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Neurociencia

Neurociencia

Los inhibidores en neurociencia son compuestos diseñados para modular la actividad de proteínas, enzimas o receptores específicos dentro del sistema nervioso. Estos inhibidores son cruciales para estudiar los mecanismos moleculares subyacentes a la función neuronal, la transmisión sináptica y las enfermedades neurodegenerativas. Al dirigirse a los receptores de neurotransmisores, canales iónicos y vías de señalización, los inhibidores en neurociencia ayudan en la exploración de la función cerebral y en el desarrollo de estrategias terapéuticas para trastornos neurológicos como el Alzheimer, Parkinson y la epilepsia. En CymitQuimica, ofrecemos una amplia gama de inhibidores de neurociencia de alta calidad para apoyar su investigación en neurobiología, neurofarmacología y ciencias cognitivas.

Subcategorías de "Neurociencia"

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Se han encontrado 5390 productos de "Neurociencia"

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  • Naftopidil dihydrochloride

    CAS:
    <p>Naftopidil dihydrochloride (KT-611 2HCl) is a selective 5-HT1A and α1-adrenergic receptor antagonist with IC50 of 0.1 μM and 0.2 μM, respectively.</p>
    Fórmula:C24H28N2O3·2HCl
    Pureza:99.76%
    Forma y color:White Solid
    Peso molecular:465.41
  • p-Hydroxybenzaldehyde

    CAS:
    1.
    Fórmula:C7H6O2
    Pureza:99.05% - 99.86%
    Forma y color:Solid
    Peso molecular:122.12
  • Tacrine hydrochloride (hydrate)

    CAS:
    <p>Tacrine hydrochloride hydrate (Tetrahydroaminacrine) is a cholinesterase inhibitor that crosses the blood-brain barrier.</p>
    Fórmula:C13H14N2·XHCl·XH2O
    Pureza:99.01% - 99.89%
    Forma y color:Solid
    Peso molecular:234.72
  • AMN082 free base

    CAS:
    <p>AMN082 free base is a metabotropic glutamate receptor 7 allosteric agonist.</p>
    Fórmula:C28H28N2
    Pureza:97.75% - 97.79%
    Forma y color:Solid
    Peso molecular:392.54
  • 4F 4PP oxalate

    CAS:
    <p>4F 4PP oxalate is a 5-HT2A antagonist.</p>
    Fórmula:C22H26FNO·C2H2O4
    Pureza:97.34%
    Forma y color:Solid
    Peso molecular:429.49
  • ARN2966

    CAS:
    <p>ARN2966 is an inhibitor of amyloid precursor protein (APP)and amyloid-β (Aβ) secretion.</p>
    Fórmula:C12H12N2O
    Pureza:99.52% - 99.86%
    Forma y color:Solid
    Peso molecular:200.24
  • AZD3839 free base

    CAS:
    <p>AZD3839 free base is a potent and selective BACE1 inhibitor with Ki of 26.1 nM, about 14-fold selectivity over BACE2. Phase 1.</p>
    Fórmula:C24H16F3N5
    Pureza:99.93% - 99.96%
    Forma y color:Solid
    Peso molecular:431.41
  • Ginsenoside Rc

    CAS:
    <p>Ginsenoside Rc (Panaxoside Rc) is one of the ginsenosides from Panax ginseng, inhibits the expression of TNF-α and IL-1β.</p>
    Fórmula:C53H90O22
    Pureza:98.83% - 99.56%
    Forma y color:White Powder
    Peso molecular:1079.27
  • ONO-8590580

    CAS:
    <p>ONO-8590580 (CS-2894) is a negative allosteric modulator of GABAA α5.</p>
    Fórmula:C21H21FN6
    Pureza:99.43%
    Forma y color:Solid
    Peso molecular:376.43
  • NAN-190 hydrobromide

    CAS:
    <p>NAN-190 hydrobromide is an antagonist of serotonin receptor 5-HT.</p>
    Fórmula:C23H28BrN3O3
    Pureza:95.20%
    Forma y color:Solid
    Peso molecular:474.39
  • SB-334867 free base

    CAS:
    <p>SB-334867 free base (SB334867A free base) is a selective orexin-1 (OX1) receptor antagonist.</p>
    Fórmula:C17H13N5O2
    Pureza:99.67% - >99.99%
    Forma y color:Solid
    Peso molecular:319.32
  • Homocarnosine acetate


