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Neurociencia

Neurociencia

Los inhibidores en neurociencia son compuestos diseñados para modular la actividad de proteínas, enzimas o receptores específicos dentro del sistema nervioso. Estos inhibidores son cruciales para estudiar los mecanismos moleculares subyacentes a la función neuronal, la transmisión sináptica y las enfermedades neurodegenerativas. Al dirigirse a los receptores de neurotransmisores, canales iónicos y vías de señalización, los inhibidores en neurociencia ayudan en la exploración de la función cerebral y en el desarrollo de estrategias terapéuticas para trastornos neurológicos como el Alzheimer, Parkinson y la epilepsia. En CymitQuimica, ofrecemos una amplia gama de inhibidores de neurociencia de alta calidad para apoyar su investigación en neurobiología, neurofarmacología y ciencias cognitivas.

Subcategorías de "Neurociencia"

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Se han encontrado 5400 productos de "Neurociencia"

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  • ACPT-II

    CAS:
    <p>metabotropic receptor antagonist</p>
    Fórmula:C8H11NO6
    Pureza:98%
    Forma y color:Solid
    Peso molecular:217.18
  • AChE-IN-15

    CAS:
    <p>AChE-IN-15 is a reversible inhibitor of huAChE and huBChE (IC50: 6.8 μM, 16.1 μM), with antioxidant activity, used in Alzheimer's research.</p>
    Fórmula:C23H24N2O7
    Forma y color:Solid
    Peso molecular:440.45
  • LY 393558

    CAS:
    <p>Dual 5-HT1B/1D receptor antagonist</p>
    Fórmula:C26H31FN4O4S2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:546.68
  • AChE/BChE-IN-9

    CAS:
    <p>Compound 7a inhibits AChE/BChE (IC50: 5.74/14.05 μM), has antioxidant effects (IC50: 57.35 μM), chelates iron, and affects amyloid β 1-42 aggregation.</p>
    Fórmula:C20H19N3O4
    Forma y color:Solid
    Peso molecular:365.38
  • Z164597606

    CAS:
    <p>Z164597606 inhibits BChE (1.3 μM equine, 1.7 μM human), binds Trp82 via π-π, potential in Alzheimer's research.</p>
    Fórmula:C20H19N3O4
    Forma y color:Solid
    Peso molecular:365.38
  • Quifenadine

    CAS:
    <p>Quifenadine, an H1-histamine receptor blocker, has antiarrhythmic properties.</p>
    Fórmula:C20H23NO
    Pureza:98%
    Forma y color:Solid
    Peso molecular:293.4
  • Tacitin

    CAS:
    <p>Tacitin (Benzoctamine Hydrochloride) shows sedative and anti-anxiety properties. Tacitin blocks the central postsynaptic serotonin receptors.</p>
    Fórmula:C18H20ClN
    Pureza:98%
    Forma y color:Solid
    Peso molecular:285.81
  • VU0652835

    CAS:
    <p>VU0652835 is a negative allosteric modulator of metabotropic glutamate receptor subtype 5 (mGlu5) (IC50: 81 nM).</p>
    Fórmula:C16H19N3O3S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:333.41
  • Iprindole

    CAS:
    <p>Iprindole, a tricyclic indole antidepressant, is a dual weak inhibitor of noradrenaline and 5-HT uptake [1].</p>
    Fórmula:C19H28N2
    Pureza:99.54%
    Forma y color:Solid
    Peso molecular:284.44
  • Metixene hydrochloride

    CAS:
    <p>Metixene hydrochloride is an anticholinergic antiparkinsonian agent.</p>
    Fórmula:C20H24ClNS
    Pureza:98%
    Forma y color:Solid
    Peso molecular:345.93
  • AVN-322

    CAS:
    <p>AVN-322 is a 5-HT6 receptor antagonist. 5-HT6R antagonists improves cognition in animal models of cognitive impairment.</p>
    Fórmula:C17H20ClN5O2S
    Pureza:>99.99%
    Forma y color:Solid
    Peso molecular:393.89
  • Darenzepine

    CAS:
    <p>Darenzepine is a muscarinic receptor inhibitor.</p>
    Fórmula:C21H21N3O2
    Pureza:99.87%
    Forma y color:Solid
    Peso molecular:347.41
  • Cinitapride Hydrogen Tartrate

    CAS:
    <p>Cinitapride Hydrogen Tartrate is a gastroprokinetic agent that acts as an antagonist of the 5-HT2 receptors and as an agonist of the 5-HT1 and 5-HT4 receptors</p>
    Fórmula:C25H36N4O10
    Pureza:98%
    Forma y color:Solid
    Peso molecular:552.581
  • MSOP

    CAS:
    MSOP is a selective antagonist of group III metabotropic glutamate receptor (KD of 51 μM for the L-AP4-sensitive presynaptic mGluR).
    Fórmula:C4H10NO6P
    Pureza:98%
    Forma y color:Solid
    Peso molecular:199.1
  • Repinotan HCl

