
Proteasas / Proteasoma
Los inhibidores de proteasas y proteasomas son compuestos que bloquean la actividad de las proteasas y del proteasoma, que están involucrados en la degradación y renovación de proteínas. Estos inhibidores son vitales para estudiar la regulación de la homeostasis proteica, el control del ciclo celular y la apoptosis. Los inhibidores de proteasas y proteasomas también se utilizan en el tratamiento de enfermedades como el cáncer, donde la degradación anormal de proteínas desempeña un papel en la progresión de la enfermedad. Al inhibir las proteasas o el proteasoma, estos compuestos pueden inducir la muerte celular en células cancerosas y son herramientas esenciales tanto en la investigación básica como en el desarrollo terapéutico. En CymitQuimica, ofrecemos una amplia gama de inhibidores de proteasas y proteasomas de alta calidad para apoyar su investigación en bioquímica, biología celular y desarrollo de fármacos.
Subcategorías de "Proteasas / Proteasoma"
- Acetil-CoA Carboxilasa(36 productos)
- Cisteína proteasa(110 productos)
- DPP-4(22 productos)
- Glutaminasa(45 productos)
- Proteasa del VIH(508 productos)
- PAI-1(26 productos)
- Inhibidores de la proteasa(50 productos)
- Receptor activado por proteasa(54 productos)
- Proteasoma(93 productos)
- Serina proteasa(55 productos)
- p97(15 productos)
Mostrar 3 subcategorías más
Se han encontrado 1066 productos de "Proteasas / Proteasoma"
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SB-3CT
CAS:SB-3CT is a potent and specific gelatinase inhibitor for MMP-2(Ki=13.9 nM) and MMP-9(Ki=600 nM).Fórmula:C15H14O3S2Pureza:98% - 99.38%Forma y color:SolidPeso molecular:306.4Ref: TM-T2009
1mg48,00€2mg65,00€5mg88,00€10mg159,00€25mg246,00€50mg368,00€100mg547,00€500mg1.198,00€1mL*10mM (DMSO)88,00€S-methyl-KE-298
CAS:S-methyl-KE-298 is the second main metabolite in plasma,is a methyl conjugate of deacetyl-KE-298.KE-298 inhibits matrix metalloproteinase (MMP-1) productionFórmula:C13H16O3SPureza:97.33%Forma y color:SolidPeso molecular:252.33Ref: TM-T4282
1mg88,00€5mg210,00€10mg338,00€25mg625,00€50mg938,00€100mg1.264,00€1mL*10mM (DMSO)188,00€Tenofovir alafenamide hemifumarate
CAS:<p>Tenofovir alafenamide hemifumarate (GS-7340 hemifumarate) is an oral phosphonoamidate prodrug of the HIV reverse transcriptase nucleotide inhibitor tenofovir.</p>Fórmula:C21H29N6O5PC4H4O4Pureza:99.33% - 99.96%Forma y color:SolidPeso molecular:534.51Trelagliptin succinate
CAS:Trelagliptin succinate (SYR-472 succinate) is a long-acting inhibitor of dipeptidyl peptidase-4 (DPP-4), being developed for the treatment of type 2 diabetes (Fórmula:C22H26FN5O6Pureza:99.27% - 99.92%Forma y color:SolidPeso molecular:475.47Ilomastat
CAS:Ilomastat (GM6001) (GM6001, Galardin) is a broad spectrum matrix metalloprotease (MMP) inhibitor.Fórmula:C20H28N4O4Pureza:97.04% - 99.51%Forma y color:SolidPeso molecular:388.46Ref: TM-T2743
1mg46,00€2mg62,00€5mg89,00€10mg145,00€25mg255,00€50mg429,00€100mg620,00€200mg880,00€1mL*10mM (DMSO)94,00€2-Benzylsuccinic acid
CAS:2-Benzylsuccinic acid (DL-Benzylsuccinic acid) is a bacterial xenobiotic metabolite.Fórmula:C11H12O4Pureza:99.01% - ≥95%Forma y color:SolidPeso molecular:208.21(R)-MG-132
CAS:(R)-MG-132 (Z-Leu-D-leu-leu-al) is the enantiomer of MG-132. (R)-MG-132 stereoisomer is a more potent proteasome inhibitor than MG-132.Fórmula:C26H41N3O5Pureza:99.90%Forma y color:SolidPeso molecular:475.62Ref: TM-T12628
