Proteasas / Proteasoma
Los inhibidores de proteasas y proteasomas son compuestos que bloquean la actividad de las proteasas y del proteasoma, que están involucrados en la degradación y renovación de proteínas. Estos inhibidores son vitales para estudiar la regulación de la homeostasis proteica, el control del ciclo celular y la apoptosis. Los inhibidores de proteasas y proteasomas también se utilizan en el tratamiento de enfermedades como el cáncer, donde la degradación anormal de proteínas desempeña un papel en la progresión de la enfermedad. Al inhibir las proteasas o el proteasoma, estos compuestos pueden inducir la muerte celular en células cancerosas y son herramientas esenciales tanto en la investigación básica como en el desarrollo terapéutico. En CymitQuimica, ofrecemos una amplia gama de inhibidores de proteasas y proteasomas de alta calidad para apoyar su investigación en bioquímica, biología celular y desarrollo de fármacos.
Subcategorías de "Proteasas / Proteasoma"
- Acetil-CoA Carboxilasa(36 productos)
- Cisteína proteasa(111 productos)
- DPP-4(24 productos)
- Glutaminasa(44 productos)
- Proteasa del VIH(501 productos)
- PAI-1(26 productos)
- Inhibidores de la proteasa(50 productos)
- Receptor activado por proteasa(54 productos)
- Proteasoma(89 productos)
- Serina proteasa(54 productos)
- p97(15 productos)
Mostrar 3 subcategorías más
Se han encontrado 993 productos de "Proteasas / Proteasoma"
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MMP13-IN-3
CAS:MMP13-IN-3 is an oral, selective MMP-13 inhibitor with IC50 of 1 nM, >1000x selective, for osteoarthritis treatment.Fórmula:C24H22N4O5Pureza:99.76%Forma y color:SolidPeso molecular:446.46Ref: TM-T16124
1mg93,00€5mg205,00€10mg334,00€25mg587,00€50mg802,00€100mg1.108,00€1mL*10mM (DMSO)227,00€MMP-7-IN-2
CAS:MMP-7-IN-2 acts as a selective and potent MMP7 inhibitor and can be used to study inflammatory responses and vascular-related diseases.Fórmula:C28H40ClF3N6O9SPureza:97.82%Forma y color:SolidPeso molecular:729.17Beclabuvir HCl
CAS:Beclabuvir (BMS-791325) is an HCV inhibitor targeting NS5B polymerase with sub-28 nM potency for genotypes 1, 3, 4, 5.Fórmula:C36H46ClN5O5SForma y color:SolidPeso molecular:696.3Paltimatrectinib
CAS:Paltimatrectinib (PBI-200) is a tyrosine kinase inhibitor with anticancer activity, and is used in the study of bladder, breast, and colorectal cancers.Fórmula:C20H15F5N6Pureza:99.96%Forma y color:SolidPeso molecular:434.37MeOSuc-AAPV-CMK
CAS:MeOSuc-AAPV-CMK (Elastase Inhibitor III) serves as an inhibitor of elastase, as well as cathepsin G and proteinase 3, and impedes leukocyte elastase-mediatedFórmula:C22H35ClN4O7Forma y color:SolidPeso molecular:502.99Cathepsin K inhibitor 3
CAS:Cathepsin K inhibitor 3: Selective, IC50 of 0.5 nM, good pharmacokinetics, potential for OA research.Fórmula:C30H31FN4O4SForma y color:SolidPeso molecular:562.65Ecallantide
CAS:Ecallantide (DX-88) is a recombinant inhibitor specifically targeting plasma kallikrein, which serves to impede the synthesis of bradykinin.Fórmula:C305H448N88O91S8Forma y color:SolidPeso molecular:7059.88MMP-9 Inhibitor I
CAS:MMP-9 inhibitor I is an inhibitor of matrix metalloproteinase-9 (MMP-9) that is selective over MMP-1 and MMP-13 (IC50s = 5, 1,050, and 113 nM, respectively).Fórmula:C27H33N3O5SForma y color:SolidPeso molecular:511.63BMS-189664 HCl
CAS:BMS-189664 HCl is a selective and orally active thrombin active site inhibitor.Fórmula:C22H35ClN6O4SPureza:98%Forma y color:SolidPeso molecular:515.07Z-DEVD-CMK
CAS:Z-DEVD-CMK irreversibly inhibits various cathepsins in vitro [1].Fórmula:C27H35ClN4O12Forma y color:SolidPeso molecular:643.04DCLK1-IN-2
CAS:DCLK1-IN-2 (Compound I-5) is a potent inhibitor of DCLK1, exhibiting an IC50 of 171.3 nM, and demonstrates significant antiproliferative effects on SW1990 cellFórmula:C26H32N8O3SForma y color:SolidPeso molecular:536.65Cardanol diene
CAS:Cardanol diene: phenol in cashew shells; anti-tyrosinase (IC50=52.5μM); used to make anti-E. coli biofilm complexes.Fórmula:C21H32OForma y color:SolidPeso molecular:300.48ASP-8497
CAS:ASP8497 is a potent DPP-IV inhibitor enhancing GLP-1, used for type 2 diabetes and glucose intolerance.Fórmula:C18H27FN4O7SForma y color:SolidPeso molecular:462.49I-XW-053
CAS:I-XW-053 is an inhibitor of capsid targeted HIV-1 replication using the hybrid structure based method to block the interface between CA N-terminal domains (NTD-Fórmula:C22H16N2O2Pureza:99.05%Forma y color:SolidPeso molecular:340.37NS5A-IN-3
CAS:NS5A-IN-3 is a potent NS5A inhibitor with high efficacy against HCV 1b, good activity on 3a, and strong metabolic stability; superior to daclatasvir.Fórmula:C44H44N6O8Pureza:98%Forma y color:SolidPeso molecular:784.86Collagen proline hydroxylase inhibitor-1
CAS:Collagen proline hydroxylase inhibitor-1 具有抗纤维增生活性。Fórmula:C24H21N5O4Pureza:99.57%Forma y color:SolidPeso molecular:443.45HIV-1 inhibitor-54
CAS:HIV-1 inhibitor-54: potent anti-HIV (EC50: 32 nM), targets WT HIV-1 IIIB in MT-4 cells for infection research.Fórmula:C27H30N6O4SPureza:98.05% - 99.39%Forma y color:SoildPeso molecular:534.63BMS-212122
CAS:BMS-212122 inhibits MTP, reduces lipids and plaque in animal tests.Fórmula:C43H36F6N4O2Pureza:99.85%Forma y color:SolidPeso molecular:754.76Ref: TM-T30506
1mg315,00€5mg745,00€10mg1.018,00€25mg1.431,00€50mg1.783,00€100mg2.250,00€500mg4.410,00€γ-Glu-Tyr
CAS:gamma-Glu-Tyr (gamma-Glutamyltyrosine) is a kokumi peptide against dipeptidyl peptidase-IV (DPP-IV) and is used in the study of diabetes mellitus.Fórmula:C14H18N2O6Pureza:98.92%Forma y color:SolidPeso molecular:310.3ZED-1227
CAS:ZED-1227 (TAK-227) is a TG2 inhibitor with anticancer activity that blocks inflammation-induced TG2 expression and activation for the treatment of Celiac Diseas
Fórmula:C26H36N6O6Pureza:99.04%Forma y color:SolidPeso molecular:528.6
