
Neurociencia
Los inhibidores en neurociencia son compuestos diseñados para modular la actividad de proteínas, enzimas o receptores específicos dentro del sistema nervioso. Estos inhibidores son cruciales para estudiar los mecanismos moleculares subyacentes a la función neuronal, la transmisión sináptica y las enfermedades neurodegenerativas. Al dirigirse a los receptores de neurotransmisores, canales iónicos y vías de señalización, los inhibidores en neurociencia ayudan en la exploración de la función cerebral y en el desarrollo de estrategias terapéuticas para trastornos neurológicos como el Alzheimer, Parkinson y la epilepsia. En CymitQuimica, ofrecemos una amplia gama de inhibidores de neurociencia de alta calidad para apoyar su investigación en neurobiología, neurofarmacología y ciencias cognitivas.
Subcategorías de "Neurociencia"
- Receptor 5-HT(939 productos)
- ACK(1 productos)
- AChR(575 productos)
- ATP Citrato Liasa(16 productos)
- Receptor adrenérgico(2.945 productos)
- BACE(36 productos)
- Beta amiloide(205 productos)
- CAMK(69 productos)
- Inhibidores de ciclooxigenasa (COX)(561 productos)
- Receptor de dopamina(407 productos)
- Receptor GABA(336 productos)
- Gamma-secretasa(59 productos)
- GluR(255 productos)
- GlyT(24 productos)
- Receptor de histamina(358 productos)
- LRRK2(33 productos)
- Receptor de melatonina(24 productos)
- NMDAR(28 productos)
- Receptor de OX(40 productos)
- Receptor de opioides(297 productos)
Mostrar 12 subcategorías más
Se han encontrado 5398 productos de "Neurociencia"
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Harmine
CAS:<p>Harmine (Telepathine) is an alkaloid isolated from seeds of Peganum harmala.</p>Fórmula:C13H12N2OPureza:98.29% - 99.92%Forma y color:Off-White SolidPeso molecular:212.25Naftopidil dihydrochloride
CAS:<p>Naftopidil dihydrochloride (KT-611 2HCl) is a selective 5-HT1A and α1-adrenergic receptor antagonist with IC50 of 0.1 μM and 0.2 μM, respectively.</p>Fórmula:C24H28N2O3·2HClPureza:99.76%Forma y color:White SolidPeso molecular:465.41Idalopirdine Hydrochloride
CAS:<p>Idalopirdine Hydrochloride (Lu AE58054 Hydrochloride) is an in-vivo binding affinity and effect, in-vitro selectivity and potency of 5-HT(6)R antagonist (Ki: 0.</p>Fórmula:C20H20ClF5N2OPureza:99.77%Forma y color:SolidPeso molecular:434.83p-Hydroxybenzaldehyde
CAS:1.Fórmula:C7H6O2Pureza:99.05% - 99.86%Forma y color:SolidPeso molecular:122.12Isocarboxazid
CAS:<p>Isocarboxazid: a monoamine oxidase inhibitor used for various depression and anxiety disorders.</p>Fórmula:C12H13N3O2Pureza:98.32% - 99.94%Forma y color:SolidPeso molecular:231.25JLK6
CAS:<p>JLK6 was a gamma-secretase inhibitor that does not interfere with Notch signalling</p>Fórmula:C10H8ClNO3Pureza:96.50%Forma y color:SolidPeso molecular:225.63MCI-225
CAS:<p>MCI-225 is a selective inhibitor of NA reuptake with 5-HT3 receptor antagonism.</p>Fórmula:C17H17FN4SPureza:99.32%Forma y color:SolidPeso molecular:328.4NS3861
