
Proteasas / Proteasoma
Los inhibidores de proteasas y proteasomas son compuestos que bloquean la actividad de las proteasas y del proteasoma, que están involucrados en la degradación y renovación de proteínas. Estos inhibidores son vitales para estudiar la regulación de la homeostasis proteica, el control del ciclo celular y la apoptosis. Los inhibidores de proteasas y proteasomas también se utilizan en el tratamiento de enfermedades como el cáncer, donde la degradación anormal de proteínas desempeña un papel en la progresión de la enfermedad. Al inhibir las proteasas o el proteasoma, estos compuestos pueden inducir la muerte celular en células cancerosas y son herramientas esenciales tanto en la investigación básica como en el desarrollo terapéutico. En CymitQuimica, ofrecemos una amplia gama de inhibidores de proteasas y proteasomas de alta calidad para apoyar su investigación en bioquímica, biología celular y desarrollo de fármacos.
Subcategorías de "Proteasas / Proteasoma"
- Acetil-CoA Carboxilasa(50 productos)
- Cisteína proteasa(120 productos)
- DPP-4(27 productos)
- Glutaminasa(46 productos)
- Proteasa del VIH(487 productos)
- PAI-1(30 productos)
- Inhibidores de la proteasa(49 productos)
- Receptor activado por proteasa(57 productos)
- Proteasoma(91 productos)
- Serina proteasa(70 productos)
- p97(15 productos)
Mostrar 3 subcategorías más
Se han encontrado 922 productos para "Proteasas / Proteasoma".
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2-Oxiranecarboxylic acid, 3-[[[(1S)-3-methyl-1-[[(3-methylbutyl)amino]carbonyl]butyl]amino]carbonyl]-, ethyl ester, (2S,3S)-
CAS:Fórmula:C17H30N2O5Pureza:98%Forma y color:SolidPeso molecular:342.4305Retagliptin Phosphate
CAS:Retagliptin Phosphate (SP 2086) is pharmaceutical composition of DPP-4 inhibitor, for treating type-2 diabetes.Fórmula:C19H21F6N4O7PPureza:98.70%Forma y color:SolidPeso molecular:562.36Ref: TM-T12710
100mgA consultar1mg34,00€2mg42,00€5mg60,00€1mL*10mM (DMSO)79,00€10mg87,00€25mg161,00€50mg245,00€RAMB4
CAS:RAMB4 (PTP1B-IN-9) is a ubiquitin-proteasome system (UPS)-stressor,with anticancer activity.Fórmula:C19H13Cl4NOPureza:98.89% - 99.38%Forma y color:Yellow SolidPeso molecular:413.12Anisindione
CAS:Anisindione, a synthetic indanedione, inhibits vitamin K, blocking factors II, VII, IX, X, and proteins C, S.Fórmula:C16H12O3Pureza:98.25%Forma y color:White SolidPeso molecular:252.26ARP-100
CAS:ARP-100 (MMP-2 Inhibitor III) is a potent and selective matrix metalloproteinase MMP-2 inhibitor (IC50=12 nM).Fórmula:C17H20N2O5SPureza:97.18%Forma y color:White SolidPeso molecular:364.42Ruzasvir
CAS:Ruzasvir (MK-8408) is a novel and potent pan-genotypic inhibitor of hepatitis C virus NS5A with antiviral activity.Fórmula:C49H55FN10O7SPureza:96.87% - 99.93%Forma y color:SolidPeso molecular:947.09DPP-IV-IN-2
CAS:DPP-IV-IN-2 (H-Lys(4-nitro-Z)-pyrrolidide) is an inhibitor of both DP8/9 and dipeptidyl peptidase IV (IC50s: 0.1 and 0.95 μM).Fórmula:C18H26N4O5Pureza:99.08% - 99.51%Forma y color:White SolidPeso molecular:378.42Avoralstat
CAS:Avoralstat (BCX4161) is an oral plasma kallikrein (PKK) inhibitor. Which is used for the treatment of hereditary angioedema.Fórmula:C28H27N5O5Pureza:99.77%Forma y color:SolidPeso molecular:513.54Saxagliptin hydrate
CAS:Saxagliptin hydrate (Onglyza hydrate) is a selective and reversible DPP4 inhibitor (IC50: 26 nM; Ki: 1.3 nM).Fórmula:C18H25N3O2·H2OPureza:99.52%Forma y color:SolidPeso molecular:333.43RA190
CAS:RA190 inhibits proteasome function by covalently binding to cysteine 88 of ubiquitin receptor RPN13.Fórmula:C28H23Cl5N2O2Pureza:97.7%Forma y color:SolidPeso molecular:596.76Ref: TM-T13858
1mg54,00€5mg109,00€1mL*10mM (DMSO)142,00€10mg159,00€25mg233,00€50mg414,00€100mg608,00€PMSF
CAS:PMSF (Phenylmethylsulfonyl fluoride) is an irreversible inhibitor of serine/cysteine protease , preparation of cell lysates. High-Quality, Low-Cost!Fórmula:C7H7FO2SPureza:97.75% - 99.88%Forma y color:White SolidPeso molecular:174.19DBPR108
CAS:DBPR108 is an orally bioavailable dipeptide-derived DPP4 inhibitor (IC50: 15 nM) and it has no inhibition on DDP8 and DPP9.Fórmula:C16H25FN4O2Pureza:99.68%Forma y color:SolidPeso molecular:324.39Ref: TM-T15079
1mg48,00€5mg100,00€1mL*10mM (DMSO)110,00€10mg133,00€25mg215,00€50mg306,00€100mg414,00€200mg573,00€Mecarbinate
CAS:Mecarbinate (Dimecarbin) is arbidol hydrochloride's chemical intermediate.Fórmula:C13H15NO3Pureza:99.28%Forma y color:Off-White Crystalline PowderPeso molecular:233.26ML604440
CAS:ML604440 is a cell permeable proteasome β1i (LMP2) subunit inhibitor.Fórmula:C17H24BF3N2O4Pureza:97.06%Forma y color:SolidPeso molecular:388.19Ref: TM-T12079
1mg109,00€2mg158,00€5mg259,00€1mL*10mM (DMSO)285,00€10mg409,00€25mg677,00€50mg954,00€100mg1.288,00€200mg1.728,00€midesteine
CAS:Midesteine (MR-889) is a small molecule neutrophil elastase inhibitor used in the treatment of bronchitis, asthma and chronic lung disease.Fórmula:C12H13NO3S3Pureza:99.87% - 99.98%Forma y color:SolidPeso molecular:315.43CL-82198
CAS:CL-82198, a selective MMP-13 inhibitor, serves as a pharmacological intervention to halt the progression of osteoarthritis (OA).Fórmula:C17H22N2O3Pureza:95.91%Forma y color:SolidPeso molecular:302.37L-Leucinamide, N-[(phenylmethoxy)carbonyl]-L-leucyl-N-[(1S)-1-formyl-3-methylbutyl]-
CAS:Fórmula:C26H41N3O5Pureza:98%Forma y color:SolidPeso molecular:475.6208Benzoic acid, 4-[[6-[(aminoiminomethyl)amino]-1-oxohexyl]oxy]-, ethylester, monomethanesulfonate
CAS:Fórmula:C17H27N3O7SPureza:98%Forma y color:SolidPeso molecular:417.4772Ref: IN-DA00IA62
10mg20,00€25mg23,00€5mg26,00€50mg27,00€100mg31,00€250mg40,00€1g72,00€5g146,00€25g691,00€1,10-Phenanthroline hydrate
CAS:Fórmula:C12H10N2OPureza:98%Forma y color:SolidPeso molecular:198.2206

