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Tirosina quinasa / adaptadores
Subcategorías de "Tirosina quinasa / adaptadores"
ALK
CSF-1R
EGFR
Receptor de efrina
FLT
Receptor del factor de crecimiento de fibroblastos (FGFR)
HER
Hck
IGF-1R
PDGFR
PYK2
Src
Receptor TAM
Tie-2
Receptor de Trk
Tirosina quinasas
VEGFR
c-Fms
c-Kit
c-Met / HGFR
c-RET
Mostrar 13 subcategorías más
Productos de "Tirosina quinasa / adaptadores"
![discount label](https://static.cymitquimica.com/public/img/discount.png)
FGFR2-IN-1
CAS:2677709-76-9
FGFR2-IN-1 is an FGFR inhibitor that inhibits FGFR1, FGFR2, and FGFR3, and can be used …
Fórmula:
C22H19N3O2
Forma y color:
Solid
Peso molecular:
357.41
Ref: TM-T61304
1mg | 60,00 € | ||
5mg | 130,00 € | ||
10mg | 198,00 € | ||
25mg | 333,00 € | ||
50mg | 495,00 € | ||
100mg | 704,00 € | ||
500mg | 1.419,00 € |
Entrega estimada en Estados Unidos, el Martes 3 de Septiembre de 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
DDR Inhibitor
CAS:1644069-80-6
DDR inhibitor is a potent discidin domain receptor (DDR) inhibitor. The IC50 of DDR2 is …
Fórmula:
C23H20FN5O2
Pureza:
97.75%
Forma y color:
Solid
Peso molecular:
417.44
Ref: TM-T10985
1mg | 114,00 € | ||
1ml | 258,00 € | ||
5mg | 230,00 € | ||
10mg | 369,00 € | ||
25mg | 741,00 € | ||
50mg | 1.179,00 € | ||
100mg | 1.597,00 € |
Entrega estimada en Estados Unidos, el Martes 3 de Septiembre de 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
c-Fms-IN-6
CAS:1628574-81-1
c-Fms-IN-6 is a potent inhibitor of c-FMS (IC50 ≤10 nM for unphosphorylated c-FMS) and also …
Fórmula:
C22H25N7O2
Pureza:
98%
Forma y color:
Solid
Peso molecular:
419.48
Ref: TM-T10645
25mg | 1.549,00 € | ||
50mg | 2.038,00 € | ||
100mg | 2.617,00 € |
Entrega estimada en Estados Unidos, el Martes 3 de Septiembre de 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Tafetinib
CAS:1032265-57-8
Tafetinib (SIM-010603) is a novel potent and orally available tyrosine kinase inhibitor with anti-angiogenic and …
Fórmula:
C24H29FN4O2
Pureza:
96.66%
Forma y color:
Solid
Peso molecular:
424.51
Ref: TM-T28911
1mg | 233,00 € | ||
5mg | 581,00 € | ||
10mg | 824,00 € | ||
25mg | 1.234,00 € | ||
50mg | 1.654,00 € | ||
100mg | 2.265,00 € | ||
500mg | 4.532,00 € |
Entrega estimada en Estados Unidos, el Martes 3 de Septiembre de 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
OD36 hydrochloride
CAS:2387510-88-3
OD36 hydrochloride (OD-36 hydrochloride) is a potent RIPK2 inhibitor with an IC50 of 5.3 nM.OD36 …
Fórmula:
C16H16Cl2N4O2
Pureza:
99.85%
Forma y color:
Solid
Peso molecular:
367.23
Ref: TM-T61424
25mg | 1.197,00 € | ||
50mg | 1.561,00 € | ||
100mg | 2.320,00 € |
Entrega estimada en Estados Unidos, el Martes 3 de Septiembre de 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
CHMFL-EGFR-202
CAS:2089381-40-6
CHMFL-EGFR-202 is a potent, irreversible inhibitor of EGFR mutant kinase (IC50s: 5.3 nM and 8.3 …
Fórmula:
C25H24ClN7O2
Pureza:
99.19%
Forma y color:
Solid
Peso molecular:
489.96
Ref: TM-T10802
1mg | 113,00 € | ||
1ml | 304,00 € | ||
2mg | 169,00 € | ||
5mg | 250,00 € | ||
10mg | 368,00 € | ||
25mg | 552,00 € | ||
50mg | 772,00 € | ||
100mg | 1.053,00 € |
Entrega estimada en Estados Unidos, el Martes 3 de Septiembre de 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Rogaratinib
CAS:1443530-05-9
Rogaratinib (BAY1163877) is an aberrant inhibitor of fibroblast growth factor receptor (FGFR).
