Proteasas / Proteasoma
Los inhibidores de proteasas y proteasomas son compuestos que bloquean la actividad de las proteasas y del proteasoma, que están involucrados en la degradación y renovación de proteínas. Estos inhibidores son vitales para estudiar la regulación de la homeostasis proteica, el control del ciclo celular y la apoptosis. Los inhibidores de proteasas y proteasomas también se utilizan en el tratamiento de enfermedades como el cáncer, donde la degradación anormal de proteínas desempeña un papel en la progresión de la enfermedad. Al inhibir las proteasas o el proteasoma, estos compuestos pueden inducir la muerte celular en células cancerosas y son herramientas esenciales tanto en la investigación básica como en el desarrollo terapéutico. En CymitQuimica, ofrecemos una amplia gama de inhibidores de proteasas y proteasomas de alta calidad para apoyar su investigación en bioquímica, biología celular y desarrollo de fármacos.
Subcategorías de "Proteasas / Proteasoma"
- Acetil-CoA Carboxilasa(34 productos)
- Cisteína proteasa(96 productos)
- DPP-4(20 productos)
- Glutaminasa(40 productos)
- Proteasa del VIH(449 productos)
- PAI-1(25 productos)
- Inhibidores de la proteasa(50 productos)
- Receptor activado por proteasa(53 productos)
- Proteasoma(94 productos)
- Serina proteasa(50 productos)
- p97(14 productos)
Mostrar 3 subcategorías más
Se han encontrado 1044 productos de "Proteasas / Proteasoma"
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Carbobenzoxyproline
CAS:<p>Carbobenzoxyproline (Carbobenzoxy-S-proline) is a prolidase inhibitor.</p>Fórmula:C13H15NO4Pureza:99.79%Forma y color:White To Light Yellow Crystal PowderPeso molecular:249.26PF-00835231
CAS:<p>PF-00835231 is a CoV-2 cysteine 3C-like protease (3CLpro) inhibitor, with IC50s of 0.27 nM and 4 nM for SARS CoV-2 and SARS CoV-1 3CLpro, respectively.PF-</p>Fórmula:C24H32N4O6Pureza:97.83%Forma y color:SolidPeso molecular:472.53CH 5450
CAS:<p>CH 5450 (Z-Ile-Glu-Pro-Phe-Ome) (Z-Ile-Glu-Pro-Phe-Ome) is a short peptide inhibitor of chymase in the human heart</p>Fórmula:C34H44N4O9Pureza:95.93%Forma y color:SolidPeso molecular:652.73Rusalatide acetate (497221-38-2 free base)
CAS:<p>Rusalatide acetate (TP508 amide acetate), a regenerated peptide, alleviates radiation-induced gastrointestinal injury by activating stem cells.</p>Fórmula:C99H151N29O37SPureza:>99.99%Forma y color:SolidPeso molecular:2371.5Hepln-13
CAS:<p>Hepln-13 is a hepsin inhibitor that acts by hindering prostate cancer bone metastasis.</p>Fórmula:C17H13BrN2Pureza:97.67%Forma y color:SolidPeso molecular:325.2(Arg)9 TFA (143413-47-2 free base)
CAS:<p>(Arg)9 TFA (Peptide R9 TFA) is a cell-penetrating peptide. (Arg)9 TFA exhibits neuroprotective activity with an IC50 of 0.78 μM in the glutamic acid model.</p>Fórmula:C56H111F3N36O12Pureza:>99.99%Forma y color:SolidPeso molecular:1537.714-Isopropylcatechol
