
Neurociencia
Los inhibidores en neurociencia son compuestos diseñados para modular la actividad de proteínas, enzimas o receptores específicos dentro del sistema nervioso. Estos inhibidores son cruciales para estudiar los mecanismos moleculares subyacentes a la función neuronal, la transmisión sináptica y las enfermedades neurodegenerativas. Al dirigirse a los receptores de neurotransmisores, canales iónicos y vías de señalización, los inhibidores en neurociencia ayudan en la exploración de la función cerebral y en el desarrollo de estrategias terapéuticas para trastornos neurológicos como el Alzheimer, Parkinson y la epilepsia. En CymitQuimica, ofrecemos una amplia gama de inhibidores de neurociencia de alta calidad para apoyar su investigación en neurobiología, neurofarmacología y ciencias cognitivas.
Subcategorías de "Neurociencia"
- Receptor 5-HT(939 productos)
- ACK(1 productos)
- AChR(575 productos)
- ATP Citrato Liasa(16 productos)
- Receptor adrenérgico(2.945 productos)
- BACE(36 productos)
- Beta amiloide(205 productos)
- CAMK(69 productos)
- Inhibidores de ciclooxigenasa (COX)(561 productos)
- Receptor de dopamina(407 productos)
- Receptor GABA(336 productos)
- Gamma-secretasa(59 productos)
- GluR(255 productos)
- GlyT(24 productos)
- Receptor de histamina(358 productos)
- LRRK2(33 productos)
- Receptor de melatonina(24 productos)
- NMDAR(28 productos)
- Receptor de OX(40 productos)
- Receptor de opioides(297 productos)
Mostrar 12 subcategorías más
Se han encontrado 5398 productos de "Neurociencia"
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NRA-0160
CAS:<p>NRA-0160 is a selective antagonist of dopamine D4 receptor(Ki of 0.48 nM)</p>Fórmula:C24H23F2N3OSPureza:98%Forma y color:SolidPeso molecular:439.52AR-R 17779 hydrochloride
CAS:<p>AR-R17779 hydrochloride: potent α7 nAChR agonist; K i : 92 nM (α7), 16,000 nM (α4β2); enhances rat cognition; anxiolytic; anti-inflammatory.</p>Fórmula:C9H15ClN2O2Forma y color:SolidPeso molecular:218.68PNU-142633
CAS:<p>PNU-142633: anti-migraine, selective 5-HT1D agonist, Ki=6 nM; >18,000 nM for 5-HT1B.</p>Fórmula:C24H30N4O3Pureza:98%Forma y color:SolidPeso molecular:422.52Etbicyphat
CAS:<p>Etbicyphat: potent GABA(A) antagonist, induces epileptiform activity, binds to GABA/benzodiazepine receptors.</p>Fórmula:C6H11O4PForma y color:SolidPeso molecular:178.12SSAO inhibitor-2
CAS:<p>SSAO inhibitor-2 targets human SSAO (<10 nM) and MAO-A (10-100 μM); useful in various diseases research.</p>Fórmula:C14H21FN4O2Forma y color:SolidPeso molecular:296.342-Methyl-5-HT maleate
CAS:<p>2-Methyl-5-HT maleate, a selective 5-HT3 agonist, shows anti-depressive effects.</p>Fórmula:C15H18N2O5Pureza:98%Forma y color:SolidPeso molecular:306.31AChE/BChE-IN-2
CAS:<p>AChE/BChE-IN-2 (Compound 13b) is a potent inhibitor of AChE/BChE with IC50 values of 0.96 ± 0.14 μM and 1.23 ± 0.23 μM for AChE and BChE, respectively.</p>Fórmula:C23H25N3O5Forma y color:SolidPeso molecular:423.46Arecaidine propargyl ester tosylate
CAS:<p>Arecaidine propargyl ester tosylate is a muscarinic receptor agonist.</p>Fórmula:C17H21NO5SPureza:98%Forma y color:SolidPeso molecular:351.425-HT3 antagonist 2
CAS:<p>5-HT3 antagonist 2 is an antagonist of 5-HT3 receptor.</p>Fórmula:C18H21N3OPureza:98%Forma y color:SolidPeso molecular:295.38MAP4
CAS:<p>metabotropic glutamate receptor modulator</p>Fórmula:C5H12NO5PPureza:98%Forma y color:White SolidPeso molecular:197.13PQCA
CAS:<p>PQCA is a selective M1 receptor modulator with EC50s of 49 nM (monkey) and 135 nM (human), potential for Alzheimer's treatment.</p>Fórmula:C22H20N4O3Pureza:99.88%Forma y color:SolidPeso molecular:388.42ADX71743