Fórmula:
C23H26N6O3S
Pureza:
99.54%
Forma y color:
Solid
Peso molecular:
466.56
Ref: TM-T16781
1mg | 147,00 € |
Entrega estimada en Estados Unidos, el Martes 3 de Septiembre de 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Selatinib
CAS:1275595-86-2
Selatinib is an orally active and potent dual inhibitor of EGFR and ErbB2 with anticancer …
Fórmula:
C29H26ClFN4O3S
Pureza:
98%
Forma y color:
Solid
Peso molecular:
565.06
Ref: TM-T34602
1mg | 96,00 € | ||
5mg | 229,00 € | ||
10mg | 345,00 € | ||
25mg | 730,00 € | ||
50mg | 1.167,00 € | ||
100mg | 1.847,00 € |
Entrega estimada en Estados Unidos, el Martes 3 de Septiembre de 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
A-770041
CAS:869748-10-7
A-770041 is selective and orally active Src-family Lck inhibitor, and the other Src family kinase …
Fórmula:
C34H39N9O3
Pureza:
98%
Forma y color:
Solid
Peso molecular:
621.73
Ref: TM-T14074
5mg | A consultar |
Entrega estimada en Estados Unidos, el Martes 3 de Septiembre de 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
SKLB 1028
CAS:1350544-93-2
SKLB 1028, an oral EGFR/FLT3/Abl inhibitor, excels in AML and CML with Abl mutations.
Fórmula:
C24H29N9
Pureza:
99.71%
Forma y color:
Solid
Peso molecular:
443.55
Ref: TM-T34656
1mg | 55,00 € | ||
1ml | 143,00 € | ||
5mg | 118,00 € | ||
10mg | 185,00 € | ||
25mg | 369,00 € | ||
50mg | 547,00 € | ||
100mg | 786,00 € | ||
500mg | 1.616,00 € |
Entrega estimada en Estados Unidos, el Martes 3 de Septiembre de 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
FGFR4-IN-8
CAS:2765240-52-4
FGFR4-IN-8 (Compound 7v) is an ATP-competitive inhibitor that covalently and highly selectively targets both the …
Fórmula:
C32H34Cl2FN7O3
Pureza:
98%
Peso molecular:
654.56
Ref: TM-T73121
25mg | 1.549,00 € | ||
50mg | 2.038,00 € | ||
100mg | 2.617,00 € |
Entrega estimada en Estados Unidos, el Lunes 16 de Septiembre de 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Ifebemtinib
CAS:1227948-82-4
Ifebemtinib (BI-853520) is an orally active and potent inhibitor of adhesion plaque kinase (FAK) (IC50=1 …
Fórmula:
C28H28F4N6O4
Pureza:
99.82%
Forma y color:
Solid
Peso molecular:
588.55
Ref: TM-T64167
1mg | 160,00 € | ||
5mg | 387,00 € | ||
10mg | 646,00 € | ||
25mg | 1.396,00 € |
Entrega estimada en Estados Unidos, el Lunes 16 de Septiembre de 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Simotinib
CAS:944258-89-3
Simotinib (AL-6802) is a selective and orally bioactive EGFR tyrosine kinase inhibitor (IC50: 19.9 nM) …
Fórmula:
C25H26ClFN4O4
Pureza:
99.7%
Forma y color:
Solid
Peso molecular:
500.95
Ref: TM-T35916
1mg | 171,00 € | ||
1ml*10 (DMSO) | 295,00 € |
Entrega estimada en Estados Unidos, el Lunes 16 de Septiembre de 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
MK-2461
CAS:917879-39-1
MK-2461 is a novel inhibitor that targets multiple proteins and competitively binds to ATP sites, …
Fórmula:
C24H25N5O5S
Pureza:
98.36%
Forma y color:
Solid
Peso molecular:
495.55
Ref: TM-T6094
1mg | 59,00 € | ||
1ml | 159,00 € | ||
2mg | 83,00 € | ||
5mg | 145,00 € | ||
10mg | 245,00 € | ||
25mg | 495,00 € | ||
50mg | 713,00 € | ||
100mg | 1.000,00 € | ||
500mg | 1.996,00 € |
Entrega estimada en Estados Unidos, el Lunes 16 de Septiembre de 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
PF-06459988
CAS:1428774-45-1
PF-06459988 is a novel, effective, orally active, irreversible, and selective epidermal growth factor receptor (EGFR) …