CAS:<p>4-Isopropylcatechol is a potent depigmenting agent and is of use in the topical therapy of selected patients with hypermelanosis.</p>Fórmula:C9H12O2Pureza:97.93%Forma y color:SolidPeso molecular:152.19Azvudine
CAS:<p>Azvudine (FNC) is a powerful NRTI effective against HIV, HBV, HCV, and resistant strains.</p>Fórmula:C9H11FN6O4Pureza:99.76% - >99.99%Forma y color:SolidPeso molecular:286.22Z-YVAD-FMK
CAS:<p>AA-Z-YVAD-FMK is a Irreversible caspase-1 inhibitor,with anti-inflammatory and anti-tumor activities.</p>Fórmula:C31H39FN4O9Pureza:98.00%Forma y color:SolidPeso molecular:630.66Enfuvirtide acetate
CAS:<p>Enfuvirtide acetate salt is a linear synthetic peptide made of 36 amino acids. It has an acetylated N-terminus and a carboxamide C-terminus.</p>Fórmula:C206H305N51O66Pureza:99.34%Forma y color:SolidPeso molecular:4552Diprotin A
CAS:<p>Diprotin A (Ile-Pro-Ile) (Ile-Pro-Ile) is a dipeptidyl peptidase IV (DPP-IV) inhibitor.</p>Fórmula:C17H31N3O4Pureza:99.29%Forma y color:White PowderPeso molecular:341.45GI254023X
CAS:<p>GI254023X is a MMP9 and ADAM10 inhibitor with IC50 values of 2.5 and 5.3 nM.Cost-effective and quality-assured.</p>Fórmula:C21H33N3O4Pureza:98.21% - 98.56%Forma y color:SolidPeso molecular:391.5Paritaprevir free base
CAS:<p>Paritaprevir (ABT-450) is an oral HCV NS3/NS4A protease inhibitor with potential against genotype 1, disrupting viral replication.</p>Fórmula:C40H43N7O7SPureza:95% - 99.26%Forma y color:SolidPeso molecular:765.89Bictegravir
CAS:<p>Bictegravir (GS-9883) is a potent inhibitor of HIV-1 integrase (IC50: 7.5 nM).</p>Fórmula:C21H18F3N3O5Pureza:97.6% - 99.51%Forma y color:SolidPeso molecular:449.38ABT530
CAS:<p>ABT530 (Pibrentasvir) is an HCV NS5A inhibitor with EC50s ranging from 1.4-5.0 pM against HCV replicons containing NS5A from genotypes 1-6.</p>Fórmula:C57H65F5N10O8Pureza:99.15% - 99.93%Forma y color:SolidPeso molecular:1113.18TMC647055 Choline Hydroxide Salt
<p>TMC647055 is a potent HCV NS5B inhibitor with low toxicity and good pharmacokinetics, under clinical evaluation.</p>Fórmula:C37H53N5O8SPureza:99.44%Forma y color:SolidPeso molecular:727.91Brensocatib
CAS:<p>Brensocatib (AZD7986) is a Dipeptidyl peptidase 1 (DPP1) inhibitor (pIC50s: 6.85, 7.7, 7.6, 7.8, and 7.8 in human, rat, mouse, rabbit, and dog, respectively).</p>Fórmula:C23H24N4O4Pureza:97.55%Forma y color:SolidPeso molecular:420.46Apelin-17 (human, bovine) acetate
<p>Apelin-17 (human, bovine) acetate is an endogenous apelin receptor agonist. Potently inhibits forskolin-stimulated cAMP accumulation (pIC50 = 9.94).</p>Fórmula:C98H160N34O22SPureza:99.36%Forma y color:SolidPeso molecular:2198.63Rilpivirine
CAS:<p>Rilpivirine (R278474) is a diarylpyrimidine derivative and reverse transcriptase inhibitor with antiviral activity against HIV-1 that is used in the treatment</p>Fórmula:C22H18N6Pureza:97.22% - 98.83%Forma y color:SolidPeso molecular:366.42CASP3 Activator 1541
