
Neurociencia
Los inhibidores en neurociencia son compuestos diseñados para modular la actividad de proteínas, enzimas o receptores específicos dentro del sistema nervioso. Estos inhibidores son cruciales para estudiar los mecanismos moleculares subyacentes a la función neuronal, la transmisión sináptica y las enfermedades neurodegenerativas. Al dirigirse a los receptores de neurotransmisores, canales iónicos y vías de señalización, los inhibidores en neurociencia ayudan en la exploración de la función cerebral y en el desarrollo de estrategias terapéuticas para trastornos neurológicos como el Alzheimer, Parkinson y la epilepsia. En CymitQuimica, ofrecemos una amplia gama de inhibidores de neurociencia de alta calidad para apoyar su investigación en neurobiología, neurofarmacología y ciencias cognitivas.
Subcategorías de "Neurociencia"
- Receptor 5-HT(985 productos)
- ACK(1 productos)
- AChR(613 productos)
- ATP Citrato Liasa(17 productos)
- Receptor adrenérgico(2.991 productos)
- BACE(36 productos)
- Beta amiloide(216 productos)
- CAMK(71 productos)
- Inhibidores de ciclooxigenasa (COX)(583 productos)
- Receptor de dopamina(433 productos)
- Receptor GABA(351 productos)
- Gamma-secretasa(63 productos)
- GluR(261 productos)
- GlyT(24 productos)
- Receptor de histamina(380 productos)
- LRRK2(41 productos)
- Receptor de melatonina(26 productos)
- NMDAR(22 productos)
- Receptor de OX(41 productos)
- Receptor de opioides(309 productos)
Mostrar 12 subcategorías más
Se han encontrado 5520 productos de "Neurociencia"
Ordenar por
Pureza (%)
0
100
|
0
|
50
|
90
|
95
|
100
Cgp 52608
CAS:CGP 52608 is a selective ligand for RAR-associated orphan receptor alpha.Fórmula:C8H12N4OS2Forma y color:SolidPeso molecular:244.34AZD-9164 bromide
CAS:AMG-221, a selective 11β-HSD1 inhibitor, suppresses enzyme activity, lowers glucose/insulin, and reduces weight in obese mice.Fórmula:C29H38BrFN2O2Forma y color:SolidPeso molecular:545.53Caramiphen hydrochloride
CAS:Caramiphen hydrochloride: antimuscarinic, anticholinergic, NMDA receptor antagonist salt.Fórmula:C18H28ClNO2Forma y color:SolidPeso molecular:325.88Metanicotine
CAS:Metanicotine is a selective nicotinic agonist with antinociceptive properties.Fórmula:C10H14N2Forma y color:SolidPeso molecular:162.23LC kinetic stabilizer-2
CAS:LC Kinetic Stabilizer-2 is a powerful stabilizer for amyloidogenic immunoglobulin light chains (LC), demonstrating significant efficacy with an EC50 of 24 nM.Fórmula:C28H31N3O3Forma y color:SolidPeso molecular:457.56N-Nitroso Fluoxetine
CAS:N-Nitroso fluoxetine is a derivative of fluoxetine.1It is genotoxic toS. typhimuriumwhen used at concentrations ranging from 0.06 to 0.12 mg/ml.Fórmula:C17H17F3N2O2Forma y color:SolidPeso molecular:338.32CFM-2
CAS:<p>CFM-2, a potent and selective non-competitive antagonist of AMPAR (AMPAR), exhibits anticonvulsant activity across various seizure models.</p>Fórmula:C17H17N3O3Pureza:99.84%Forma y color:SolidPeso molecular:311.34Octamylamine sulfamate
CAS:Octamylamine sulfamate is a P450 inhibitor.Fórmula:C13H32N2O3SForma y color:SolidPeso molecular:296.47Zimelidine
CAS:Zimelidine, a withdrawn antidepressant, posed Guillain-Barre risk.Fórmula:C16H17BrN2Pureza:98%Forma y color:SolidPeso molecular:317.22Fonazine mesylate
CAS:Fonazine mesylate is a phenothiazine drug used for the treatment of migraine. It is a serotonin antagonist and histamine antagonist.Fórmula:C20H29N3O5S3Forma y color:SolidPeso molecular:487.65Hadacidin sodium