Fórmula:
C19H22ClN7O3
Pureza:
98%
Forma y color:
Solid
Peso molecular:
431.88
Ref: TM-T16492
1mg | 143,00 € |
Entrega estimada en Estados Unidos, el Lunes 16 de Septiembre de 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
LX7101
CAS:1192189-69-7
LX7101 is an effective inhibitor of LIMK and ROCK2 (IC50: 24, 1.6, and 10 nM …
Fórmula:
C23H29N7O3
Pureza:
98.42%
Forma y color:
Solid
Peso molecular:
451.52
Ref: TM-T15798
1mg | 61,00 € | ||
5mg | 159,00 € | ||
50mg | 931,00 € | ||
1ml*10 (DMSO) | 222,00 € |
Entrega estimada en Estados Unidos, el Lunes 16 de Septiembre de 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
EGFR-IN-1
CAS:1625677-63-5
EGFR-IN-1, an orally active and irreversible selective inhibitor targeting L858R/T790M mutant EGFR, exhibits strong antiproliferative …
Fórmula:
C28H30N6O4
Pureza:
98%
Forma y color:
Solid
Peso molecular:
514.58
Ref: TM-T11157
25mg | 1.688,00 € | ||
50mg | 2.225,00 € | ||
100mg | 2.897,00 € |
Entrega estimada en Estados Unidos, el Lunes 16 de Septiembre de 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
JND3229
CAS:2260886-64-2
JND3229 inhibits EGFRC797S; IC50: 5.8-30.5 nM; halts cell growth; effective in non-small cell lung cancer …
Fórmula:
C33H41ClN8O2
Pureza:
97.35%
Forma y color:
Solid
Peso molecular:
617.18
Ref: TM-T15615
1mg | 123,00 € | ||
1ml | 419,00 € | ||
5mg | 303,00 € | ||
10mg | 456,00 € | ||
25mg | 754,00 € | ||
50mg | 1.049,00 € |
Entrega estimada en Estados Unidos, el Lunes 16 de Septiembre de 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Tyrphostin AG1433
CAS:168835-90-3
Tyrphostin AG1433 (AG1433) is an inhibitor of tyrosine kinases and also a dual inhibitor of …
Fórmula:
C16H14N2O2
Pureza:
97.51%
Forma y color:
Solid
Peso molecular:
266.29
Ref: TM-T13238
1mg | 52,00 € | ||
1ml | 111,00 € | ||
5mg | 95,00 € | ||
10mg | 157,00 € | ||
25mg | 266,00 € | ||
50mg | 407,00 € | ||
100mg | 607,00 € | ||
500mg | 1.255,00 € |
Entrega estimada en Estados Unidos, el Lunes 16 de Septiembre de 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
PAT-505
CAS:1782070-22-7
PAT-505 is an orally available, selective and potent inhibitor of autologous epidermal growth factor (IC50 …
Fórmula:
C23H18ClF2N3O2S
Pureza:
98.84%
Forma y color:
Solid
Peso molecular:
473.92
Ref: TM-T12372
1mg | 243,00 € | ||
1ml*10 (DMSO) | 455,00 € |
Entrega estimada en Estados Unidos, el Lunes 16 de Septiembre de 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
KB SRC 4
CAS:1380088-03-8
KB SRC 4 is a selective and potent c-Src inhibitor with antitumour activity that inhibits …
Fórmula:
C32H23ClN8
Pureza:
99.66%
Forma y color:
Solid
Peso molecular:
555.03
Ref: TM-T11745
1mg | 147,00 € |
Entrega estimada en Estados Unidos, el Lunes 16 de Septiembre de 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Brepocitinib
CAS:1883299-62-4
Brepocitinib (PF-06700841) is a potent dual JAK1/TYK2 inhibitor (IC50s: 17 nM/23 nM). Brepocitinib also inhibits …
Fórmula:
C18H21F2N7O
Pureza:
98%
Forma y color:
Solid
Peso molecular:
389.4
Ref: TM-TQ0010
1mg | 35,00 € | ||
1ml | 117,00 € | ||
5mg | 69,00 € | ||
10mg | 102,00 € | ||
25mg | 212,00 € | ||
50mg | 383,00 € | ||
100mg | 614,00 € | ||
200mg | 859,00 € | ||
500mg | 1.270,00 € |
Entrega estimada en Estados Unidos, el Lunes 16 de Septiembre de 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
BMS-935177
CAS:1231889-53-4
BMS-935177 is a reversible BTK inhibitor with IC50 value of 3 nM.