CAS:<p>NS3861 is a selective agonist for α3β4/α4β2 nAChRs, preferring β-subunits, with no effect on α4-based receptors.</p>Fórmula:C12H14BrNSPureza:99.853%Forma y color:SolidPeso molecular:284.224F 4PP oxalate
CAS:<p>4F 4PP oxalate is a 5-HT2A antagonist.</p>Fórmula:C22H26FNO·C2H2O4Pureza:97.34%Forma y color:SolidPeso molecular:429.49Tasimelteon
CAS:<p>Tasimelteon (BMS-214778) is a melatonin receptor agonist that is used for the treatment of non-24 hour sleep-wake disorder in blind individuals.</p>Fórmula:C15H19NO2Pureza:98.93% - 99.93%Forma y color:SolidPeso molecular:245.32Fluralaner
CAS:<p>Fluralaner (A1443) is an isoxazoline ectoparasiticide.</p>Fórmula:C22H17Cl2F6N3O3Pureza:99.72% - 99.90%Forma y color:Solid PowderPeso molecular:556.29Ginsenoside Rc
CAS:<p>Ginsenoside Rc (Panaxoside Rc) is one of the ginsenosides from Panax ginseng, inhibits the expression of TNF-α and IL-1β.</p>Fórmula:C53H90O22Pureza:98.83% - 99.56%Forma y color:White PowderPeso molecular:1079.27NS11394
CAS:<p>NS11394 is a effective and subtype-selective GABA(A) receptor-positive modulator; possesses a functional efficacy selectivity profile of α(5) > α(3) > α(2) > α(</p>Fórmula:C23H19N3OPureza:99.44% - 99.86%Forma y color:SolidPeso molecular:353.42Fenchlorphos
CAS:<p>Fenchlorphos (Dermafos) is a cholinesterase inhibitor, used as an insecticide.</p>Fórmula:C8H8Cl3O3PSPureza:98% - >99.99%Forma y color:Colorless CrystalsPeso molecular:321.55ONO-8590580
CAS:<p>ONO-8590580 (CS-2894) is a negative allosteric modulator of GABAA α5.</p>Fórmula:C21H21FN6Pureza:99.43%Forma y color:SolidPeso molecular:376.43PHA 568487 free base
CAS:<p>PHA 568487 free base, an α7 nicotinic receptor agonist, designed to reduce bioactivation and improve in vivo tolerability.</p>Fórmula:C16H20N2O3Pureza:99.74%Forma y color:SolidPeso molecular:288.34VU-29
CAS:<p>VU-29 is a positive allosteric mGlu5 receptor modulator with EC50=9 nM and Ki=244 nM for rmGluR5. It is selective for mGluR5 relative to other mGluR subtypes.</p>Fórmula:C22H16N4O3Pureza:99.63%Forma y color:SolidPeso molecular:384.39L-701324
CAS:<p>L-701324 is an NMDA receptor with high affinity and selectivity for the glycine site, used as an orally active and long-acting anticonvulsant.</p>Fórmula:C21H14ClNO3Pureza:98.63% - >99.99%Forma y color:SolidPeso molecular:363.79Jujuboside A
CAS:<p>Jujuboside A: glycoside from Semen Ziziphi Spinosae, may treat Alzheimer's, has neuro-inhibitory effects.</p>Fórmula:C58H94O26Pureza:98% - >99.99%Forma y color:SolidPeso molecular:1207.35Perospirone hydrochloride
CAS:<p>Perospirone hydrochloride (Perospirone HCl) is an atypical antipsychotic agent for the treatment of schizophrenia.</p>Fórmula:C23H31ClN4O2SPureza:99.37%Forma y color:White SolidPeso molecular:463RAGE antagonist peptide acetate
<p>RAGE antagonist peptide acetate blocks RAGE-ligands like HMGB-1, has anti-tumor, and anti-inflammatory effects.</p>Fórmula:C59H105N13O19SPureza:97.17%Forma y color:SolidPeso molecular:1332.61FTIDC
