
Neurociencia
Los inhibidores en neurociencia son compuestos diseñados para modular la actividad de proteínas, enzimas o receptores específicos dentro del sistema nervioso. Estos inhibidores son cruciales para estudiar los mecanismos moleculares subyacentes a la función neuronal, la transmisión sináptica y las enfermedades neurodegenerativas. Al dirigirse a los receptores de neurotransmisores, canales iónicos y vías de señalización, los inhibidores en neurociencia ayudan en la exploración de la función cerebral y en el desarrollo de estrategias terapéuticas para trastornos neurológicos como el Alzheimer, Parkinson y la epilepsia. En CymitQuimica, ofrecemos una amplia gama de inhibidores de neurociencia de alta calidad para apoyar su investigación en neurobiología, neurofarmacología y ciencias cognitivas.
Subcategorías de "Neurociencia"
- Receptor 5-HT(942 productos)
- ACK(1 productos)
- AChR(575 productos)
- ATP Citrato Liasa(16 productos)
- Receptor adrenérgico(2.948 productos)
- BACE(36 productos)
- Beta amiloide(205 productos)
- CAMK(69 productos)
- Inhibidores de ciclooxigenasa (COX)(565 productos)
- Receptor de dopamina(409 productos)
- Receptor GABA(336 productos)
- Gamma-secretasa(59 productos)
- GluR(255 productos)
- GlyT(24 productos)
- Receptor de histamina(359 productos)
- LRRK2(33 productos)
- Receptor de melatonina(24 productos)
- NMDAR(27 productos)
- Receptor de OX(40 productos)
- Receptor de opioides(298 productos)
Mostrar 12 subcategorías más
Se han encontrado 5390 productos de "Neurociencia"
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A 582941 HCl (848591-90-2(free base))
<p>A-582941 is a alpha7 neuronal nicotinic receptor agonist with broad spectrum cognition-enhancing properties</p>Fórmula:C17H21ClN4Pureza:99.83%Forma y color:SolidPeso molecular:316.83Imidazenil
CAS:<p>Imidazenil is an modulator of GABA-A that blocks the sedative effects without lowering the convulsion threshold.</p>Fórmula:C18H12BrFN4OPureza:98.4%Forma y color:SolidPeso molecular:399.22Lurasidone hydrochloride
CAS:Lurasidone HCl: Atypical antipsychotic, treats schizophrenia & bipolar, affects dopamine, serotonin & adrenergic receptors.Fórmula:C28H36N4O2S·HClPureza:99.51%Forma y color:SolidPeso molecular:529.14RO-3
CAS:<p>RO3 is a selective antagonist of homomeric P2X3 and heteromeric P2X2/3 receptor</p>Fórmula:C16H22N4O2Pureza:99.63%Forma y color:SolidPeso molecular:302.37XAP044
CAS:<p>XAP044 blocks mGlu7, inhibiting long-term potentiation in mouse brain with a half-maximal effect at 88nm.</p>Fórmula:C15H9IO4Pureza:97.41%Forma y color:SolidPeso molecular:380.13Brexpiprazole
CAS:<p>Brexpiprazole (OPC-34712) is a partial agonist of human 5-hydroxytryptamine (5-HT) 5-HT1A and dopamine D2 receptors.</p>Fórmula:C25H27N3O2SPureza:99.06% - 99.96%Forma y color:SolidPeso molecular:433.57Melitracen
CAS:<p>Melitracen is a tricyclic antidepressant.</p>Fórmula:C21H25NForma y color:SolidPeso molecular:291.43MDL 72527
CAS:<p>MDL 72527 (N1,N4-Di(buta-2,3-dien-1-yl)butane-1,4-diamine dihydrochloride) is a polyamine oxidase (POA) inhibitor</p>Fórmula:C12H22Cl2N2Pureza:98.98%Forma y color:SolidPeso molecular:265.22Cromoglicic acid
