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Neurociencia

Neurociencia

Los inhibidores en neurociencia son compuestos diseñados para modular la actividad de proteínas, enzimas o receptores específicos dentro del sistema nervioso. Estos inhibidores son cruciales para estudiar los mecanismos moleculares subyacentes a la función neuronal, la transmisión sináptica y las enfermedades neurodegenerativas. Al dirigirse a los receptores de neurotransmisores, canales iónicos y vías de señalización, los inhibidores en neurociencia ayudan en la exploración de la función cerebral y en el desarrollo de estrategias terapéuticas para trastornos neurológicos como el Alzheimer, Parkinson y la epilepsia. En CymitQuimica, ofrecemos una amplia gama de inhibidores de neurociencia de alta calidad para apoyar su investigación en neurobiología, neurofarmacología y ciencias cognitivas.

Subcategorías de "Neurociencia"

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Se han encontrado 5557 productos de "Neurociencia"

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  • SCH-23390 hydrochloride

    CAS:
    SCH-23390 hydrochloride (R-(+)-SCH23390 hydrochloride) is an effective dopamine receptor antagonist, and for the D1(Ki=0.2 nM) and D5(Ki=0.3 nM).
    Fórmula:C17H19Cl2NO
    Pureza:98% - 99.83%
    Forma y color:Solid
    Peso molecular:324.24
  • Syk Inhibitor II dihydrochloride

    CAS:
    Syk inhibitor II selectively blocks Syk (IC50 = 41 nM), impacting platelet function and inflammation, with lower potency against other kinases.
    Fórmula:C14H17Cl2F3N6O
    Pureza:98.53%
    Forma y color:Solid
    Peso molecular:413.22
  • F-15599

    CAS:
    <p>F-15599 is a highly selective G-protein biased 5-HT1A receptor agonist(Ki : 3.4 nM).</p>
    Fórmula:C19H21ClF2N4O
    Pureza:98.72%
    Forma y color:Solid
    Peso molecular:394.85
  • γ-Acetylenic GABA

    CAS:
    <p>γ-Acetylenic GABA (4-Aminohex-5-ynoic acid) is a potent, irreversible inhibitor of GABA-transaminase.</p>
    Fórmula:C6H9NO2
    Forma y color:Solid
    Peso molecular:127.143
  • Piperidolate hydrochloride

    CAS:
    Piperidolate hydrochloride, an antimuscarinic, reduces acetylcholine-induced intestinal spasms in rats and dogs.
    Fórmula:C21H26ClNO2
    Pureza:99.5%
    Forma y color:Solid
    Peso molecular:359.89
  • PF-06447475

    CAS:
    PF-06447475 is a highly effective, specific, brain penetrant LRRK2 inhibitor with IC0 of 3/11 nM for wild type LRRK2 and G2019S LRRK2 respectively.
    Fórmula:C17H15N5O
    Pureza:98.61% - 99.62%
    Forma y color:Solid
    Peso molecular:305.33
  • GNE-9605

    CAS:
    <p>GNE-9605 is a highly effective, specifical, and brain-penetrant LRRK2 inhibitor (IC50: 19 nM).</p>
    Fórmula:C17H20ClF4N7O
    Pureza:98.55% - 98.75%
    Forma y color:Solid
    Peso molecular:449.83
  • Sertindole

    CAS:
    <p>Sertindole, atypical antipsychotic, targets D2, 5-HT1D, 5-HT2A, 5-HT2C receptors (Kds: 2.7, 20, 0.14, 6 nM).</p>
    Fórmula:C24H26ClFN4O
    Pureza:99.87% - 99.92%
    Forma y color:Off-White To Pale Yellow Solid
    Peso molecular:440.94
  • SQ22536

    CAS:
    SQ22536, a tetrahydrofuryl adenosine analogue, inhibits adenylate cyclase in catfish and rat hepatocytes non-competitively.
    Fórmula:C9H11N5O
    Pureza:99.18%
    Forma y color:Off-White Solid
    Peso molecular:205.22
  • Ralmitaront

    CAS:
    <p>Ralmitaront (RO6889450) is a potent, orally active partial agonist of the trace amine-associated receptor 1 (TAAR1).</p>
    Fórmula:C17H22N4O2
    Pureza:99.71% - 99.79%
    Forma y color:Solid
    Peso molecular:314.38
  • BRL-15572 dihydrochloride

    CAS:
    BRL-15572 dihydrochloride: 5-HT1D antagonist, pKi 7.9, also binds 5-HT1A/2B, 60x selective over 5-HT1B.
    Fórmula:C25H27ClN2O·2HCl
    Pureza:99.74%
    Forma y color:Solid
    Peso molecular:479.87
  • Ziprasidone mesylate

    CAS:
    Ziprasidone mesylate (CP-88059), an oral 5-HT & dopamine blocker, binds D2, 5-HT2A, 5-HT1A with Ki values: 4.8, 0.42, 3.4 nM.
    Fórmula:C22H25ClN4O4S2
    Forma y color:Solid
    Peso molecular:509.04
  • (RS)-3-Hydroxyphenylglycine

    CAS:
    (RS)-3-Hydroxyphenylglycine is a PI-linked metabotropic glutamate receptors agonist.
    Fórmula:C8H9NO3
    Pureza:99.29%
    Forma y color:Solid
    Peso molecular:167.16
  • SSR504734

    CAS:
    SSR504734 is a novel potent glycine transporter 1 (GlyT1) inhibitor.
    Fórmula:C20H20ClF3N2O
    Forma y color:Solid
    Peso molecular:396.83
  • 6-fluoro-DL-Tryptophan

    CAS:
    6-fluoro-DL-Tryptophan is an inhibitor of serotonin (5-HT) synthesis.
    Fórmula:C11H11FN2O2
    Pureza:99.25%
    Forma y color:Off-White Powder
    Peso molecular:222.22
  • β-Amyloid 15-21 acetate


    β-Amyloid 15-21 acetate (Beta-Amyloid (15-21) acetate) is a fragment of Amyloid-β peptide, maybe used in the research of neurological disease.
    Fórmula:C45H69N9O11
    Pureza:99.62%
    Forma y color:Solid
    Peso molecular:912.1
  • LY2119620

    CAS:
    LY2119620 is a specific, and allosteric agonist of human M2 and M4 muscarinic acetylcholine receptors.
    Fórmula:C19H24ClN5O3S
    Pureza:99.7%
    Forma y color:Solid
    Peso molecular:437.94
  • Pimavanserin tartrate

    CAS:
    Pimavanserin tartrate is a potent 5-HT 2A receptor inverse agonist used to treat Parkinson's disease-related psychosis.Cost-effective and quality-assured.
    Fórmula:C50H68F2N6O4·C4H6O6
    Pureza:99.24% - 99.98%
    Forma y color:Solid
    Peso molecular:1005.2
  • (S)-3-Hydroxyphenylglycine

    CAS:
    (S)-3-Hydroxyphenylglycine is an agonist of group I metabotropic glutamate receptors (mGluRs).
    Fórmula:C8H9NO3
    Pureza:99.65%
    Forma y color:Solid
    Peso molecular:167.16
  • RS-127445

    CAS:
    <p>RS-127445 (MT500) is a selective 5-HT2B receptor antagonist with pKi of 9.5 and pIC50 of 10.4, exhibits &gt;1000-fold selectivity against other 5-HT receptors.</p>
    Fórmula:C17H16FN3
    Pureza:99.32%
    Forma y color:Solid
    Peso molecular:281.33