
Neurociencia
Los inhibidores en neurociencia son compuestos diseñados para modular la actividad de proteínas, enzimas o receptores específicos dentro del sistema nervioso. Estos inhibidores son cruciales para estudiar los mecanismos moleculares subyacentes a la función neuronal, la transmisión sináptica y las enfermedades neurodegenerativas. Al dirigirse a los receptores de neurotransmisores, canales iónicos y vías de señalización, los inhibidores en neurociencia ayudan en la exploración de la función cerebral y en el desarrollo de estrategias terapéuticas para trastornos neurológicos como el Alzheimer, Parkinson y la epilepsia. En CymitQuimica, ofrecemos una amplia gama de inhibidores de neurociencia de alta calidad para apoyar su investigación en neurobiología, neurofarmacología y ciencias cognitivas.
Subcategorías de "Neurociencia"
- Receptor 5-HT(939 productos)
- ACK(1 productos)
- AChR(574 productos)
- ATP Citrato Liasa(16 productos)
- Receptor adrenérgico(2.943 productos)
- BACE(36 productos)
- Beta amiloide(204 productos)
- CAMK(68 productos)
- Inhibidores de ciclooxigenasa (COX)(561 productos)
- Receptor de dopamina(407 productos)
- Receptor GABA(336 productos)
- Gamma-secretasa(59 productos)
- GluR(255 productos)
- GlyT(24 productos)
- Receptor de histamina(358 productos)
- LRRK2(33 productos)
- Receptor de melatonina(24 productos)
- NMDAR(28 productos)
- Receptor de OX(40 productos)
- Receptor de opioides(297 productos)
Mostrar 12 subcategorías más
Se han encontrado 5397 productos de "Neurociencia"
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DSS30
CAS:<p>DSS30 is a P25/CDK5 inhibitor that reduces β-amyloid secretion to help prevent Alzheimer's.</p>Fórmula:C16H14ClNO3S2Pureza:99.19% - 99.4%Forma y color:SolidPeso molecular:367.872-BFI hydrochloride
CAS:<p>2-BFI hydrochloride: High-affinity I2 agonist; used in researching stroke and immune disease protection.</p>Fórmula:C11H11ClN2OPureza:99.94%Forma y color:SolidPeso molecular:222.67E6801
CAS:<p>E6801: selective 5-HT6 agonist for research in dementia, Parkinson's, depression, obesity, epilepsy, anxiety, etc.</p>Fórmula:C17H18ClN5O2S2Pureza:96.32% - 99.53%Forma y color:SolidPeso molecular:423.94SCH-900271
CAS:<p>SCH-900271 treats dyslipidemia by targeting nicotinic acid receptors, addressing hyperlipidaemia.</p>Fórmula:C14H16N2O4Pureza:98.82% - 99.93%Forma y color:SolidPeso molecular:276.29Desformylflustrabromine hydrochloride
CAS:<p>Desformylflustrabromine hydrochloride (dFBr hydrochloride) is a selective agonist of nicotinic acetylcholine receptor (nAChR) in α4β2 neurons, with pEC50 of 6.</p>Fórmula:C17H12INO5Pureza:98.12%Forma y color:SolidPeso molecular:437.19Iperoxo
CAS:<p>Iperoxo (Iperoxo iodide) is an agonist of Muscarinic AChR and can be used to probe activation-related conformational transitions of muscarinic receptors.</p>Fórmula:C10H17IN2O2Pureza:99.81%Forma y color:SolidPeso molecular:324.16Ricasetron
CAS:<p>Ricasetron (Brl 46470) is a 5-HT3 receptor antagonist with pro-axonal lysing properties and is used in the study of anxiety disorders and anxiety disorders.</p>Fórmula:C19H27N3OPureza:99.52%Forma y color:SolidPeso molecular:313.44ALX-1393
