
Neurociencia
Los inhibidores en neurociencia son compuestos diseñados para modular la actividad de proteínas, enzimas o receptores específicos dentro del sistema nervioso. Estos inhibidores son cruciales para estudiar los mecanismos moleculares subyacentes a la función neuronal, la transmisión sináptica y las enfermedades neurodegenerativas. Al dirigirse a los receptores de neurotransmisores, canales iónicos y vías de señalización, los inhibidores en neurociencia ayudan en la exploración de la función cerebral y en el desarrollo de estrategias terapéuticas para trastornos neurológicos como el Alzheimer, Parkinson y la epilepsia. En CymitQuimica, ofrecemos una amplia gama de inhibidores de neurociencia de alta calidad para apoyar su investigación en neurobiología, neurofarmacología y ciencias cognitivas.
Subcategorías de "Neurociencia"
- Receptor 5-HT(942 productos)
- ACK(1 productos)
- AChR(576 productos)
- ATP Citrato Liasa(16 productos)
- Receptor adrenérgico(2.949 productos)
- BACE(36 productos)
- Beta amiloide(205 productos)
- CAMK(69 productos)
- Inhibidores de ciclooxigenasa (COX)(565 productos)
- Receptor de dopamina(410 productos)
- Receptor GABA(337 productos)
- Gamma-secretasa(59 productos)
- GluR(255 productos)
- GlyT(24 productos)
- Receptor de histamina(359 productos)
- LRRK2(33 productos)
- Receptor de melatonina(24 productos)
- NMDAR(26 productos)
- Receptor de OX(40 productos)
- Receptor de opioides(298 productos)
Mostrar 12 subcategorías más
Se han encontrado 5389 productos de "Neurociencia"
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Nerispirdine HCl
CAS:Nerispirdine enhances acetylcholine, blocks Na+ channels (IC50 11.9µM) and K(v) 1.1/1.2 channels (IC50 3.6/3.7µM).Fórmula:C17H19ClFN3Pureza:98%Forma y color:SolidPeso molecular:319.8AC260584
CAS:AC260584 is an M1 muscarinic receptor allosteric agonist (pEC50: 7.6).Fórmula:C20H29FN2O2Forma y color:SolidPeso molecular:348.45LY487379 hydrochloride
CAS:Positive allosteric modulator of mGlu2 receptorsFórmula:C21H20ClF3N2O4SPureza:98%Forma y color:SolidPeso molecular:488.91PF-4479745
CAS:<p>PF-4479745 ia a potent and selective agonist of 5-HT2C receptor.</p>Fórmula:C17H22N4Pureza:98%Forma y color:SolidPeso molecular:282.38hMAO-B-IN-2
CAS:<p>hMAO-B-IN-2: selective oral hMAO-B inhibitor, crosses BBB, IC50=4 nM, potential for Alzheimer's research, neuroprotective, low toxicity.</p>Fórmula:C18H23NO3Forma y color:SolidPeso molecular:301.38LY 2365109 hydrochloride
CAS:<p>glycine transporter 1 (GlyT1) inhibitor</p>Fórmula:C22H27NO5Pureza:98%Forma y color:SolidPeso molecular:385.45Alaproclate (hydrochloride)
CAS:<p>Alaproclate, an SSRI, enhances serotonin and SIRT1, hinders NMDA and K+ currents in neurons, and shows antidepressant-like effects in rats.</p>Fórmula:C13H19Cl2NO2Forma y color:SolidPeso molecular:292.2Anxiolytic/nonsedative agent-1
CAS:<p>TCS 1205: Selective GABAA agonist, BzR affinity in bovine brain (Kis: 14-239 nM), α2 efficacy in vitro, anxioselective in vivo.</p>Fórmula:C18H15N3O4Pureza:98.61%Forma y color:SolidPeso molecular:337.33MPDC
CAS:<p>MPDC acts as a competitive inhibitor against the Na+-dependent high-affinity glutamate transporter within forebrain synaptosomes.</p>Fórmula:C7H9NO4Pureza:98%Forma y color:SolidPeso molecular:171.15Levemopamil HCl
CAS:Levemopamil HCl is used as a calcium channel blocker.Fórmula:C23H31ClN2Pureza:98%Forma y color:SolidPeso molecular:370.96SB-269970
CAS:SB-269970 is a antagonist of 5-HT7 receptor(pKi of 8.3).Fórmula:C18H28N2O3SPureza:98%Forma y color:SolidPeso molecular:352.49SB 206553 hydrochloride
