
Neurociencia
Los inhibidores en neurociencia son compuestos diseñados para modular la actividad de proteínas, enzimas o receptores específicos dentro del sistema nervioso. Estos inhibidores son cruciales para estudiar los mecanismos moleculares subyacentes a la función neuronal, la transmisión sináptica y las enfermedades neurodegenerativas. Al dirigirse a los receptores de neurotransmisores, canales iónicos y vías de señalización, los inhibidores en neurociencia ayudan en la exploración de la función cerebral y en el desarrollo de estrategias terapéuticas para trastornos neurológicos como el Alzheimer, Parkinson y la epilepsia. En CymitQuimica, ofrecemos una amplia gama de inhibidores de neurociencia de alta calidad para apoyar su investigación en neurobiología, neurofarmacología y ciencias cognitivas.
Subcategorías de "Neurociencia"
- Receptor 5-HT(942 productos)
- ACK(1 productos)
- AChR(575 productos)
- ATP Citrato Liasa(16 productos)
- Receptor adrenérgico(2.948 productos)
- BACE(36 productos)
- Beta amiloide(205 productos)
- CAMK(69 productos)
- Inhibidores de ciclooxigenasa (COX)(565 productos)
- Receptor de dopamina(409 productos)
- Receptor GABA(336 productos)
- Gamma-secretasa(59 productos)
- GluR(255 productos)
- GlyT(24 productos)
- Receptor de histamina(359 productos)
- LRRK2(33 productos)
- Receptor de melatonina(24 productos)
- NMDAR(27 productos)
- Receptor de OX(40 productos)
- Receptor de opioides(298 productos)
Mostrar 12 subcategorías más
Se han encontrado 5390 productos de "Neurociencia"
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DS1
CAS:<p>DS1 is a GABAA receptor agonist which can stimulate gonadotropin subunit gene expression in mouse.</p>Fórmula:C18H10Br2ClN3OSForma y color:SolidPeso molecular:511.62(R)-Viloxazine Hydrochloride
CAS:<p>(R)-Viloxazine Hydrochloride, the R-isomer of Viloxazine.</p>Fórmula:C13H20ClNO3Pureza:99.88% - 99.94%Forma y color:SolidPeso molecular:273.76PRX-08066 Maleic acid
CAS:<p>PRX-08066 Maleic acid is the salt form of PRX-08066.PRX-08066 is a 5-HT receptor 2B antagonist that induces selective vasodilation of the pulmonary artery.</p>Fórmula:C23H21ClFN5O4SPureza:97.59%Forma y color:SolidPeso molecular:517.96Iprindole
CAS:<p>Iprindole, a tricyclic indole antidepressant, is a dual weak inhibitor of noradrenaline and 5-HT uptake [1].</p>Fórmula:C19H28N2Pureza:99.54%Forma y color:SolidPeso molecular:284.44Iloperidone hydrochloride
CAS:<p>Iloperidone hydrochloride is a D(2)/5-HT(2) receptor antagonist. It is also an atypical antipsychotic for the treatment of schizophrenia symptoms.</p>Fórmula:C24H28ClFN2O4Pureza:98%Forma y color:SolidPeso molecular:462.95SB 258719 hydrochloride
CAS:<p>Selective 5-HT7 receptor antagonist</p>Fórmula:C18H31ClN2O2SPureza:98%Forma y color:SolidPeso molecular:374.97AVN-322
CAS:<p>AVN-322 is a 5-HT6 receptor antagonist. 5-HT6R antagonists improves cognition in animal models of cognitive impairment.</p>Fórmula:C17H20ClN5O2SPureza:>99.99%Forma y color:SolidPeso molecular:393.89Alaproclate hydrochloride, (S)-
CAS:<p>Alaproclate hydrochloride, (S)- is a selective inhibitor of serotonin reuptake.</p>Fórmula:C13H19Cl2NO2Pureza:98%Forma y color:SolidPeso molecular:292.2NFPS
CAS:<p>NFPS exerts neuroprotection via glyR alpha1 subunit in the rat model of transient focal cerebral ischaemia and reperfusion.</p>Fórmula:C24H24FNO3Pureza:98%Forma y color:SolidPeso molecular:393.45YIAD-0205
CAS:<p>YIAD-0205, an orally administered inhibitor of Aβ(1-42) aggregation, has exhibited in vivo efficacy in a 5XFAD transgenic mouse model that harbors five familial</p>Fórmula:C26H16Br2ClN3Forma y color:SolidPeso molecular:565.69VU0652835
