydrochloride: selective h5-HT1D antagonist with high affinity; useful for studying h5-HT1D responses.</p>Fórmula:C25H28Cl2N2OForma y color:SolidPeso molecular:443.41Loreclezole hydrochloride
CAS:<p>Loreclezole hydrochloride is an antiepileptic, enhancing GABA A receptors with β2/β3 subunits.</p>Fórmula:C10H7Cl4N3Forma y color:SolidPeso molecular:310.99Volinanserin
CAS:<p>Volinanserin (MDL100907) is a potent 5-HT2 receptor antagonist with a Ki of 0.36 nM, 300x selective over 5-HT1c, alpha-1, and sigma receptors.</p>Fórmula:C22H28FNO3Pureza:98.94% - 99.95%Forma y color:SolidPeso molecular:373.46TA-03
CAS:<p>TA-03 (7-Meota) is a potent inhibitor of AChE in treatment of cognitive manifestation of AD.</p>Fórmula:C14H16N2OPureza:99.22%Forma y color:SolidPeso molecular:228.29ARC-239
CAS:<p>ARC-239 is an agonist of α2-adrenergic receptor.</p>Fórmula:C24H29N3O3Forma y color:SolidPeso molecular:407.51LP-922761 hydrate
<p>LP-922761 hydrate: selective AAK1 inhibitor; IC50: 4.8 nM (enzyme), 7.6 nM (cellular); also inhibits BIKE (IC50: 24 nM); inert to GAK, opioids, α2, GABAa.</p>Fórmula:C21H28N6O4Forma y color:SolidPeso molecular:414.98Isocorynoxeine
CAS:<p>Isocorynoxeine reduces blood pressure, dilates vessels, and guards neurons against ischemia and glutamate toxicity.</p>Fórmula:C22H26N2O4Pureza:98% - 99.9%Forma y color:SolidPeso molecular:382.45Tianeptine
CAS:<p>Tianeptine (Tianeptine sodium) 是一种选择性5-HT 摄取促进剂,具有抗抑郁、抗焦虑和神经保护作用,可用于缓解疼痛的研究。</p>Fórmula:C21H25ClN2O4SPureza:99.04%Forma y color:SolidPeso molecular:436.95Milnacipran
CAS:<p>Milnacipran, an SNRI with 85% bioavailability, treats fibromyalgia and is well absorbed orally.</p>Fórmula:C15H22N2OForma y color:SolidPeso molecular:246.35Pipequaline hydrochloride
CAS:<p>Pipequaline hydrochloride (PK-8165 hydrochloride) is an anticonflict & anticonvulsant quinoline derivative.</p>Fórmula:C22H25ClN2Pureza:99.46%Forma y color:SolidPeso molecular:352.9Quipazine maleate
CAS:<p>Quipazine maleate is a 5-HT agonist affecting L-02 hepatocytes and raphe neurons, causing smooth muscle contracture and bronchospasm.</p>Fórmula:C17H19N3O4Forma y color:SolidPeso molecular:329.36Tiagabine hydrochloride hydrate
CAS:<p>Tiagabine HCl hydrate, IC50: 67-446 nM, selectively inhibits GABA uptake, acts as an anticonvulsant.</p>Fórmula:C20H28ClNO3S2Forma y color:SolidPeso molecular:430.02Duloxetine
CAS:<p>Duloxetine is an inhibitor of serotonin-norepinephrine reuptake(Ki of 4.6 nM),with treatment of major depressive disorder and generalized anxiety disorder.</p>Fórmula:C18H19NOSPureza:99.71% - 99.89%Forma y color:SolidPeso molecular:297.41Ansofaxine
CAS:<p>Ansofaxine, an SNRI compound, is commonly utilized in depression research as a serotonin-norepinephrine reuptake inhibitor.</p>Fórmula:C24H31NO3Forma y color:SolidPeso molecular:381.516GNE-7915 tosylate
CAS:<p>GNE-7915 tosylate is a potent, selective, and brain-penetrant LRRK2 inhibitor, boasting an IC50 value of 9 nM.</p>Fórmula:C26H29F4N5O6SForma y color:SolidPeso molecular:615.6(S)-Amisulpride
CAS:<p>(S)-Amisulpride ((S) Amisulpride) (Esamisulpride) is a potent dopamine D2/D3 receptor antagonist.</p>Fórmula:C17H27N3O4SPureza:98.38%Forma y color:SolidPeso molecular:369.48TCN238
CAS:<p>TCN238 is an orally bioavailable positive allosteric modulator of the metabotropic glutamate receptor 4 (mGluR4with an EC50 of 1 μM).</p>Fórmula:C12H11N3Pureza:99.9% - 99.92%Forma y color:SolidPeso molecular:197.241-BCP