CAS:<p>ALX-1393 is a selective GlyT2 inhibitor that effectively reduces neuronal action potential activity in a concentration-dependent manner and inhibits the</p>Fórmula:C23H22FNO4Pureza:99.83%Forma y color:SolidPeso molecular:395.42ABP688
CAS:<p>ABP688 is a non-competitive and selective mGluR5 antagonist(Ki = 1.7 nM). ABP688 can be used as a PET tracer for clinical imaging.</p>Fórmula:C15H16N2OPureza:98.63%Forma y color:SolidPeso molecular:240.3BPDBA
CAS:<p>BPDBA is an effective, selective, and non-competitive inhibitor of the betaine/GABA transporter (BGT-1), displaying inhibitory activity against human BGT-1 and</p>Fórmula:C19H20Cl2N2OPureza:99.37% - 99.95%Forma y color:SolidPeso molecular:363.28Alpidem
CAS:<p>Alpidem (Ananxyl), a non-sedative imidazopyridine anxiolytic, treats anxiety with high benzodiazepine receptor affinity.</p>Fórmula:C21H23Cl2N3OPureza:99.56% - 99.97%Forma y color:White To Off-White SolidPeso molecular:404.33Lesopitron
CAS:<p>Lesopitron: anxiolytic, 5-HT1A agonist, treats rodent anxiety, counters benzodiazepine withdrawal, low toxicity, no alcohol/barbiturate interaction.</p>Fórmula:C15H21ClN6Pureza:99.15% - 99.38%Forma y color:SolidPeso molecular:320.82Ezeprogind disulfate
CAS:<p>Ezeprogind disulfate: neurotrophic inducer targeting neurodegeneration causes like Abeta, tau; for neurological disorder research.</p>Fórmula:C25H48N6O8S2Pureza:99.72%Forma y color:SolidPeso molecular:624.81Selurampanel
CAS:<p>Selurampanel (BGG492), an oral AMPA antagonist for epilepsy, migraine, and tinnitus studies.</p>Fórmula:C16H19N5O4SPureza:99.60% - 99.78%Forma y color:SolidPeso molecular:377.42MK-3328
CAS:<p>MK-3328, a potential Alzheimer's drug, binds β-Amyloid with strong affinity (IC50:10.5 nM) and may serve as a PET ligand to gauge plaque load.</p>Fórmula:C14H9FN4OPureza:99.70% - >99.99%Forma y color:SolidPeso molecular:268.25BL-1020 Mesylate
CAS:<p>BL-1020 Mesylate (CYP-1020 Mesylate) is a GABA A receptor agonist and D2 antagonist used in studies of neurodegeneration.</p>Fórmula:C28H45ClN4O11S4Pureza:>99.99%Forma y color:SolidPeso molecular:777.39Felcisetrag
CAS:<p>Felcisetrag (TD-8954), an oral 5-HT4 agonist with GI prokinetic effects, has a high affinity (pKi 9.4) for h5-HT4(c) receptors.</p>Fórmula:C25H37N5O3Pureza:99.99%Forma y color:SolidPeso molecular:455.59Suriclone
CAS:<p>Suriclone (RP 31264), a cyclic pyrrolidone for anxiety, modulates GABA-A receptors without major sedation.</p>Fórmula:C20H20ClN5O3S2Pureza:99.21% - 99.73%Forma y color:SolidPeso molecular:477.99Agomelatine hydrochloride
CAS:<p>Agomelatine HCl is a MT1/MT2 receptor agonist (Ki: 0.1-0.27 nM) and a 5-HT2C antagonist (pKi: 6.2-6.4).</p>Fórmula:C15H18ClNO2Pureza:99.57%Forma y color:SolidPeso molecular:279.76W-9 hydrochloride
CAS:<p>W-9 hydrochloride is a calmodulin antagonist.</p>Fórmula:C16H22Cl2N2O2SPureza:98.9%Forma y color:SolidPeso molecular:377.33RWJ-51204
CAS:<p>RWJ-51204: potent adenosine A2A blocker, GABA(A) partial agonist (IC50: 0.2-2 nM), neuroprotective, may treat Parkinson's.</p>Fórmula:C21H19F2N3O3Pureza:99.57% - 99.95%Forma y color:SolidPeso molecular:399.39CGP 37849