CAS:<p>VU0652835 is a negative allosteric modulator of metabotropic glutamate receptor subtype 5 (mGlu5) (IC50: 81 nM).</p>Fórmula:C16H19N3O3SPureza:98%Forma y color:SolidPeso molecular:333.41SKF 97541
CAS:<p>GABAB agonist</p>Fórmula:C4H12NO2PPureza:98%Forma y color:SolidPeso molecular:137.12T 82
CAS:<p>T 82 is an antagonist of 5-HT3 and inhibitor of acetylcholinesterase (AChE) and used for the treatment of Alzheimer's Disease.</p>Fórmula:C56H62N6O8Pureza:98%Forma y color:SolidPeso molecular:947.146CP-601932
CAS:<p>CP-601932 (free base) is a selective base α( 4) β( 2) Nicotinic acetylcholine receptor agonist.</p>Fórmula:C12H12F3NForma y color:SolidPeso molecular:227.23OAB-14
CAS:<p>OAB-14, a Bexarotene derivative, enhances β-amyloid clearance and cognitive function in APP/PS1 mice, improving Alzheimer's symptoms.</p>Fórmula:C32H46N4O2Forma y color:SolidPeso molecular:518.73Ro15-4513
CAS:<p>Ro15-4513 is imidazobenzodiazepinone derivative and is a partial inverse agonist of benzodiazepine receptors. Ro15-4513 is an effective ethanol antagonist.</p>Fórmula:C15H14N6O3Pureza:98%Forma y color:SolidPeso molecular:326.31Ambenonium chloride tetrahydrate
CAS:<p>Ambenonium chloride, a salt with cholinesterase inhibiting properties, treats myasthenia gravis by enhancing acetylcholine activity.</p>Fórmula:C28H50Cl4N4O6Forma y color:SolidPeso molecular:680.53T761-0184
CAS:<p>T761-0184 is a potent antagonist of α7 nicotinic receptor (nAChR) [1].</p>Fórmula:C16H20FN3OForma y color:SolidPeso molecular:289.35UPF-523
CAS:group I metabotropic glutamate receptors (mGlu1a) antagonistFórmula:C11H11NO4Pureza:98%Forma y color:White SolidPeso molecular:221.21DAU 5884 hydrochloride
CAS:muscarinic M3 receptor antagonistFórmula:C17H22ClN3O3Pureza:98%Forma y color:SolidPeso molecular:351.83K 01-162
CAS:K 01-162 binds and destabilizes AβO (β-amyloid), with an EC50 of 80 nM.Fórmula:C15H14BrNForma y color:SolidPeso molecular:288.18Zaldaride maleate
CAS:Zaldaride maleate blocks Ca2+, Na+, K+ currents, and nAChR; inhibits CaM cAMP PDE (IC50: 3.3 nM) and estrogen signaling.Fórmula:C30H32N4O6Pureza:98%Forma y color:SolidPeso molecular:544.6AChE-IN-15
CAS:<p>AChE-IN-15 is a reversible inhibitor of huAChE and huBChE (IC50: 6.8 μM, 16.1 μM), with antioxidant activity, used in Alzheimer's research.</p>Fórmula:C23H24N2O7Forma y color:SolidPeso molecular:440.45Alvameline
CAS:Alvameline (Lu25-109) is a partial M1 agonist. Alvameline (Lu25-109) also is a M2/M3 antagonist.Fórmula:C9H15N5Pureza:98%Forma y color:SolidPeso molecular:193.25Lilly 51641
CAS:<p>Lilly 51641 is used as a MAO inhibitor.</p>Fórmula:C11H14ClNOPureza:98%Forma y color:SolidPeso molecular:211.69Trimipramine
CAS:<p>Trimipramine is an antidepressant with an anxiety-reducing sedative component to its action.</p>Fórmula:C20H26N2Pureza:98%Forma y color:SolidPeso molecular:294.432-Hydroxysaclofen
CAS:2-Hydroxysaclofen is a GABAB receptor antagonist.Fórmula:C9H12ClNO4SPureza:98%Forma y color:White SolidPeso molecular:265.71VU0090157
CAS:<p>VU0090157, a novel allosteric potentiators of M1 muscarinic receptor, may provide novel treatments for schizophrenia and Alzheimer's disease.</p>Fórmula:C19H21N3O7Pureza:98%Forma y color:SolidPeso molecular:403.39ACPT-II
CAS:<p>metabotropic receptor antagonist</p>Fórmula:C8H11NO6Pureza:98%Forma y color:SolidPeso molecular:217.18W-5 hydrochloride
CAS:<p>W-5 hydrochloride (N-(6-Aminohexyl)-1-naphthalenesulfonamide HCl) is a potent calmodulin antagonist.</p>Fórmula:C16H23ClN2O2SPureza:99.35%Forma y color:Off-White Crystalline SolidPeso molecular:342.88Org-25935
