CymitQuimica logo
Neurociencia

Neurociencia

Los inhibidores en neurociencia son compuestos diseñados para modular la actividad de proteínas, enzimas o receptores específicos dentro del sistema nervioso. Estos inhibidores son cruciales para estudiar los mecanismos moleculares subyacentes a la función neuronal, la transmisión sináptica y las enfermedades neurodegenerativas. Al dirigirse a los receptores de neurotransmisores, canales iónicos y vías de señalización, los inhibidores en neurociencia ayudan en la exploración de la función cerebral y en el desarrollo de estrategias terapéuticas para trastornos neurológicos como el Alzheimer, Parkinson y la epilepsia. En CymitQuimica, ofrecemos una amplia gama de inhibidores de neurociencia de alta calidad para apoyar su investigación en neurobiología, neurofarmacología y ciencias cognitivas.

Subcategorías de "Neurociencia"

Mostrar 12 subcategorías más

Se han encontrado 5398 productos de "Neurociencia"

Ordenar por

Pureza (%)
0
100
|
0
|
50
|
90
|
95
|
100
productos por página.
  • Harmine

    CAS:
    <p>Harmine (Telepathine) is an alkaloid isolated from seeds of Peganum harmala.</p>
    Fórmula:C13H12N2O
    Pureza:98.29% - 99.92%
    Forma y color:Off-White Solid
    Peso molecular:212.25
  • Naftopidil dihydrochloride

    CAS:
    <p>Naftopidil dihydrochloride (KT-611 2HCl) is a selective 5-HT1A and α1-adrenergic receptor antagonist with IC50 of 0.1 μM and 0.2 μM, respectively.</p>
    Fórmula:C24H28N2O3·2HCl
    Pureza:99.76%
    Forma y color:White Solid
    Peso molecular:465.41
  • Idalopirdine Hydrochloride

    CAS:
    <p>Idalopirdine Hydrochloride (Lu AE58054 Hydrochloride) is an in-vivo binding affinity and effect, in-vitro selectivity and potency of 5-HT(6)R antagonist (Ki: 0.</p>
    Fórmula:C20H20ClF5N2O
    Pureza:99.77%
    Forma y color:Solid
    Peso molecular:434.83
  • p-Hydroxybenzaldehyde

    CAS:
    1.
    Fórmula:C7H6O2
    Pureza:99.05% - 99.86%
    Forma y color:Solid
    Peso molecular:122.12
  • Isocarboxazid

    CAS:
    <p>Isocarboxazid: a monoamine oxidase inhibitor used for various depression and anxiety disorders.</p>
    Fórmula:C12H13N3O2
    Pureza:98.32% - 99.94%
    Forma y color:Solid
    Peso molecular:231.25
  • JLK6

    CAS:
    <p>JLK6 was a gamma-secretase inhibitor that does not interfere with Notch signalling</p>
    Fórmula:C10H8ClNO3
    Pureza:96.50%
    Forma y color:Solid
    Peso molecular:225.63
  • MCI-225

    CAS:
    <p>MCI-225 is a selective inhibitor of NA reuptake with 5-HT3 receptor antagonism.</p>
    Fórmula:C17H17FN4S
    Pureza:99.32%
    Forma y color:Solid
    Peso molecular:328.4
  • NS3861

    CAS:
    <p>NS3861 is a selective agonist for α3β4/α4β2 nAChRs, preferring β-subunits, with no effect on α4-based receptors.</p>
    Fórmula:C12H14BrNS
    Pureza:99.853%
    Forma y color:Solid
    Peso molecular:284.22
  • 4F 4PP oxalate

    CAS:
    <p>4F 4PP oxalate is a 5-HT2A antagonist.</p>
    Fórmula:C22H26FNO·C2H2O4
    Pureza:97.34%
    Forma y color:Solid
    Peso molecular:429.49
  • Tasimelteon

    CAS:
    <p>Tasimelteon (BMS-214778) is a melatonin receptor agonist that is used for the treatment of non-24 hour sleep-wake disorder in blind individuals.</p>
    Fórmula:C15H19NO2
    Pureza:98.93% - 99.93%
    Forma y color:Solid
    Peso molecular:245.32
  • Fluralaner