    <p>Homocarnosine acetate is a dipeptide unique to brain consisting of γ-aminobutyric acid (GABA) and histidine.</p>
    Fórmula:C12H20N4O5
    Pureza:99.52%
    Forma y color:Solid
    Peso molecular:300.31
  • Eliprodil

    CAS:
    <p>Eliprodil (SL-820715), NR2B-NMDA receptor blocker (IC50: 1 uM), less potent on NR2A/NR2C (IC50&gt;100 uM), explored for Parkinson's and movement issues.</p>
    Fórmula:C20H23ClFNO
    Pureza:99.53% - 99.77%
    Forma y color:Solid
    Peso molecular:347.85
  • GNE-7915

    CAS:
    <p>GNE-7915 is a highly potent, selective and brain-penetrable leucine-rich repeat kinase 2 (LRRK2) inhibitor.</p>
    Fórmula:C19H21F4N5O3
    Pureza:98% - ≥95%
    Forma y color:Solid
    Peso molecular:443.4
  • MK-0752

    CAS:
    <p>MK-0752, a γ-secretase inhibitor, reduces Aβ40 production(IC50=5 nM).</p>
    Fórmula:C21H21ClF2O4S
    Pureza:98% - 99.55%
    Forma y color:Solid
    Peso molecular:442.9
  • JHU37160

    CAS:
    JHU37160 is a DREADD agonist with Ki of 1.9 nM for hM3Dq, 3.6 nM for hM4Di, and EC50 of 18.5 nM (hM3Dq), 0.2 nM (hM4Di) in HEK-293 cell assays.
    Fórmula:C19H20ClFN4
    Pureza:99.87%
    Forma y color:Solid
    Peso molecular:358.84
  • CZC-25146

    CAS:
    <p>CZC-25146, a stable LRRK2 inhibitor, IC50: 4.76 nM (wild-type), 6.87 nM (G2019S).</p>
    Fórmula:C22H25FN6O4S
    Pureza:97.68%
    Forma y color:Solid
    Peso molecular:488.54
  • Imidafenacin

    CAS:
    <p>Imidafenacin (KRP-197)(KRP-197; ONO-8025) is a potent and selective inhibitor of M3 receptors with Kb of 0.317 nM.</p>
    Fórmula:C20H21N3O
    Pureza:99.17%
    Forma y color:Solid
    Peso molecular:319.4
  • Indophagolin

    CAS:
    <p>Indophagolin: autophagy inhibitor, IC50 140 nM; blocks P2X4, P2X1, P2X3 receptors, IC50s 2.71, 2.40, 3.49 μM.</p>
    Fórmula:C19H15BrClF3N2O3S
    Pureza:99.76%
    Forma y color:Solid
    Peso molecular:523.75
  • Eltoprazine hydrochloride

    CAS:
    <p>Eltoprazine hydrochloride (DU 28853 hydrochloride) is a partial agonist at serotonin 5-HT1A, 5-HT1B, and 5-HT2B receptors (Ki value of 40, 52, and 81 nM,</p>
    Fórmula:C12H17ClN2O2
    Pureza:99.35%
    Forma y color:Solid
    Peso molecular:256.73
  • VU-1545

    CAS:
    <p>VU-1545 is mGlu5 positive allosteric modulator.</p>
    Fórmula:C22H15FN4O3
    Pureza:98.8%
    Forma y color:Solid
    Peso molecular:402.38
  • PE859

    CAS:
    <p>PE859 is a potent inhibitor of both tau and Aβ aggregation.</p>
    Fórmula:C28H24N4O2
    Pureza:98.8% - 99.09%
    Forma y color:Solid
    Peso molecular:448.52
  • Loreclezole

    CAS:
    <p>Loreclezole is a selective GABAA receptor modulator and acts as a positive allosteric modulator of β2 or β3-subunit-containing receptors.</p>
    Fórmula:C10H6Cl3N3
    Pureza:99.78%
    Forma y color:Solid
    Peso molecular:274.53
  • MK-1064

    CAS:
    <p>MK-1064 (Urokinase inhibitor 1) is a selective orexin 2 receptor antagonist (2-SORA).</p>
    Fórmula:C24H20ClN5O3
    Pureza:99.19% - 99.82%
    Forma y color:Solid
    Peso molecular:461.9
  • Azaphen dihydrochloride monohydrate

