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Neurociencia

Neurociencia

Los inhibidores en neurociencia son compuestos diseñados para modular la actividad de proteínas, enzimas o receptores específicos dentro del sistema nervioso. Estos inhibidores son cruciales para estudiar los mecanismos moleculares subyacentes a la función neuronal, la transmisión sináptica y las enfermedades neurodegenerativas. Al dirigirse a los receptores de neurotransmisores, canales iónicos y vías de señalización, los inhibidores en neurociencia ayudan en la exploración de la función cerebral y en el desarrollo de estrategias terapéuticas para trastornos neurológicos como el Alzheimer, Parkinson y la epilepsia. En CymitQuimica, ofrecemos una amplia gama de inhibidores de neurociencia de alta calidad para apoyar su investigación en neurobiología, neurofarmacología y ciencias cognitivas.

Subcategorías de "Neurociencia"

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Se han encontrado 5514 productos de "Neurociencia"

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  • Flufiprole

    CAS:
    Flufiprole is used as a phenylpyrazole pesticide. It has enantioselective metabolism in human and rat liver microsomes.
    Fórmula:C16H10Cl2F6N4OS
    Forma y color:Solid
    Peso molecular:491.24

    Ref: TM-T25428

    25mg
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    50mg
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    100mg
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  • hAChE-IN-5


    hAChE-IN-5 (compound 49) is a dual inhibitor of human acetylcholinesterase (hAChE) and human butyrylcholinesterase (hBuChE), exhibiting inhibitory potency with
    Pureza:98%
    Forma y color:Odour Solid

    Ref: TM-T82243

    5mg
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    50mg
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  • 8-hydroxy Amoxapine

    CAS:

    8-hydroxy Amoxapine is a metabolite of the tetracyclic antidepressant amoxapine .1,2

    Fórmula:C17H16ClN3O2
    Forma y color:Solid
    Peso molecular:329.78

    Ref: TM-T37161

    1mg
    725,00€
  • 5-HT6R antagonist 1


    Compound 8 (5-HT6R antagonist 1), a 5-HT6R antagonist (K i : 5 nM), not only demonstrates inhibition of platelet aggregation and excellent metabolic stability
    Fórmula:C17H22F2N6O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:364.39

    Ref: TM-T79684

    5mg
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    50mg
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  • MmTx1 toxin


    Micrurotoxin 1 (MmTx1 toxin) acts as an allosteric modulator of GABA A receptors, enhancing the receptor's sensitivity to its agonist [1].
    Fórmula:C295H455N95O97S10
    Pureza:98%
    Forma y color:Solid
    Peso molecular:7205

    Ref: TM-T80489

    5mg
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    50mg
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  • CaMKIIα-PHOTAC


    CaMKIIα-PHOTAC is a photochemically targeted chimera (PHOTAC) that specifically targets Ca2+/calmodulin-dependent protein kinase II α (CaMKIIα).
    Fórmula:C54H58Cl2N10O11
    Pureza:98%
    Forma y color:Solid
    Peso molecular:1094

    Ref: TM-T79718

    5mg
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    50mg
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  • GAD65(247-266) epitope TFA


    GAD65(247-266) epitope TFA, a T cell epitope derived from islet antigens, exhibits competitive binding to the type I diabetes-associated molecule I-A g7, albeit
    Fórmula:C111H174F3N27O29S4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:2535.99

    Ref: TM-T80218

    5mg
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    50mg
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  • COX-1/2-IN-5


    COX-1/2-IN-5 (compound 2a) functions as a dual inhibitor of COX1/2, demonstrating inhibitory concentrations (IC50) of 2.650 μM and 0.958 μM, respectively, and

    Fórmula:C21H22N2O5S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:414.47

    Ref: TM-T79594

    5mg
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    50mg
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  • Calmodulin Kinase IINtide, Myristoylated