    CAS:
    <p>Repinotan HCl (Bay-x-3702) is a 5-HT1A receptor agonist with potent neuroprotective effects for the study of ischemic stroke and traumatic brain injury.</p>
    Fórmula:C21H25ClN2O4S
    Pureza:99.57%
    Forma y color:Solid
    Peso molecular:436.95
  • EMDT

    CAS:
    <p>EMDT oxalate is a selective 5-HT6 agonist, and has antidepressant effects.</p>
    Fórmula:C15H22N2O
    Pureza:97.66% - 99.78%
    Forma y color:Solid
    Peso molecular:246.35
  • A-794282

    CAS:
    <p>A-794282 is a selective antagonist of mGluR1.</p>
    Fórmula:C19H18N4OS
    Pureza:99.87%
    Forma y color:Solid
    Peso molecular:350.44
  • CGS8216

    CAS:
    <p>CGS8216 shows analgesic activity at high doses, has anxiolytic activity, and can be used to study immune system disorders.</p>
    Fórmula:C16H11N3O
    Pureza:98.53%
    Forma y color:Solid
    Peso molecular:261.28
  • (1S,3R)-ACPD

    CAS:
    <p>(1S,3R)-ACPD is a group I and II mGlu receptor agonist.</p>
    Fórmula:C7H11NO4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:173.17
  • DS2

    CAS:
    <p>Positive allosteric modulator of δ-subunit containing GABAA receptors</p>
    Fórmula:C18H12ClN3OS
    Pureza:98%
    Forma y color:Solid
    Peso molecular:353.83
  • Foliglurax monohydrochloride

    CAS:
    <p>Foliglurax monohydrochloride, an antiparkinsonian, is a selective brain-penetrant mGluR4 PAM with an EC50 of 79 nM.</p>
    Fórmula:C23H24ClN3O3S
    Forma y color:Solid
    Peso molecular:457.97
  • 17-PA

    CAS:
    <p>17-PA is a GABAA receptor antagonist.</p>
    Fórmula:C25H34O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:350.54
  • Prenylamine lactate

    CAS:
    <p>Prenylamine lactate, an ex-angina drug, depletes heart catecholamines and blocks calcium channels.</p>
    Fórmula:C27H33NO3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:419.56
  • UCSF678

    CAS:
    <p>UCSF678: selective 42 nM partial agonist at 5-HT5AR, fewer off-target effects, and lower assay risks than SB-699551.</p>
    Fórmula:C15H18N2O2S
    Forma y color:Solid
    Peso molecular:290.38
  • CGP11952

    CAS:
    <p>CGP11952 is same the benzodiazepines in its pharmacological action and it also is an experimental benzodiazepine derivative.</p>
    Fórmula:C21H21Cl2N5O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:446.33
  • Itameline

    CAS:
    <p>RU 47213 can be used to inhibit scopolamine-induced working memory impairment in rats.</p>
    Fórmula:C14H15ClN2O3
    Pureza:99.55%
    Forma y color:Solid
    Peso molecular:294.73
  • VU0361747

    CAS:
    <p>VU0361747 is a positive allosteric modulators (PAM) of metabotropic glutamate receptor subtype 5 (mGlu5).</p>
    Fórmula:C19H17FN2O2
    Forma y color:Solid
    Peso molecular:324.35
  • TC 2559 difumarate

    CAS:
    <p>partial agonist of α4β2 nicotinic acetylcholine receptor</p>
    Fórmula:C12H18N2OC4H404
    Pureza:98%
    Forma y color:Solid
    Peso molecular:380.39
  • mGAT3/4-IN-1

    CAS:
    <p>mGAT3/4-IN-1 inhibits mGAT3/4 with pIC50: 5.31/5.24, reduces neuropathic pain in diabetic mice.</p>
    Fórmula:C26H31ClN2O2S2
    Forma y color:Solid
    Peso molecular:503.12
  • JNJ-55308942

    CAS:
    <p>JNJ-55308942: selective, brain-penetrant P2X7 antagonist; IC50s: 10nM (human), 15nM (rat); Kis: 7.1nM (h), 2.9nM (r).</p>
    Fórmula:C17H12F5N7O
    Pureza:99.94%
    Forma y color:Solid
    Peso molecular:425.32
  • Org 24598

    CAS:
    <p>Potent GlyT1b inhibitor, IC50 = 6.9 nM; little effect on GlyT-2, adrenoceptors, dopamine, 5HT receptors, GABA transporters.</p>
    Fórmula:C19H20F3NO3
    Forma y color:Solid
    Peso molecular:367.36
  • GABAA receptor agent 4

    CAS:
    <p>Compound 1e is a potent γ-GABAAR antagonist with a Ki of 0.18 µM, offering immunomodulatory effects on T cell proliferation.</p>
    Fórmula:C17H24N2O
    Forma y color:Solid
    Peso molecular:272.39
  • ML169

    CAS:
    <p>ML169 is a selective and brain penetrant M1 positive allosteric modulator (PAM).</p>
    Fórmula:C21H17BrFN3O4S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:506.34
  • Aβ42-IN-2

