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Neurociencia

Neurociencia

Los inhibidores en neurociencia son compuestos diseñados para modular la actividad de proteínas, enzimas o receptores específicos dentro del sistema nervioso. Estos inhibidores son cruciales para estudiar los mecanismos moleculares subyacentes a la función neuronal, la transmisión sináptica y las enfermedades neurodegenerativas. Al dirigirse a los receptores de neurotransmisores, canales iónicos y vías de señalización, los inhibidores en neurociencia ayudan en la exploración de la función cerebral y en el desarrollo de estrategias terapéuticas para trastornos neurológicos como el Alzheimer, Parkinson y la epilepsia. En CymitQuimica, ofrecemos una amplia gama de inhibidores de neurociencia de alta calidad para apoyar su investigación en neurobiología, neurofarmacología y ciencias cognitivas.

Subcategorías de "Neurociencia"

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Se han encontrado 5398 productos de "Neurociencia"

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  • Almotriptan Malate

    CAS:
    <p>Almotriptan Malate (PNU180638), a selective 5-HT1B/1D receptor agonist, is used in the therapy of Migraine attacks in adults.</p>
    Fórmula:C17H25N3O2S·C4H6O5
    Pureza:99.95%
    Forma y color:Pale Yellow Solid
    Peso molecular:469.55
  • SKF89976A hydrochloride

    CAS:
    <p>SKF89976A hydrochloride (d,l-SKF89976A hydrochloride) is a selective inhibitor GABA transporter such as GAT-1 (IC50s = 0.28 μM), GAT-2 (IC50s = 137.34 μM) and</p>
    Fórmula:C22H26ClNO2
    Pureza:98.02%
    Forma y color:Solid
    Peso molecular:371.9
  • 3-MATIDA

    CAS:
    <p>3-MATIDA is an effective mGluR-1 antagonist (IC50: 6.3 μM, rat mGluR-1a).</p>
    Fórmula:C8H9NO4S
    Pureza:99.75% - 99.96%
    Forma y color:Solid
    Peso molecular:215.23
  • Homocarnosine acetate


    <p>Homocarnosine acetate is a dipeptide unique to brain consisting of γ-aminobutyric acid (GABA) and histidine.</p>
    Fórmula:C12H20N4O5
    Pureza:99.52%
    Forma y color:Solid
    Peso molecular:300.31
  • Demecarium bromide

    CAS:
    <p>Demecarium bromide (BC-48) is a potent cholinesterase inhibitor,and is treatment glaucoma agent.</p>
    Fórmula:C32H52Br2N4O4
    Pureza:98%
    Forma y color:White Powder Solid
    Peso molecular:716.59
  • Revefenacin

    CAS:
    <p>Revefenacin (TD-4208) is a mAChR antagonist has a high affinity on M3 receptor( Ki : 0.18 nM),and potentially useful for the treatment of respiratory disease.</p>
    Fórmula:C35H43N5O4
    Pureza:98.12%
    Forma y color:Solid
    Peso molecular:597.75
  • Tiaprofenic acid

    CAS:
    <p>Tiaprofenic acid (Acido tiaprofenico) is a non-steroidal anti-inflammatory drug used to treat pain, especially arthritic pain.</p>
    Fórmula:C14H12O3S
    Pureza:99.51%
    Forma y color:Solid
    Peso molecular:260.31
  • Rebamipide mofetil

    CAS:
    <p>Rebamipide mofetil is an orally active prodrug of Rebamipide which is a mucoprotective agent.</p>
    Fórmula:C25H26ClN3O5
    Pureza:98.17%
    Forma y color:Solid
    Peso molecular:483.94
  • (S)-UFR2709

    CAS:
    <p>(S)-UFR2709, a nAChR competitive antagonist, favors α4β2 over α7, reduces anxiety and alcohol use in rats.</p>
    Fórmula:C13H17NO2
    Forma y color:Solid
    Peso molecular:219.284
  • Ipratropium Bromide

    CAS:
    <p>Ipratropium Bromide (Sch 1000) is an antagonist of muscarinic receptors and is used in COPD and asthma studies.</p>
    Fórmula:C20H30BrNO3
    Pureza:99.92%
    Forma y color:Solid
    Peso molecular:412.37
  • SB-334867 free base

