
Neurociencia
Los inhibidores en neurociencia son compuestos diseñados para modular la actividad de proteínas, enzimas o receptores específicos dentro del sistema nervioso. Estos inhibidores son cruciales para estudiar los mecanismos moleculares subyacentes a la función neuronal, la transmisión sináptica y las enfermedades neurodegenerativas. Al dirigirse a los receptores de neurotransmisores, canales iónicos y vías de señalización, los inhibidores en neurociencia ayudan en la exploración de la función cerebral y en el desarrollo de estrategias terapéuticas para trastornos neurológicos como el Alzheimer, Parkinson y la epilepsia. En CymitQuimica, ofrecemos una amplia gama de inhibidores de neurociencia de alta calidad para apoyar su investigación en neurobiología, neurofarmacología y ciencias cognitivas.
Subcategorías de "Neurociencia"
- Receptor 5-HT(939 productos)
- ACK(1 productos)
- AChR(575 productos)
- ATP Citrato Liasa(16 productos)
- Receptor adrenérgico(2.945 productos)
- BACE(36 productos)
- Beta amiloide(205 productos)
- CAMK(69 productos)
- Inhibidores de ciclooxigenasa (COX)(561 productos)
- Receptor de dopamina(407 productos)
- Receptor GABA(336 productos)
- Gamma-secretasa(59 productos)
- GluR(255 productos)
- GlyT(24 productos)
- Receptor de histamina(358 productos)
- LRRK2(33 productos)
- Receptor de melatonina(24 productos)
- NMDAR(28 productos)
- Receptor de OX(40 productos)
- Receptor de opioides(297 productos)
Mostrar 12 subcategorías más
Se han encontrado 5398 productos de "Neurociencia"
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Spiperone hydrochloride
CAS:<p>5-HT2A serotonin and selective D2-like dopamine receptor antagonist</p>Fórmula:C23H27ClFN3O2Pureza:98%Forma y color:SolidPeso molecular:431.93DNQX disodium salt
CAS:<p>DNQX disodium salt is a water-soluble form of selective antagonist of non-NMDA receptor</p>Fórmula:C8H2N4Na2O6Pureza:98.93%Forma y color:SolidPeso molecular:296.1(E)-3,4,5-Trimethoxycinnamic acid
CAS:<p>(E)-3,4,5-Trimethoxycinnamic acid (O-Methylsinapic acid) is a natural product from the roots and rhizomes of Notopterygium incisum.</p>Fórmula:C12H14O5Pureza:99.83%Forma y color:SolidPeso molecular:238.24Eptapirone
CAS:<p>Eptapirone (F 11440) is a highly effective and selective 5-HT1A receptor agonist with marked antidepressant and anxiolytic potential.</p>Fórmula:C16H23N7O2Pureza:99.39% - 99.65%Forma y color:SolidPeso molecular:345.4RU 24969 free base
CAS:<p>RU 24969 (5-methoxy-3-(1,2,3,6-tetrahydropyridin-4-yl)-1H-indole) is a selective agonist of 5-HT1A and 5-HT1B receptors.</p>Fórmula:C14H16N2OPureza:97.38%Forma y color:SolidPeso molecular:228.29Farampator
CAS:<p>Farampator (CX-691) (CX-691;Org24448) is a positive modulator of AMPA receptor.</p>Fórmula:C12H13N3O2Pureza:99.84% - >99.99%Forma y color:SolidPeso molecular:231.25α-Thujone
CAS:<p>α-Thujone is an inhibitor of ACh with an IC50 value of 24.7μM.</p>Fórmula:C10H16OPureza:97.02% - 98.41%Forma y color:Less Or Almost Colorless Liquid With A Menthol- Like Odor (Albert-Puleo 1978; Budavari 1996) Colorless Or Almost Colorless Liquid With A Menthol- Like Odor (Albert-Puleo 1978; Budavari 1996)Peso molecular:152.23PHA 568487