CAS:<p>CGP 37849: oral NMDA antagonist (Ki=35 nM), anticonvulsant, with antidepressant/anxiolytic effects.</p>Fórmula:C6H12NO5PPureza:99.87%Forma y color:White SolidPeso molecular:209.14Buntanetap
CAS:<p>Buntanetap ((+)-Phenserine) is an inhibitor of TINAPs used in the study of neurological disorders, endocrine and metabolic disorders, and cardiovascular disease</p>Fórmula:C20H23N3O2Pureza:98.2%Forma y color:SolidPeso molecular:337.42Tedatioxetine
CAS:<p>Tedatioxetine (Lu AA24530) is a serotonin-norepinephrine-dopamine reuptake inhibitor (SNDRI) with antidepressant properties.</p>Fórmula:C18H21NSPureza:99.76% - >99.99%Forma y color:SolidPeso molecular:283.43Sarmazenil
CAS:<p>Sarmazenil (Ro 15-3505) is a partial inverse agonist at the benzodiazepine receptor and is used in the study of chronic hepatic encephalopathy.</p>Fórmula:C15H14ClN3O3Pureza:99.46%Forma y color:SolidPeso molecular:319.74Aplindore Fumarate
CAS:<p>Aplindore Fumarate (DAB-452), a selective dopamine D2/D3 partial agonist, is used in Parkinson's and schizophrenia research.</p>Fórmula:C22H22N2O7Pureza:>99.99%Forma y color:SolidPeso molecular:426.42JNJ-54175446
CAS:<p>JNJ-54175446 (JNJ-5446) is a P2X7 receptor antagonist that attenuates the release of IL-1β/IL-18 from microglia and is used in the study of depression.</p>Fórmula:C18H13ClF4N6OPureza:97.98% - 99.79%Forma y color:SolidPeso molecular:440.78DSP-0565
CAS:<p>DSP-0565 is a broad-spectrum anti-epileptic with a high safety margin and effectiveness in several convulsant models.</p>Fórmula:C14H12FNOPureza:99.51% - 99.56%Forma y color:SolidPeso molecular:229.25VU 0285683
CAS:<p>VU 0285683 is a specific negative allosteric modulator of mGluR5 with a high affinity for the MPEP binding site. VU 0285683 shows anxiolytic-like activity.</p>Fórmula:C14H7FN4OPureza:99.98%Forma y color:SolidPeso molecular:266.23LRRK2-IN-7
CAS:<p>LRRK2-IN-7: potent, selective CNS-active LRRK2 inhibitor, IC50 0.9 nM, >1000x selectivity vs kinases/channels/CYPs.</p>Fórmula:C24H26N6OPureza:99.26%Forma y color:SolidPeso molecular:414.5Adoprazine
CAS:<p>Adoprazine (SLV313) is a potential atypical antipsychotic bearing potent D2 receptor antagonist and 5-HT1A receptor agonist properties.</p>Fórmula:C24H24FN3O2Pureza:99.83%Forma y color:SolidPeso molecular:405.46Cyamemazine
CAS:<p>Cyamemazine is an antipsychotic compound with sedative and anxiolytic activity.Cyamemazine is a 5-HT3, 5-HT2A, and 5-HT2C receptor antagonist.</p>Fórmula:C19H21N3SPureza:97.01%Forma y color:SolidPeso molecular:323.46Lecozotan HCl
CAS:<p>Lecozotan HCl is a selective 5-HT antagonist boosting glutamate and acetylcholine release without causing 5-HT(1A) tolerance.</p>Fórmula:C28H30ClN5O3Pureza:99.04%Forma y color:SolidPeso molecular:520.02DMCM hydrochloride
CAS:<p>DMCM hydrochloride is a non-selective fully inverse agonist of benzodiazepine.</p>Fórmula:C17H19ClN2O4Pureza:99.56%Forma y color:SolidPeso molecular:350.8Tribendimidine
CAS:<p>Tribendimidine: broad-spectrum oral anthelmintic, nAChR agonist, effective against A. lumbricoides and N. americanus.</p>Fórmula:C28H32N6Pureza:≥98%Forma y color:SolidPeso molecular:452.59Eltenac
CAS:<p>Eltenac, a cyclooxygenase (COX) inhibitor, is used potentially for the treatment of pain.</p>Fórmula:C12H9Cl2NO2SPureza:98.53%Forma y color:SolidPeso molecular:302.18PHA 543613