    CAS:
    <p>SB-334867 free base (SB334867A free base) is a selective orexin-1 (OX1) receptor antagonist.</p>
    Fórmula:C17H13N5O2
    Pureza:99.67% - >99.99%
    Forma y color:Solid
    Peso molecular:319.32
  • Abaperidone Hydrochloride

    CAS:
    <p>Abaperidone Hydrochloride is an atypical antipsychotic, potently binging to5-HT2 receptors and D2 receptors.</p>
    Fórmula:C25H26ClFN2O5
    Forma y color:Solid
    Peso molecular:488.94
  • KN-62

    CAS:
    <p>KN-62 is a potent and specific Ca2+/calmodulin-dependent protein kinase II (CaMKII) inhibitor with Ki of 0.9 μM.</p>
    Fórmula:C38H35N5O6S2
    Pureza:99.80% - >99.99%
    Forma y color:White Solid
    Peso molecular:721.84
  • Temgicoluril

    CAS:
    <p>Temgicoluril (mebikar) acts on GABA Receptor.</p>
    Fórmula:C8H14N4O2
    Pureza:99.8%
    Forma y color:Solid
    Peso molecular:198.22
  • Isocorynoxeine

    CAS:
    <p>Isocorynoxeine reduces blood pressure, dilates vessels, and guards neurons against ischemia and glutamate toxicity.</p>
    Fórmula:C22H26N2O4
    Pureza:98% - 99.9%
    Forma y color:Solid
    Peso molecular:382.45
  • 3-AQC

    CAS:
    <p>3-AQC is a competitive antagonist of 5-HT3.</p>
    Fórmula:C20H21N5O4
    Pureza:99.45%
    Forma y color:Solid
    Peso molecular:395.41
  • JH-II-127

    CAS:
    <p>JH-II-127 is an oral LRRK2 inhibitor with IC50s: 6.6 nM (WT), 2.2 nM (G2019S), 47.7 nM (A2016T).</p>
    Fórmula:C19H21ClN6O3
    Pureza:98.32%
    Forma y color:Solid
    Peso molecular:416.86
  • Medetomidine hydrochloride

    CAS:
    <p>Medetomidine hydrochloride (MPV785) is a selective α2-adrenoceptor agonist, with Ki of 1.08 nM, exhibts 1620-fold selectivity over α1-adrenoceptor.</p>
    Fórmula:C13H16N2·HCl
    Pureza:99.96%
    Forma y color:White Or Off White Crystalline Powder
    Peso molecular:236.74
  • MDL 72527

    CAS:
    <p>MDL 72527 (N1,N4-Di(buta-2,3-dien-1-yl)butane-1,4-diamine dihydrochloride) is a polyamine oxidase (POA) inhibitor</p>
    Fórmula:C12H22Cl2N2
    Pureza:98.98%
    Forma y color:Solid
    Peso molecular:265.22
  • Donepezil Hydrochloride

    CAS:
    <p>Donepezil HCl(Aricept) is a selective and effective AChE inhibitor for bAChE and hAChE (IC50: 8.12/11.6 nM).</p>
    Fórmula:C24H29NO3·HCl
    Pureza:99.55% - 99.8%
    Forma y color:White To Off-White Crystalline Solid
    Peso molecular:415.96
  • Sofpironium bromide

    CAS:
    <p>Sofpironium bromide (BBI4000) belongs to a class of drugs called anticholinergics, which exert their effect by blocking the action of acetylcholine.</p>
    Fórmula:C22H32BrNO5
    Pureza:98.85%
    Forma y color:Solid
    Peso molecular:470.4
  • MK-3697

    CAS:
    <p>MK-3697, an isonicotinamide small molecule, acts as a potent and selective Orexin 2 receptor antagonist (Ki: 0.95 nM).</p>
    Fórmula:C23H21N5O3S
    Pureza:97.69% - 98.15%
    Forma y color:Solid
    Peso molecular:447.51
  • Cariprazine

    CAS:
    <p>Cariprazine (RGH-188) is a novel antipsychotic drug candidate that exhibits high affinity for the D3 (Ki=0.085 nM) and D2 (Ki=0.49 nM) receptors, and moderate</p>
    Fórmula:C21H32Cl2N4O
    Pureza:99.68% - 99.87%
    Forma y color:Solid
    Peso molecular:427.41
  • PNU-120596

