
Neurociencia
Los inhibidores en neurociencia son compuestos diseñados para modular la actividad de proteínas, enzimas o receptores específicos dentro del sistema nervioso. Estos inhibidores son cruciales para estudiar los mecanismos moleculares subyacentes a la función neuronal, la transmisión sináptica y las enfermedades neurodegenerativas. Al dirigirse a los receptores de neurotransmisores, canales iónicos y vías de señalización, los inhibidores en neurociencia ayudan en la exploración de la función cerebral y en el desarrollo de estrategias terapéuticas para trastornos neurológicos como el Alzheimer, Parkinson y la epilepsia. En CymitQuimica, ofrecemos una amplia gama de inhibidores de neurociencia de alta calidad para apoyar su investigación en neurobiología, neurofarmacología y ciencias cognitivas.
Subcategorías de "Neurociencia"
- Receptor 5-HT(939 productos)
- ACK(1 productos)
- AChR(575 productos)
- ATP Citrato Liasa(16 productos)
- Receptor adrenérgico(2.945 productos)
- BACE(36 productos)
- Beta amiloide(205 productos)
- CAMK(69 productos)
- Inhibidores de ciclooxigenasa (COX)(561 productos)
- Receptor de dopamina(407 productos)
- Receptor GABA(336 productos)
- Gamma-secretasa(59 productos)
- GluR(255 productos)
- GlyT(24 productos)
- Receptor de histamina(358 productos)
- LRRK2(33 productos)
- Receptor de melatonina(24 productos)
- NMDAR(28 productos)
- Receptor de OX(40 productos)
- Receptor de opioides(297 productos)
Mostrar 12 subcategorías más
Se han encontrado 5400 productos de "Neurociencia"
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VU0409106
CAS:<p>VU0409106 is a potent, mGlu5-selective inhibitor.</p>Fórmula:C15H11FN4O2SPureza:98%Forma y color:SolidPeso molecular:330.34CGS 12066B dimaleate
CAS:<p>5-HT1B full agonist</p>Fórmula:C25H25F3N4O8Pureza:98%Forma y color:SolidPeso molecular:566.48AChE-IN-12
CAS:<p>AChE-IN-12 inhibited rat/eel AChE, crossed BBB, prevented Aβ1-42 aggregation, and has potential for Alzheimer's research.</p>Fórmula:C33H41NO7Forma y color:SolidPeso molecular:563.68CP 135807
CAS:<p>CP 135807 is a 5-HT1D receptor agonist.</p>Fórmula:C19H21N5O2Pureza:98%Forma y color:SolidPeso molecular:351.4ZK93423
CAS:<p>ZK93423: potent benzodiazepine agonist, IC50=1nM, non-selective, Ki=4.1-6nM for α1-α5 GABAA subunits.</p>Fórmula:C23H22N2O4Forma y color:SolidPeso molecular:390.43VU0463841
CAS:<p>VU0463841 is a mGlu5 negative allosteric modulators.</p>Fórmula:C13H8ClFN4OForma y color:SolidPeso molecular:290.68VU 0360172 hydrochloride
CAS:<p>positive allosteric modulator of mGlu5 receptors</p>Fórmula:C18H16ClFN2OPureza:98%Forma y color:SolidPeso molecular:330.78RLH 033
CAS:<p>RLH 033 is a selective ligand for the sigma 1 recognition site.</p>Fórmula:C25H31ClN2O4Pureza:98%Forma y color:SolidPeso molecular:458.98COX-2-IN-2
CAS:<p>COX-2-IN-2 selectively inhibits COX2 (IC50: 0.24 μM); COX-2-IN-1 offers anti-inflammatory and pain relief.</p>Fórmula:C17H12FN3O2SPureza:97.62%Forma y color:SolidPeso molecular:341.36Territrem B
CAS:<p>Territrem B: A mycotoxin that irreversibly blocks AChE, causes tremors in mice at 0.21 mg/kg.</p>Fórmula:C29H34O9Forma y color:SolidPeso molecular:526.57AChE-IN-20
CAS:<p>AChE-IN-20: AChE inhibitor (IC50: 397.32 nM), hCA-I/II blocker (IC50: ~77 nM avg), α GLY suppressor (IC50: 52.08 nM).</p>Fórmula:C22H20N8O6S2Forma y color:SolidPeso molecular:556.57AChE/BChE/MAO-B-IN-3
<p>AChE/BChE/MAO-B-IN-3: potent MAO-B, AChE & BChE inhibitor; IC50: 0.0359μM (MAO-B), 0.0473/0.0782μM (AChE/BChE); possible Alzheimer's research use.</p>Fórmula:C25H31N3O3Forma y color:SolidPeso molecular:421.53Bopindolol (malonate)