Fórmula:
C31H26N4O3
Pureza:
99.89%
Forma y color:
Solid
Peso molecular:
502.56
Ref: TM-T14681
1mg | 42,00 € | ||
1ml | 166,00 € | ||
2mg | 67,00 € | ||
10mg | A consultar | ||
50mg | A consultar |
Entrega estimada en Estados Unidos, el Lunes 16 de Septiembre de 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
PF-06250112
CAS:1609465-89-5
PF-06250112 is an effective and highly selective BTK inhibitor (IC50: 0.5 nM.
Fórmula:
C22H20F2N6O2
Pureza:
98%
Forma y color:
Solid
Peso molecular:
438.43
Ref: TM-T12673L
25mg | 1.827,00 € | ||
50mg | 2.412,00 € | ||
100mg | 3.178,00 € |
Entrega estimada en Estados Unidos, el Lunes 16 de Septiembre de 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
APG-2449
CAS:2196186-84-0
APG-2449 is an orally active inhibitor targeting ALK, ROS1, and FAK, demonstrating antitumor efficacy in …
Fórmula:
C33H42ClN5O4S
Pureza:
98%
Peso molecular:
640.24
Ref: TM-T79363
25mg | 1.410,00 € | ||
50mg | 1.851,00 € | ||
100mg | 2.337,00 € |
Entrega estimada en Estados Unidos, el Lunes 16 de Septiembre de 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
AXL-IN-14
CAS:2947506-65-0
AXL-IN-14 is a potent, orally active inhibitor of AXL with an IC50 of 0.8 nM …
Fórmula:
C32H24F2N4O4
Pureza:
98%
Peso molecular:
566.55
Ref: TM-T73310
25mg | 1.688,00 € | ||
50mg | 2.225,00 € | ||
100mg | 2.897,00 € |
Entrega estimada en Estados Unidos, el Lunes 16 de Septiembre de 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
CP-547632 TFA
CAS:2805804-54-8
CP-547632 TFA is an orally active, ATP-competitive inhibitor that potently targets VEGFR-2 and FGF kinases …
Fórmula:
C22H25BrF5N5O5S
Pureza:
98%
Peso molecular:
646.43
Ref: TM-T74000
25mg | 1.827,00 € | ||
50mg | 2.412,00 € | ||
100mg | 3.178,00 € |
Entrega estimada en Estados Unidos, el Lunes 16 de Septiembre de 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
TL02-59
CAS:1315330-17-6
TL02-59: Fgr inhibitor (IC50=0.03nM), also targets Lyn (0.1nM), Hck (160nM), halts acute myelogenous leukemia growth.