    CAS:
    <p>PNU-120596 (NSC-216666) is a positive allosteric modulator of α7 nAChR with EC50 of 216 nM.</p>
    Fórmula:C13H14ClN3O4
    Pureza:99.82%
    Forma y color:Solid
    Peso molecular:311.72
  • IKK 16

    CAS:
    <p>IKK 16 (IKK Inhibitor VII) is a selective IκB kinase (IKK) inhibitor for IKK-2, IKK complex and IKK-1 with IC50 of 40 nM, 70 nM and 200 nM, respectively.</p>
    Fórmula:C28H29N5OS
    Pureza:98.76% - 99.61%
    Forma y color:Solid
    Peso molecular:483.63
  • Ocaperidone

    CAS:
    <p>Ocaperidona (Ocaperidone (Ocaperidona)), a very high affinity dopamine D2 antagonist.</p>
    Fórmula:C24H25FN4O2
    Pureza:99.33%
    Forma y color:Solid
    Peso molecular:420.48
  • Bromfenac Sodium

    CAS:
    <p>Bromfenac Sodium (AHR 10282R) is a nonsteroidal anti-inflammatory drug (NSAID) and an orally available COX inhibitor, which has anti-inflammatory activity.</p>
    Fórmula:C15H11BrNO3·Na
    Pureza:99.93%
    Forma y color:Solid
    Peso molecular:356.15
  • IPSU

    CAS:
    <p>IPSU is an antagonist of OX2 receptor. IPSU Exhibits approximately six-fold selectivity for OX2 versus OX1 receptors.</p>
    Fórmula:C23H27N5O2
    Pureza:97.05%
    Forma y color:Solid
    Peso molecular:405.49
  • Dinotefuran

    CAS:
    <p>Dinotefuran (MTI-446), a neonicotinoid insecticide, targets pests by blocking their nervous system.</p>
    Fórmula:C7H14N4O3
    Pureza:99.89%
    Forma y color:White Crystalline Powder
    Peso molecular:202.21
  • RS-127445

    CAS:
    <p>RS-127445 (MT500) is a selective 5-HT2B receptor antagonist with pKi of 9.5 and pIC50 of 10.4, exhibits &gt;1000-fold selectivity against other 5-HT receptors.</p>
    Fórmula:C17H16FN3
    Pureza:99.32%
    Forma y color:Solid
    Peso molecular:281.33
  • Bestim

    CAS:
    <p>Bestim is an immunomodulatory dipeptide that is synthetic.</p>
    Fórmula:C16H19N3O5
    Pureza:99.76%
    Forma y color:Solid
    Peso molecular:333.34
  • FTIDC

    CAS:
    <p>FTIDC: potent, selective mGluR1 allosteric antagonist, weak on mGluR5. IC50: human 5.8 nM, mouse 3.1 nM. Noncompetitive.</p>
    Fórmula:C18H23FN6O
    Pureza:94.58%
    Forma y color:Solid
    Peso molecular:358.41
  • Milnacipran

    CAS:
    <p>Milnacipran, an SNRI with 85% bioavailability, treats fibromyalgia and is well absorbed orally.</p>
    Fórmula:C15H22N2O
    Forma y color:Solid
    Peso molecular:246.35
  • IC87201

    CAS:
    <p>IC87201 is a nNOS-PDZ/PSD-95-PDZ inhibitor. IC87201 showed great promise in cellular experiments and animal models of ischemic stroke and pain.</p>
    Fórmula:C13H10Cl2N4O
    Pureza:97.44%
    Forma y color:Solid
    Peso molecular:309.15
  • Oxyphenonium bromide

    CAS:
    <p>Oxyphenonium bromide is an anticholinergic used to study and treat ulcers and relieve visceral spasms.</p>
    Fórmula:C21H34BrNO3
    Pureza:98.96%
    Forma y color:Solid
    Peso molecular:428.404
  • RAGE antagonist peptide acetate


    <p>RAGE antagonist peptide acetate blocks RAGE-ligands like HMGB-1, has anti-tumor, and anti-inflammatory effects.</p>
    Fórmula:C59H105N13O19S
    Pureza:97.17%
    Forma y color:Solid
    Peso molecular:1332.61
  • Pipequaline hydrochloride

    CAS:
    <p>Pipequaline hydrochloride (PK-8165 hydrochloride) is an anticonflict &amp; anticonvulsant quinoline derivative.</p>
    Fórmula:C22H25ClN2
    Pureza:99.46%
    Forma y color:Solid
    Peso molecular:352.9
  • Perospirone hydrochloride