    CAS:
    <p>Azaphen dihydrochloride monohydrate is a 5-hydroxytryptamine reabsorption inhibitor with antidepressant activity and can be used to study neurological diseases.</p>
    Fórmula:C16H23Cl2N5O2
    Pureza:99.85%
    Forma y color:Solid
    Peso molecular:388.29
  • RS-67333

    CAS:
    <p>RS-67333 is a partial agonist of 5-HT4R with neuroprotective effects.</p>
    Fórmula:C19H29ClN2O2
    Pureza:99.24%
    Forma y color:Solid
    Peso molecular:352.9
  • Isocorynoxeine

    CAS:
    <p>Isocorynoxeine reduces blood pressure, dilates vessels, and guards neurons against ischemia and glutamate toxicity.</p>
    Fórmula:C22H26N2O4
    Pureza:98% - 99.9%
    Forma y color:Solid
    Peso molecular:382.45
  • Milnacipran

    CAS:
    <p>Milnacipran, an SNRI with 85% bioavailability, treats fibromyalgia and is well absorbed orally.</p>
    Fórmula:C15H22N2O
    Forma y color:Solid
    Peso molecular:246.35
  • Pipequaline hydrochloride

    CAS:
    <p>Pipequaline hydrochloride (PK-8165 hydrochloride) is an anticonflict &amp; anticonvulsant quinoline derivative.</p>
    Fórmula:C22H25ClN2
    Pureza:99.46%
    Forma y color:Solid
    Peso molecular:352.9
  • Prifinium bromide

    CAS:
    <p>Prifinium bromide is a quaternary ammon antimuscarinic. It inhibits hyperkinesia of the digestive organs and urinary tract and has a spasmolytic action.</p>
    Fórmula:C22H28BrN
    Pureza:97.99%
    Forma y color:Solid
    Peso molecular:386.37
  • Teriflunomide impurity 3

    CAS:
    <p>Teriflunomide impurity 3 (4-Amino-N-(4-trifluoromethylphenyl)benzamide) is a selective COX-1 inhibitor(IC50 of 30 μM).</p>
    Fórmula:C14H11F3N2O
    Pureza:99.62%
    Forma y color:Solid
    Peso molecular:280.25
  • Ziprasidone mesylate

    CAS:
    <p>Ziprasidone mesylate (CP-88059), an oral 5-HT &amp; dopamine blocker, binds D2, 5-HT2A, 5-HT1A with Ki values: 4.8, 0.42, 3.4 nM.</p>
    Fórmula:C22H25ClN4O4S2
    Forma y color:Solid
    Peso molecular:509.04
  • Dolasetron Mesylate hydrate

    CAS:
    <p>Dolasetron Mesylate hydrate blocks 5HT3 to prevent chemo and radiotherapy nausea.</p>
    Fórmula:C20H26N2O7S
    Pureza:99.86% - 99.9%
    Forma y color:Solid
    Peso molecular:438.49
  • Frentizole

    CAS:
    <p>Frentizole, an immunosuppressive agent, is an inhibitor of the Aβ-ABAD interaction</p>
    Fórmula:C15H13N3O2S
    Pureza:99.82%
    Forma y color:Solid
    Peso molecular:299.35
  • SB 242084

    CAS:
    <p>SB 242084 dihydrochloride hydrate is a psychoactive drug and research chemical which acts as a selective antagonist for the 5HT2C receptor.</p>
    Fórmula:C21H19ClN4O2
    Pureza:99.75% - ≥98%
    Forma y color:Solid
    Peso molecular:394.85
  • MK-3697

    CAS:
    <p>MK-3697, an isonicotinamide small molecule, acts as a potent and selective Orexin 2 receptor antagonist (Ki: 0.95 nM).</p>
    Fórmula:C23H21N5O3S
    Pureza:97.69% - 98.15%
    Forma y color:Solid
    Peso molecular:447.51
  • (S)-Amisulpride

    CAS:
    <p>(S)-Amisulpride ((S) Amisulpride) (Esamisulpride) is a potent dopamine D2/D3 receptor antagonist.</p>
    Fórmula:C17H27N3O4S
    Pureza:98.38%
    Forma y color:Solid
    Peso molecular:369.48
  • A-582941 dihydrochloride