CAS:<p>Cromoglicic acid prevents the release of inflammatory chemicals such as histamine from mast cells.</p>Fórmula:C23H16O11Pureza:99.55% - >99.99%Forma y color:Colorless Crystals From Ethanol + Ether Physical Description Solid (Ntp 1992)Peso molecular:468.37Tiagabine hydrochloride
CAS:<p>Tiagabine hydrochloride, a nipecotic acid derivative, is an anticonvulsant and selective GABA reuptake inhibitor.</p>Fórmula:C20H25NO2S2·HClPureza:99.09% - 99.77%Forma y color:White To Off-White SolidPeso molecular:412.01LRRK2-IN-1
CAS:<p>LRRK2-IN-1 is an effective and selective LRRK2 inhibitor.</p>Fórmula:C31H38N8O3Pureza:98% - 98.82%Forma y color:SolidPeso molecular:570.69Encenicline
CAS:<p>Encenicline (EVP-6124), a selective α7 nAChRs agonist, targets cognitive impairment in schizophrenia and Alzheimer's.</p>Fórmula:C16H17ClN2OSPureza:99.20%Forma y color:SolidPeso molecular:320.842'MeO6MF
CAS:<p>2'MeO6MF is a brain-penetrant positive allosteric modulator at α2β1γ2L and all α1-containing GABAA receptors.It offers neuroprotection and improved functional</p>Fórmula:C17H14O3Pureza:99.28% - 99.63%Forma y color:SolidPeso molecular:266.29BRL 54443
CAS:<p>BRL 54443 is a potent 5-HT1E/1F receptor agonist (pKi values are 8.7 and 8.9 respectively).</p>Fórmula:C14H18N2OPureza:98.07%Forma y color:SolidPeso molecular:230.31VU0155041
CAS:<p>VU0155041 is an effective and positive allosteric modulator/allosteric agonist at mGlu4 receptors (EC50: 798/693 nM, at human/rat).</p>Fórmula:C14H15Cl2NO3Pureza:99.52% - 99.56%Forma y color:SolidPeso molecular:316.18Isopropamide Iodide
CAS:<p>Isopropamide iodide: long-acting anticholinergic, treats peptic ulcers, GI disorders, Alzheimer's.</p>Fórmula:C23H33IN2OPureza:99.67%Forma y color:SolidPeso molecular:480.43ML380
CAS:<p>ML380 is a highly potent and the first CNS penetrant M5 positive allosteric modulator (PAM).</p>Fórmula:C23H25F3N4O3SPureza:99.69%Forma y color:SolidPeso molecular:494.53α-Conotoxin PIA acetate
α-Conotoxin PIA acetate is an antagonist of nicotinic acetylcholine receptor (nAChR) mainly targeting α6 and α3 subunits.Pureza:98%Forma y color:LiquidPeso molecular:N/APirenperone
CAS:<p>Pirenperone is a putative 5-HT2 receptor antagonist with the central antiserotonergic and antidopaminergic action.</p>Fórmula:C23H24FN3O2Pureza:99.2%Forma y color:SolidPeso molecular:393.45Buclizine dihydrochloride
CAS:<p>Buclizine dihydrochloride (Buclina) is the hydrochloride salt form of buclizine, a piperazine histamine H1 receptor antagonist with primarily antiemetic and</p>Fórmula:C28H33ClN2·2HClPureza:98.05%Forma y color:Off-White PowderPeso molecular:505.95FPS-ZM1
CAS:<p>FPS-ZM1 is a high-affinity RAGE specific inhibitor that blocks Aβ binding to the V domain of RAGE.</p>Fórmula:C20H22ClNOPureza:99.32% - 99.52%Forma y color:SolidPeso molecular:327.85RU 24969 free base
CAS:<p>RU 24969 (5-methoxy-3-(1,2,3,6-tetrahydropyridin-4-yl)-1H-indole) is a selective agonist of 5-HT1A and 5-HT1B receptors.</p>Fórmula:C14H16N2OPureza:97.38%Forma y color:SolidPeso molecular:228.29NMDAR antagonist 1