    CAS:
    <p>Perospirone hydrochloride (Perospirone HCl) is an atypical antipsychotic agent for the treatment of schizophrenia.</p>
    Fórmula:C23H31ClN4O2S
    Pureza:99.37%
    Forma y color:White Solid
    Peso molecular:463
  • Pimavanserin tartrate

    CAS:
    <p>Pimavanserin tartrate is a potent 5-HT 2A receptor inverse agonist used to treat Parkinson's disease-related psychosis.Cost-effective and quality-assured.</p>
    Fórmula:C50H68F2N6O4·C4H6O6
    Pureza:99.24% - 99.98%
    Forma y color:Solid
    Peso molecular:1005.2
  • SB 242084

    CAS:
    <p>SB 242084 dihydrochloride hydrate is a psychoactive drug and research chemical which acts as a selective antagonist for the 5HT2C receptor.</p>
    Fórmula:C21H19ClN4O2
    Pureza:99.75% - ≥98%
    Forma y color:Solid
    Peso molecular:394.85
  • SB-203186 hydrochloride

    CAS:
    <p>SB 203186 hydrochloride is a potent 5-HT4 receptor antagonist</p>
    Fórmula:C16H20N2O2·HCl
    Pureza:99.64%
    Forma y color:Solid
    Peso molecular:308.81
  • Jujuboside A

    CAS:
    <p>Jujuboside A: glycoside from Semen Ziziphi Spinosae, may treat Alzheimer's, has neuro-inhibitory effects.</p>
    Fórmula:C58H94O26
    Pureza:98% - >99.99%
    Forma y color:Solid
    Peso molecular:1207.35
  • L-701324

    CAS:
    <p>L-701324 is an NMDA receptor with high affinity and selectivity for the glycine site, used as an orally active and long-acting anticonvulsant.</p>
    Fórmula:C21H14ClNO3
    Pureza:98.63% - >99.99%
    Forma y color:Solid
    Peso molecular:363.79
  • Escitalopram Oxalate

    CAS:
    <p>Escitalopram Oxalate ((S)-(+)Citalopram oxalate) is a selective serotonin (5-HT) reuptake inhibitor (SSRI) with Ki of 0.89 nM.</p>
    Fórmula:C22H23FN2O5
    Pureza:97.39% - 99.73%
    Forma y color:White Solid
    Peso molecular:414.43
  • A-804598

    CAS:
    <p>A-804598 is a competitive and selective P2X7 receptor antagonist (IC50: 10 nM, rat; 9 nM, mouse; 11 nM, human).</p>
    Fórmula:C19H17N5
    Pureza:99.57%
    Forma y color:Solid
    Peso molecular:315.37
  • A 582941 HCl (848591-90-2(free base))


    <p>A-582941 is a alpha7 neuronal nicotinic receptor agonist with broad spectrum cognition-enhancing properties</p>
    Fórmula:C17H21ClN4
    Pureza:99.83%
    Forma y color:Solid
    Peso molecular:316.83
  • Aripiprazole monohydrate

    CAS:
    <p>Aripiprazole (OPC-14597) is a potent D2 partial agonist and inverse agonist of 5-HT2 receptors, used for schizophrenia and COVID-19 studies.</p>
    Fórmula:C23H29Cl2N3O3
    Forma y color:Solid
    Peso molecular:466.4
  • LY310762

    CAS:
    <p>LY310762 is a 5-HT1D receptor antagonist with Ki of 249 nM.</p>
    Fórmula:C24H27FN2O2·HCl
    Pureza:99.8%
    Forma y color:Solid
    Peso molecular:430.94
  • EUK-134

    CAS:
    <p>EUK-134, a synthetic SOD/catalase mimetic, exhibits potent antioxidant activities, and inhibits the formation of β-amyloid and related amyloid fibril.</p>
    Fórmula:C18H18ClMnN2O4
    Pureza:98.39%
    Forma y color:Solid
    Peso molecular:416.74
  • Azeliragon

    CAS:
    <p>Azeliragon (TTP488) is an antagonist at the Receptor for Advanced Glycation End products; is evaluated as a potential treatment for patients with mild-to-</p>
    Fórmula:C32H38ClN3O2
    Pureza:96.7% - 98.33%
    Forma y color:Solid
    Peso molecular:532.12