    CAS:
    <p>Fluralaner (A1443) is an isoxazoline ectoparasiticide.</p>
    Fórmula:C22H17Cl2F6N3O3
    Pureza:99.72% - 99.90%
    Forma y color:Solid Powder
    Peso molecular:556.29
  • Ginsenoside Rc

    CAS:
    <p>Ginsenoside Rc (Panaxoside Rc) is one of the ginsenosides from Panax ginseng, inhibits the expression of TNF-α and IL-1β.</p>
    Fórmula:C53H90O22
    Pureza:98.83% - 99.56%
    Forma y color:White Powder
    Peso molecular:1079.27
  • NS11394

    CAS:
    <p>NS11394 is a effective and subtype-selective GABA(A) receptor-positive modulator; possesses a functional efficacy selectivity profile of α(5) &gt; α(3) &gt; α(2) &gt; α(</p>
    Fórmula:C23H19N3O
    Pureza:99.44% - 99.86%
    Forma y color:Solid
    Peso molecular:353.42
  • Fenchlorphos

    CAS:
    <p>Fenchlorphos (Dermafos) is a cholinesterase inhibitor, used as an insecticide.</p>
    Fórmula:C8H8Cl3O3PS
    Pureza:98% - >99.99%
    Forma y color:Colorless Crystals
    Peso molecular:321.55
  • ONO-8590580

    CAS:
    <p>ONO-8590580 (CS-2894) is a negative allosteric modulator of GABAA α5.</p>
    Fórmula:C21H21FN6
    Pureza:99.43%
    Forma y color:Solid
    Peso molecular:376.43
  • PHA 568487 free base

    CAS:
    <p>PHA 568487 free base, an α7 nicotinic receptor agonist, designed to reduce bioactivation and improve in vivo tolerability.</p>
    Fórmula:C16H20N2O3
    Pureza:99.74%
    Forma y color:Solid
    Peso molecular:288.34
  • VU-29

    CAS:
    <p>VU-29 is a positive allosteric mGlu5 receptor modulator with EC50=9 nM and Ki=244 nM for rmGluR5. It is selective for mGluR5 relative to other mGluR subtypes.</p>
    Fórmula:C22H16N4O3
    Pureza:99.63%
    Forma y color:Solid
    Peso molecular:384.39
  • L-701324

    CAS:
    <p>L-701324 is an NMDA receptor with high affinity and selectivity for the glycine site, used as an orally active and long-acting anticonvulsant.</p>
    Fórmula:C21H14ClNO3
    Pureza:98.63% - >99.99%
    Forma y color:Solid
    Peso molecular:363.79
  • Jujuboside A

    CAS:
    <p>Jujuboside A: glycoside from Semen Ziziphi Spinosae, may treat Alzheimer's, has neuro-inhibitory effects.</p>
    Fórmula:C58H94O26
    Pureza:98% - >99.99%
    Forma y color:Solid
    Peso molecular:1207.35
  • Perospirone hydrochloride

    CAS:
    <p>Perospirone hydrochloride (Perospirone HCl) is an atypical antipsychotic agent for the treatment of schizophrenia.</p>
    Fórmula:C23H31ClN4O2S
    Pureza:99.37%
    Forma y color:White Solid
    Peso molecular:463
  • RAGE antagonist peptide acetate


    <p>RAGE antagonist peptide acetate blocks RAGE-ligands like HMGB-1, has anti-tumor, and anti-inflammatory effects.</p>
    Fórmula:C59H105N13O19S
    Pureza:97.17%
    Forma y color:Solid
    Peso molecular:1332.61
  • FTIDC

    CAS:
    <p>FTIDC: potent, selective mGluR1 allosteric antagonist, weak on mGluR5. IC50: human 5.8 nM, mouse 3.1 nM. Noncompetitive.</p>
    Fórmula:C18H23FN6O
    Pureza:94.58%
    Forma y color:Solid
    Peso molecular:358.41
  • NAN-190 hydrobromide

    CAS:
    <p>NAN-190 hydrobromide is an antagonist of serotonin receptor 5-HT.</p>
    Fórmula:C23H28BrN3O3
    Pureza:95.20%
    Forma y color:Solid
    Peso molecular:474.39
  • ACH-000143

    CAS:
    <p>ACH-000143 是一种可口服的褪黑素受体激动剂,对 MT1 和 MT2 的EC50值分别为0.06 和0.32 nM。</p>
    Fórmula:C13H16ClN3O3
    Pureza:98.15%
    Forma y color:Solid
    Peso molecular:297.74
  • Medetomidine hydrochloride