CAS:<p>SB 206553 hydrochloride is a 5-HT2C inverse agonist and a 5-HT2C/5-HT2B receptor antagonist with anxiolytic activity, useful for studying neurological disorders</p>Fórmula:C17H17ClN4OPureza:99.56%Forma y color:SolidPeso molecular:328.8Ro 19-4603
CAS:<p>Benzodiazepine inverse agonist</p>Fórmula:C15H17N3O3SPureza:98%Forma y color:SolidPeso molecular:319.38AR-A 2
CAS:<p>AR-A 2, a selective 5-HT1B antagonist; high guinea pig 5-HT1B/1D affinity (Ki: 0.24, 0.47 nM); 10x less for 5-HT1D (Ki: 5 nM).</p>Fórmula:C27H36N4O2Pureza:98%Forma y color:SolidPeso molecular:448.6Telenzepine
CAS:<p>Telenzepine is a potent and selective M1 antimuscarinic.</p>Fórmula:C19H22N4O2SPureza:98%Forma y color:SolidPeso molecular:370.47BChE-IN-14
CAS:<p>BChE-IN-14 reverses cognitive decline, is safe for primary cells, crosses the blood-brain barrier, and selectively inhibits BChE (IC50: 0.011 μM for hBChE).</p>Fórmula:C24H29NForma y color:SolidPeso molecular:331.49BNC375
CAS:BNC375 is a α7 nAChRs type I positive allosteric modulator (EC50: 1.9 μM).Fórmula:C19H23ClN2O3SPureza:98%Forma y color:SolidPeso molecular:394.92NCS-382
CAS:<p>γ-Hydroxybutyric acid antagonist</p>Fórmula:C13H14O3Pureza:98%Forma y color:SolidPeso molecular:218.25Pregabalin arenacarbil
CAS:<p>Pregabalin arenacarbil is a gabamimetic.</p>Fórmula:C15H27NO6Forma y color:SolidPeso molecular:317.38HZ166
CAS:<p>HZ-166 is a positive GABAA receptor modulator and a GABAA receptor subtype-selective benzodiazepine site ligand.</p>Fórmula:C21H16N4O2Pureza:98%Forma y color:SolidPeso molecular:356.38VU0410425
CAS:VU0410425 is a metabotropic glutamate receptor subtype 1 negative allosteric modulator.Fórmula:C19H16ClN3O3Pureza:98%Forma y color:SolidPeso molecular:369.8T 82
CAS:<p>T 82 is an antagonist of 5-HT3 and inhibitor of acetylcholinesterase (AChE) and used for the treatment of Alzheimer's Disease.</p>Fórmula:C56H62N6O8Pureza:98%Forma y color:SolidPeso molecular:947.146γ-secretase modulator 2
CAS:<p>Gamma-secretase modulator 2 selectively targets Alzheimer's by reducing Aβ(1-42), aiding in prevention and treatment.</p>Fórmula:C25H22F4N6O2Pureza:98%Forma y color:SolidPeso molecular:514.47SKF-83566 hydrobromide
CAS:<p>D1-like dopamine receptor antagonist</p>Fórmula:C17H19BrClNOPureza:98%Forma y color:SolidPeso molecular:368.7Ro 04-6790
CAS:<p>Ro 04-6790 is a 5-HT6 receptor antagonist.</p>Fórmula:C12H16N6O2SPureza:98%Forma y color:SolidPeso molecular:308.36(S)-3,5-DHPG
CAS:<p>group I mGlu receptor agonist</p>Fórmula:C8H9NO4Pureza:98%Forma y color:SolidPeso molecular:183.16S 16924
CAS:S 16924 is a 5-HT 1A agonist with potential anxiolytic effects and may be useful in the study of neurologic disorders.Fórmula:C22H24FNO4Pureza:99.35% - 99.6%Forma y color:SolidPeso molecular:385.43RS 39604
CAS:<p>potent and selective 5-HT4 antagonist</p>Fórmula:C26H37Cl2N3O6SPureza:98%Forma y color:SolidPeso molecular:590.56TC-N 22A
CAS:TC-N 22A is a strong, selective, oral active mGlu4 forward allosteric regulator (PAM) that can cross the blood-brain barrier.Fórmula:C14H13N5SPureza:99.95%Forma y color:SolidPeso molecular:283.35TPMPA
CAS:<p>GABAA-ρ antagonist</p>Fórmula:C6H12NO2PPureza:98%Forma y color:SolidPeso molecular:161.14CPPHA
CAS:<p>CPPHA, a positive allosteric modulator of glutamate receptors mGluR5 and mGluR1, is commonly used in development for central nervous system diseases.</p>Fórmula:C22H15ClN2O4Pureza:98.07%Forma y color:SolidPeso molecular:406.82Depramine
