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Neurociencia

Neurociencia

Los inhibidores en neurociencia son compuestos diseñados para modular la actividad de proteínas, enzimas o receptores específicos dentro del sistema nervioso. Estos inhibidores son cruciales para estudiar los mecanismos moleculares subyacentes a la función neuronal, la transmisión sináptica y las enfermedades neurodegenerativas. Al dirigirse a los receptores de neurotransmisores, canales iónicos y vías de señalización, los inhibidores en neurociencia ayudan en la exploración de la función cerebral y en el desarrollo de estrategias terapéuticas para trastornos neurológicos como el Alzheimer, Parkinson y la epilepsia. En CymitQuimica, ofrecemos una amplia gama de inhibidores de neurociencia de alta calidad para apoyar su investigación en neurobiología, neurofarmacología y ciencias cognitivas.

Subcategorías de "Neurociencia"

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Se han encontrado 5532 productos de "Neurociencia"

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  • Cyclopiazonic acid

    CAS:
    <p>Cyclopiazonic acid (CPA) is a neurotoxic secondary metabolite (SM) made by A.</p>
    Fórmula:C20H20N2O3
    Pureza:99.27% - 99.80%
    Forma y color:Solid
    Peso molecular:336.38
  • Escitalopram Oxalate

    CAS:
    <p>Escitalopram Oxalate ((S)-(+)Citalopram oxalate) is a selective serotonin (5-HT) reuptake inhibitor (SSRI) with Ki of 0.89 nM.</p>
    Fórmula:C22H23FN2O5
    Pureza:97.39% - 99.73%
    Forma y color:White Solid
    Peso molecular:414.43
  • A-867744

    CAS:
    <p>A-867744 is an effective and selective type II positive allosteric modulator of the α7 nAChR (EC50: 1.0 μM).</p>
    Fórmula:C20H19ClN2O3S
    Pureza:95.66%
    Forma y color:Solid
    Peso molecular:402.89
  • Piboserod hydrochloride

    CAS:
    Piboserod HCl is a selective antagonist of 5-HT4 and muscarinic receptor.
    Fórmula:C22H32ClN3O2
    Forma y color:Solid
    Peso molecular:405.96
  • TAT-GluA2 3Y acetate(1404188-93-7 free base)


    TAT-GluA2 3Y acetate is an inhibitor of AMPA receptor endocytosis.Systemic administration of Tat-GluA2(3Y) during the induction phase of d-amphetamine blocked
    Fórmula:C115H185N43O29
    Pureza:99.43%
    Forma y color:Solid
    Peso molecular:2634.02
  • Revefenacin

    CAS:
    Revefenacin (TD-4208) is a mAChR antagonist has a high affinity on M3 receptor( Ki : 0.18 nM),and potentially useful for the treatment of respiratory disease.
    Fórmula:C35H43N5O4
    Pureza:98.12%
    Forma y color:Solid
    Peso molecular:597.75
  • SKF89976A hydrochloride

    CAS:
    <p>SKF89976A hydrochloride (d,l-SKF89976A hydrochloride) is a selective inhibitor GABA transporter such as GAT-1 (IC50s = 0.28 μM), GAT-2 (IC50s = 137.34 μM) and</p>
    Fórmula:C22H26ClNO2
    Pureza:98.02%
    Forma y color:Solid
    Peso molecular:371.9
  • CRANAD 2

    CAS:
    <p>CRANAD-2, a near-infrared probe, detects amyloid-beta in vivo, increasing fluorescence 70x and shifting blue 90 nm upon binding.</p>
    Fórmula:C23H25BF2N2O2
    Pureza:99.44%
    Forma y color:Dark Blue To Black Powder
    Peso molecular:410.27
  • PNU-282987 S enantiomer free base

    CAS:
    PNU-282987 S enantiomer free base is an agonist of α7 nicotinic acetylcholine receptor (α7 nAChR).
    Fórmula:C14H17ClN2O
    Pureza:99.74%
    Forma y color:Solid
    Peso molecular:264.75
  • GALANTHAMINONE

    CAS:
    <p>Galanthaminone ((-)-Narwedine) is a cholinesterase (AChE) inhibitor, used for the treatment of mild to moderate Alzheimer's disease and other memory impairments</p>
    Fórmula:C17H19NO3
    Pureza:99.93%
    Forma y color:White To Off-White Chemical
    Peso molecular:285.34
  • Rivanicline hemioxalate


    <p>Rivanicline hemioxalate is a selective α4β2 nicotinic receptor agonist (K i =26 nM), over 1,000x preference to α7 (K i =3.6 μM), with limited side effects.</p>
    Fórmula:C12H16N2O4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:207.23
  • Lu AF21934

    CAS:
    <p>Lu AF21934 is a brain-penetrant and selective mGlu4 receptor positive allosteric modulator (IC50: 500 nM, human).</p>
    Fórmula:C14H16Cl2N2O2
    Pureza:99.79%
    Forma y color:Solid
    Peso molecular:315.2
  • Autocamtide 2 TFA(129198-88-5 free base)


    <p>Autocamtide 2 TFA, selective CaMKII peptide substrate, used in its activity assay.</p>
    Fórmula:C67H119F3N22O22
    Pureza:98%
    Forma y color:Solid
    Peso molecular:1641.79
  • Prucalopride Succinate

    CAS:
    Prucalopride Succinate is a 5-HT4 receptor agonist with Ki 2.5 nM (5-HT4a) and 8 nM (5-HT4b).
    Fórmula:C18H26ClN3O3·C4H6O4
    Pureza:99.24%
    Forma y color:Solid
    Peso molecular:485.96
  • Naratriptan

    CAS:
    <p>Naratriptan is a selective agonist of 5-HT1 receptor and is is used for the treatment of migraine headaches.</p>
    Fórmula:C17H25N3O2S
    Pureza:99.08%
    Forma y color:Solid
    Peso molecular:335.47
  • SB-200646

    CAS:
    SB-200646 is a selective and potent antagonist of 5-HT2B/5-HT2C receptor
    Fórmula:C15H14N4O
    Pureza:99.61%
    Forma y color:Solid
    Peso molecular:266.3
  • Amitriptyline

    CAS:
    <p>Amitriptyline: a tricyclic antidepressant used for depression and neuropathic pain.</p>
    Fórmula:C20H23N
    Pureza:98.24% - 99.64%
    Forma y color:Crystals Solid
    Peso molecular:277.4
  • pyridostigmine

    CAS:
    <p>Pyridostigmine(Regonol) is an acetylcholinesterase inhibitor that can treat myasthenia gravis by increasing acetylcholine at the postsynaptic motor endplate.</p>
    Fórmula:C9H13N2O2
    Pureza:98.10%
    Forma y color:Solid
    Peso molecular:181.21
  • GW791343 dihydrochloride

    CAS:
    <p>GW791343 dihydrochloride (GW791343 (HCl)) is a P2X7 allosteric modulator.</p>
    Fórmula:C20H26Cl2F2N4O
    Pureza:>99.99%
    Forma y color:Solid
    Peso molecular:447.35
  • VU0364770

    CAS:
    VU0364770 (VU 0364770)(EC50=1.1 μM), a positive allosteric modulator(PAM) of mGlu4, shows insignificant activity at 68 other receptors, including other mGlu
    Fórmula:C12H9ClN2O
    Pureza:99.65% - >99.99%
    Forma y color:Solid
    Peso molecular:232.67