CAS:<p>PHA 568487: α-7 nAChR agonist, rapid brain uptake, lessens oxidative stress & neuroinflammation.</p>Fórmula:C20H24N2O7Forma y color:SolidPeso molecular:404.419OXA (17-33) acetate
<p>OXA (17-33) acetate is a more potent agonist of orexin-1 receptor (OX1, EC50 = 8.29 nM)) over OX2 (EC50 = 187 nM).</p>Fórmula:C79H125N23O22Pureza:98.52%Forma y color:SolidPeso molecular:1748.98(2S)-6-Prenylnaringenin
CAS:<p>(2S)-6-Prenylnaringenin (6-Prenylnaringenin) is an isomer of the potent phytoestrogen, 8-prenylnaringenin.</p>Fórmula:C20H20O5Pureza:99.47%Forma y color:SolidPeso molecular:340.37Tebanicline hydrochloride
CAS:<p>Tebanicline hydrochloride (Ebanicline hydrochloride) , is an effective synthetic nicotinic (non-opioid) analgesic drug.</p>Fórmula:C9H12Cl2N2OPureza:91.74% - 98.71%Forma y color:SolidPeso molecular:235.11Tiaprofenic acid
CAS:<p>Tiaprofenic acid (Acido tiaprofenico) is a non-steroidal anti-inflammatory drug used to treat pain, especially arthritic pain.</p>Fórmula:C14H12O3SPureza:99.51%Forma y color:SolidPeso molecular:260.31Piperacetazine
CAS:<p>Piperacetazine (Piperacetazinum), an antipsychotic prodrug, is used forschizophrenia.</p>Fórmula:C24H30N2O2SPureza:99.9% - 99.92%Forma y color:SolidPeso molecular:410.57Verubecestat TFA
CAS:<p>Verubecestat (MK-8931/SCH 900931), a potent BACE1 inhibitor, shows promise for Alzheimer's, cuts Aβ CSF levels by 92%.</p>Fórmula:C19H18F5N5O5SForma y color:SolidPeso molecular:523.435MPEP
CAS:<p>MPEP is a selective mGlu5 receptor antagonist with IC50 of 36 nM, exhibits no appreciable activity at mGlu1b/2/3/4a/7b/8a/6 receptors.</p>Fórmula:C14H11NPureza:99.54%Forma y color:SolidPeso molecular:193.24Almotriptan Malate
CAS:<p>Almotriptan Malate (PNU180638), a selective 5-HT1B/1D receptor agonist, is used in the therapy of Migraine attacks in adults.</p>Fórmula:C17H25N3O2S·C4H6O5Pureza:99.95%Forma y color:Pale Yellow SolidPeso molecular:469.55SAX-187 hydrochloride
CAS:<p>WAY-181187 is a potent, selective 5-HT6 agonist with high affinity (2.2-4.8 nM), and increases GABA in rat cortex at 3-30 mg/kg s.c.</p>Fórmula:C15H14Cl2N4O2S2Forma y color:SolidPeso molecular:417.33NGB 2904
CAS:<p>NGB 2904 is a potent and selective antagonist of dopamine D3 receptor. NGB2904 potently antagonizes mitogenesis stimulated by quinpirole (IC50 = 6.8 nM).</p>Fórmula:C28H29Cl2N3OPureza:98.79%Forma y color:SolidPeso molecular:494.46Temgicoluril
CAS:<p>Temgicoluril (mebikar) acts on GABA Receptor.</p>Fórmula:C8H14N4O2Pureza:99.8%Forma y color:SolidPeso molecular:198.22Verubecestat
CAS:<p>Verubecestat (MK-8931) (MK-8931) is an effective and specific β-secretase inhibitor and β-site APP-cleaving enzyme 1 inhibitor or BACE1 protein inhibitor.</p>Fórmula:C17H17F2N5O3SPureza:92.24% - 99.55%Forma y color:SolidPeso molecular:409.41NS3861
CAS:<p>NS3861 is a selective agonist for α3β4/α4β2 nAChRs, preferring β-subunits, with no effect on α4-based receptors.</p>Fórmula:C12H14BrNSPureza:99.853%Forma y color:SolidPeso molecular:284.22Semax acetate(80714-61-0 free base)
CAS:<p>Semax acetate is a synthetic peptide analog of adrenocorticotropic hormone (ACTH) that has neuroprotective, analgesic, and anxiolytic properties.</p>Fórmula:C39H55N9O12SPureza:99.46%Forma y color:SolidPeso molecular:873.98VU0364770