CAS:<p>CASP3 Activator 1541 is an activator of the proenzyme forms of caspase-3, and induces cell death.</p>Fórmula:C24H17N3O4Pureza:98.84%Forma y color:SolidPeso molecular:411.41EIDD-1931
CAS:<p>EIDD-1931 (Beta-d-N4-hydroxycytidine) is a ribonucleoside analog with antiviral activity. It inhibits replication of SARS-CoV, MERS-CoV, and SARS-CoV-2.</p>Fórmula:C9H13N3O6Pureza:99.14% - 99.73%Forma y color:SolidPeso molecular:259.22GSK-690693
CAS:<p>GSK-690693 is a pan-Akt inhibitor targeting Akt1/2/3 with IC50 of 2 nM/13 nM/9 nM, also sensitive to the AGC kinase family: PKA, PrkX and PKC isozymes. Phase 1.</p>Fórmula:C21H27N7O3Pureza:98.07% - 99.77%Forma y color:SolidPeso molecular:425.483-O-Ethyl-L-ascorbic acid
CAS:3-O-Ethyl-L-ascorbic acid is a cosmetic tyrosinase inhibitor with whitening ability and is a stabilized vitamin C derivative.Fórmula:C8H12O6Pureza:97.35% - 99.99%Forma y color:White To Very Pale Yellow Crystalline Powder Solid PowderPeso molecular:204.18PSI-6130
CAS:<p>PSI-6130 (R 1656) is a potent and selective HCV NS5B polymerase inhibitor. PSI-6130 inhibits HCV replication with a mean IC50 of 0.6 μM.</p>Fórmula:C10H14FN3O4Pureza:98.63% - 99.79%Forma y color:SolidPeso molecular:259.23Asunaprevir
CAS:<p>Asunaprevir (BMS-650032) is an effective hepatitis C virus (HCV) NS3 protease inhibitor.</p>Fórmula:C35H46ClN5O9SPureza:99.34% - 99.8%Forma y color:SolidPeso molecular:748.29PTACH
CAS:<p>PTACH (Cpd 51) (NCH-51) is a SAHA-based inhibitor of human HDAC. It can potently inhibit the growth of various human Y cells (EC50: 1 to 10 μM).</p>Fórmula:C20H26N2O2S2Pureza:87.44% - 99.74%Forma y color:SolidPeso molecular:390.56Daclatasvir
CAS:<p>Daclatasvir (EBP 883/BMS-790052) is a potent HCV NS5A inhibitor with EC50 9-50 pM across various genotypes. Phase 3.</p>Fórmula:C40H50N8O6Pureza:99.81%Forma y color:SolidPeso molecular:738.88CA-074 methyl ester
CAS:<p>CA-074 methyl ester (Cathepsin B Inhibitor IV) is a selective inhibitor of Cathepsin B (IC50=36.3 nM). neuroprotective effect. High-Quality, Low-Cost!</p>Fórmula:C19H31N3O6Pureza:97.26% - 99.58%Forma y color:SolidPeso molecular:397.47Peptide T acetate(106362-32-7 free base)
<p>Peptide T acetate is an octapeptide from the V2 region of HIV-1 gp120.</p>Fórmula:C37H59N9O18Pureza:99.47%Forma y color:SolidPeso molecular:917.91Letermovir
CAS:<p>Letermovir (AIC246) (AIC246) is a novel anti-CMV compound (EC50: about 5 nM in fibroblast cells). It targets the pUL56 subunit of the viral terminase complex.</p>Fórmula:C29H28F4N4O4Pureza:99.85% - 99.87%Forma y color:SolidPeso molecular:572.55Bemnifosbuvir
CAS:<p>Bemnifosbuvir (AT-511) is a novel phosphoramidate prodrug of 2'-fluoro-2'-C-methylguanosine-5'-monophosphate that has potent in vitro activity against HCV.</p>Fórmula:C24H33FN7O7PPureza:99.35% - 99.54%Forma y color:SolidPeso molecular:581.53LY 3000328
CAS:<p>LY 3000328 (Cathepsin S inhibitor) is a selective inhibitor of cathepsin S.Cost-effective and quality-assured.</p>Fórmula:C25H29FN4O5Pureza:97.83% - 99.54%Forma y color:SolidPeso molecular:484.524-Butylresorcinol