CAS:Hadacidin sodium is an inhibitor of AMP synthesis. Hadacidin and hadacidin analogues have anticancer activity and activity against adenylosuccinate synthetase.Fórmula:C3H4NNaO4Forma y color:SolidPeso molecular:141.06RJR-2429
CAS:RJR-2429 is a potent AChR agonist.Fórmula:C12H16N2Forma y color:SolidPeso molecular:188.27VER-3323
CAS:VER-3323 is a selective agonist for the 5-HT2B and 5-HT2C serotonin receptor with potent anorectic effects in animal studies.Fórmula:C11H15BrN2Pureza:98%Forma y color:SolidPeso molecular:255.15Iferanserin HCl
CAS:Iferanserin HCl is a selective serotonin receptor antagonist.Fórmula:C23H29ClN2OForma y color:SolidPeso molecular:384.95Echothiophate chloride
CAS:Echothiophate: long-lasting cholinesterase inhibitor for chronic glaucoma treatment; binds irreversibly, inactivating the enzyme.Fórmula:C9H23ClNO3PSForma y color:SolidPeso molecular:291.7708PF-06663195
CAS:PF-06663195 is a potent inhibitor of β-site amyloid precursor protein (APP) Cleaving Enzyme 1 (BACE1, β-Secretase 1).Fórmula:C18H18F3N3O2SForma y color:SolidPeso molecular:397.41A-850002
CAS:A-850002 is a bioactive chemical.Fórmula:C18H16N4OSForma y color:SolidPeso molecular:336.41SH-053-S-CH3-2'F
CAS:SH-053-S-CH3-2'F is a potent and selective agonist of GABAA receptors.Fórmula:C23H18FN3O2Forma y color:SolidPeso molecular:387.41Milacemide HCl
CAS:Milacemide HCl is an MAO-B inhibitor and glycine prodrug.Fórmula:C7H17ClN2OPureza:98%Forma y color:SolidPeso molecular:180.68DH-97
CAS:DH-97 is a potent MT2 melatonin receptor antagonist (pKi value = 8.03).Fórmula:C22H26N2OForma y color:SolidPeso molecular:334.45Methacholine iodide
CAS:Methacholine iodide is a muscarinic acetylcholine receptor agonist.Fórmula:C8H18INO2Forma y color:SolidPeso molecular:287.14(R,R)-Glycopyrrolate
CAS:(R,R)-Glycopyrrolate is an agent of anticholinergic, has the ability to reduce the frequency of drooling in vivo with developmental disabilities.Fórmula:C19H28BrNO3Pureza:98%Forma y color:SolidPeso molecular:398.34VU0486321
CAS:VU0486321: potent mGlu1 PAM, rat PK CLp 13.3 mL/min/kg, t1/2 54 min, human fu 0.05, rat fu 0.03, great CNS penetration Kp 1.02.Fórmula:C20H12ClFN2O4Forma y color:SolidPeso molecular:398.77Neopterin, L-erythro-
CAS:Neopterin, L-erythro- can be used as a cholinergic receptor.Fórmula:C9H11N5O4Forma y color:SolidPeso molecular:253.21Asoxime dichloride
CAS:<p>Asoxime dichloride (HI-6) blocks AChRs, including α7 nAChR, and boosts vaccination in the nervous system.</p>Fórmula:C14H16Cl2N4O3Pureza:99.86%Forma y color:SolidPeso molecular:359.21Thiothixene hydrochloride
CAS:Thiothixene hydrochloride is an antipsychotic agent that can be used in the study of schizophrenia and bipolar mania.Fórmula:C23H30ClN3O2S2Forma y color:SolidPeso molecular:480.08Hadacidin
CAS:Hadacidin is an inhibitor of AMP synthesis. Hadacidin and hadacidin analogues have anticancer activity and activity against adenylosuccinate synthetase.Fórmula:C3H5NO4Forma y color:SolidPeso molecular:119.08VRX 03011 Potassium salt
CAS:VRX 03011, a 5-HT4 partial agonist, is used potentially for the treatment of Alzheimer's disease.Fórmula:C19H27KN3O3SPureza:98%Forma y color:SolidPeso molecular:416.6PF-06767832
CAS:PF-06767832: selective M1 PAM (EC50=60 nM), no M2-M5 activity, good CNS penetration, but has GI and cardiovascular risks.Fórmula:C22H23N3O3SForma y color:SolidPeso molecular:409.5q-FTAA
CAS:q-FTAA targets Aβ1-42 fibrils (330-630 nM) and ADPBC (300-500 nM), useful in Alzheimer's disease research.Fórmula:C21H14O6S4Forma y color:SolidPeso molecular:490.59MD 780236
CAS:MD 780236 is a monoamine oxidase-B inhibitor.Fórmula:C18H19ClN2O3Forma y color:SolidPeso molecular:346.81Almoxatone