CAS:<p>VU0364770 (VU 0364770)(EC50=1.1 μM), a positive allosteric modulator(PAM) of mGlu4, shows insignificant activity at 68 other receptors, including other mGlu</p>Fórmula:C12H9ClN2OPureza:99.65% - >99.99%Forma y color:SolidPeso molecular:232.67FITM
CAS:<p>FITM is a potent negative allosteric modulator of mGlu1 receptor(Ki : 2.5 nM).</p>Fórmula:C18H18FN5OSPureza:97.25%Forma y color:SolidPeso molecular:371.43LOX-IN-3 dihydrochloride monohydrate
CAS:<p>LOX-IN-3 dihydrochloride monohydrate is an oral lysyl oxidase inhibitor for research in fibrosis, cancer, and angiogenesis.</p>Fórmula:C13H17Cl2FN2O3SForma y color:SolidPeso molecular:371.25VU0357017 hydrochloride
CAS:<p>VU0357017 hydrochloride (ML071 hydrochloride) is highly selective M1 agonists act at an allosteric site to activate the receptor (EC50: 477 ± 172 nM; Pec50: 6.</p>Fórmula:C18H28ClN3O3Pureza:99% - 99.97%Forma y color:SolidPeso molecular:369.89FPS-ZM1
CAS:<p>FPS-ZM1 is a high-affinity RAGE specific inhibitor that blocks Aβ binding to the V domain of RAGE.</p>Fórmula:C20H22ClNOPureza:99.32% - 99.52%Forma y color:SolidPeso molecular:327.85A 582941 HCl (848591-90-2(free base))
<p>A-582941 is a alpha7 neuronal nicotinic receptor agonist with broad spectrum cognition-enhancing properties</p>Fórmula:C17H21ClN4Pureza:99.83%Forma y color:SolidPeso molecular:316.83TBPB
CAS:<p>TBPB is an allosteric M1 mAChR agonist.</p>Fórmula:C25H32N4OPureza:97.87% - 99.9%Forma y color:SolidPeso molecular:404.55Propiverine
CAS:<p>Propiverine reduces muscle spasms by limiting calcium influx, targeting bladder smooth muscles, aiding OAB research.</p>Fórmula:C23H29NO3Forma y color:SolidPeso molecular:367.483-MATIDA
CAS:<p>3-MATIDA is an effective mGluR-1 antagonist (IC50: 6.3 μM, rat mGluR-1a).</p>Fórmula:C8H9NO4SPureza:99.75% - 99.96%Forma y color:SolidPeso molecular:215.23Umibecestat HCl
CAS:<p>Umibecestat HCl (CNP520 HCl) is an efficient β-secretase (BACE1/BACE2) inhibitor that reduces Aβ levels in mice and rats.</p>Fórmula:C19H16Cl2F7N5O2Pureza:99.92%Forma y color:SolidPeso molecular:550.26Demecarium bromide
CAS:<p>Demecarium bromide (BC-48) is a potent cholinesterase inhibitor,and is treatment glaucoma agent.</p>Fórmula:C32H52Br2N4O4Pureza:98%Forma y color:White Powder SolidPeso molecular:716.59Semagacestat
CAS:<p>Semagacestat (LY450139) (LY450139) is a γ-secretase blocker for Aβ42/Aβ40/Aβ38 (IC50: 10.9/12.1/12.0 nM) and also inhibits Notch signaling (IC50: 14.1 nM).</p>Fórmula:C19H27N3O4Pureza:97.1% - 99.9%Forma y color:SolidPeso molecular:361.44(-)-(S)-B-973B
CAS:<p>(-)-(S)-B-973B is an effective allosteric agonist and a positive allosteric modulator of α7 nAChR.</p>Fórmula:C24H26F2N6OPureza:99.52%Forma y color:SolidPeso molecular:452.52'MeO6MF
CAS:<p>2'MeO6MF is a brain-penetrant positive allosteric modulator at α2β1γ2L and all α1-containing GABAA receptors.It offers neuroprotection and improved functional</p>Fórmula:C17H14O3Pureza:99.28% - 99.63%Forma y color:SolidPeso molecular:266.29Azeliragon