CAS:<p>4-Butylresorcinol (Butylresorcinol) is a potent inhibitor of tyrosinase(IC50 : 11.27 μM), and is used in cosmetics as a depigmenting agent.</p>Fórmula:C10H14O2Pureza:98.64% - ≥95%Forma y color:Light Beige Solid PowderPeso molecular:166.22Daclatasvir dihydrochloride
CAS:<p>Daclatasvir dihydrochloride is an oral antiviral that treats chronic hepatitis C by inhibiting HCV's NS5A; rare liver enzyme elevation, seldom causes jaundice.</p>Fórmula:C40H52Cl2N8O6Pureza:99.67%Forma y color:SolidPeso molecular:811.8Ixazomib citrate
CAS:<p>Ixazomib citrate (MLN9708), a prodrug of Ixazomib (MMLN-2238), is an oral 2nd-gen proteasome inhibitor with anti-cancer potential (IC50: 3.4 nM).</p>Fórmula:C20H23BCl2N2O9Pureza:98.37% - >99.99%Forma y color:SolidPeso molecular:517.12Paritaprevir
CAS:<p>Paritaprevir (ABT450) 是一种非结构蛋白 3/4A 蛋白酶抑制剂，对 HCV 1a 和 HCV 1b 的 EC50 值分别为 1 和 0.21 nM。它也是SARS-CoV 3CLpro 的抑制剂，IC50为 1.31 μM。</p>Fórmula:C40H43N7O7SPureza:99.72%Forma y color:SolidPeso molecular:765.88Avatrombopag
CAS:<p>Avatrombopag (YM477) is a new oral thrombopoietin (TPO) receptor agonist, activating TPO receptor and increasing megakaryocytic proliferation/differentiation</p>Fórmula:C29H34Cl2N6O3S2Pureza:99.01% - 99.63%Forma y color:SolidPeso molecular:649.65S 3304
CAS:<p>S 3304 is a novel matrix metalloproteinases inhibitor which is specific for MMP-2 and MMP-9.</p>Fórmula:C24H20N2O4S2Pureza:98.09%Forma y color:SolidPeso molecular:464.56Velpatasvir
CAS:<p>Velpatasvir (GS-5816), also known as GS-5816, is a potent and selective Hepatitis C virus NS5A inhibitor.</p>Fórmula:C49H54N8O8Pureza:99.17% - 99.83%Forma y color:SolidPeso molecular:883Boc-Asp(OMe)-fluoromethyl ketone
CAS:<p>Boc-Asp(OMe)-FMK is a broad-spectrum caspase inhibitor that blocks Fas-mediated processes without affecting IL-8 chemotaxis.</p>Fórmula:C11H18FNO5Pureza:≥98%Forma y color:SolidPeso molecular:263.26Obefazimod
CAS:<p>Obefazimod (ABX-464) is a potent anti-HIV agent. ABX464 inhibits HIV-1 replication in stimulated peripheral blood mononuclear cells (PBMCs).</p>Fórmula:C16H10ClF3N2OPureza:99.86%Forma y color:SolidPeso molecular:338.71KKI-5 acetate(97145-43-2 free base)
<p>KKI-5 acetate: Serine protease inhibitor, targets kallikrein/plasmin, potential anticancer and angioedema therapy.</p>Fórmula:C37H59N11O11Pureza:99.44%Forma y color:SolidPeso molecular:833.95Tris(4-aminophenyl)methane
CAS:<p>Tris(4-aminophenyl)methane (Leucopararosaniline), a triphenylmethane dye, is a weak HCV helicase inhibitor.</p>Fórmula:C19H19N3Pureza:95.73%Forma y color:Beige Solid CrystallinePeso molecular:289.37JNJ0966
CAS:<p>JNJ0966 is a highly selective MMP-9 zymogen inhibitor (IC50: 440 nM).</p>Fórmula:C16H16N4O2S2Pureza:99.46% - 99.62%Forma y color:SolidPeso molecular:360.45Omarigliptin
CAS:<p>Omarigliptin is a potent and selective oral dipeptidyl peptidase 4 (DPP4) inhibitor with IC50 value of 1.6 nM. Cost-effective and quality-assured.</p>Fórmula:C17H20F2N4O3SPureza:99.68% - 99.77%Forma y color:SolidPeso molecular:398.43Thiamine disulfide