CAS:Almoxatone, also known as MD 780236, is a monoamine oxidase (MAO) inhibitor.Fórmula:C18H19ClN2O3Forma y color:SolidPeso molecular:346.81Levomepromazine Maleate
CAS:Levomepromazine Maleate: TCA and SNRI with antihistamine, antiadrenergic, and anticholinergic properties.Fórmula:C23H28N2O5SForma y color:SolidPeso molecular:444.546F-15599 tosylate
CAS:F-15599 tosylate is a selective 5-HT(1A) agonist.Fórmula:C26H29ClF2N4O4SForma y color:SolidPeso molecular:567.05Neostigmine hydroxide
CAS:Neostigmine hydroxide, a cholinesterase inhibitor, treats myasthenia gravis and reverses muscle relaxants; doesn't cross the blood-brain barrier.Fórmula:C12H20N2O3Forma y color:SolidPeso molecular:240.3Atropine Oxide Hydrochloride
CAS:Atropine Oxide, a derivative of anticholinergic Atropine, treats poisonings, slow heart rate, and reduces saliva during surgery.Fórmula:C17H24ClNO4Forma y color:SolidPeso molecular:341.83Tropatepine
CAS:Tropatepine: oral anticholinergic, treats extrapyramidal symptoms, anti-Parkinson's.Fórmula:C22H23NSForma y color:SolidPeso molecular:333.49Ethybenztropine HBr
CAS:Ethybenztropine HBr is an anticholinergic which is used as an antiparkinsonian agent. Ethybenztropine may also act as a dopamine reuptake inhibitor.Fórmula:C22H28BrNOForma y color:SolidPeso molecular:402.37SCH-23390 maleate
CAS:<p>SCH-23390 maleate (R-(+)-SCH-23390 maleate) is a potent and selective antagonist of dopamine D1-like receptor (1 and D5 receptor with Kis of 0.2 nM and 0.3 nM,</p>Fórmula:C21H22ClNO5Pureza:98%Forma y color:SolidPeso molecular:403.86Ciclotizolam
CAS:Ciclotizolam, a thienotriazolodiazepine derivative and partial GABAA receptor agonist, has low efficacy but similar affinity as brotizolam.Fórmula:C20H18BrClN4SForma y color:SolidPeso molecular:461.81(E/Z)-VU0029767
CAS:VU0029767 enhances M1 muscarinic receptor function, increasing acetylcholine potency and efficacy.Fórmula:C21H21N3O3Forma y color:SolidPeso molecular:363.41Dexetimide HCl
CAS:Dexetimide HCl is a muscarinic antagonist that has been used to treat neuroleptic-induced parkinsonism. Benzetimide is the (-)-enantimorph of dexetimide.Fórmula:C23H27ClN2O2Forma y color:SolidPeso molecular:398.93NW-1772 free base
CAS:NW-1772 free base is a monoamine oxidase B inhibitor.Fórmula:C18H16ClNO3Forma y color:SolidPeso molecular:329.78UH-AH 37
CAS:UH-AH 37 is a antagonist of human muscarinic acetylcholine receptor.Fórmula:C21H23Cl2N3O2Pureza:98%Forma y color:SolidPeso molecular:420.33CC4
CAS:Selective α6β2/α4β2 partial agonist; Ki: 12/26nM (rat); poor α3β4/α7 affinity; stimulates dopamine release; reduces nicotine self-admin in rats.Fórmula:C24H30N4O2Forma y color:SolidPeso molecular:406.52Fonazine hydrochloride
CAS:Fonazine hydrochloride is a phenothiazine drug used for the treatment of migraine. It is a serotonin antagonist and histamine antagonist.Fórmula:C19H26ClN3O2S2Forma y color:SolidPeso molecular:428.01Pd 158771
CAS:Pd 158771 is a D2 and 5-HT1A agonist.Fórmula:C22H31N5Forma y color:SolidPeso molecular:365.52SC 53116 Hydrochloride
CAS:SC 53116 Hydrochloride is selective agonist of the newly identified serotonin 5-HT4 receptor subtype.Fórmula:C16H23Cl2N3O2Forma y color:SolidPeso molecular:360.28Way 100135
CAS:WAY-100135: research drug, phenylpiperazine, potent 5-HT1A antagonist, partial 5-HT1D agonist, minor 5-HT1B activity.Fórmula:C24H33N3O2Forma y color:SolidPeso molecular:395.54AQ-RA 721
CAS:AQ-RA 721 is a selective muscarinic antagonist with high affinity for M1- and M3-receptors. AQ-RA 721 may be used as a bronchodilator.Fórmula:C22H23N3O2Forma y color:SolidPeso molecular:361.44