2mg40,00€5mg60,00€10mg84,00€25mg127,00€50mg187,00€100mg283,00€200mg419,00€1mL*10mM (DMSO)74,00€NBD-557
CAS:NBD-557 is a potentially HIV-1 inhibitor.Fórmula:C17H24BrN3O2Pureza:99.52%Forma y color:SolidPeso molecular:382.3Ref: TM-T7382
1mg35,00€5mg74,00€10mg109,00€25mg210,00€50mg306,00€100mg434,00€200mg590,00€1mL*10mM (DMSO)82,00€Sofosbuvir
CAS:Sofosbuvir (GS 7977) is a uridine monophosphate analog inhibitor of hepatitis C virus (HCV) polymerase NS5B that is used as an antiviral agent in the treatmentFórmula:C22H29FN3O9PPureza:99.77% - 99.82%Forma y color:SolidPeso molecular:529.45Vesnarinone
CAS:Vesnarinone (Arkin) (INN) is a mixed phosphodiesterase 3 inhibitor and ion-channel modifier that has modest, dose-dependent, positive inotropic activity, butFórmula:C22H25N3O4Pureza:96.69% - 98.13%Forma y color:SolidPeso molecular:395.45Ref: TM-T3465
2mg35,00€5mg52,00€10mg80,00€25mg117,00€100mg313,00€200mg452,00€1mL*5mM (DMSO)49,00€50mg*5mM (DMSO)210,00€Lersivirine
CAS:Lersivirine (UK-453061)(UK 453061) is a second-generation non-nucleoside reverse transcriptase inhibitor (NNRTI) under development for HIV infection therapy.Fórmula:C17H18N4O2Pureza:98.01%Forma y color:SolidPeso molecular:310.35Boceprevir
CAS:Boceprevir (SCH 503034), an oral HCV NS3 protease inhibitor, has a Ki of 14 nM and EC90 of 350 nM.Fórmula:C27H45N5O5Pureza:95% - 99.16%Forma y color:SolidPeso molecular:519.68Ref: TM-T4988
1mg35,00€5mg70,00€10mg96,00€25mg144,00€50mg187,00€100mg274,00€200mg378,00€1mL*10mM (DMSO)80,00€HCV-IN-31
CAS:HCV-IN-31 is a HCV inhibitor with an EC50/EC95 of 15.7 μM.Fórmula:C12H17FN6O3Pureza:99.83%Forma y color:SolidPeso molecular:312.3VCH-916
CAS:VCH-916 is a new nonnucleoside inhibitor of HCV NS5B polymerase.Fórmula:C26H36KNO4SPureza:98%Forma y color:SolidPeso molecular:497.732-PMPA
CAS:2-PMPA (2-(Phosphonomethyl)pentanedioic acid) is a potent and selective inhibitor of glutamate carboxypeptidase II (GCPII) (IC50=300 pM).Fórmula:C6H11O7PPureza:97.4% - 99.5%Forma y color:SolidPeso molecular:226.12Bz-RS-ISer(3-Ph)-Ome
CAS:<p>Bz-RS-ISer(3-Ph)-Ome (Methyl (2R,3S)-3-(benzoylamino)-2-hydroxy-3-phenylpropanoate) is a paclitaxel derivative that inhibits the HSV replication cycle.</p>Fórmula:C17H17NO4Pureza:99.36% - 99.89%Forma y color:White CrystalPeso molecular:299.32Ledipasvir (acetone)
CAS:Ledipasvir (acetone) (GS-5885 acetone) is an HCV NS5A polymerase inhibitor, used for the treatment of hepatitis C virus infection.Fórmula:C52H60F2N8O7Pureza:99.72%Forma y color:SolidPeso molecular:947.08Ref: TM-T4203
1mg35,00€2mg48,00€5mg70,00€10mg93,00€25mg153,00€50mg235,00€100mg359,00€200mgA consultar1mL*10mM (DMSO)96,00€Teneligliptin
CAS:Teneligliptin (MP-513), potent DPP-4 inhibitor, IC50 ~1 nM, blocks DPP-4 in human/rat plasma and recombinant forms.Fórmula:C22H30N6OSPureza:99.73%Forma y color:SolidPeso molecular:426.58KP-457
CAS:KP-457 is a ADAM17 and a TNFα converting enzyme TACE inhibitor that blocks the production of soluble TNF (sTNF).Fórmula:C21H24N2O7S2Pureza:98.33%Forma y color:SolidPeso molecular:480.56Ref: TM-T77778
1mg92,00€5mg216,00€10mg354,00€25mg655,00€50mg1.035,00€100mg1.406,00€1mL*10mM (DMSO)230,00€Rilpivirine HCl
CAS:Rilpivirine HCl (Rilpivirine hydrochloride) is an NNRTI inhibitor with antiviral activity that inhibits the HIV virus.Fórmula:C22H19ClN6Pureza:99.48%Forma y color:SolidPeso molecular:402.88