    CAS:
    <p>Aβ42-IN-2 is a γ-secretase modulator. Aβ42-IN-2 has an IC 50 of 6.5 nM for Αβ 42. Aβ42-IN-2 can be used for the Alzheimer's disease research[1].</p>
    Fórmula:C24H26N6O2
    Pureza:98.09% - 99.87%
    Forma y color:Solid
    Peso molecular:430.5
  • Glemanserin

    CAS:
    <p>Glemanserin (MDL11939) is a specific 5-HT2A antagonist with Ki values of 0.54 nM, 2.5 nM and 2.89 nM for rabbit, human and rat 5-HT2A.</p>
    Fórmula:C20H25NO
    Pureza:99.93%
    Forma y color:Solid
    Peso molecular:295.42
  • hMAO-B-IN-2

    CAS:
    <p>hMAO-B-IN-2: selective oral hMAO-B inhibitor, crosses BBB, IC50=4 nM, potential for Alzheimer's research, neuroprotective, low toxicity.</p>
    Fórmula:C18H23NO3
    Forma y color:Solid
    Peso molecular:301.38
  • LY 2365109 hydrochloride

    CAS:
    <p>glycine transporter 1 (GlyT1) inhibitor</p>
    Fórmula:C22H27NO5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:385.45
  • Alaproclate (hydrochloride)

    CAS:
    <p>Alaproclate, an SSRI, enhances serotonin and SIRT1, hinders NMDA and K+ currents in neurons, and shows antidepressant-like effects in rats.</p>
    Fórmula:C13H19Cl2NO2
    Forma y color:Solid
    Peso molecular:292.2
  • MPDC

    CAS:
    <p>MPDC acts as a competitive inhibitor against the Na+-dependent high-affinity glutamate transporter within forebrain synaptosomes.</p>
    Fórmula:C7H9NO4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:171.15
  • Levemopamil HCl

    CAS:
    <p>Levemopamil HCl is used as a calcium channel blocker.</p>
    Fórmula:C23H31ClN2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:370.96
  • SB 206553 hydrochloride

    CAS:
    <p>SB 206553 hydrochloride is a 5-HT2C inverse agonist and a 5-HT2C/5-HT2B receptor antagonist with anxiolytic activity, useful for studying neurological disorders</p>
    Fórmula:C17H17ClN4O
    Pureza:99.56%
    Forma y color:Solid
    Peso molecular:328.8
  • RLH 033

    CAS:
    <p>RLH 033 is a selective ligand for the sigma 1 recognition site.</p>
    Fórmula:C25H31ClN2O4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:458.98
  • AChE/BChE/MAO-B-IN-2


    <p>AChE/BChE/MAO-B-IN-2 inhibits AChE (48.2 nM), BChE (83.9 nM), MAO-B (31.2 nM), has antioxidant activity, and aids Parkinson's research.</p>
    Fórmula:C25H31N3O3
    Forma y color:Solid
    Peso molecular:421.53
  • SV5

    CAS:
    <p>SV5: potent anti-Alzheimer's, protects SHSY-5Y from Aβ1-42 death, stable with optimal pharmacology in plasma, antioxidant, neuroprotective.</p>
    Fórmula:C21H30N2O4S2
    Forma y color:Solid
    Peso molecular:438.6
  • S 14063

    CAS:
    <p>S 14063 is a potent 5-HT1A receptor antagonist devoid of beta-adrenoceptor blocking properties.</p>
    Fórmula:C22H29Cl2N3O2S
    Forma y color:Solid
    Peso molecular:470.45
  • Bradanicline

    CAS:
    <p>Bradanicline: potent α7 nAChR agonist, EC50=17 nM, Ki=1.4 nM, used in cognitive disorder research.</p>
    Fórmula:C22H23N3O2
    Forma y color:Solid
    Peso molecular:361.44
  • hMAO-B-IN-6

    CAS:
    <p>Compound 17d (hMAO-B-IN-6) is an effective and selective hMAO-B inhibitor, demonstrating an IC 50 of 67.02 nM. It significantly ameliorates cognitive deficits induced by Scopolamine in Alzheimer's disease (AD) mice [1].</p>
    Fórmula:C19H20N2O5
    Forma y color:Solid
    Peso molecular:356.37
  • CP94253 hydrochloride

    CAS:
    <p>CP94253 hydrochloride: selective 5-HT1B agonist, Ki=2 nM; less active on 5-HT1A/D/C/2 (Ki=89/49/860/1600 nM).</p>
    Fórmula:C15H20ClN3O
    Pureza:99.78%
    Forma y color:Solid
    Peso molecular:293.79
  • JNJ1930942

    CAS:
    <p>JNJ1930942 is a novel positive allosteric modulator of the α7 nicotinic acetylcholine receptor.</p>
    Fórmula:C16H11F4N3OS
    Forma y color:Solid
    Peso molecular:369.34
  • Carburazepam

    CAS:
    <p>Carburazepam is a derivate of benzodiazepines. Benzodiazepines are a class of psychoactive drugs.</p>
    Fórmula:C17H16ClN3O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:329.78