CAS:<p>Depramine (GP 31406), a tricyclic antidepressant, exhibits pharmacological activity by inhibiting acetylcholinesterase, Mg^2+-ATPase, and Na^+/K^+ ATPase</p>Fórmula:C19H22N2Forma y color:SolidPeso molecular:278.39Alniditan dihydrochloride
CAS:<p>Alniditan dihydrochloride is a potent 5-HT1D agonist and migraine-abortive agent.</p>Fórmula:C17H28Cl2N4OForma y color:SolidPeso molecular:375.34ZAPA sulfate
CAS:<p>GABAA receptors agonist</p>Fórmula:C4H8N2O6S2Pureza:98%Forma y color:SolidPeso molecular:244.25TASP0433864
CAS:<p>TASP0433864 enhances mGlu2 activity; EC50: 199 nM (human), 206 nM (rat); not an agonist.</p>Fórmula:C18H23N3O3Pureza:98%Forma y color:SolidPeso molecular:329.39GABAA receptor agent 8
CAS:<p>Compound 5e, a GABAA receptor modulator, shows potent anticonvulsant effects with low neurotoxicity for epilepsy research.</p>Fórmula:C19H16N4OForma y color:SolidPeso molecular:316.36Piperilate
CAS:<p>Piperilate (Pipethanate), a hetrazepine PAF antagonist and anticholinergic used in asthma studies, counters organophosphate toxicity.</p>Fórmula:C21H25NO3Forma y color:SolidPeso molecular:339.43JNJ-40068782
CAS:<p>JNJ-40068782 is a potent, selective and systemically active positive allosteric modulator of the mGlu2 receptor.</p>Fórmula:C21H23N3OPureza:98%Forma y color:SolidPeso molecular:333.43Distigmine Bromide
CAS:<p>Distigmine Bromide is an acetylcholinesterase inhibitor. It is used for the treatment of underactive neurogenic bladder and myasthenia gravis.</p>Fórmula:C22H32BrN4O4Pureza:98%Forma y color:SolidPeso molecular:496.42LY 2087101
CAS:<p>Allosteric potentiator of α7, α4β2 and α4β4 nAChRs</p>Fórmula:C15H11FN2OS2Pureza:98%Forma y color:SolidPeso molecular:318.39ML289
CAS:<p>ML289 is a potent CNS-penetrant mGlu3 modulator with IC50 of 0.66 μM, >15-fold selectivity over mGlu2, and inactive against mGlu5.</p>Fórmula:C22H23NO3Pureza:99.54%Forma y color:SolidPeso molecular:349.42Pruvanserin hydrochloride
CAS:<p>Pruvanserin hydrochloride (EMD 281014 HCl) is a selective 5-HT2A receptor antagonist, inhibits GTP-gamma-S accumulation and alleviates tactile allodynia.</p>Fórmula:C22H22ClFN4OPureza:99.6%Forma y color:SolidPeso molecular:412.895-Iodo-A-85380 dihydrochloride
CAS:α4β2 and α6β2 nicotinic acetylcholine receptors agonistFórmula:C9H13Cl2IN2OPureza:98%Forma y color:SolidPeso molecular:363.02BChE-IN-4
CAS:<p>BChE-IN-4, a potent butyrylcholinesterase inhibitor, crosses blood-brain barrier, improves memory in mice; promising for Alzheimer's research.</p>Fórmula:C24H37N3OForma y color:SolidPeso molecular:383.57Irindalone
CAS:<p>IrindaloneIrindalone is a potent serotonin (5-HT2) antagonist.</p>Fórmula:C24H29FN4OPureza:98%Forma y color:SolidPeso molecular:408.51LY456066
CAS:<p>LY456066 is a mGluR1 receptor-selective, negative allosteric modulator.</p>Fórmula:C19H23N3OSPureza:98%Forma y color:SolidPeso molecular:341.47BuChE-IN-4
CAS:<p>BuChE-IN-4 is a potent inhibitor of BuChE (IC50: 7.7 nM) and exhibits mild antioxidant capacity, non-toxicity, lipophilicity and neuroprotective effects.</p>Fórmula:C21H21BrFN3O4SForma y color:SolidPeso molecular:510.38F13714 fumarate
CAS:<p>F13714 fumarate is a 5-HT1A receptor-biased agonist.</p>Fórmula:C25H29ClF2N4O5Pureza:98.86%Forma y color:SolidPeso molecular:538.97Z-Cyclopentyl-AP4
CAS:Group III mGlu receptor agonistFórmula:C6H12NO5PPureza:98%Forma y color:SolidPeso molecular:209.14PNU-282987 S enantiomer hydrochloride
CAS:<p>(S)-PNU-282987, selective α7 nAChR agonist; Ki=26 nM (rat), weak on other receptors except 5-HT3; Ki=930 nM.</p>Fórmula:C14H18Cl2N2OPureza:98%Forma y color:SolidPeso molecular:301.21