CAS:<p>1-BCP (Piperonylic acid piperidide) is a centrally active drug that modulates AMPA receptor gated currents.</p>Fórmula:C13H15NO3Pureza:99.60%Forma y color:SolidPeso molecular:233.26Piperazine
CAS:<p>Piperazine (1,4-Diazacyclohexane), a gamma-aminobutyric acid (GABA) agonist, serves as a crucial building block and core component in a wide range of marketed drugs known for their varied pharmacological activities.</p>Fórmula:C4H10N2Forma y color:SolidPeso molecular:86.14Ziprasidone mesylate
CAS:<p>Ziprasidone mesylate (CP-88059), an oral 5-HT & dopamine blocker, binds D2, 5-HT2A, 5-HT1A with Ki values: 4.8, 0.42, 3.4 nM.</p>Fórmula:C22H25ClN4O4S2Forma y color:SolidPeso molecular:509.04Aclidinium bromide
CAS:<p>Aclidinium bromide (LAS-W 330) is a synthetic anticholinergic agent that is used as an inhalant for treatment of acute bronchospasm due to chronic bronchitis.</p>Fórmula:C26H30NO4S2·BrPureza:99.53% - 99.69%Forma y color:SolidPeso molecular:564.55Prifinium bromide
CAS:<p>Prifinium bromide is a quaternary ammon antimuscarinic. It inhibits hyperkinesia of the digestive organs and urinary tract and has a spasmolytic action.</p>Fórmula:C22H28BrNPureza:97.99%Forma y color:SolidPeso molecular:386.37NPS ALX Compound 4a
CAS:<p>NPS ALX Compound 4a is a potent and selective antagonist of 5-HT6 receptor (IC50 of 7.2 nM)</p>Fórmula:C25H25N3O2SPureza:98%Forma y color:SolidPeso molecular:431.55S1RA hydrochloride
CAS:<p>S1RA hydrochloride (E-52862 hydrochloride) is an effective and specific sigma-1 receptor(σ1R, Ki: 17 nM) antagonist, and has good selectivity against σ2R (Ki ></p>Fórmula:C20H24ClN3O2Pureza:98% - 99.84%Forma y color:SolidPeso molecular:373.87Indomethacin heptyl ester
CAS:<p>Indomethacin heptyl ester is a non-selective inhibitor of both COX-1 and COX-2</p>Fórmula:C26H30ClNO4Pureza:99.86%Forma y color:SolidPeso molecular:455.97Clothianidin
CAS:<p>Clothianidin (TI 435), an insecticide, stimulates nAChR as acetylcholine agonist, not AChE inhibitor.</p>Fórmula:C6H8ClN5O2SPureza:99.71% - 99.87%Forma y color:Solid PowderPeso molecular:249.68Risperidone hydrochloride
CAS:<p>Risperidone hydrochloride blocks 5-HT2, inhibits P-glycoprotein, and antagonizes D2 receptors (Ki: 5-HT2A - 4.8 nM, D2 - 5.9 nM).</p>Fórmula:C23H28ClFN4O2Forma y color:SolidPeso molecular:446.95Cinanserin
CAS:<p>Cinanserin is a serotonin 5-HT2 antagonist.</p>Fórmula:C20H24N2OSForma y color:SolidPeso molecular:340.48Azeliragon HCl
CAS:<p>Azeliragon: potent oral RAGE inhibitor, blocks Alzheimer's-linked amyloid brain entry.</p>Fórmula:C32H40Cl3N3O2Forma y color:SolidPeso molecular:605.04Oxyphencyclimine
CAS:<p>Oxyphencyclimine is a muscarinic receptor antagonist (MRA) anticholinergic drug used to treat peptic ulcers.</p>Fórmula:C20H28N2O3Forma y color:SolidPeso molecular:344.45S 14506 HCl
CAS:<p>S 14506 HCl: Strong 5-HT1A agonist; pKi - 9.0 (5-HT1A), 6.6 (5-HT1B/C), <6.0 (5-HT3).</p>Fórmula:C24H26FN3O2Forma y color:SolidPeso molecular:407.48Teriflunomide impurity 3
CAS:<p>Teriflunomide impurity 3 (4-Amino-N-(4-trifluoromethylphenyl)benzamide) is a selective COX-1 inhibitor(IC50 of 30 μM).</p>Fórmula:C14H11F3N2OPureza:99.62%Forma y color:SolidPeso molecular:280.25Urapidil
CAS:<p>Urapidil (Ebrantil), a sympatholytic antihypertensive drug, acts as a 5-HT1A receptor agonist and as an α1-adrenoceptor antagonist.</p>Fórmula:C20H29N5O3Pureza:99.85% - >99.99%Forma y color:SolidPeso molecular:387.48Arecaidine hydrochloride