CAS:<p>NMDAR antagonist 1 is an orally active, NR2B-selective NMDAR antagonist.</p>Fórmula:C20H20BrN3O2Pureza:98%Forma y color:SolidPeso molecular:414.3Escitalopram Oxalate
CAS:<p>Escitalopram Oxalate ((S)-(+)Citalopram oxalate) is a selective serotonin (5-HT) reuptake inhibitor (SSRI) with Ki of 0.89 nM.</p>Fórmula:C22H23FN2O5Pureza:97.39% - 99.73%Forma y color:White SolidPeso molecular:414.43SKF89976A hydrochloride
CAS:<p>SKF89976A hydrochloride (d,l-SKF89976A hydrochloride) is a selective inhibitor GABA transporter such as GAT-1 (IC50s = 0.28 μM), GAT-2 (IC50s = 137.34 μM) and</p>Fórmula:C22H26ClNO2Pureza:98.02%Forma y color:SolidPeso molecular:371.9Miltirone
CAS:<p>Miltirone is a CYPs inhibitor, it has been characterized as a low-affinity ligand for central benzodiazepine receptors.</p>Fórmula:C19H22O2Pureza:99.22% - 99.66%Forma y color:SolidPeso molecular:282.38PNU-282987 S enantiomer free base
CAS:<p>PNU-282987 S enantiomer free base is an agonist of α7 nicotinic acetylcholine receptor (α7 nAChR).</p>Fórmula:C14H17ClN2OPureza:99.74%Forma y color:SolidPeso molecular:264.75Autocamtide 2 TFA(129198-88-5 free base)
<p>Autocamtide 2 TFA, selective CaMKII peptide substrate, used in its activity assay.</p>Fórmula:C67H119F3N22O22Pureza:98%Forma y color:SolidPeso molecular:1641.79Prucalopride Succinate
CAS:Prucalopride Succinate is a 5-HT4 receptor agonist with Ki 2.5 nM (5-HT4a) and 8 nM (5-HT4b).Fórmula:C18H26ClN3O3·C4H6O4Pureza:99.24%Forma y color:SolidPeso molecular:485.96AC-90179 HCl
CAS:<p>AC-90179 HCl: selective 5-HT2A inverse agonist, atypical antipsychotic, reduces hallucinogen-induced vasoconstriction.</p>Fórmula:C23H31ClN2O2Pureza:99.71%Forma y color:SolidPeso molecular:402.96CFMTI
CAS:<p>CFMTI: potent mGluR1 allosteric antagonist, 2000x selectivity over mGluR5, IC50: 2.6 nM.</p>Fórmula:C19H16FN5OPureza:97.23%Forma y color:SolidPeso molecular:349.36Tariquidar
CAS:<p>Tariquidar (XR9576)(Kd=5.1 nM) is a specific and effective non-competitive inhibitor of P-glycoprotein. It can reverse drug resistance in MDR cell Lines.</p>Fórmula:C38H38N4O6Pureza:98.07% - 99.45%Forma y color:SolidPeso molecular:646.73Lurasidone
CAS:<p>Lurasidone (SM-13496) is an antagonist of both dopamine D2 and 5-HT7(IC50=1.68 and 0.495 nM, respectively).It also a partial agonist of 5-HT1A receptor(IC50 : 6</p>Fórmula:C28H36N4O2SPureza:99.78% - 99.91%Forma y color:SolidPeso molecular:492.68NS9283
CAS:<p>NS9283, a positive allosteric modulator selective for the α4β2 form, reduces ethanol consumption.</p>Fórmula:C14H8N4OPureza:99.12%Forma y color:SolidPeso molecular:248.24CGP52432
CAS:<p>CGP52432 is a very potent antagonist of GABAB receptors (IC50 = 85 nM).</p>Fórmula:C15H24Cl2NO4PPureza:98.75%Forma y color:SolidPeso molecular:384.24Dasotraline hydrochloride
CAS:Dasotraline hydrochloride, a dopamine, norepinephrine, and serotonin reuptake inhibitor with IC50s: 4, 6, 11 nM.Fórmula:C16H16Cl3NPureza:98.92% - 99.6%Forma y color:SolidPeso molecular:328.66Gefapixant
