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Neurociencia

Neurociencia

Los inhibidores en neurociencia son compuestos diseñados para modular la actividad de proteínas, enzimas o receptores específicos dentro del sistema nervioso. Estos inhibidores son cruciales para estudiar los mecanismos moleculares subyacentes a la función neuronal, la transmisión sináptica y las enfermedades neurodegenerativas. Al dirigirse a los receptores de neurotransmisores, canales iónicos y vías de señalización, los inhibidores en neurociencia ayudan en la exploración de la función cerebral y en el desarrollo de estrategias terapéuticas para trastornos neurológicos como el Alzheimer, Parkinson y la epilepsia. En CymitQuimica, ofrecemos una amplia gama de inhibidores de neurociencia de alta calidad para apoyar su investigación en neurobiología, neurofarmacología y ciencias cognitivas.

Subcategorías de "Neurociencia"

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Se han encontrado 5400 productos de "Neurociencia"

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  • Baclofen hydrochloride

    CAS:
    <p>Baclofen HCL, a GABA-B agonist, treats muscle spasticity by reducing excitatory transmission.</p>
    Fórmula:C10H13Cl2NO2
    Pureza:99.55%
    Forma y color:Solid
    Peso molecular:250.122
  • Tiagabine hydrochloride hydrate

    CAS:
    <p>Tiagabine HCl hydrate, IC50: 67-446 nM, selectively inhibits GABA uptake, acts as an anticonvulsant.</p>
    Fórmula:C20H28ClNO3S2
    Forma y color:Solid
    Peso molecular:430.02
  • Ramosetron hydrochloride

    CAS:
    <p>Ramosetron hydrochloride (YM-060) is a serotonin 5-HT3 receptor antagonist. It is used to treat diarrhea-predominant irritable bowel syndrome and nausea.</p>
    Fórmula:C17H18ClN3O
    Pureza:99.95%
    Forma y color:Solid
    Peso molecular:315.8
  • LP-211

    CAS:
    <p>LP-211 is a brain penetrant selective agonist for a 5-HT7 receptor (Ki: 0.58 nM), and &gt;300-fold selectivity over the 5-HT1A receptor.</p>
    Fórmula:C30H34N4O
    Pureza:98.65%
    Forma y color:Solid
    Peso molecular:466.62
  • A-740003

    CAS:
    <p>A-740003 is a potent P2X7 receptor blocker, inhibiting rat/human receptors (IC50: 18/40 nM), lessens pain in animals, and shrinks mouse neuroblastoma.</p>
    Fórmula:C26H30N6O3
    Pureza:96.53% - 99.68%
    Forma y color:Solid
    Peso molecular:474.55
  • CX516

    CAS:
    <p>CX516 (Ampalex), an ampakine and nootropic, acts as an AMPA receptor positive allosteric modulator as a therapy for Alzheimer's disease, schizophrenia and MCI.</p>
    Fórmula:C14H15N3O
    Pureza:99.04% - ≥95%
    Forma y color:Tan Solid
    Peso molecular:241.29
  • FK 3311

    CAS:
    <p>FK 3311 (COX-2 Inhibitor V) is a cell permeable and orally available sulfonanilide that acts as a COX-2 inhibitor and non-steroidal anti-inflammatory drug (</p>
    Fórmula:C15H13F2NO4S
    Pureza:97.98%
    Forma y color:Solid
    Peso molecular:341.33
  • Piboserod hydrochloride

    CAS:
    <p>Piboserod HCl is a selective antagonist of 5-HT4 and muscarinic receptor.</p>
    Fórmula:C22H32ClN3O2
    Forma y color:Solid
    Peso molecular:405.96
  • NS 1738

    CAS:
    <p>NS 1738 (NSC-213859) is a positive allosteric modulator of the α7-containing neuronal nicotinic acetylcholine receptors (nAChRs)</p>
    Fórmula:C14H9Cl2F3N2O2
    Pureza:99.11%
    Forma y color:Solid
    Peso molecular:365.13
  • Melitracen hydrochloride

    CAS:
    Melitracen hydrochloride (Thymeol hydrochloride) , an antidepressant, is used as potential dopamine D1/2 receptor antagonist to treat depression.
    Fórmula:C21H26ClN
    Pureza:99.99%
    Forma y color:Crystalline Solid
    Peso molecular:327.90
  • Rizatriptan benzoate