    CAS:
    <p>Medetomidine hydrochloride (MPV785) is a selective α2-adrenoceptor agonist, with Ki of 1.08 nM, exhibts 1620-fold selectivity over α1-adrenoceptor.</p>
    Fórmula:C13H16N2·HCl
    Pureza:99.96%
    Forma y color:White Or Off White Crystalline Powder
    Peso molecular:236.74
  • JH-II-127

    CAS:
    <p>JH-II-127 is an oral LRRK2 inhibitor with IC50s: 6.6 nM (WT), 2.2 nM (G2019S), 47.7 nM (A2016T).</p>
    Fórmula:C19H21ClN6O3
    Pureza:98.32%
    Forma y color:Solid
    Peso molecular:416.86
  • 3-AQC

    CAS:
    <p>3-AQC is a competitive antagonist of 5-HT3.</p>
    Fórmula:C20H21N5O4
    Pureza:99.45%
    Forma y color:Solid
    Peso molecular:395.41
  • VU 0238429

    CAS:
    <p>VU 0238429 (SCR-1481B1) is positive allosteric modulator of muscarinic acetylcholine receptor subtype 5 (mAChR5 or M5)( EC50 : 1.16 μM).</p>
    Fórmula:C17H12F3NO4
    Pureza:>99.99%
    Forma y color:Solid
    Peso molecular:351.28
  • SB-334867 free base

    CAS:
    <p>SB-334867 free base (SB334867A free base) is a selective orexin-1 (OX1) receptor antagonist.</p>
    Fórmula:C17H13N5O2
    Pureza:99.67% - >99.99%
    Forma y color:Solid
    Peso molecular:319.32
  • Ipratropium Bromide

    CAS:
    <p>Ipratropium Bromide (Sch 1000) is an antagonist of muscarinic receptors and is used in COPD and asthma studies.</p>
    Fórmula:C20H30BrNO3
    Pureza:99.92%
    Forma y color:Solid
    Peso molecular:412.37
  • Homocarnosine acetate


    <p>Homocarnosine acetate is a dipeptide unique to brain consisting of γ-aminobutyric acid (GABA) and histidine.</p>
    Fórmula:C12H20N4O5
    Pureza:99.52%
    Forma y color:Solid
    Peso molecular:300.31
  • Mosapride

    CAS:
    <p>Mosapride (AS-4370) is a selective 5HT4 agonist</p>
    Fórmula:C21H25ClFN3O3
    Pureza:99.56%
    Forma y color:White To Off-White Crystalline Solid
    Peso molecular:421.89
  • Eliprodil

    CAS:
    <p>Eliprodil (SL-820715), NR2B-NMDA receptor blocker (IC50: 1 uM), less potent on NR2A/NR2C (IC50&gt;100 uM), explored for Parkinson's and movement issues.</p>
    Fórmula:C20H23ClFNO
    Pureza:99.53% - 99.77%
    Forma y color:Solid
    Peso molecular:347.85
  • TCN 201

    CAS:
    <p>TCN 201 is a selective antagonist of NMDA receptors containing the NR2A subunit.</p>
    Fórmula:C21H17ClFN3O4S
    Pureza:98.5%
    Forma y color:Solid
    Peso molecular:461.89
  • Xaliproden hydrochloride

    CAS:
    <p>Xaliproden is a compound that mimics the effects of nerve growth factor and is also a serotonin 5-HT1A receptor agonist.</p>
    Fórmula:C24H23ClF3N
    Pureza:99.99%
    Forma y color:Solid
    Peso molecular:417.89
  • GNE-7915

    CAS:
    <p>GNE-7915 is a highly potent, selective and brain-penetrable leucine-rich repeat kinase 2 (LRRK2) inhibitor.</p>
    Fórmula:C19H21F4N5O3
    Pureza:98% - ≥95%
    Forma y color:Solid
    Peso molecular:443.4
  • MK-0752

    CAS:
    <p>MK-0752, a γ-secretase inhibitor, reduces Aβ40 production(IC50=5 nM).</p>
    Fórmula:C21H21ClF2O4S
    Pureza:98% - 99.55%
    Forma y color:Solid
    Peso molecular:442.9
  • Tianeptine sodium salt