CAS:<p>Thiamine disulfide (Algoneurina) , also known as thiamin or vitamin B1, is a vitamin found in food and manufactured as a dietary supplement and medication.</p>Fórmula:C24H34N8O4S2Pureza:99.81%Forma y color:CoaPeso molecular:562.71Y-29794 Tosylate
CAS:<p>Y-29794 Tosylate (Y-29794) is an orally active, effective, and specific non-peptide-prolyl endopeptidase (PPCE) inhibitor.</p>Fórmula:C30H42N2O4S3Pureza:99.86%Forma y color:SolidPeso molecular:590.86GK921
CAS:<p>GK921 is a transglutaminase 2 (TGase) inhibitor.</p>Fórmula:C21H20N4OPureza:97.44% - 99.49%Forma y color:SolidPeso molecular:344.41HIV-1 Inhibitor 18A
CAS:<p>HIV-1 Inhibitor 18A (HIV-1 Inhibitor-18A) specifically inhibits the entry of multiple HIV-1 isolates.</p>Fórmula:C14H11N5O2SPureza:99.79%Forma y color:SolidPeso molecular:313.33CTTHWGFTLC, CYCLIC acetate(244082-19-7 free base)
<p>CTTHWGFTLC, CYCLIC acetate is an inhibitor for matrix metalloproteinases (MMP)-2 and MMP-9.</p>Fórmula:C54H75N13O16S2Pureza:99.71%Forma y color:SolidPeso molecular:1226.39Dabigatran
CAS:<p>Dabigatran (BIBR 953ZW), a thrombin inhibitor, prevents thrombus formation, reducing stroke and embolism risk in nonvalvular atrial fibrillation patients.</p>Fórmula:C25H25N7O3Pureza:97.44% - 98.7%Forma y color:Tan SolidPeso molecular:471.51CeMMEC13
CAS:<p>CeMMEC13 is an isoquinolinone that selectively inhibits the second bromodomain of TAF1 (IC50 = 2.1 μM).</p>Fórmula:C19H16N2O4Pureza:98.52%Forma y color:SolidPeso molecular:336.34Doravirine
CAS:<p>Doravirine (MK-1439) is a non-nucleoside reverse transcriptase inhibitor, used in the treatment of HIV/AIDS.</p>Fórmula:C17H11ClF3N5O3Pureza:99.65% - 99.79%Forma y color:SolidPeso molecular:425.75L-Albizziin
CAS:<p>L-Albizziin (L-beta-Ureidoalanine) is a glutamase inhibitor and is a glutaminyl-tRNA synthetase inhibitor.</p>Fórmula:C4H9N3O3Pureza:99.98%Forma y color:White PowderPeso molecular:147.13Anagliptin
CAS:<p>Anagliptin (SK-0403) is a potent Inhibitor of DPP-4(IC50 of 3.8 nM), for the treatment of type 2 diabetes mellitus.</p>Fórmula:C19H25N7O2Pureza:97.59% - 99.98%Forma y color:SolidPeso molecular:383.45P-113 acetate
<p>P-113 acetate: AMP from histatin 5, treats gingivitis and HIV-related oral candidiasis safely and effectively.</p>Fórmula:C73H114N28O15Pureza:97.4%Forma y color:SolidPeso molecular:1623.86Samatasvir
CAS:<p>Samatasvir (ATOLIHZIXHZSBA-BTSKBWHGSA-N) is a pan-genotypic inhibitor of the HCV non-structural protein 5A.</p>Fórmula:C47H48N8O6S2Pureza:98.03%Forma y color:SolidPeso molecular:885.06Glutaminase C-IN-1
CAS:<p>Glutaminase C-IN-1 (Compound 968) is a Glutaminase C allosteric inhibitor.</p>Fórmula:C27H27BrN2OPureza:99.68% - >99.99%Forma y color:SolidPeso molecular:475.422,4-Dioxaspiro(5.5)undec-8-ene, 3-(2-furanyl)-
