
Neurociencia
Los inhibidores en neurociencia son compuestos diseñados para modular la actividad de proteínas, enzimas o receptores específicos dentro del sistema nervioso. Estos inhibidores son cruciales para estudiar los mecanismos moleculares subyacentes a la función neuronal, la transmisión sináptica y las enfermedades neurodegenerativas. Al dirigirse a los receptores de neurotransmisores, canales iónicos y vías de señalización, los inhibidores en neurociencia ayudan en la exploración de la función cerebral y en el desarrollo de estrategias terapéuticas para trastornos neurológicos como el Alzheimer, Parkinson y la epilepsia. En CymitQuimica, ofrecemos una amplia gama de inhibidores de neurociencia de alta calidad para apoyar su investigación en neurobiología, neurofarmacología y ciencias cognitivas.
Subcategorías de "Neurociencia"
- Receptor 5-HT(942 productos)
- ACK(1 productos)
- AChR(575 productos)
- ATP Citrato Liasa(16 productos)
- Receptor adrenérgico(2.946 productos)
- BACE(36 productos)
- Beta amiloide(205 productos)
- CAMK(69 productos)
- Inhibidores de ciclooxigenasa (COX)(562 productos)
- Receptor de dopamina(408 productos)
- Receptor GABA(336 productos)
- Gamma-secretasa(59 productos)
- GluR(255 productos)
- GlyT(24 productos)
- Receptor de histamina(359 productos)
- LRRK2(33 productos)
- Receptor de melatonina(24 productos)
- NMDAR(28 productos)
- Receptor de OX(40 productos)
- Receptor de opioides(298 productos)
Mostrar 12 subcategorías más
Se han encontrado 5400 productos de "Neurociencia"
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ACPT-II
CAS:<p>metabotropic receptor antagonist</p>Fórmula:C8H11NO6Pureza:98%Forma y color:SolidPeso molecular:217.18AChE-IN-15
CAS:<p>AChE-IN-15 is a reversible inhibitor of huAChE and huBChE (IC50: 6.8 μM, 16.1 μM), with antioxidant activity, used in Alzheimer's research.</p>Fórmula:C23H24N2O7Forma y color:SolidPeso molecular:440.45LY 393558
CAS:<p>Dual 5-HT1B/1D receptor antagonist</p>Fórmula:C26H31FN4O4S2Pureza:98%Forma y color:SolidPeso molecular:546.68AChE/BChE-IN-9
CAS:<p>Compound 7a inhibits AChE/BChE (IC50: 5.74/14.05 μM), has antioxidant effects (IC50: 57.35 μM), chelates iron, and affects amyloid β 1-42 aggregation.</p>Fórmula:C20H19N3O4Forma y color:SolidPeso molecular:365.38Z164597606
CAS:<p>Z164597606 inhibits BChE (1.3 μM equine, 1.7 μM human), binds Trp82 via π-π, potential in Alzheimer's research.</p>Fórmula:C20H19N3O4Forma y color:SolidPeso molecular:365.38Quifenadine
CAS:<p>Quifenadine, an H1-histamine receptor blocker, has antiarrhythmic properties.</p>Fórmula:C20H23NOPureza:98%Forma y color:SolidPeso molecular:293.4Tacitin
CAS:<p>Tacitin (Benzoctamine Hydrochloride) shows sedative and anti-anxiety properties. Tacitin blocks the central postsynaptic serotonin receptors.</p>Fórmula:C18H20ClNPureza:98%Forma y color:SolidPeso molecular:285.81VU0652835
CAS:<p>VU0652835 is a negative allosteric modulator of metabotropic glutamate receptor subtype 5 (mGlu5) (IC50: 81 nM).</p>Fórmula:C16H19N3O3SPureza:98%Forma y color:SolidPeso molecular:333.41Iprindole
CAS:<p>Iprindole, a tricyclic indole antidepressant, is a dual weak inhibitor of noradrenaline and 5-HT uptake [1].</p>Fórmula:C19H28N2Pureza:99.54%Forma y color:SolidPeso molecular:284.44Metixene hydrochloride
CAS:<p>Metixene hydrochloride is an anticholinergic antiparkinsonian agent.</p>Fórmula:C20H24ClNSPureza:98%Forma y color:SolidPeso molecular:345.93AVN-322
CAS:<p>AVN-322 is a 5-HT6 receptor antagonist. 5-HT6R antagonists improves cognition in animal models of cognitive impairment.</p>Fórmula:C17H20ClN5O2SPureza:>99.99%Forma y color:SolidPeso molecular:393.89Darenzepine
CAS:<p>Darenzepine is a muscarinic receptor inhibitor.</p>Fórmula:C21H21N3O2Pureza:99.87%Forma y color:SolidPeso molecular:347.41Cinitapride Hydrogen Tartrate