    CAS:
    <p>Tianeptine sodium salt 是一种选择性5-HT 摄取促进剂,具有抗抑郁、抗焦虑和神经保护作用,可用于缓解疼痛的研究。</p>
    Fórmula:C21H24ClN2NaO4S
    Pureza:99.82%
    Forma y color:Solid
    Peso molecular:458.93
  • JHU37160

    CAS:
    JHU37160 is a DREADD agonist with Ki of 1.9 nM for hM3Dq, 3.6 nM for hM4Di, and EC50 of 18.5 nM (hM3Dq), 0.2 nM (hM4Di) in HEK-293 cell assays.
    Fórmula:C19H20ClFN4
    Pureza:99.87%
    Forma y color:Solid
    Peso molecular:358.84
  • RO4929097

    CAS:
    <p>RO4929097 (RG-4733), a γ secretase inhibitor (IC50: 4 nM), inhibits cellular processing of Aβ40 and Notch (EC50: 14/5 nM).</p>
    Fórmula:C22H20F5N3O3
    Pureza:98.5% - 99.51%
    Forma y color:Solid
    Peso molecular:469.4
  • E4CPG

    CAS:
    <p>E4CPG is a novel group I/II metabotropic glutamate receptor antagonist, more potent than (RS)-MCPG.</p>
    Fórmula:C11H13NO4
    Pureza:99.96%
    Forma y color:Solid
    Peso molecular:223.23
  • Radiprodil

    CAS:
    <p>Radiprodil (RGH-896) is an oral NMDA NR2B antagonist for potential DPNP neuropathic pain treatment.</p>
    Fórmula:C21H20FN3O4
    Pureza:99.74%
    Forma y color:Solid
    Peso molecular:397.4
  • Cariprazine hydrochloride

    CAS:
    <p>Cariprazine hydrochloride (RGH188 hydrochloride) is an antipsychotic drug, is a D3 and D2 receptor partial agonist((Ki of 0.085 nM and 0.49 nM, respectively)</p>
    Fórmula:C21H33Cl3N4O
    Pureza:99.78% - >99.99%
    Forma y color:Solid
    Peso molecular:463.87
  • Polmacoxib

    CAS:
    <p>Polmacoxib, a first-class NSAID, dual inhibitor of CA and COX-2, may hinder colorectal cancer growth in mice.</p>
    Fórmula:C18H16FNO4S
    Pureza:97.88%
    Forma y color:Solid
    Peso molecular:361.39
  • Methylbenactyzium Bromide

    CAS:
    <p>Methylbenactyzium Bromide (Semulgin) is an anticonvulsant that is the active metabolite of trimethadione.</p>
    Fórmula:C21H28BrNO3
    Pureza:99.29%
    Forma y color:Solid
    Peso molecular:422.36
  • CZC-54252

    CAS:
    <p>CZC-54252 is a potent inhibitor of LRRK2.</p>
    Fórmula:C22H25ClN6O4S
    Pureza:99.39%
    Forma y color:Solid
    Peso molecular:504.99
  • DORA-22

    CAS:
    <p>DORA-22 is a dual orexin receptor antagonist, improves mild stress-induced insomnia with minimal effect on memory</p>
    Fórmula:C23H22F2N4O2
    Pureza:97.67%
    Forma y color:Solid
    Peso molecular:424.44
  • Chelidamic acid

    CAS:
    <p>Chelidamic acid is a heterocyclic organic acid with a pyran skeleton. Chelidamic acid is inhibitors of glutamate decarboxylase, with a Ki of 33 μM.</p>
    Fórmula:C7H5NO5
    Pureza:98.11%
    Forma y color:Pale Yellow Powder
    Peso molecular:183.12
  • Suprofen

    CAS:
    <p>Suprofen (Suprol) is an IBUPROFEN-type anti-inflammatory analgesic and antipyretic.</p>
    Fórmula:C14H12O3S
    Pureza:99.23% - 99.33%
    Forma y color:Solid
    Peso molecular:260.31
  • Tinoridine hydrochloride

    CAS:
    <p>Tinoridine HCl is an NSAID that inhibits lipid peroxides and renin release, unlike indomethacin and corticosteroids.</p>
    Fórmula:C17H21ClN2O2S
    Pureza:97.49%
    Forma y color:Solid
    Peso molecular:352.88