CAS:<p>2,4-Dioxaspiro(5.5)undec-8-ene, 3-(2-furanyl)- (Ulinastatin) ,as an urinary trypsin inhibitor (UTI), is a glycoprotein that is isolated from healthy human urine</p>Fórmula:C13H16O3Pureza:99.53% - 99.81%Forma y color:SolidPeso molecular:220.26Ixazomib
CAS:<p>Ixazomib (MLN2238) is a boron-based peptide proteasome inhibitor targeting β5 site (IC50: 3.4 nM), also affecting β1 and β2 sites.</p>Fórmula:C14H19BCl2N2O4Pureza:98% - 98.92%Forma y color:SolidPeso molecular:361.03Batimastat
CAS:<p>Batimastat (BB94) (BB-94) is an effective, broad-spectrum matrix metalloprotease (MMP) inhibitor.</p>Fórmula:C23H31N3O4S2Pureza:98.15% - 99.5%Forma y color:SolidPeso molecular:477.64Elvitegravir
CAS:<p>Elvitegravir (JTK-303) is an HIV integrase inhibitor and CYP2C9 inducer.</p>Fórmula:C23H23ClFNO5Pureza:98.43% - 99.57%Forma y color:SolidPeso molecular:447.88Telaprevir
CAS:<p>Telaprevir (Incivek) (VX-950) is an effective inhibitor of HCV NS3-4A serine protease (IC50: 0.35 μM).</p>Fórmula:C36H53N7O6Pureza:96.9% - 98.89%Forma y color:SolidPeso molecular:679.854-Chloro-2-(trifluoroacetyl)aniline hydrochloride
CAS:<p>4-Chloro-2-(trifluoroacetyl)aniline hydrochloride is an inhibitor of HIV-1 RT (HIV reverse transcriptase) .</p>Fórmula:C8H6Cl2F3NOPureza:97.15%Forma y color:SolidPeso molecular:260.04Ceritinib
CAS:<p>Ceritinib (LDK378) is an ALK inhibitor with selective, ATP-competitive, and oral activity. Ceritinib has antitumor activity. Cost-effective and quality-assured.</p>Fórmula:C28H36ClN5O3SPureza:98.52% - 99.77%Forma y color:SolidPeso molecular:558.14CGS 27023A
CAS:<p>CGS 27023A is a non-peptidic, potent, and orally active stromelysin inhibitor.</p>Fórmula:C18H24ClN3O5SPureza:99.08%Forma y color:SolidPeso molecular:429.92Picolamine
CAS:<p>Picolamine acts as a potential inhibitor of DPP-4.</p>Fórmula:C6H8N2Pureza:98.3%Forma y color:Light Yellow LiquidPeso molecular:108.14SB-3CT
CAS:<p>SB-3CT is a potent and specific gelatinase inhibitor for MMP-2(Ki=13.9 nM) and MMP-9(Ki=600 nM).</p>Fórmula:C15H14O3S2Pureza:98% - 99.38%Forma y color:SolidPeso molecular:306.4S-methyl-KE-298
CAS:S-methyl-KE-298 is the second main metabolite in plasma,is a methyl conjugate of deacetyl-KE-298.KE-298 inhibits matrix metalloproteinase (MMP-1) productionFórmula:C13H16O3SPureza:97.33%Forma y color:SolidPeso molecular:252.33Tenofovir alafenamide hemifumarate
CAS:<p>Tenofovir alafenamide hemifumarate (GS-7340 hemifumarate) is an oral phosphonoamidate prodrug of the HIV reverse transcriptase nucleotide inhibitor tenofovir.</p>Fórmula:C21H29N6O5PC4H4O4Pureza:99.33% - 99.96%Forma y color:SolidPeso molecular:534.51Trelagliptin succinate
CAS:<p>Trelagliptin succinate (SYR-472 succinate) is a long-acting inhibitor of dipeptidyl peptidase-4 (DPP-4), being developed for the treatment of type 2 diabetes (</p>Fórmula:C22H26FN5O6Pureza:99.27% - 99.92%Forma y color:SolidPeso molecular:475.47Ilomastat
CAS:<p>Ilomastat (GM6001) (GM6001, Galardin) is a broad spectrum matrix metalloprotease (MMP) inhibitor.</p>Fórmula:C20H28N4O4Pureza:97.04% - 99.51%Forma y color:SolidPeso molecular:388.462-Benzylsuccinic acid