    CAS:
    <p>Rizatriptan benzoate (MK-462 Benzoate) selectively binds to and activates serotonin (5-HT) 1B receptors and 5-HT 1D receptors providing relief of migraine</p>
    Fórmula:C22H25N5O2
    Pureza:99% - 99.79%
    Forma y color:White To Off-White Crystalline Powder
    Peso molecular:391.47
  • CRANAD 2

    CAS:
    <p>CRANAD-2, a near-infrared probe, detects amyloid-beta in vivo, increasing fluorescence 70x and shifting blue 90 nm upon binding.</p>
    Fórmula:C23H25BF2N2O2
    Pureza:99.44%
    Forma y color:Dark Blue To Black Powder
    Peso molecular:410.27
  • PU02

    CAS:
    <p>PU02 (6-[(1-Naphthalenylmethyl)thio]-9H-purine) is a potent and selective antagonist of 5-HT3 receptor.</p>
    Fórmula:C16H12N4S
    Pureza:99.35%
    Forma y color:Solid
    Peso molecular:292.36
  • Bitopertin

    CAS:
    <p>Bitopertin (Paliflutine) (RG1678, RO-4917838) is a potent inhibitor of glycine transporter 1 (GlyT1), with Ki of 8.1 nM for human hGlyT1b and IC50 of 22-25 nM</p>
    Fórmula:C21H20F7N3O4S
    Pureza:98.57% - 98.71%
    Forma y color:Solid
    Peso molecular:543.46
  • Succinylcholine Chloride Dihydrate

    CAS:
    <p>Succinylcholine Chloride Dihydrate (Succinyldicholine dichloride) is a nicotinic AChR agonist and also acts as a depolarizing neuromuscular blocker.</p>
    Fórmula:C14H30N2O4·2Cl·2H2O
    Pureza:99.87%
    Forma y color:White Solid
    Peso molecular:397.34
  • Ritanserin

    CAS:
    <p>Ritanserin (R 55667) is a long-acting, highly potent, relatively selective, orally bioavailable 5-HT2 receptor antagonist.Cost-effective and quality-assured.</p>
    Fórmula:C27H25F2N3OS
    Pureza:99.77% - 99.89%
    Forma y color:Solid
    Peso molecular:477.57
  • JHU37152

    CAS:
    <p>JHU37152 is a DREADD agonist; Ki: 1.8 nM at hM3Dq, 8.7 nM at hM4Di; EC50: 5 nM (hM3Dq), 0.5 nM (hM4Di) in HEK-293 cell assays.</p>
    Fórmula:C19H20ClFN4
    Pureza:99.72%
    Forma y color:Solid
    Peso molecular:358.84
  • Ethyl (triphenylphosphoranylidene) acetate

    CAS:
    <p>Ethyl (triphenylphosphoranylidene) acetate ((Carbethoxymethylene)triphenylphosphorane) may act as an cholinesterase inhibitor that inhibits AChE and BChE.</p>
    Fórmula:C22H21O2P
    Pureza:97.985%
    Forma y color:White Or Slight Yellow Powder
    Peso molecular:348.37
  • Ro0711401

    CAS:
    <p>Ro0711401 is an agonist of mGlu1 receptor.</p>
    Fórmula:C18H11F3N2O3
    Pureza:97.57%
    Forma y color:Solid
    Peso molecular:360.29
  • GNE-7915 tosylate

    CAS:
    <p>GNE-7915 tosylate is a potent, selective, and brain-penetrant LRRK2 inhibitor, boasting an IC50 value of 9 nM.</p>
    Fórmula:C26H29F4N5O6S
    Forma y color:Solid
    Peso molecular:615.6
  • VU0467154

    CAS:
    <p>VU0467154 is a positive allosteric modulator of the M4 muscarinic acetylcholine receptor.</p>
    Fórmula:C17H15F3N4O3S2
    Pureza:98.28% - 99.51%
    Forma y color:Solid
    Peso molecular:444.45
  • (S)-Flurbiprofen

    CAS:
    <p>Esflurbiprofen is an inhibitor of COX-1 and COX-2.</p>
    Fórmula:C15H13FO2
    Pureza:99.99%
    Forma y color:White To Yellowish Crystalline Powder
    Peso molecular:244.26
  • Traxoprodil

    CAS:
    <p>Traxoprodil (CP101606) is a selective NMDA antagonist and protects hippocampal neurons (IC50: 10 nM).</p>
    Fórmula:C20H25NO3
    Pureza:99.89%
    Forma y color:Solid
    Peso molecular:327.42
  • 6-Methylflavone