CAS:<p>Bopindolol is a non-selective β-adrenergic receptor antagonist.</p>Fórmula:C26H32N2O7Forma y color:SolidPeso molecular:484.549Naronapride
CAS:<p>Naronapride (ATI-7505) is a potent agonist of the prokinetic 5-HT4receptor and can be used to study gastrointestinal disorders.</p>Fórmula:C27H41ClN4O5Forma y color:SolidPeso molecular:537.09SSAO inhibitor-3
CAS:<p>SSAO inhibitor-3 targets human AOC1/SSAO in atherosclerosis, diabetes, obesity, CKD, and more, with IC50s of 0.1-10 μM/<10 nM.</p>Fórmula:C15H23FN4O3Forma y color:SolidPeso molecular:326.37BuChE-IN-6
CAS:<p>BuChE-IN-6 inhibits BuChE (IC50: 0.46 μM eqBuChE, 0.51 μM hBuChE) and prevents Aβ 42 self-aggregation.</p>Fórmula:C21H26N4O2Forma y color:SolidPeso molecular:366.46MDL-29951
CAS:<p>MDL-29951 is a novel glycine antagonist of NMDA receptor activation.</p>Fórmula:C12H9Cl2NO4Pureza:98.79% - 99.49%Forma y color:SolidPeso molecular:302.11SC58451
CAS:<p>SC58451 is a novel potent, orally active and selective COX-2 inhibitor.SC58451 showed anti-inflammatory activity in a rat model of arthritis.</p>Fórmula:C20H19FO2SPureza:>99.99%Forma y color:SolidPeso molecular:342.43S 14506 hydrochloride
CAS:<p>S 14506 hydrochloride is a 5-HT1A receptor full agonist.</p>Fórmula:C24H27ClFN3O2Pureza:99.92%Forma y color:SolidPeso molecular:443.94Timegadine
CAS:<p>Timegadine is a competitive inhibitor of COX and lipo-oxygenase, with IC50s ranging from 5 nM (washed rabbit platelets) to 20 μM (rat brain) for COX and 100 μM</p>Fórmula:C20H23N5SPureza:98%Forma y color:SolidPeso molecular:365.5Prifuroline
CAS:<p>Prifuroline is an agent of antiarrhythmic.</p>Fórmula:C14H16N2OPureza:98%Forma y color:SolidPeso molecular:228.29LY2607540
CAS:<p>LY2607540 is a metabotropic glutamate 2 potentiator with potential anxiolytic/antidepressant properties (EC(50) = 23 and 13 nM, respectively).</p>Fórmula:C24H24F3N3O4Pureza:98%Forma y color:SolidPeso molecular:475.46NGX-267
CAS:<p>NGX-267, a muscarinic M1 agonist, is used potentially for the treatment of Xerostomia, Alzheimer's disease and cognitive.</p>Fórmula:C10H18N2OSForma y color:SolidPeso molecular:214.33HUHS2002
CAS:<p>HUHS2002 is a free fatty acid derivative that works as a potentiator of GluA1 AMPA receptor responses and α7 ACh receptor responses.</p>Fórmula:C17H24O3Pureza:98%Forma y color:SolidPeso molecular:276.37RGH 1756
CAS:<p>RGH 1756 is an atypical antipsychotic with high affinity to dopamine D(3) receptors that leads to c-Fos induction in a unique pattern.</p>Fórmula:C26H30N4O2SPureza:98%Forma y color:SolidPeso molecular:462.615-Nonyloxytryptamine oxalate
CAS:<p>5-HT1B agonist</p>Fórmula:C21H32N2O5Pureza:98%Forma y color:SolidPeso molecular:392.49Thiazinamium chloride
CAS:<p>Thiazinamium chloride possesses potent anticholinergic and antiallergic activity and inhibits synthesis of TxB2(IC50 value of 0.2 μM).</p>Fórmula:C18H23ClN2SPureza:98%Forma y color:SolidPeso molecular:334.91CPP-115
CAS:<p>CPP-115 is a GABA-aminotransferase inhibitor and a high-affinity vigabatrin analogue.</p>Fórmula:C7H9F2NO2Forma y color:SolidPeso molecular:177.15Epibatidine 2HCl
CAS:<p>Epibatidine 2HCl is a potent nicotinic agonist.</p>Fórmula:C11H15Cl3N2Pureza:98%Forma y color:SolidPeso molecular:281.61LP 20 hydrochloride
CAS:<p>ligand of the 5-HT7 receptor</p>Fórmula:C17H21ClN2OPureza:98%Forma y color:SolidPeso molecular:304.81Siltenzepine