CAS:<p>2-Benzylsuccinic acid (DL-Benzylsuccinic acid) is a bacterial xenobiotic metabolite.</p>Fórmula:C11H12O4Pureza:99.01% - ≥95%Forma y color:SolidPeso molecular:208.21(R)-MG-132
CAS:<p>(R)-MG-132 (Z-Leu-D-leu-leu-al) is the enantiomer of MG-132. (R)-MG-132 stereoisomer is a more potent proteasome inhibitor than MG-132.</p>Fórmula:C26H41N3O5Pureza:98.45%Forma y color:SolidPeso molecular:475.62NBD-557
CAS:<p>NBD-557 is a potentially HIV-1 inhibitor.</p>Fórmula:C17H24BrN3O2Pureza:99.52%Forma y color:SolidPeso molecular:382.3Sofosbuvir
CAS:<p>Sofosbuvir (GS 7977) is a uridine monophosphate analog inhibitor of hepatitis C virus (HCV) polymerase NS5B that is used as an antiviral agent in the treatment</p>Fórmula:C22H29FN3O9PPureza:99.77% - 99.82%Forma y color:SolidPeso molecular:529.45Vesnarinone
CAS:<p>Vesnarinone (Arkin) (INN) is a mixed phosphodiesterase 3 inhibitor and ion-channel modifier that has modest, dose-dependent, positive inotropic activity, but</p>Fórmula:C22H25N3O4Pureza:96.69% - 98.13%Forma y color:SolidPeso molecular:395.45Lersivirine
CAS:<p>Lersivirine (UK-453061)(UK 453061) is a second-generation non-nucleoside reverse transcriptase inhibitor (NNRTI) under development for HIV infection therapy.</p>Fórmula:C17H18N4O2Pureza:98.01%Forma y color:SolidPeso molecular:310.35Boceprevir
CAS:<p>Boceprevir (SCH 503034), an oral HCV NS3 protease inhibitor, has a Ki of 14 nM and EC90 of 350 nM.</p>Fórmula:C27H45N5O5Pureza:95% - 99.16%Forma y color:SolidPeso molecular:519.68Trovirdine
CAS:<p>Trovirdine (LY300046) is a thiourea non-nucleoside reverse transcriptase inhibitor.</p>Fórmula:C13H13BrN4SPureza:98.12% - 98.50%Forma y color:SolidPeso molecular:337.24HCV-IN-31
CAS:<p>HCV-IN-31 is a HCV inhibitor with an EC50/EC95 of 15.7 μM.</p>Fórmula:C12H17FN6O3Pureza:99.83%Forma y color:SolidPeso molecular:312.3VCH-916
CAS:<p>VCH-916 is a new nonnucleoside inhibitor of HCV NS5B polymerase.</p>Fórmula:C26H36KNO4SPureza:98%Forma y color:SolidPeso molecular:497.732-PMPA
CAS:<p>2-PMPA (2-(Phosphonomethyl)pentanedioic acid) is a potent and selective inhibitor of glutamate carboxypeptidase II (GCPII) (IC50=300 pM).</p>Fórmula:C6H11O7PPureza:97.4% - 99.5%Forma y color:SolidPeso molecular:226.12Bz-RS-ISer(3-Ph)-Ome
CAS:<p>Bz-RS-ISer(3-Ph)-Ome (Methyl (2R,3S)-3-(benzoylamino)-2-hydroxy-3-phenylpropanoate) is a paclitaxel derivative that inhibits the HSV replication cycle.</p>Fórmula:C17H17NO4Pureza:99.36% - 99.89%Forma y color:White CrystalPeso molecular:299.32Ledipasvir (acetone)
CAS:<p>Ledipasvir (acetone) (GS-5885 acetone) is an HCV NS5A polymerase inhibitor, used for the treatment of hepatitis C virus infection.</p>Fórmula:C52H60F2N8O7Pureza:99.72%Forma y color:SolidPeso molecular:947.08Methylchloroisothiazolinone/Methylisothiazolinone Mixture