CAS:<p>Azeliragon (TTP488) is an antagonist at the Receptor for Advanced Glycation End products; is evaluated as a potential treatment for patients with mild-to-</p>Fórmula:C32H38ClN3O2Pureza:96.7% - 98.33%Forma y color:SolidPeso molecular:532.12Solifenacin hydrochloride
CAS:<p>Solifenacin Hcl is a muscarinic receptor antagonist.</p>Fórmula:C23H27ClN2O2Pureza:98%Forma y color:SolidPeso molecular:398.93Sivopixant
CAS:<p>Sivopixant (S-600918), a potent P2X3 receptor antagonist, has a high analgesic effect (P2X3 IC50=4.2 nM, P2X2/3 IC50=1100 nM).</p>Fórmula:C25H22ClN5O5Pureza:99.34%Forma y color:SolidPeso molecular:507.93Pergolide mesylate
CAS:<p>Pergolide mesylate (LY127809), a dopamine agonist for Parkinson's and hyperprolactinemia, was withdrawn for heart valve risk.</p>Fórmula:C20H30N2O3S2Pureza:99.70%Forma y color:White To Off-White SolidPeso molecular:410.59Imidazenil
CAS:<p>Imidazenil is an modulator of GABA-A that blocks the sedative effects without lowering the convulsion threshold.</p>Fórmula:C18H12BrFN4OPureza:98.4%Forma y color:SolidPeso molecular:399.22MK-3697
CAS:<p>MK-3697, an isonicotinamide small molecule, acts as a potent and selective Orexin 2 receptor antagonist (Ki: 0.95 nM).</p>Fórmula:C23H21N5O3SPureza:97.69% - 98.15%Forma y color:SolidPeso molecular:447.51Cariprazine
CAS:<p>Cariprazine (RGH-188) is a novel antipsychotic drug candidate that exhibits high affinity for the D3 (Ki=0.085 nM) and D2 (Ki=0.49 nM) receptors, and moderate</p>Fórmula:C21H32Cl2N4OPureza:99.68% - 99.87%Forma y color:SolidPeso molecular:427.41Ocaperidone
CAS:<p>Ocaperidona (Ocaperidone (Ocaperidona)), a very high affinity dopamine D2 antagonist.</p>Fórmula:C24H25FN4O2Pureza:99.33%Forma y color:SolidPeso molecular:420.48GSK163090
CAS:<p>GSK163090 is a specific and orally active 5-HT1A/B/D receptor antagonist (pKis: 9.4/8.5/9.7, and 6.3/6.7 for 5-HT1A/B/D, and dopamine D2/D3).</p>Fórmula:C25H29N5OPureza:99.2%Forma y color:SolidPeso molecular:415.53Dasotraline hydrochloride
CAS:<p>Dasotraline hydrochloride, a dopamine, norepinephrine, and serotonin reuptake inhibitor with IC50s: 4, 6, 11 nM.</p>Fórmula:C16H16Cl3NPureza:98.92% - 99.6%Forma y color:SolidPeso molecular:328.661,1'-Methylenedi-2-naphthol
CAS:<p>1,1'-Methylenedi-2-naphthol target CYP2C19 - cytochrome P450 family 2 subfamily C member 19 (human).</p>Fórmula:C21H16O2Pureza:98.91%Forma y color:Light Pink To Light Brown Crystalline PowderPeso molecular:300.35RS-127445
CAS:<p>RS-127445 (MT500) is a selective 5-HT2B receptor antagonist with pKi of 9.5 and pIC50 of 10.4, exhibits >1000-fold selectivity against other 5-HT receptors.</p>Fórmula:C17H16FN3Pureza:99.32%Forma y color:SolidPeso molecular:281.33Pimavanserin tartrate
CAS:<p>Pimavanserin tartrate is a potent 5-HT 2A receptor inverse agonist used to treat Parkinson's disease-related psychosis.Cost-effective and quality-assured.</p>Fórmula:C50H68F2N6O4·C4H6O6Pureza:99.24% - 99.98%Forma y color:SolidPeso molecular:1005.2Acephate
CAS:<p>Acephate (Orthene) is an anticholinesterase insecticide with a weak inhibitory effect on AChE in rats, but it can effectively inhibit AChE in cockroaches.</p>Fórmula:C4H10NO3PSPureza:≥98%Forma y color:Colorless Crystals Acephate Is A White Solid Used As A Contact And Systemic InsecticidePeso molecular:183.17