CAS:<p>Siltenzepine is an agent of anti-acid agent,and used in the treatment of peptic ulcers.</p>Fórmula:C19H20ClN3O4Pureza:98%Forma y color:SolidPeso molecular:389.83RS 45041-190 hydrochloride
CAS:<p>Highly selective I2 imidazoline receptor ligand</p>Fórmula:C11H13Cl2N3Pureza:98%Forma y color:SolidPeso molecular:258.15NPS ALX Compound 4a dihydrochloride
CAS:<p>NPS ALX Compound 4a dihydrochloride is a potent and selective antagonist of 5-HT6 receptor (IC50 of 7.2 nM)</p>Fórmula:C25H27Cl2N3O2SPureza:98%Forma y color:SolidPeso molecular:504.47LSP1-2111
CAS:<p>LSP1-2111 is a mGlu4 receptor subtype agonist.</p>Fórmula:C12H17N2O9PForma y color:SolidPeso molecular:364.25Benactyzine
CAS:<p>Benactyzine is a centrally acting muscarinic antagonist.</p>Fórmula:C20H25NO3Pureza:98%Forma y color:Crystals SolidPeso molecular:327.42Lu-AF11205
CAS:<p>Lu-AF11205 is a potent positive allosteric modulator (PAM) of mGlu5 receptor.</p>Fórmula:C17H16N2OSPureza:98%Forma y color:SolidPeso molecular:296.39Fluoroclorgyline
CAS:<p>Fluoroclorgyline is a specific inhibitor of monoamine oxidase A (MAO-A).</p>Fórmula:C13H15ClFNOPureza:98%Forma y color:SolidPeso molecular:255.72(S)-HexylHIBO
CAS:<p>Group I mGlu receptor antagonist</p>Fórmula:C12H20N2O4Pureza:98%Forma y color:SolidPeso molecular:256.3CUMI-101
CAS:<p>CUMI-101 is an agonist of 5-HT1A receptor.</p>Fórmula:C19H27N5O3Forma y color:SolidPeso molecular:373.45Mimopezil
CAS:<p>Mimopezil is an acetylcholinesterase (AChE) inhibitor.</p>Fórmula:C23H23ClN2O3Pureza:98%Forma y color:SolidPeso molecular:410.89(1R,2S)-VU0155041
CAS:<p>(1R,2S)-VU0155041 is the cis regioisomer of VU0155041 and a partial agonist of mGluR4.</p>Fórmula:C14H15Cl2NO3Pureza:98.85%Forma y color:SolidPeso molecular:316.18AS19
CAS:<p>AS19 is a potent, selective 5-HT7 receptor agonist (IC50: 0.83 nM; Ki: 0.6 nM).</p>Fórmula:C18H25N3Pureza:98%Forma y color:SolidPeso molecular:283.41COX-2-IN-1
CAS:<p>COX-2-IN-1 is a potent and selective COX-2 inhibitor (IC50: 3.9 μM).</p>Fórmula:C18H14ClF3N4O2SPureza:>99.99%Forma y color:SolidPeso molecular:442.84PF-184298
CAS:<p>PF-184298 is a serotonin and norepinephrine monoamine reuptake inhibitor (SNRI) that inhibits dopamine reuptake.</p>Fórmula:C15H20Cl2N2OPureza:98.67%Forma y color:SolidPeso molecular:315.24Tedatioxetine hydrobromide
CAS:<p>Tedatioxetine hydrobromide (Lu AA 24530 hydrobromide) is a serotonin-norepinephrine-dopamine reuptake inhibitor and 5-HT2A receptor antagonist.</p>Fórmula:C18H22BrNSPureza:99.65%Forma y color:SolidPeso molecular:364.34Lintopride
CAS:<p>Lintopride is an antagonist of 5HT4. It has moderate 5HT3 antagonist properties.</p>Fórmula:C14H19ClN4O2Pureza:98%Forma y color:SolidPeso molecular:310.78PD-102807
CAS:<p>PD-102807 is a selective and competitive M4 muscarinic receptor antagonist for Parkinson's disease research, inhibit airway smooth muscle (ASM) contraction.</p>Fórmula:C23H24N2O4Pureza:98.90%Forma y color:SolidPeso molecular:392.45E2730
CAS:<p>E2730 is a non-competitive GABA transporter 1 (GAT1) inhibitor with anti-epileptic activity, useful in studying neurological disorders.</p>Fórmula:C9H8F4N2O2SPureza:98.22% - 98.54%Forma y color:SolidPeso molecular:284.23U-89843A
CAS:<p>U-89843A is an allosteric modulator of the GABA_A receptor, known to enhance GABA-induced Cl^- currents [1].</p>Fórmula:C16H24ClN5Pureza:98%Forma y color:SolidPeso molecular:321.85SCH 50911
CAS:<p>SCH 50911 is a selective GABA(B) receptor antagonist with IC50: 1.1 μM, boosting 3H overflow at IC50: 3 μM.</p>Fórmula:C8H15NO3Pureza:98%Forma y color:SolidPeso molecular:173.21