CAS:<p>Cinitapride Hydrogen Tartrate is a gastroprokinetic agent that acts as an antagonist of the 5-HT2 receptors and as an agonist of the 5-HT1 and 5-HT4 receptors</p>Fórmula:C25H36N4O10Pureza:98%Forma y color:SolidPeso molecular:552.581MSOP
CAS:MSOP is a selective antagonist of group III metabotropic glutamate receptor (KD of 51 μM for the L-AP4-sensitive presynaptic mGluR).Fórmula:C4H10NO6PPureza:98%Forma y color:SolidPeso molecular:199.1Repinotan HCl
CAS:<p>Repinotan HCl (Bay-x-3702) is a 5-HT1A receptor agonist with potent neuroprotective effects for the study of ischemic stroke and traumatic brain injury.</p>Fórmula:C21H25ClN2O4SPureza:99.57%Forma y color:SolidPeso molecular:436.95EMDT
CAS:<p>EMDT oxalate is a selective 5-HT6 agonist, and has antidepressant effects.</p>Fórmula:C15H22N2OPureza:97.66% - 99.78%Forma y color:SolidPeso molecular:246.35A-794282
CAS:<p>A-794282 is a selective antagonist of mGluR1.</p>Fórmula:C19H18N4OSPureza:99.87%Forma y color:SolidPeso molecular:350.44CGS8216
CAS:<p>CGS8216 shows analgesic activity at high doses, has anxiolytic activity, and can be used to study immune system disorders.</p>Fórmula:C16H11N3OPureza:98.53%Forma y color:SolidPeso molecular:261.28(1S,3R)-ACPD
CAS:<p>(1S,3R)-ACPD is a group I and II mGlu receptor agonist.</p>Fórmula:C7H11NO4Pureza:98%Forma y color:SolidPeso molecular:173.17DS2
CAS:<p>Positive allosteric modulator of δ-subunit containing GABAA receptors</p>Fórmula:C18H12ClN3OSPureza:98%Forma y color:SolidPeso molecular:353.83Foliglurax monohydrochloride
CAS:<p>Foliglurax monohydrochloride, an antiparkinsonian, is a selective brain-penetrant mGluR4 PAM with an EC50 of 79 nM.</p>Fórmula:C23H24ClN3O3SForma y color:SolidPeso molecular:457.9717-PA
CAS:<p>17-PA is a GABAA receptor antagonist.</p>Fórmula:C25H34OPureza:98%Forma y color:SolidPeso molecular:350.54Prenylamine lactate
CAS:<p>Prenylamine lactate, an ex-angina drug, depletes heart catecholamines and blocks calcium channels.</p>Fórmula:C27H33NO3Pureza:98%Forma y color:SolidPeso molecular:419.56UCSF678
CAS:<p>UCSF678: selective 42 nM partial agonist at 5-HT5AR, fewer off-target effects, and lower assay risks than SB-699551.</p>Fórmula:C15H18N2O2SForma y color:SolidPeso molecular:290.38CGP11952
CAS:<p>CGP11952 is same the benzodiazepines in its pharmacological action and it also is an experimental benzodiazepine derivative.</p>Fórmula:C21H21Cl2N5O2Pureza:98%Forma y color:SolidPeso molecular:446.33Itameline
CAS:<p>RU 47213 can be used to inhibit scopolamine-induced working memory impairment in rats.</p>Fórmula:C14H15ClN2O3Pureza:99.55%Forma y color:SolidPeso molecular:294.73VU0361747
CAS:<p>VU0361747 is a positive allosteric modulators (PAM) of metabotropic glutamate receptor subtype 5 (mGlu5).</p>Fórmula:C19H17FN2O2Forma y color:SolidPeso molecular:324.35TC 2559 difumarate
CAS:<p>partial agonist of α4β2 nicotinic acetylcholine receptor</p>Fórmula:C12H18N2OC4H404Pureza:98%Forma y color:SolidPeso molecular:380.39mGAT3/4-IN-1
CAS:<p>mGAT3/4-IN-1 inhibits mGAT3/4 with pIC50: 5.31/5.24, reduces neuropathic pain in diabetic mice.</p>Fórmula:C26H31ClN2O2S2Forma y color:SolidPeso molecular:503.12JNJ-55308942
CAS:<p>JNJ-55308942: selective, brain-penetrant P2X7 antagonist; IC50s: 10nM (human), 15nM (rat); Kis: 7.1nM (h), 2.9nM (r).</p>Fórmula:C17H12F5N7OPureza:99.94%Forma y color:SolidPeso molecular:425.32Org 24598
CAS:<p>Potent GlyT1b inhibitor, IC50 = 6.9 nM; little effect on GlyT-2, adrenoceptors, dopamine, 5HT receptors, GABA transporters.</p>Fórmula:C19H20F3NO3Forma y color:SolidPeso molecular:367.36GABAA receptor agent 4
CAS:<p>Compound 1e is a potent γ-GABAAR antagonist with a Ki of 0.18 µM, offering immunomodulatory effects on T cell proliferation.</p>Fórmula:C17H24N2OForma y color:SolidPeso molecular:272.39ML169