CAS:<p>FTIDC: potent, selective mGluR1 allosteric antagonist, weak on mGluR5. IC50: human 5.8 nM, mouse 3.1 nM. Noncompetitive.</p>Fórmula:C18H23FN6OPureza:94.58%Forma y color:SolidPeso molecular:358.41NAN-190 hydrobromide
CAS:<p>NAN-190 hydrobromide is an antagonist of serotonin receptor 5-HT.</p>Fórmula:C23H28BrN3O3Pureza:95.20%Forma y color:SolidPeso molecular:474.39ACH-000143
CAS:<p>ACH-000143 是一种可口服的褪黑素受体激动剂,对 MT1 和 MT2 的EC50值分别为0.06 和0.32 nM。</p>Fórmula:C13H16ClN3O3Pureza:98.15%Forma y color:SolidPeso molecular:297.74Medetomidine hydrochloride
CAS:<p>Medetomidine hydrochloride (MPV785) is a selective α2-adrenoceptor agonist, with Ki of 1.08 nM, exhibts 1620-fold selectivity over α1-adrenoceptor.</p>Fórmula:C13H16N2·HClPureza:99.96%Forma y color:White Or Off White Crystalline PowderPeso molecular:236.74JH-II-127
CAS:<p>JH-II-127 is an oral LRRK2 inhibitor with IC50s: 6.6 nM (WT), 2.2 nM (G2019S), 47.7 nM (A2016T).</p>Fórmula:C19H21ClN6O3Pureza:98.32%Forma y color:SolidPeso molecular:416.863-AQC
CAS:<p>3-AQC is a competitive antagonist of 5-HT3.</p>Fórmula:C20H21N5O4Pureza:99.45%Forma y color:SolidPeso molecular:395.41VU 0238429
CAS:<p>VU 0238429 (SCR-1481B1) is positive allosteric modulator of muscarinic acetylcholine receptor subtype 5 (mAChR5 or M5)( EC50 : 1.16 μM).</p>Fórmula:C17H12F3NO4Pureza:>99.99%Forma y color:SolidPeso molecular:351.28SB-334867 free base
CAS:<p>SB-334867 free base (SB334867A free base) is a selective orexin-1 (OX1) receptor antagonist.</p>Fórmula:C17H13N5O2Pureza:99.67% - >99.99%Forma y color:SolidPeso molecular:319.32Ipratropium Bromide
CAS:<p>Ipratropium Bromide (Sch 1000) is an antagonist of muscarinic receptors and is used in COPD and asthma studies.</p>Fórmula:C20H30BrNO3Pureza:99.92%Forma y color:SolidPeso molecular:412.37Homocarnosine acetate
<p>Homocarnosine acetate is a dipeptide unique to brain consisting of γ-aminobutyric acid (GABA) and histidine.</p>Fórmula:C12H20N4O5Pureza:99.52%Forma y color:SolidPeso molecular:300.31Mosapride
CAS:<p>Mosapride (AS-4370) is a selective 5HT4 agonist</p>Fórmula:C21H25ClFN3O3Pureza:99.56%Forma y color:White To Off-White Crystalline SolidPeso molecular:421.89Eliprodil
CAS:<p>Eliprodil (SL-820715), NR2B-NMDA receptor blocker (IC50: 1 uM), less potent on NR2A/NR2C (IC50>100 uM), explored for Parkinson's and movement issues.</p>Fórmula:C20H23ClFNOPureza:99.53% - 99.77%Forma y color:SolidPeso molecular:347.85TCN 201
CAS:<p>TCN 201 is a selective antagonist of NMDA receptors containing the NR2A subunit.</p>Fórmula:C21H17ClFN3O4SPureza:98.5%Forma y color:SolidPeso molecular:461.89Xaliproden hydrochloride
CAS:<p>Xaliproden is a compound that mimics the effects of nerve growth factor and is also a serotonin 5-HT1A receptor agonist.</p>Fórmula:C24H23ClF3NPureza:99.99%Forma y color:SolidPeso molecular:417.89GNE-7915
CAS:<p>GNE-7915 is a highly potent, selective and brain-penetrable leucine-rich repeat kinase 2 (LRRK2) inhibitor.</p>Fórmula:C19H21F4N5O3Pureza:98% - ≥95%Forma y color:SolidPeso molecular:443.4MK-0752