CAS:<p>PHA 543613 is a specific agonist of α7 nAChR (Ki = 8.8 nM) and can be used in studies about the cognitive deficits of Alzheimer's disease and schizophrenia.</p>Fórmula:C15H17N3O2Pureza:99.43% - 99.96%Forma y color:SolidPeso molecular:271.31PAT-1251
CAS:<p>PAT-1251 is an inhibitor of LOXL2 with IC50s of 10, 0.12, and 0.16 μM for the mouse, rat, and dog and can be used in studies about fibrotic diseases.</p>Fórmula:C18H17F4N3O3Pureza:97.27% - 98.46%Forma y color:SolidPeso molecular:399.34GSK-1482160
CAS:<p>GSK-1482160 is a CNS-penetrant negative allosteric modulator of P2X7 receptor with oral activity.</p>Fórmula:C14H14ClF3N2O2Pureza:99.57%Forma y color:SolidPeso molecular:334.72NS-2710
CAS:<p>NS-2710, a GABA receptor agonist, is used potentially for the treatment of anxiety.</p>Fórmula:C22H20N4OPureza:99.7% - 99.82%Forma y color:SolidPeso molecular:356.42Anpirtoline hydrochloride
CAS:<p>Anpirtoline hydrochloride (D-16949 hydrochloride) is a 5-HT1B receptor agonist and 5-HT3 receptor antagonist used in the study of dyskinesia.</p>Fórmula:C10H14Cl2N2SPureza:>99.99% - >99.99%Forma y color:SolidPeso molecular:265.20Glutaminyl Cyclase Inhibitor 1
CAS:<p>Glutaminyl Cyclase Inhibitor 1 is a glutaminyl cyclase inhibitor (IC50: 0.5 μM) that can be used to study neurological disorders.</p>Fórmula:C21H24FN3O2Pureza:99.81%Forma y color:SolidPeso molecular:369.43ASM-024
CAS:<p>ASM-024, a synthetic piperazine, activates nicotinic and β2-adrenergic receptors for potential asthma and bronchitis treatment with anti-inflammatory effects.</p>Fórmula:C15H25N2Pureza:99.74%Forma y color:SolidPeso molecular:233.37Divaplon
CAS:<p>Divaplon is a GABA receptor agonist (IC50: 0.056 µM) that displays non-sedating anxiolytic behavioral characteristics in a rat model of anxiety.</p>Fórmula:C17H17N3O2Pureza:97.44% - 98.25%Forma y color:SolidPeso molecular:295.34NKY80
CAS:<p>NKY80 regulates the adenylyl cyclase catalytic activity in heart and lung tissues.</p>Fórmula:C12H11N3O2Pureza:99.88%Forma y color:SolidPeso molecular:229.23Mibampator
CAS:<p>Mibampator (LY451395) is an effective and selective AMPA receptor potentiator.</p>Fórmula:C21H30N2O4S2Pureza:99.34%Forma y color:SolidPeso molecular:438.6SB-215505
CAS:<p>SB215505: potent 5-HT2B/2C blocker, enhances rat wakefulness/motor activity. (pKi: 5-HT2B - 8.3, 5-HT2C - 7.66, 5-HT2A - 6.77).</p>Fórmula:C19H16ClN3OPureza:98.33%Forma y color:SolidPeso molecular:337.85HT6-ligand-1
CAS:<p>5HT6-ligand-1 is an orally active ligand of 5-HT6 receptor (Ki = 1.43 nM).</p>Fórmula:C20H22BrN3O2SPureza:99.24% - 99.93%Forma y color:SolidPeso molecular:448.38Rilapine
CAS:<p>Rilapine (Rilapinum) is an antipsychotic compound that shows high affinity for 5-HT6 receptors and can be used to study neurological disorders.</p>Fórmula:C22H20ClN3Pureza:97.76% - 99.20%Forma y color:SolidPeso molecular:361.87CBiPES hydrochloride
CAS:<p>CBiPES hydrochloride (CBiPES HCl) is an orthosteric modulator of the mGlu2 receptor and is used to study neurological disorders like epilepsy.</p>Fórmula:C21H20ClN3O2SPureza:99.66%Forma y color:SolidPeso molecular:413.92
