
Neurociencia
Los inhibidores en neurociencia son compuestos diseñados para modular la actividad de proteínas, enzimas o receptores específicos dentro del sistema nervioso. Estos inhibidores son cruciales para estudiar los mecanismos moleculares subyacentes a la función neuronal, la transmisión sináptica y las enfermedades neurodegenerativas. Al dirigirse a los receptores de neurotransmisores, canales iónicos y vías de señalización, los inhibidores en neurociencia ayudan en la exploración de la función cerebral y en el desarrollo de estrategias terapéuticas para trastornos neurológicos como el Alzheimer, Parkinson y la epilepsia. En CymitQuimica, ofrecemos una amplia gama de inhibidores de neurociencia de alta calidad para apoyar su investigación en neurobiología, neurofarmacología y ciencias cognitivas.
Subcategorías de "Neurociencia"
- Receptor 5-HT(942 productos)
- ACK(1 productos)
- AChR(576 productos)
- ATP Citrato Liasa(16 productos)
- Receptor adrenérgico(2.949 productos)
- BACE(36 productos)
- Beta amiloide(205 productos)
- CAMK(69 productos)
- Inhibidores de ciclooxigenasa (COX)(565 productos)
- Receptor de dopamina(410 productos)
- Receptor GABA(337 productos)
- Gamma-secretasa(59 productos)
- GluR(255 productos)
- GlyT(24 productos)
- Receptor de histamina(359 productos)
- LRRK2(33 productos)
- Receptor de melatonina(24 productos)
- NMDAR(26 productos)
- Receptor de OX(40 productos)
- Receptor de opioides(298 productos)
Mostrar 12 subcategorías más
Se han encontrado 5389 productos de "Neurociencia"
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WAY208466 dihydrochloride
CAS:<p>WAY208466 dihydrochloride is a 5-HT6 receptor agonist (EC50=7.3 nM) with antidepressant and anxiolytic activity.</p>Fórmula:C17H20Cl2FN3O2SPureza:98.43%Forma y color:SolidPeso molecular:420.33VU0463841
CAS:<p>VU0463841 is a mGlu5 negative allosteric modulators.</p>Fórmula:C13H8ClFN4OForma y color:SolidPeso molecular:290.68Lesogaberan
CAS:<p>Lesogaberan: selective GABAB agonist, EC50 8.6 nM, Ki 5.1 nM in rats, weak GABAA affinity (Ki 1.4 μM).</p>Fórmula:C3H9FNO2PPureza:98%Forma y color:SolidPeso molecular:141.08VU 0360172 hydrochloride
CAS:<p>positive allosteric modulator of mGlu5 receptors</p>Fórmula:C18H16ClFN2OPureza:98%Forma y color:SolidPeso molecular:330.78BChE-IN-6
CAS:<p>BChE-IN-6 inhibits BChE with a Ki of 0.182 μM and chelates Zn 2+, useful in AD research.</p>Fórmula:C24H29N3O2Forma y color:SolidPeso molecular:391.51Alvameline
CAS:Alvameline (Lu25-109) is a partial M1 agonist. Alvameline (Lu25-109) also is a M2/M3 antagonist.Fórmula:C9H15N5Pureza:98%Forma y color:SolidPeso molecular:193.252-Iodomelatonin
CAS:<p>2-Iodomelatonin, Ki 28 pM, is an MT1 agonist, >5x selective over MT2, used to map melatonin sites in brain/tissues.</p>Fórmula:C13H15IN2O2Pureza:99.7%Forma y color:SolidPeso molecular:358.17Tracazolate hydrochloride
CAS:<p>Tracazolate hydrochloride (Tracazolate (hydrochloride)) is a modulator of the GABAA receptor with anxiolytic and anticonvulsant activity.</p>Fórmula:C16H25ClN4O2Pureza:99.52%Forma y color:SolidPeso molecular:340.85CBP501
CAS:<p>CBP501 peptide inhibits kinases like MAPKAP-K2/C-Tak1/CHK1, preventing Cdc25C function and blocking the entry into mitosis.</p>Fórmula:C86H122F5N29O17Forma y color:SolidPeso molecular:1929.06DREADD agonist 21 dihydrochloride
CAS:<p>DREADD agonist 21 dihydrochloride is a potent human muscarinic acetylcholine M3 receptors ( hM3Dq ) agonist with EC 50 of 1.7 nM [1].</p>Fórmula:C17H20Cl2N4Pureza:98%Forma y color:SolidPeso molecular:351.27CIA-1 hcl(452087-38-6 Free base)
CAS:<p>CIA-1 inhibits the nuclear receptor COUP-TFII, with IC50s ranging from 1.2 μM to 7.6 μM in prostate cancer cell lines.CIA-1 inhibits the growth of a variety of</p>Fórmula:C17H20ClN3O2SPureza:99.02%Forma y color:SolidPeso molecular:365.88Lilly 51641