CAS:<p>Arecaidine hydrochloride may have carcinogenesis.</p>Fórmula:C7H12ClNO2Pureza:99.69% - ≥95%Forma y color:SolidPeso molecular:177.63Syn-Ake acetate
CAS:<p>Syn-Ake acetate (Dipeptide diaminobutyroyl benzylamide) is a muscarinic acetylcholine receptor antagonist.</p>Fórmula:C19H29N5O3·2(C2H4O2)Pureza:99.60%Forma y color:SolidPeso molecular:495.58CNQX
CAS:<p>CNQX (FG9065) is a competitive, non-NMDA glutamate receptor antagonist (IC50s = 0.3 and 1.5 μM for AMPA and kainate receptors, respectively)</p>Fórmula:C9H4N4O4Pureza:99.70%Forma y color:Pale Yellow SolidPeso molecular:232.15(-)-Securinine
CAS:<p>(-)-Securinine (Securinine) is plant-derived alkaloid and also a GABAA receptor antagonist.</p>Fórmula:C13H15NO2Pureza:99.58% - 99.87%Forma y color:SolidPeso molecular:217.26Edonerpic maleate
CAS:<p>Edonerpic maleate (T-817 maleate) is a neurotrophic agent which can inhibit amyloid-β peptides (Aβ).</p>Fórmula:C20H25NO6SPureza:98.24%Forma y color:SolidPeso molecular:407.48β-Amyloid (31-35)
CAS:<p>β-Amyloid (31-35) (β-Amyloid 31-35) is the shortest sequence of native Amyloid-β peptide.</p>Fórmula:C25H47N5O6SPureza:>99.99%Forma y color:SolidPeso molecular:545.74Benzetimide hydrochloride
CAS:<p>Benzetimide hydrochloride (R4929) is an antagonist of muscarinic acetylcholine receptor.treatment neuroleptic-induced parkinsonism.</p>Fórmula:C23H27ClN2O2Pureza:99.32%Forma y color:Off-White PowderPeso molecular:398.93QNZ46
CAS:<p>QNZ46 is a NR2C/NR2D-selective NMDA receptor non-competitive antagonist.</p>Fórmula:C24H17N3O6Pureza:99.65%Forma y color:SolidPeso molecular:443.41Edrophonium chloride
CAS:<p>Edrophonium chloride is an acetylcholinesterase (AChE) inhibitor that is known to prevent the breakdown of the neurotransmitter acetylcholine by binding</p>Fórmula:C10H16ClNOPureza:97.41%Forma y color:LiquidPeso molecular:201.69TCS 1102
CAS:<p>TCS 1102 is an effective, dual orexin receptor antagonist (Ki: 0.2/3 nM for OX2/1 receptors).</p>Fórmula:C27H26N4O2SPureza:99.35% - 99.52%Forma y color:SolidPeso molecular:470.59Methiothepin mesylate
CAS:<p>Methiothepin mesylate (Metitepine mesylate) is a potent and non-selective 5-HT2 receptor antagonist, used as an antipsychotic.</p>Fórmula:C21H28N2O3S3Pureza:98% - 99.92%Forma y color:SolidPeso molecular:452.65MTEP
CAS:<p>MTEP: potent, selective mGluR5 antagonist; IC50=5 nM, Ki=16 nM; may have antidepressant/anxiolytic effects; useful in Parkinson's research.</p>Fórmula:C11H8N2SForma y color:SolidPeso molecular:200.26Guvacine hydrochloride
CAS:<p>Guvacine hydrochloride is an inhibits of GABA uptake (IC50 : 10 μM)</p>Fórmula:C6H10ClNO2Pureza:98.42%Forma y color:SolidPeso molecular:163.602SC-560
CAS:<p>SC-560 is a member of the diaryl heterocycle class of cyclooxygenase (COX) inhibitors.</p>Fórmula:C17H12ClF3N2OPureza:99.97%Forma y color:SolidPeso molecular:352.74Rotundine
CAS:<p>Rotundine (Gindarine) (L-tetrahydropalmatine, L-THP) is a selective dopamine D1 receptor antagonist with IC50 of 166 nM.</p>Fórmula:C21H25NO4Pureza:99.8% - 99.91%Forma y color:Off-White SolidPeso molecular:355.43ML 10302
CAS:<p>ML 10302 is a potent 5-HT4 agonist with Ki of 1.07 nM, boosts bowel movement, and may aid in neurology research.</p>Fórmula:C15H21ClN2O3Forma y color:SolidPeso molecular:312.79