CAS:<p>ADX71743 is a potent and selective negative allosteric modulator of metabotropic glutamate receptor 7.</p>Fórmula:C17H19NO2Forma y color:SolidPeso molecular:269.34GABA-AT-IN-1
CAS:<p>GABA-AT-IN-1 (Compound 6) is an inhibitor of γ-aminobutyric acid transaminase (GABA-AT) that crosses the blood-brain barrier.</p>Fórmula:C23H18N2O6Forma y color:SolidPeso molecular:418.4SB-221284
CAS:<p>5-HT2C/2B receptor antagonist</p>Fórmula:C16H14F3N3OSPureza:98%Forma y color:SolidPeso molecular:353.36LY 125180
CAS:<p>LY 125180 is a serotonin antagonist.</p>Fórmula:C18H24ClNOPureza:98%Forma y color:SolidPeso molecular:305.84Cinitapride Hydrogen Tartrate
CAS:<p>Cinitapride Hydrogen Tartrate is a gastroprokinetic agent that acts as an antagonist of the 5-HT2 receptors and as an agonist of the 5-HT1 and 5-HT4 receptors</p>Fórmula:C25H36N4O10Pureza:98%Forma y color:SolidPeso molecular:552.581ML375
CAS:<p>ML375 is a potent, selective and CNS penetrant M5 negative allosteric modulator (NAM).</p>Fórmula:C23H15ClF2N2O2Forma y color:SolidPeso molecular:424.83Rapacuronium bromide
CAS:Rapacuronium bromide is an allosteric muscarinic acetylcholine receptor (mAChR) modulator.Fórmula:C37H61BrN2O4Pureza:98%Forma y color:SolidPeso molecular:677.8LY 334370 hydrochloride
CAS:<p>5-HT1F receptor agonist</p>Fórmula:C21H23ClFN3OPureza:98%Forma y color:SolidPeso molecular:387.88Org-12962
CAS:<p>Org-12962: 5-HT2C agonist (pEC50: 7.01), anti-panic in rats, affects 5-HT2A/B (pEC50: 6.38/6.28).</p>Fórmula:C10H11ClF3N3Pureza:98.34%Forma y color:SolidPeso molecular:265.66Dimethyl-W84 (dibromide)
CAS:<p>Dimethyl-W84, selective M2 muscarinic receptor modulator; slows N-methylscopolamine release, EC50=3 nM.</p>Fórmula:C34H48Br2N4O4Forma y color:SolidPeso molecular:736.59p-MPPF dihydrochloride
CAS:<p>p-MPPF dihydrochloride is a 5-HT antagonist that can be used to study neurological diseases.</p>Fórmula:C25H29Cl2FN4O2Pureza:99.55%Forma y color:SolidPeso molecular:507.43Pivalylbenzhydrazine
CAS:<p>Pivhydrazine: strong MAO inhibitor, stunts rat cartilage growth, used in depression research.</p>Fórmula:C12H18N2OForma y color:SolidPeso molecular:206.28Aβ42-IN-1 free base
CAS:<p>Aβ42-IN-1 free base (compound 1v), an orally active γ-secretase modulator with high brain exposure, effectively lowers Aβ42 levels, exhibiting an IC 50 of 0.091</p>Fórmula:C29H26N4O2Pureza:98%Forma y color:SolidPeso molecular:462.54(R)-Baclofen hydrochloride
CAS:<p>Arbaclofen HCl, a GABA-B agonist, treats spasticity from spinal injury by reducing excitatory transmission.</p>Fórmula:C10H13Cl2NO2Pureza:98%Forma y color:SolidPeso molecular:250.12VU 6008667
CAS:VU 6008667 is a selective negative allosteric M5 NAM modulator (IC50s: 1.2 μM and 1.6 μM for human M5 and rat M5, respectively).Fórmula:C24H17ClF2N2O2Pureza:98%Forma y color:SolidPeso molecular:438.85Obidoxime dichloride
CAS:<p>Obidoxime dichloride is an antidote for organophosphate poisoning that enhances the positive inotropic effect of phosphamidon on isolated working rat hearts.</p>Fórmula:C14H16Cl2N4O3Pureza:98%Forma y color:SolidPeso molecular:359.21MSOP
CAS:MSOP is a selective antagonist of group III metabotropic glutamate receptor (KD of 51 μM for the L-AP4-sensitive presynaptic mGluR).Fórmula:C4H10NO6PPureza:98%Forma y color:SolidPeso molecular:199.1Repinotan HCl
CAS:<p>Repinotan HCl (Bay-x-3702) is a 5-HT1A receptor agonist with potent neuroprotective effects for the study of ischemic stroke and traumatic brain injury.</p>Fórmula:C21H25ClN2O4SPureza:99.57%Forma y color:SolidPeso molecular:436.95EMDT
CAS:<p>EMDT oxalate is a selective 5-HT6 agonist, and has antidepressant effects.</p>Fórmula:C15H22N2OPureza:97.66% - 99.78%Forma y color:SolidPeso molecular:246.35PF-184298