CAS:<p>Lilly 51641 is used as a MAO inhibitor.</p>Fórmula:C11H14ClNOPureza:98%Forma y color:SolidPeso molecular:211.69GR 113808
CAS:<p>GR 113808 is a 5-HT4 receptor antagonist that inhibits 5-HT1B and 5-HT3 receptors and attenuates morphine-stimulated dopamine release in the rat striatum.</p>Fórmula:C19H27N3O4SPureza:98.16%Forma y color:SolidPeso molecular:393.5Foliglurax
CAS:Foliglurax is a highly selective brain-penetrant metabotropic glutamate receptor 4 positive allosteric modulator (mGluR4 PAM) (EC50: 79 nM).Fórmula:C23H23N3O3SPureza:98%Forma y color:SolidPeso molecular:421.51TIK-301
CAS:<p>TIK-301 is a chlorinated melatonin derivative and a potent, high-affinity, and orally active melatonin MT1 and MT2 receptors agonist (Kis: 0.081 nM and 0.042 nM</p>Fórmula:C14H17ClN2O2Pureza:98%Forma y color:SolidPeso molecular:280.75DL-AP4 Sodium salt
CAS:Broad spectrum EAA ligandFórmula:C4H10NNaO5PPureza:98%Forma y color:SolidPeso molecular:206.09Trimipramine
CAS:<p>Trimipramine is an antidepressant with an anxiety-reducing sedative component to its action.</p>Fórmula:C20H26N2Pureza:98%Forma y color:SolidPeso molecular:294.432-Hydroxysaclofen
CAS:2-Hydroxysaclofen is a GABAB receptor antagonist.Fórmula:C9H12ClNO4SPureza:98%Forma y color:White SolidPeso molecular:265.71VU6001376
CAS:<p>VU6001376 is an effective and selective positive allosteric modulator of the metabotropic glutamate receptor 4 (EC50: 50.1 nM).</p>Fórmula:C18H14F2N6OSPureza:98%Forma y color:SolidPeso molecular:400.41VU0090157
CAS:<p>VU0090157, a novel allosteric potentiators of M1 muscarinic receptor, may provide novel treatments for schizophrenia and Alzheimer's disease.</p>Fórmula:C19H21N3O7Pureza:98%Forma y color:SolidPeso molecular:403.39(S)-VQW-765
<p>(S)-VQW-765, oral α7 nAChR partial agonist, may improve cognition in Alzheimer's and schizophrenia.</p>Fórmula:C19H22N2OForma y color:SolidPeso molecular:294.39PRX933 hydrochloride
CAS:<p>PRX933 hydrochloride (GW876167 hydrochloride) is an agonist of 5-HT2C receptor and can be used in studies about hypertension acute treatment.</p>Fórmula:C16H22ClN5O2Pureza:99.51% - 99.89%Forma y color:SolidPeso molecular:351.848-M-PDOT
CAS:<p>8-M-PDOT (AH-002) is an MT2 receptor agonist that inhibits MT1.8-M-PDOT has anxiolytic activity and may be used in the study of neuropathic pain.</p>Fórmula:C14H19NO2Pureza:99.54% - 99.54%Forma y color:SolidPeso molecular:233.31Thiochrome
CAS:<p>Thiochrome is a selective enhancer of M4 muscarinic receptor of acetylcholine (ACh) affinity.</p>Fórmula:C12H14N4OSPureza:98%Forma y color:SolidPeso molecular:262.33S-22153
CAS:<p>S22153 is an antagonist of melatonin receptor.</p>Fórmula:C14H17NOSForma y color:SolidPeso molecular:247.362-PAT
CAS:<p>2-PAT: reversible MAO-A inhib., IC50=0.721 µM; MAO-B inactivator, IC50=14.6 µM; potential in Parkinson's/depression study.</p>Fórmula:C13H15NForma y color:SolidPeso molecular:185.26GR 128107
CAS:<p>GR 128107 is an antagonist of melatonin receptor.</p>Fórmula:C16H20N2O2Forma y color:SolidPeso molecular:272.34Cimetropium Bromide
CAS:<p>Cimetropium Bromide is a mAChR antagonist used for long-term treatment of irritable bowel syndrome.</p>Fórmula:C21H28BrNO4Forma y color:SolidPeso molecular:438.36SGC-AAK1-1N
CAS:<p>SGC-AAK1-1N is a potent and selective inhibitor of AAK1 (AP2 associated kinase 1) with an IC 50 of 1.8 μM [1].</p>Fórmula:C20H22N4O3SForma y color:SolidPeso molecular:398.48Chrysamine G
CAS:<p>Chrysamine G, Congo red analog, blocks Aβ toxicity, probes Alzheimer's amyloid.</p>Fórmula:C26H16N4Na2O6Forma y color:SolidPeso molecular:526.416CGS 20625