    CAS:
    <p>6-Methylflavone is an activator of α1β2γ2L and α1β2 GABAA receptors.</p>
    Fórmula:C16H12O2
    Pureza:99.69%
    Forma y color:Solid
    Peso molecular:236.27
  • Dolasetron

    CAS:
    <p>Dolasetron (MDL-73147)(MDL-73147) is a serotonin 5-HT3 receptor antagonist. Dolasetron is used to treat nausea and vomiting following chemotherapy.</p>
    Fórmula:C19H20N2O3
    Pureza:99.84% - 99.86%
    Forma y color:White Powder
    Peso molecular:324.37
  • BPAM344

    CAS:
    <p>BPAM344 is a potent positive allosteric modulator (PAM) of the KAR subunits GluK1b, GluK2a, and GluK3a.</p>
    Fórmula:C10H11FN2O2S
    Pureza:99.53%
    Forma y color:Solid
    Peso molecular:242.27
  • Eptapirone

    CAS:
    <p>Eptapirone (F 11440) is a highly effective and selective 5-HT1A receptor agonist with marked antidepressant and anxiolytic potential.</p>
    Fórmula:C16H23N7O2
    Pureza:99.39% - 99.65%
    Forma y color:Solid
    Peso molecular:345.4
  • DNQX

    CAS:
    <p>DNQX (FG 9041) is a competitive, non-NMDA glutamate receptor antagonist (IC50s = 0.5 and 0.1 μM for AMPA and kainate receptors, respectively)</p>
    Fórmula:C8H4N4O6
    Pureza:97.27% - 99.1%
    Forma y color:Off-White Powder With A Yellow Tinge
    Peso molecular:252.14
  • YM90K

    CAS:
    <p>YM90K (6-(1H-imidazol-1-yl)-7-nitro-2,3(1H,4H)-) hydrochloride is an antagonist of AMPA receptor.</p>
    Fórmula:C11H8ClN5O4
    Pureza:98.23%
    Forma y color:Solid
    Peso molecular:309.66
  • Oxyphencyclimine Hydrochloride

    CAS:
    <p>Oxyphencyclimine Hydrochloride (Ulcociclinina) is a synthetic tertiary amine and antimuscarinic agent with antispasmodic and antisecretory activities.</p>
    Fórmula:C20H29ClN2O3
    Pureza:99.55%
    Forma y color:Solid
    Peso molecular:380.91
  • Xanthotoxol

    CAS:
    <p>Xanthotoxol (Psoralen) is a bioactive furocoumarin with anti-inflammatory, antioxidant, 5-HT antagonist, and neuroprotective properties.</p>
    Fórmula:C11H6O4
    Pureza:99.97%
    Forma y color:Solid
    Peso molecular:202.16
  • Piperazine

    CAS:
    <p>Piperazine (1,4-Diazacyclohexane), a gamma-aminobutyric acid (GABA) agonist, serves as a crucial building block and core component in a wide range of marketed drugs known for their varied pharmacological activities.</p>
    Fórmula:C4H10N2
    Forma y color:Solid
    Peso molecular:86.14
  • Orexin B, rat, mouse Acetate


    Orexin B, rat, mouse Acetate (Rat orexin B) is an endogenous agonist at Orexin receptor with Kis of 420 and 36 nM for OX1 and OX2, respectively.
    Fórmula:C128H219N45O36S
    Pureza:94.61%
    Forma y color:Solid
    Peso molecular:2996.45
  • AZD7325

    CAS:
    <p>AZD7325 (AZD-7325) is a GABA-Aα2,3 -selective receptor modulator.</p>
    Fórmula:C19H19FN4O2
    Pureza:99.83%
    Forma y color:Solid
    Peso molecular:354.38
  • Ralmitaront

    CAS:
    <p>Ralmitaront (RO6889450) is a potent, orally active partial agonist of the trace amine-associated receptor 1 (TAAR1).</p>
    Fórmula:C17H22N4O2
    Pureza:99.71% - 99.79%
    Forma y color:Solid
    Peso molecular:314.38
  • FITM

    CAS:
    <p>FITM is a potent negative allosteric modulator of mGlu1 receptor(Ki : 2.5 nM).</p>
    Fórmula:C18H18FN5OS
    Pureza:97.25%
    Forma y color:Solid
    Peso molecular:371.43
  • L-745870 trihydrochloride

    CAS:
    <p>L-745870 trihydrochloride is a highly potent and selective D4 dopamine receptor antagonist.</p>
    Fórmula:C18H22Cl4N4
    Pureza:97.52%
    Forma y color:Solid
    Peso molecular:436.21
  • N-Desmethylclozapine