CAS:<p>Gefapixant (AF219) is a P2X3 receptor (P2X3R) antagonist with IC50 of ~30 nM at recombinant hP2X3 homotrimers and 100-250 nM at hP2X2/3 heterotrimeric receptors</p>Fórmula:C14H19N5O4SPureza:99.28% - 99.50%Forma y color:SolidPeso molecular:353.4BPAM344
CAS:BPAM344 is a potent positive allosteric modulator (PAM) of the KAR subunits GluK1b, GluK2a, and GluK3a.Fórmula:C10H11FN2O2SPureza:99.53%Forma y color:SolidPeso molecular:242.27VU0467154
CAS:<p>VU0467154 is a positive allosteric modulator of the M4 muscarinic acetylcholine receptor.</p>Fórmula:C17H15F3N4O3S2Pureza:98.28% - 99.51%Forma y color:SolidPeso molecular:444.45Succinylcholine Chloride Dihydrate
CAS:<p>Succinylcholine Chloride Dihydrate (Succinyldicholine dichloride) is a nicotinic AChR agonist and also acts as a depolarizing neuromuscular blocker.</p>Fórmula:C14H30N2O4·2Cl·2H2OPureza:99.87%Forma y color:White SolidPeso molecular:397.34PU02
CAS:<p>PU02 (6-[(1-Naphthalenylmethyl)thio]-9H-purine) is a potent and selective antagonist of 5-HT3 receptor.</p>Fórmula:C16H12N4SPureza:99.35%Forma y color:SolidPeso molecular:292.36Rizatriptan benzoate
CAS:<p>Rizatriptan benzoate (MK-462 Benzoate) selectively binds to and activates serotonin (5-HT) 1B receptors and 5-HT 1D receptors providing relief of migraine</p>Fórmula:C22H25N5O2Pureza:99% - 99.79%Forma y color:White To Off-White Crystalline PowderPeso molecular:391.47LP-211
CAS:<p>LP-211 is a brain penetrant selective agonist for a 5-HT7 receptor (Ki: 0.58 nM), and >300-fold selectivity over the 5-HT1A receptor.</p>Fórmula:C30H34N4OPureza:98.65%Forma y color:SolidPeso molecular:466.62Harmine
CAS:<p>Harmine (Telepathine) is an alkaloid isolated from seeds of Peganum harmala.</p>Fórmula:C13H12N2OPureza:98.29% - 99.92%Forma y color:Off-White SolidPeso molecular:212.25Idalopirdine Hydrochloride
CAS:<p>Idalopirdine Hydrochloride (Lu AE58054 Hydrochloride) is an in-vivo binding affinity and effect, in-vitro selectivity and potency of 5-HT(6)R antagonist (Ki: 0.</p>Fórmula:C20H20ClF5N2OPureza:99.77%Forma y color:SolidPeso molecular:434.83Puerarin
CAS:<p>Puerarin (Kakonein), also known as Kakonein, is a member of the class of compounds known as isoflavonoid C-glycosides. It is a 5-HT2C receptor antagonist.</p>Fórmula:C21H20O9Pureza:98.90% - 99.21%Forma y color:Yellow Brown Fine PowderPeso molecular:416.38MCI-225
CAS:<p>MCI-225 is a selective inhibitor of NA reuptake with 5-HT3 receptor antagonism.</p>Fórmula:C17H17FN4SPureza:99.32%Forma y color:SolidPeso molecular:328.4NS3861
CAS:<p>NS3861 is a selective agonist for α3β4/α4β2 nAChRs, preferring β-subunits, with no effect on α4-based receptors.</p>Fórmula:C12H14BrNSPureza:99.853%Forma y color:SolidPeso molecular:284.224F 4PP oxalate
CAS:<p>4F 4PP oxalate is a 5-HT2A antagonist.</p>Fórmula:C22H26FNO·C2H2O4Pureza:97.34%Forma y color:SolidPeso molecular:429.49Melatonin
CAS:<p>Melatonin (Melatonine) is a natural hormone that activates melatonin receptors. Melatonin regulates the biological clock. Cost-effective and quality-assured.</p>Fórmula:C13H16N2O2Pureza:98% - 99.89%Forma y color:Pale Yellow Leaflets From Benzene SolidPeso molecular:232.28