CAS:<p>MK-0752, a γ-secretase inhibitor, reduces Aβ40 production(IC50=5 nM).</p>Fórmula:C21H21ClF2O4SPureza:98% - 99.55%Forma y color:SolidPeso molecular:442.9Tianeptine sodium salt
CAS:<p>Tianeptine sodium salt 是一种选择性5-HT 摄取促进剂,具有抗抑郁、抗焦虑和神经保护作用,可用于缓解疼痛的研究。</p>Fórmula:C21H24ClN2NaO4SPureza:99.82%Forma y color:SolidPeso molecular:458.93JHU37160
CAS:JHU37160 is a DREADD agonist with Ki of 1.9 nM for hM3Dq, 3.6 nM for hM4Di, and EC50 of 18.5 nM (hM3Dq), 0.2 nM (hM4Di) in HEK-293 cell assays.Fórmula:C19H20ClFN4Pureza:99.87%Forma y color:SolidPeso molecular:358.84RO4929097
CAS:<p>RO4929097 (RG-4733), a γ secretase inhibitor (IC50: 4 nM), inhibits cellular processing of Aβ40 and Notch (EC50: 14/5 nM).</p>Fórmula:C22H20F5N3O3Pureza:98.5% - 99.51%Forma y color:SolidPeso molecular:469.4E4CPG
CAS:<p>E4CPG is a novel group I/II metabotropic glutamate receptor antagonist, more potent than (RS)-MCPG.</p>Fórmula:C11H13NO4Pureza:99.96%Forma y color:SolidPeso molecular:223.23Radiprodil
CAS:<p>Radiprodil (RGH-896) is an oral NMDA NR2B antagonist for potential DPNP neuropathic pain treatment.</p>Fórmula:C21H20FN3O4Pureza:99.74%Forma y color:SolidPeso molecular:397.4Cariprazine hydrochloride
CAS:<p>Cariprazine hydrochloride (RGH188 hydrochloride) is an antipsychotic drug, is a D3 and D2 receptor partial agonist((Ki of 0.085 nM and 0.49 nM, respectively)</p>Fórmula:C21H33Cl3N4OPureza:99.78% - >99.99%Forma y color:SolidPeso molecular:463.87Polmacoxib
CAS:<p>Polmacoxib, a first-class NSAID, dual inhibitor of CA and COX-2, may hinder colorectal cancer growth in mice.</p>Fórmula:C18H16FNO4SPureza:97.88%Forma y color:SolidPeso molecular:361.39Methylbenactyzium Bromide
CAS:<p>Methylbenactyzium Bromide (Semulgin) is an anticonvulsant that is the active metabolite of trimethadione.</p>Fórmula:C21H28BrNO3Pureza:99.29%Forma y color:SolidPeso molecular:422.36CZC-54252
CAS:<p>CZC-54252 is a potent inhibitor of LRRK2.</p>Fórmula:C22H25ClN6O4SPureza:99.39%Forma y color:SolidPeso molecular:504.99DORA-22
CAS:<p>DORA-22 is a dual orexin receptor antagonist, improves mild stress-induced insomnia with minimal effect on memory</p>Fórmula:C23H22F2N4O2Pureza:97.67%Forma y color:SolidPeso molecular:424.44Chelidamic acid
CAS:<p>Chelidamic acid is a heterocyclic organic acid with a pyran skeleton. Chelidamic acid is inhibitors of glutamate decarboxylase, with a Ki of 33 μM.</p>Fórmula:C7H5NO5Pureza:98.11%Forma y color:Pale Yellow PowderPeso molecular:183.12Suprofen
CAS:<p>Suprofen (Suprol) is an IBUPROFEN-type anti-inflammatory analgesic and antipyretic.</p>Fórmula:C14H12O3SPureza:99.23% - 99.33%Forma y color:SolidPeso molecular:260.31Tinoridine hydrochloride
CAS:<p>Tinoridine HCl is an NSAID that inhibits lipid peroxides and renin release, unlike indomethacin and corticosteroids.</p>Fórmula:C17H21ClN2O2SPureza:97.49%Forma y color:SolidPeso molecular:352.88