    CAS:
    <p>A-582941 dihydrochloride (A 582941) is a Selective agonist of α7 nAChR partial</p>
    Fórmula:C17H22Cl2N4
    Pureza:99.55%
    Forma y color:Solid
    Peso molecular:353.29
  • Suritozole

    CAS:
    <p>Suritozole (MDL-26479) is a negative modulator at the gamma-aminobutyric acidA (GABAA) receptor</p>
    Fórmula:C10H10FN3S
    Pureza:99.25%
    Forma y color:Solid
    Peso molecular:223.27
  • Cerlapirdine

    CAS:
    <p>Cerlapirdine (PF-05212365), a 5-HT6 receptor antagonist, is in trials for Alzheimer's and schizophrenia cognition issues.</p>
    Fórmula:C22H23N3O3S
    Pureza:98.77%
    Forma y color:Solid
    Peso molecular:409.5
  • Pipamperone HCl

    CAS:
    <p>Pipamperone blocks 5-HT2A/B/C, D2/D3/D4, α1/α2 receptors; favors 5-HT2A/D4 over D2; negligible affinity for H1, mACh. Highly selective at low doses.</p>
    Fórmula:C21H31ClFN3O2
    Forma y color:Solid
    Peso molecular:411.95
  • Vilazodone Hydrochloride

    CAS:
    <p>Vilazodone Hydrochloride (EMD 68843) , a partial agonist of 5-HT1A receptors and specific serotonin reuptake inhibitor (SSRI), is utilized in treating of the</p>
    Fórmula:C26H27N5O2·HCl
    Pureza:99.56% - >99.99%
    Forma y color:Solid
    Peso molecular:477.99
  • RO4929097

    CAS:
    <p>RO4929097 (RG-4733), a γ secretase inhibitor (IC50: 4 nM), inhibits cellular processing of Aβ40 and Notch (EC50: 14/5 nM).</p>
    Fórmula:C22H20F5N3O3
    Pureza:98.5% - 99.51%
    Forma y color:Solid
    Peso molecular:469.4
  • CNQX disodium

    CAS:
    <p>CNQX disodium is a competitive non-NMDA receptor antagonist and competitive AMPA/kainate receptor antagonist in neuronal cultures.</p>
    Fórmula:C9H2N4Na2O4
    Pureza:97.77%
    Forma y color:Solid
    Peso molecular:276.12
  • A-804598

    CAS:
    <p>A-804598 is a competitive and selective P2X7 receptor antagonist (IC50: 10 nM, rat; 9 nM, mouse; 11 nM, human).</p>
    Fórmula:C19H17N5
    Pureza:99.57%
    Forma y color:Solid
    Peso molecular:315.37
  • Tianeptine sodium salt

    CAS:
    <p>Tianeptine sodium salt 是一种选择性5-HT 摄取促进剂,具有抗抑郁、抗焦虑和神经保护作用,可用于缓解疼痛的研究。</p>
    Fórmula:C21H24ClN2NaO4S
    Pureza:99.82%
    Forma y color:Solid
    Peso molecular:458.93
  • Xaliproden hydrochloride

    CAS:
    <p>Xaliproden is a compound that mimics the effects of nerve growth factor and is also a serotonin 5-HT1A receptor agonist.</p>
    Fórmula:C24H23ClF3N
    Pureza:99.99%
    Forma y color:Solid
    Peso molecular:417.89
  • (RS)-3-Hydroxyphenylglycine

    CAS:
    <p>(RS)-3-Hydroxyphenylglycine is a PI-linked metabotropic glutamate receptors agonist.</p>
    Fórmula:C8H9NO3
    Pureza:99.29%
    Forma y color:Solid
    Peso molecular:167.16
  • SQ22536

    CAS:
    <p>SQ22536, a tetrahydrofuryl adenosine analogue, inhibits adenylate cyclase in catfish and rat hepatocytes non-competitively.</p>
    Fórmula:C9H11N5O
    Pureza:99.18%
    Forma y color:Off-White Solid
    Peso molecular:205.22
  • Mosapride

    CAS:
    <p>Mosapride (AS-4370) is a selective 5HT4 agonist</p>
    Fórmula:C21H25ClFN3O3
    Pureza:99.56%
    Forma y color:White To Off-White Crystalline Solid
    Peso molecular:421.89