CAS:<p>Org-25935, a GlyT-1 inhibitor, is used potentially for the treatment of schizophrenia and alcohol dependence.</p>Fórmula:C21H26ClNO3Forma y color:SolidPeso molecular:375.89Chrysamine G
CAS:<p>Chrysamine G, Congo red analog, blocks Aβ toxicity, probes Alzheimer's amyloid.</p>Fórmula:C26H16N4Na2O6Forma y color:SolidPeso molecular:526.416ZLWH-23
CAS:<p>ZLWH-23: AChE inhibitor (IC50: 0.27μM), GSK-3β (6.78μM), BChE (20.82μM), potential in Alzheimer's research.</p>Fórmula:C30H32FN5O2Forma y color:SolidPeso molecular:513.61CGS 20625
CAS:<p>partial agonist for the benzodiazepine binding site of the GABAA receptor</p>Fórmula:C18H19N3O2Pureza:99.61%Forma y color:SolidPeso molecular:309.36SX-3228
CAS:SX-3228 is a selective agonist of benzodiazepine1 (BZ1) receptor(IC50 of 17 nM).Fórmula:C18H18N4O3Pureza:98%Forma y color:SolidPeso molecular:338.36Penbutolol
CAS:<p>Penbutolol is a nonselective beta-blocker utilized as an antihypertensive and an antianginal.</p>Fórmula:C18H29NO2Pureza:98%Forma y color:SolidPeso molecular:291.43ENS-163 phosphate
CAS:<p>Ens-163 phosphate is a muscarinic M1 receptor agonist. It is selective.</p>Fórmula:C11H19N2O5PSPureza:98%Forma y color:SolidPeso molecular:322.32Bifeprunox Mesylate
CAS:<p>Bifeprunox: partial dopamine/serotonin agonist for schizophrenia; suppresses VTA neurons via D2; affects rat nicotine-seeking.</p>Fórmula:C25H27N3O5SPureza:98%Forma y color:SolidPeso molecular:481.56Org 20599
CAS:<p>GABAA receptor agonist</p>Fórmula:C25H40ClNO3Pureza:98%Forma y color:SolidPeso molecular:438.04Opiranserin
CAS:<p>Opiranserin is a development as an injectable agent for the treatment of postoperative pain.</p>Fórmula:C21H34N2O5Pureza:98%Forma y color:SolidPeso molecular:394.51ML352
CAS:ML352 inhibits choline transporter noncompetitively; Ki of 92 nM in human CHT, 166 nM in mouse synaptosomes.Fórmula:C21H29N3O4Pureza:99.15%Forma y color:SolidPeso molecular:387.47Rivanicline oxalate
CAS:<p>Rivanicline oxalate is an agonist of neuronal nicotinic receptor, showing high selectivity for the α4β2 subtype (Ki=26 nM).</p>Fórmula:C12H16N2O4Pureza:98%Forma y color:SolidPeso molecular:252.27Hexafluronium Bromide
CAS:<p>Hexafluronium bromide enhances muscle relaxation in surgery by blocking acetylcholine receptors.</p>Fórmula:C36H42BrN2Forma y color:SolidPeso molecular:582.649TC299423
CAS:<p>TC299423 is a novel agonist for nicotinic acetylcholine receptors (nAChRs). TC299423 modestly selectively targets α6β2 subtype.</p>Fórmula:C11H15N3Forma y color:SolidPeso molecular:189.26BTM-1086
CAS:BTM-1086 is a potent gastric secretory inhibitor and an anti-ulcer agent.Fórmula:C21H25N3OSPureza:98%Forma y color:SolidPeso molecular:367.51TMPH hydrochloride
CAS:<p>neuronal nicotinic ACh receptors (nAChRs) antagonist</p>Fórmula:C16H32ClNO2Pureza:98%Forma y color:SolidPeso molecular:305.88BACE1/2-IN-1
CAS:<p>BACE1/2-IN-1 inhibits BACE1/2 with IC50s of 0.01μM/0.0053μM, has better permeability and lower Pgp efflux but reduced metabolic stability.</p>Fórmula:C21H31N5OSForma y color:SolidPeso molecular:401.57MAO-B-IN-16
CAS:<p>MAO-B-IN-16 selectively inhibits MAO-B with IC50 of 1.55 μM, useful in studying central nervous disorders like Parkinson's.</p>Fórmula:C18H19NO3Forma y color:SolidPeso molecular:297.35SL-25.1188
CAS:<p>SL-25.1188: Reversible MAO-B inhibitor with high brain uptake & slow plasma metabolism.</p>Fórmula:C16H17F3N2O5Forma y color:SolidPeso molecular:374.31NPS ALX Compound 4a dihydrochloride
CAS:<p>NPS ALX Compound 4a dihydrochloride is a potent and selective antagonist of 5-HT6 receptor (IC50 of 7.2 nM)</p>Fórmula:C25H27Cl2N3O2SPureza:98%Forma y color:SolidPeso molecular:504.47