CAS:<p>partial agonist for the benzodiazepine binding site of the GABAA receptor</p>Fórmula:C18H19N3O2Pureza:99.61%Forma y color:SolidPeso molecular:309.36Pralidoxime
CAS:<p>Pralidoxime reactivates AChE blocked by nerve agents, aiding as an organophosphate poisoning antidote.</p>Fórmula:C7H9N2OForma y color:SolidPeso molecular:137.16SX-3228
CAS:SX-3228 is a selective agonist of benzodiazepine1 (BZ1) receptor(IC50 of 17 nM).Fórmula:C18H18N4O3Pureza:98%Forma y color:SolidPeso molecular:338.36SC58451
CAS:<p>SC58451 is a novel potent, orally active and selective COX-2 inhibitor.SC58451 showed anti-inflammatory activity in a rat model of arthritis.</p>Fórmula:C20H19FO2SPureza:>99.99%Forma y color:SolidPeso molecular:342.43Beperidium iodide
CAS:<p>Beperidium iodide is a competitive antagonist of the acetylcholine receptor (pA2: 7.93).</p>Fórmula:C23H34IN3O3Forma y color:SolidPeso molecular:527.44Penbutolol
CAS:<p>Penbutolol is a nonselective beta-blocker utilized as an antihypertensive and an antianginal.</p>Fórmula:C18H29NO2Pureza:98%Forma y color:SolidPeso molecular:291.43Eucatropine
CAS:<p>Eucatropine, an anticholinergic agent, acts as a potent inhibitor of the muscarinic acetylcholine receptor (mAChR) with an IC 50 value of 0.583 μM.</p>Fórmula:C17H25NO3Forma y color:SolidPeso molecular:291.39AZ-4217
CAS:<p>AZ-4217: potent BACE inhibitor, reduces amyloid in mice, IC50 160 pM in SH-SY5Y cells, effective in vivo.</p>Fórmula:C30H25FN4OForma y color:SolidPeso molecular:476.54AChE/BuChE-IN-1
CAS:<p>AChE/BuChE-IN-1: BuChE inhibitor (IC50=0.48µM), weaker AChE blocker (IC50=7.16µM), ·OH scavenger (IC50=0.1674µM), may aid in AD research.</p>Fórmula:C19H19NO4Forma y color:SolidPeso molecular:325.36PF-04781340
CAS:PF-04781340 is an effective, selective, and CNS penetrant agonist of 5-HT2C receptor.Fórmula:C17H21N3Pureza:98%Forma y color:SolidPeso molecular:267.37BMS-902483
CAS:<p>BMS-902483: potent α7 partial agonist; enhances rodent cognition; α7 EC50=9.3nM; 5-HT3A IC50=480nM.</p>Fórmula:C18H20N4OPureza:98%Forma y color:SolidPeso molecular:308.38RLH 033
CAS:<p>RLH 033 is a selective ligand for the sigma 1 recognition site.</p>Fórmula:C25H31ClN2O4Pureza:98%Forma y color:SolidPeso molecular:458.98Bradanicline HCl
CAS:<p>Bradanicline(TC-5619) is the agonist of Alpha-7 Nicotinic Receptor.</p>Fórmula:C22H24ClN3O2Forma y color:SolidPeso molecular:397.9AChE/MAO-B-IN-3
<p>AChE/MAO-B-IN-3: dual inhibitor for AChE (IC50 = 0.0257 µM) and MAO-B (IC50 = 0.0456 µM), researched for Alzheimer's.</p>Fórmula:C24H28N2O4Forma y color:SolidPeso molecular:408.49AT-1001
CAS:<p>AT-1001 is an α3β4 nAChR partial agonist reducing nicotine relapse and withdrawal with negligible impact on food response and dopamine release.</p>Fórmula:C15H21BrN2Forma y color:SolidPeso molecular:309.24Cyclopenin
CAS:<p>Cyclopenin is an inhibitor of acetylcholinesterase (AChE; IC50 = 2.04 μM for human recombinant AChE).</p>Fórmula:C17H14N2O3Forma y color:SolidPeso molecular:294.35-HT2A receptor agonist-2
CAS:<p>Potent 5-HT2A receptor agonist-2 targets 5-HT2A/B/C with EC50 1.7, 0.58, 0.50 nM.</p>Fórmula:C20H21ClN2O3Forma y color:SolidPeso molecular:372.85COX-2-IN-2
CAS:<p>COX-2-IN-2 selectively inhibits COX2 (IC50: 0.24 μM); COX-2-IN-1 offers anti-inflammatory and pain relief.</p>Fórmula:C17H12FN3O2SPureza:97.62%Forma y color:SolidPeso molecular:341.36Territrem B
CAS:<p>Territrem B: A mycotoxin that irreversibly blocks AChE, causes tremors in mice at 0.21 mg/kg.</p>Fórmula:C29H34O9Forma y color:SolidPeso molecular:526.57AChE-IN-20
CAS:<p>AChE-IN-20: AChE inhibitor (IC50: 397.32 nM), hCA-I/II blocker (IC50: ~77 nM avg), α GLY suppressor (IC50: 52.08 nM).</p>Fórmula:C22H20N8O6S2Forma y color:SolidPeso molecular:556.57