CAS:<p>PF-184298 is a serotonin and norepinephrine monoamine reuptake inhibitor (SNRI) that inhibits dopamine reuptake.</p>Fórmula:C15H20Cl2N2OPureza:98.67%Forma y color:SolidPeso molecular:315.24Oxetorone fumarate
CAS:<p>Oxetorone fumarate is a non-selective, orally active antagonist of serotonin and 5-HT receptors,used for migraine treatment.</p>Fórmula:C25H25NO6Pureza:99.809%Forma y color:SolidPeso molecular:435.48Bibn 99
CAS:<p>Bibn 99, a lipophilic and selective muscarinic M2 receptor antagonist, has applications in cognitive performance and Alzheimer's Disease.</p>Fórmula:C31H42ClN5O3Forma y color:SolidPeso molecular:568.15RJR 2429 dihydrochloride
CAS:<p>nAChR agonist that displays selectivity for α4β2</p>Fórmula:C12H18Cl2N2Pureza:98%Forma y color:SolidPeso molecular:261.19Methoxy-PEPy
CAS:<p>Methoxy-PEPy is a potent and selective mGlu5 receptor inhibitor with an IC50 value of 1 nM.</p>Fórmula:C13H10N2OPureza:99.22%Forma y color:SolidPeso molecular:210.23ELN318463 racemate
CAS:<p>ELN318463 racemate (ELN 318463 racemate) is the racemate of ELN318463 which is an amyloid precursor protein (APP) selective γ-secretase inhibitor.</p>Fórmula:C19H20BrClN2O3SPureza:99.69%Forma y color:SolidPeso molecular:471.8BChE-IN-15
<p>BChE-IN-15 is a compound characterized as a pseudo-irreversible, covalent inhibitor of butyrylcholinesterase (BChE), demonstrating potent activity with an</p>Fórmula:C22H33N3O2Forma y color:SolidPeso molecular:371.52(R,R)-Glycopyrrolate
CAS:<p>(R,R)-Glycopyrrolate is an agent of anticholinergic, has the ability to reduce the frequency of drooling in vivo with developmental disabilities.</p>Fórmula:C19H28BrNO3Pureza:98%Forma y color:SolidPeso molecular:398.34BisQ
CAS:<p>BisQ is an agonist of photochromic. It used for the muscle-type nAChR.</p>Fórmula:C20H30IN4Pureza:98%Forma y color:SolidPeso molecular:453.392EMD 386088 hydrochloride
CAS:<p>EMD 386088 hydrochloride is a 5-HT6 receptor agonist.</p>Fórmula:C14H16Cl2N2Pureza:98%Forma y color:SolidPeso molecular:283.2SCH-23390 maleate
CAS:<p>SCH-23390 maleate (R-(+)-SCH-23390 maleate) is a potent and selective antagonist of dopamine D1-like receptor (1 and D5 receptor with Kis of 0.2 nM and 0.3 nM,</p>Fórmula:C21H22ClNO5Pureza:98%Forma y color:SolidPeso molecular:403.86CGS-12066 maleate salt
CAS:<p>CGS-12066 maleate salt is an agonist of 5-HT1B serotonin receptor.</p>Fórmula:C21H21F3N4O4Forma y color:SolidPeso molecular:450.41Org37684
CAS:<p>5-HT2 receptors agonist</p>Fórmula:C14H20ClNO2Pureza:98%Forma y color:SolidPeso molecular:269.77Tedatioxetine hydrobromide
CAS:<p>Tedatioxetine hydrobromide (Lu AA 24530 hydrobromide) is a serotonin-norepinephrine-dopamine reuptake inhibitor and 5-HT2A receptor antagonist.</p>Fórmula:C18H22BrNSPureza:99.65%Forma y color:SolidPeso molecular:364.34SR 16584
CAS:<p>α3β4 nAChR antagonist</p>Fórmula:C17H22N2OPureza:99.84%Forma y color:SolidPeso molecular:270.37GR 55562 dihydrochloride
CAS:<p>5-HT1B (5-HT1Dβ) silent antagonist</p>Fórmula:C23H27Cl2N3O2Pureza:99.45%Forma y color:SolidPeso molecular:448.39VU0366248
CAS:<p>VU0366248 is a mGlu5 negative allosteric modulator.</p>Fórmula:C14H7ClF2N2OPureza:98%Forma y color:SolidPeso molecular:292.67PF-3246799
CAS:<p>PF-3246799 is an effective and selective agonist of the 5-HT2C receptor.</p>Fórmula:C15H17N3Pureza:98%Forma y color:SolidPeso molecular:239.32Amitriptylinoxide
CAS:<p>Amitriptylinoxide is an antidepressant.</p>Fórmula:C20H23NOPureza:98%Forma y color:SolidPeso molecular:293.4Pirenzepine
CAS:<p>Pirenzepine targets M1 mAChR, curbs acid secretion, eases spasms, and has anti-cancer properties.</p>Fórmula:C19H21N5O2Forma y color:SolidPeso molecular:351.4