    Myristoylated Calmodulin Kinase IINtide (Myr-CaMKIINtide) serves as a selective and noncompetitive inhibitor of CaMKII [1].
    Fórmula:C156H275N47O43
    Pureza:98%
    Forma y color:Solid
    Peso molecular:3497.14

    Ref: TM-T80549

    5mg
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    50mg
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  • IHC3


    IHC3 is a competitive and reversible monoamine oxidase B (MAO-B) inhibitor with an IC50 of 1.672 μM, which targets Cys172 within the enzyme's active site.
    Fórmula:C17H12FN3O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:293.3

    Ref: TM-T78821

    5mg
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    50mg
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  • MAOA-IN-1


    MAOA-IN-1 (compound 15) is an orally-active inhibitor of monoamine oxidase A (MAOA) that exhibits cytotoxic effects on prostate cancer cells.
    Fórmula:C13H16Cl2N2O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:303.18

    Ref: TM-T78793

    5mg
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    50mg
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  • GABA receptor Antagonist 1


    GABA receptor Antagonist 1 (compound 7w) effectively inhibits the Px RDL1 GABAR at an IC50 of 7.08 nmol/L and demonstrates insecticidal efficacy against P.
    Pureza:98%
    Forma y color:Odour Solid

    Ref: TM-T82357

    5mg
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    50mg
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  • TC-2559 difumarate

    CAS:
    TC-2559 difumarate: Oral α4β2 nAChR partial agonist, CNS-selective, EC50 0.18 μM, prefers α4β2 over α2β4/α4β4/α3β4, antinociceptive.
    Fórmula:C20H26N2O9
    Forma y color:Solid
    Peso molecular:438.43

    Ref: TM-T40119

    10mg
    927,00€
    50mg
    3.705,00€
  • MAO-B-IN-3


    MAO-B-IN-3 is a reversible, selective inhibitor of monoamine oxidase B (MAO-B) with an IC50 of 96 nM and demonstrates affinity for the 5-HT6 receptor with a Ki
    Fórmula:C24H25N3O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:387.47

    Ref: TM-T78648

    5mg
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    50mg
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  • TIP 39, Tuberoinfundibular Neuropeptide

    CAS:
    TIP39 is a synthetic neuropeptide agonist for human and rat PTH2 receptors from the hypothalamus.
    Fórmula:C202H325N61O54S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:4504.2

    Ref: TM-TP1688

    100mg
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    500mg
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  • Calmodulin Binding Peptide 1

    CAS:
    Calmodulin Binding Peptide 1, a high-affinity MLCK-derived inhibitor, blocks IP3-induced Ca2+ release.
    Fórmula:C231H373N69O70S2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:5301.1

    Ref: TM-TP1710

    100mg
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    500mg
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  • MAO-B-IN-18


    MAO-B-IN-18 is a potent, selective inhibitor of MAO B, demonstrating IC50 values of 52 nM for hMAO B and 14 μM for hMAO A.
    Fórmula:C25H22N4O5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:458.47

    Ref: TM-T78690

    5mg
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    50mg
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  • 5-HT6 agonist 1


    Compound 19, a 5-HT6 agonist with an affinity (K i : 5 nM), exhibits antidepressant-like effects and enhances cognitive function while also inhibiting platelet
    Fórmula:C17H22Cl2N6S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:413.37

    Ref: TM-T79325

    5mg
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    50mg
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  • MRS7925


    MRS7925 (Compound 43) serves as a potent antagonist of the 5-HT2B receptor, with an inhibition constant (Ki) of 17 nM, and is utilized in the study of fibrosis
    Fórmula:C20H26IN5O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:511.36

    Ref: TM-T79326

    5mg
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    50mg
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  • Epiboxidine

    CAS:
    Epiboxidine: Potent, selective nAChR agonist; Ki 0.46/1.2 nM for rat/human α4β2; analogous to Epibatidine and ABT 418.
    Fórmula:C10H14N2O
    Forma y color:Solid
    Peso molecular:178.23

    Ref: TM-T74130

    5mg
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    50mg
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