    CAS:
    <p>N-Desmethylclozapine: 5-HT2C antagonist (IC50: 7.1 nM), dopamine D4 antagonist, δ-opioid agonist.</p>
    Fórmula:C17H17ClN4
    Pureza:97.25% - 99.83%
    Forma y color:Yellow Crystalline Solid
    Peso molecular:312.8
  • Ziprasidone mesylate

    CAS:
    <p>Ziprasidone mesylate (CP-88059), an oral 5-HT &amp; dopamine blocker, binds D2, 5-HT2A, 5-HT1A with Ki values: 4.8, 0.42, 3.4 nM.</p>
    Fórmula:C22H25ClN4O4S2
    Forma y color:Solid
    Peso molecular:509.04
  • Dasotraline hydrochloride

    CAS:
    <p>Dasotraline hydrochloride, a dopamine, norepinephrine, and serotonin reuptake inhibitor with IC50s: 4, 6, 11 nM.</p>
    Fórmula:C16H16Cl3N
    Pureza:98.92% - 99.6%
    Forma y color:Solid
    Peso molecular:328.66
  • PRX-07034 hydrochloride

    CAS:
    <p>PRX-07034 hydrochloride is a selective antagonist of 5-HT6 receptor. It has cognition and memory-enhancing properties and decreases body weight in rodents.</p>
    Fórmula:C21H29Cl2N3O4S
    Pureza:98.5%
    Forma y color:Solid
    Peso molecular:490.44
  • Prifinium bromide

    CAS:
    <p>Prifinium bromide is a quaternary ammon antimuscarinic. It inhibits hyperkinesia of the digestive organs and urinary tract and has a spasmolytic action.</p>
    Fórmula:C22H28BrN
    Pureza:97.99%
    Forma y color:Solid
    Peso molecular:386.37
  • PF-06447475

    CAS:
    <p>PF-06447475 is a highly effective, specific, brain penetrant LRRK2 inhibitor with IC0 of 3/11 nM for wild type LRRK2 and G2019S LRRK2 respectively.</p>
    Fórmula:C17H15N5O
    Pureza:98.61% - 99.62%
    Forma y color:Solid
    Peso molecular:305.33
  • A-804598

    CAS:
    <p>A-804598 is a competitive and selective P2X7 receptor antagonist (IC50: 10 nM, rat; 9 nM, mouse; 11 nM, human).</p>
    Fórmula:C19H17N5
    Pureza:99.57%
    Forma y color:Solid
    Peso molecular:315.37
  • 5-Benzyloxygramine

    CAS:
    <p>5-Benzyloxygramine blocks the Dopamin receptors and antagonizes the effects of 5-HT on the rat uterus and the rabbit ear.</p>
    Fórmula:C18H20N2O
    Pureza:99.13%
    Forma y color:Solid
    Peso molecular:280.36
  • Nemifitide acetate(173240-15-8 free base)


    <p>Nemifitide acetate, synthetic 5-amino acid antidepressant, has quick effect, mimics MIF.</p>
    Fórmula:C35H47FN10O8
    Pureza:97.97%
    Forma y color:Solid
    Peso molecular:754.85
  • Amyloid β-Protein 10-20 acetate


    <p>Amyloid β-Protein 10-20 acetate (Amyloid β-Protein 10-20 acetate (152286-31-2 free base)) is a fragment of Amyloid-β peptide, maybe used in the research of</p>
    Fórmula:C73H103N17O18
    Pureza:97.23%
    Forma y color:Solid
    Peso molecular:1506.65
  • SR 57227 hydrochloride

    CAS:
    <p>SR 57227A (SR 57227 hydrochloride) is a potent, orally active and selective 5-HT3 receptor agonist. It with ability to cross the blood brain barrier.</p>
    Fórmula:C10H14ClN3·HCl
    Pureza:99.89%
    Forma y color:Solid
    Peso molecular:248.15
  • VUF 10166

    CAS:
    <p>VUF10166 is a novel, potent and competitive antagonist for 5-HT3A receptor with Ki of 0.04 nM, its affinity at 5-HT3AB receptor is significantly lower.</p>
    Fórmula:C13H15ClN4
    Pureza:99.66%
    Forma y color:Solid
    Peso molecular:262.74
  • 4-Acetamidobutanoic acid

    CAS:
    <p>4-Acetamidobutanoic acid, a GABA derivative in eukaryotes, found in blood, feces, urine, and human prostate.</p>
    Fórmula:C6H11NO3
    Pureza:98.51%
    Forma y color:Solid
    Peso molecular:145.16