CAS:<p>Methylchloroisothiazolinone/Methylisothiazolinone Mixture (Kathon 886MW),a preservative, activates MMPs in human bronchial epithelial cells.</p>Fórmula:C8H9ClN2O2S2Forma y color:SolidPeso molecular:264.75KP-457
CAS:<p>KP-457 is a ADAM17 and a TNFα converting enzyme TACE inhibitor that blocks the production of soluble TNF (sTNF).</p>Fórmula:C21H24N2O7S2Pureza:98.33%Forma y color:SolidPeso molecular:480.56Sitagliptin phosphate monohydrate
CAS:<p>Sitagliptin phosphate monohydrate (MK-0431 phosphate monohydrate) is a potent inhibitor of DPP-IV with IC50 of 19 nM in Caco-2 cell extracts.</p>Fórmula:C16H15F6N5O·H3PO4·H2OPureza:99.85% - 99.98%Forma y color:White Or Almost White Crystalline PowderPeso molecular:523.33(1S,2R)-Alicapistat
CAS:<p>(1S,2R)-Alicapistat inhibits calpains 1 and 2, shows promise for Alzheimer's, and has an IC50 of 395 nM.</p>Fórmula:C25H27N3O4Pureza:99.60%Forma y color:SoildPeso molecular:433.5Ledipasvir
CAS:<p>Ledipasvir (GS-5885) is a Hepatitis C Virus NS5A Inhibitor.</p>Fórmula:C49H54F2N8O6Pureza:99.96%Forma y color:SolidPeso molecular:889Rilpivirine HCl
CAS:<p>Rilpivirine HCl (Rilpivirine hydrochloride) is an NNRTI inhibitor with antiviral activity that inhibits the HIV virus.</p>Fórmula:C22H19ClN6Pureza:99.48%Forma y color:SolidPeso molecular:402.88(R)-Trolox
CAS:<p>(R)-Trolox is a selective tyrosinase inhibitor used in food, cosmetics, and pharmaceutical products.</p>Fórmula:C14H18O4Pureza:99.88%Forma y color:SolidPeso molecular:250.29Teneligliptin
CAS:<p>Teneligliptin (MP-513), potent DPP-4 inhibitor, IC50 ~1 nM, blocks DPP-4 in human/rat plasma and recombinant forms.</p>Fórmula:C22H30N6OSPureza:99.73%Forma y color:SolidPeso molecular:426.58Nelfinavir
CAS:<p>Nelfinavir (AG1341), with Ki=2 nM, is an HIV treatment and broad-spectrum anticancer drug.</p>Fórmula:C32H45N3O4SPureza:98.16% - 99.5%Forma y color:White To Off-White Crystalline PowderPeso molecular:567.78Danoprevir
CAS:<p>Danoprevir (RG7227) is a peptidomimetic inhibitor of the NS3/4A protease(IC50=0.2-3.5 nM) of hepatitis C virus (HCV).</p>Fórmula:C35H46FN5O9SPureza:98% - 99.35%Forma y color:SolidPeso molecular:731.83PSI
CAS:<p>PSI is a proteasome inhibitor.</p>Fórmula:C32H50N4O8Pureza:97% - 98.33%Forma y color:SolidPeso molecular:618.76Lanadelumab
CAS:<p>Lanadelumab (SHP643), a humanized IgG1 antibody, inhibits plasma kallikrein and its interaction with HMWK, supporting hereditary angioedema research.</p>Pureza:95% - 95%Forma y color:LiquidGalegenimab
CAS:<p>Galegenimab (FHTR 2163; RG 6147; RO 7171009) is an HTRA1 antibody fragment for AMD research.</p>Pureza:95% - 95%Forma y color:LiquidKZR-504
CAS:KZR-504 is a selective inhibitor of immunoproteasome low molecular mass polypeptide 2 (LMP2) (IC50s: 51 nM, 4.274 μM for LMP2 and LMP7, respectively).Fórmula:C21H23N3O6Forma y color:SolidPeso molecular:413.42Triton X-45(n=4)
CAS:<p>Triton X-45: nonionic, low HLB surfactant, dispersible in water, high Krafft point, relevant for HCV research.</p>Fórmula:C22H38O5Forma y color:SolidPeso molecular:382.53