CAS:<p>ML169 is a selective and brain penetrant M1 positive allosteric modulator (PAM).</p>Fórmula:C21H17BrFN3O4SPureza:98%Forma y color:SolidPeso molecular:506.34Aβ42-IN-2
CAS:<p>Aβ42-IN-2 is a γ-secretase modulator. Aβ42-IN-2 has an IC 50 of 6.5 nM for Αβ 42. Aβ42-IN-2 can be used for the Alzheimer's disease research[1].</p>Fórmula:C24H26N6O2Pureza:98.09% - 99.87%Forma y color:SolidPeso molecular:430.5Glemanserin
CAS:<p>Glemanserin (MDL11939) is a specific 5-HT2A antagonist with Ki values of 0.54 nM, 2.5 nM and 2.89 nM for rabbit, human and rat 5-HT2A.</p>Fórmula:C20H25NOPureza:99.93%Forma y color:SolidPeso molecular:295.42hMAO-B-IN-2
CAS:<p>hMAO-B-IN-2: selective oral hMAO-B inhibitor, crosses BBB, IC50=4 nM, potential for Alzheimer's research, neuroprotective, low toxicity.</p>Fórmula:C18H23NO3Forma y color:SolidPeso molecular:301.38LY 2365109 hydrochloride
CAS:<p>glycine transporter 1 (GlyT1) inhibitor</p>Fórmula:C22H27NO5Pureza:98%Forma y color:SolidPeso molecular:385.45Alaproclate (hydrochloride)
CAS:<p>Alaproclate, an SSRI, enhances serotonin and SIRT1, hinders NMDA and K+ currents in neurons, and shows antidepressant-like effects in rats.</p>Fórmula:C13H19Cl2NO2Forma y color:SolidPeso molecular:292.2MPDC
CAS:<p>MPDC acts as a competitive inhibitor against the Na+-dependent high-affinity glutamate transporter within forebrain synaptosomes.</p>Fórmula:C7H9NO4Pureza:98%Forma y color:SolidPeso molecular:171.15Levemopamil HCl
CAS:<p>Levemopamil HCl is used as a calcium channel blocker.</p>Fórmula:C23H31ClN2Pureza:98%Forma y color:SolidPeso molecular:370.96SB 206553 hydrochloride
CAS:<p>SB 206553 hydrochloride is a 5-HT2C inverse agonist and a 5-HT2C/5-HT2B receptor antagonist with anxiolytic activity, useful for studying neurological disorders</p>Fórmula:C17H17ClN4OPureza:99.56%Forma y color:SolidPeso molecular:328.8RLH 033
CAS:<p>RLH 033 is a selective ligand for the sigma 1 recognition site.</p>Fórmula:C25H31ClN2O4Pureza:98%Forma y color:SolidPeso molecular:458.98AChE/BChE/MAO-B-IN-2
<p>AChE/BChE/MAO-B-IN-2 inhibits AChE (48.2 nM), BChE (83.9 nM), MAO-B (31.2 nM), has antioxidant activity, and aids Parkinson's research.</p>Fórmula:C25H31N3O3Forma y color:SolidPeso molecular:421.53SV5
CAS:<p>SV5: potent anti-Alzheimer's, protects SHSY-5Y from Aβ1-42 death, stable with optimal pharmacology in plasma, antioxidant, neuroprotective.</p>Fórmula:C21H30N2O4S2Forma y color:SolidPeso molecular:438.6S 14063
CAS:<p>S 14063 is a potent 5-HT1A receptor antagonist devoid of beta-adrenoceptor blocking properties.</p>Fórmula:C22H29Cl2N3O2SForma y color:SolidPeso molecular:470.45Bradanicline
CAS:<p>Bradanicline: potent α7 nAChR agonist, EC50=17 nM, Ki=1.4 nM, used in cognitive disorder research.</p>Fórmula:C22H23N3O2Forma y color:SolidPeso molecular:361.44hMAO-B-IN-6
CAS:<p>Compound 17d (hMAO-B-IN-6) is an effective and selective hMAO-B inhibitor, demonstrating an IC 50 of 67.02 nM. It significantly ameliorates cognitive deficits induced by Scopolamine in Alzheimer's disease (AD) mice [1].</p>Fórmula:C19H20N2O5Forma y color:SolidPeso molecular:356.37CP94253 hydrochloride
CAS:<p>CP94253 hydrochloride: selective 5-HT1B agonist, Ki=2 nM; less active on 5-HT1A/D/C/2 (Ki=89/49/860/1600 nM).</p>Fórmula:C15H20ClN3OPureza:99.78%Forma y color:SolidPeso molecular:293.79JNJ1930942
CAS:<p>JNJ1930942 is a novel positive allosteric modulator of the α7 nicotinic acetylcholine receptor.</p>Fórmula:C16H11F4N3OSForma y color:SolidPeso molecular:369.34Carburazepam
CAS:<p>Carburazepam is a derivate of benzodiazepines. Benzodiazepines are a class of psychoactive drugs.</p>Fórmula:C17H16ClN3O2Pureza:98%Forma y color:SolidPeso molecular:329.78