Fórmula:
C32H34F3N5O4
Pureza:
98%
Forma y color:
Solid
Peso molecular:
609.64
Ref: TM-T13186
1mg | 104,00 € | ||
1ml | 281,00 € | ||
5mg | 212,00 € | ||
10mg | 347,00 € | ||
25mg | 584,00 € | ||
50mg | 832,00 € | ||
100mg | 1.132,00 € |
Entrega estimada en Estados Unidos, el Lunes 16 de Septiembre de 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
DYRKs-IN-2
CAS:1386980-04-6
DYRKs-IN-2 has antitumor activity. DYRKs-IN-2 is a potent DYRKs inhibitor with IC50s of 30.6 nM …
Fórmula:
C32H38ClN9O3
Pureza:
98%
Forma y color:
Solid
Peso molecular:
632.16
Ref: TM-T11133
25mg | 1.967,00 € | ||
50mg | 2.592,00 € | ||
100mg | 3.450,00 € |
Entrega estimada en Estados Unidos, el Lunes 16 de Septiembre de 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
DZD1516
CAS:2387570-00-3
DZD1516, a potent and selective HER2 inhibitor (IC50 = 0.56 nM), demonstrates good blood-brain barrier …
Fórmula:
C28H27F2N7O3
Pureza:
98%
Peso molecular:
547.56
Ref: TM-T79297
25mg | 1.549,00 € | ||
50mg | 2.038,00 € | ||
100mg | 2.617,00 € |
Entrega estimada en Estados Unidos, el Lunes 16 de Septiembre de 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
2′-Thioadenosine
CAS:136904-69-3
2'-Thioadenosine (PD157432) serves as a selective and irreversible inhibitor of ErbB-1 and ErbB-2 tyrosine kinases, …
Fórmula:
C10H13N5O3S
Pureza:
98%
Peso molecular:
283.31
Ref: TM-T78634
25mg | 1.549,00 € | ||
50mg | 2.038,00 € | ||
100mg | 2.617,00 € |
Entrega estimada en Estados Unidos, el Lunes 16 de Septiembre de 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
MCHR1 antagonist 2
CAS:863115-70-2
MCHR1 antagonist 2 is an antagonist of melanin-concentratin hormone receptor 1(MCH1-R, IC50 = 65 nM) …
Fórmula:
C23H21FN2O5
Pureza:
98%
Forma y color:
Solid
Peso molecular:
424.42
Ref: TM-T11966
1mg | 142,00 € | ||
1ml | 326,00 € | ||
5mg | 291,00 € | ||
10mg | 432,00 € | ||
25mg | 708,00 € | ||
50mg | 1.000,00 € | ||
100mg | 1.327,00 € | ||
500mg | 2.675,00 € |
Entrega estimada en Estados Unidos, el Lunes 16 de Septiembre de 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Tyrosine kinase-IN-6
CAS:2377507-01-0
Tyrosine kinase-IN-6 is a potent inhibitor of RON splice variants, demonstrating significant anticancer and antineoplastic …
Fórmula:
C37H31F2N5O5S
Pureza:
98%
Peso molecular:
695.73
Ref: TM-T79612
25mg | 1.688,00 € | ||
50mg | 2.225,00 € | ||
100mg | 2.897,00 € |
Entrega estimada en Estados Unidos, el Lunes 16 de Septiembre de 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
YK-029A
CAS:2064269-82-3
YK-029A, an orally active EGFR mutant inhibitor, targets both EGFR T790M and EGFRex20ins mutations. It …
Fórmula:
C27H32N8O2
Pureza:
98%
Peso molecular:
500.6
Ref: TM-T79461
25mg | 1.549,00 € | ||
50mg | 2.038,00 € | ||
100mg | 2.617,00 € |
Entrega estimada en Estados Unidos, el Lunes 16 de Septiembre de 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
ALK/EGFR-IN-1
CAS:2730430-08-5
ALK/EGFR-IN-1 (Compound 8l) is a dual inhibitor targeting both ALK and EGFR, effectively blocking their …
Fórmula:
C27H34ClN7O3S
Pureza:
98%
Peso molecular:
572.12
Ref: TM-T79392
25mg | 1.549,00 € | ||
50mg | 2.038,00 € | ||
100mg | 2.617,00 € |
Entrega estimada en Estados Unidos, el Lunes 16 de Septiembre de 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
FGFR-IN-11
CAS:2658488-68-5
FGFR-IN-11 (compound I-5) is an orally active, covalent inhibitor of FGFR, exhibiting IC50 values of …
Fórmula:
C28H29ClN4O4
Pureza:
98%
Peso molecular:
521.01
Ref: TM-T79257
25mg | 1.688,00 € | ||
50mg | 2.225,00 € | ||
100mg | 2.897,00 € |
Entrega estimada en Estados Unidos, el Lunes 16 de Septiembre de 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
EGFR-IN-85
CAS:1956378-29-2
EGFR-IN-85 (Compound 1), an EGFR inhibitor, exhibits potent activity with an IC50 of 0.19 μM …
Fórmula:
C26H30N8O2
Pureza:
98%
Peso molecular:
486.57
Ref: TM-T78574
25mg | 1.410,00 € | ||
50mg | 1.851,00 € | ||
100mg | 2.337,00 € |
Entrega estimada en Estados Unidos, el Lunes 16 de Septiembre de 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
EGFR-IN-61
CAS:2890261-81-9
EGFR-IN-61 (compound 22a), a potent EGFR kinase inhibitor, exhibits IC50 values of 42 nM for …
Fórmula:
C33H37ClN8O3
Pureza:
98%
Peso molecular:
629.15
Ref: TM-T73128
25mg | 1.410,00 € | ||
50mg | 1.851,00 € | ||
100mg | 2.337,00 € |
Entrega estimada en Estados Unidos, el Lunes 16 de Septiembre de 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Lifirafenib
CAS:1446090-79-4
Lifirafenib (Beigene-283) is a potent inhibitor of RAF family kinases and EGFR in biochemical assays …
Fórmula:
C25H17F3N4O3
Pureza:
98.25%
Forma y color:
Solid
Peso molecular:
478.42
Ref: TM-T22272
1mg | 35,00 € | ||
1ml | 89,00 € | ||
5mg | 68,00 € | ||
10mg | 95,00 € | ||
25mg | 185,00 € | ||
50mg | A consultar | ||
100mg | A consultar |
Entrega estimada en Estados Unidos, el Lunes 16 de Septiembre de 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
VEGFR-2-IN-9
CAS:408502-06-7
VEGFR-2-IN-9 (KDR-in-4) is a potent KDR/VEGFR2 inhibitor (IC50: 7 nM). It can be used to …
Fórmula:
C23H25N3O3
Pureza:
97.19%
Forma y color:
Solid
Peso molecular:
391.46
Ref: TM-T10123
1mg | 650,00 € | ||
5mg | 1.671,00 € |
Entrega estimada en Estados Unidos, el Lunes 16 de Septiembre de 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
IN-1130
CAS:868612-83-3
IN-1130: ALK5 inhibitor, IC50 - 5.3 nM (Smad3), 36 nM (casein), 4.3 μM (p38α MAPK).
Fórmula:
C25H20N6O
Pureza:
98.08%
Forma y color:
Solid
Peso molecular:
420.47
Ref: TM-T15572
1ml | 58,00 € | ||
5mg | 52,00 € | ||
10mg | 90,00 € | ||
25mg | 167,00 € | ||
50mg | 255,00 € | ||
100mg | 368,00 € |
Entrega estimada en Estados Unidos, el Lunes 16 de Septiembre de 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
WAY-600
CAS:1062159-35-6
WAY-600 is a potent, ATP-competitive and selective inhibitor of mTOR with IC50 of 9 nM; …
Fórmula:
C28H30N8O
Pureza:
99.63%
Forma y color:
Solid
Peso molecular:
494.59
Ref: TM-T6730
1mg | 38,00 € | ||
1ml | 111,00 € | ||
2mg | 63,00 € | ||
5mg | 95,00 € | ||
10mg | 138,00 € | ||
25mg | 240,00 € | ||
50mg | 355,00 € | ||
100mg | 495,00 € | ||
500mg | A consultar |
Entrega estimada en Estados Unidos, el Lunes 16 de Septiembre de 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
TG 100572 Hydrochloride
CAS:867331-64-4
TG 100572 Hydrochloride is a inhibitor of multi-targeted kinase which inhibits receptor tyrosine kinases and …
Fórmula:
C26H27Cl2N5O2
Pureza:
98%
Forma y color:
Solid
Peso molecular:
512.43
Ref: TM-T13156L
1mg | 370,00 € |
Entrega estimada en Estados Unidos, el Lunes 16 de Septiembre de 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
PF-06733804
CAS:1873373-33-1
PF-06733804 is a potent inhibitor of pan-Trk in cell-based assays (IC50s: 8.4 nM, 6.2 nM, …
Fórmula:
C20H19F5N4O4
Pureza:
98%
Forma y color:
Solid
Peso molecular:
474.38
Ref: TM-T13207
25mg | 1.688,00 € | ||
50mg | 2.225,00 € | ||
100mg | 2.897,00 € |
Entrega estimada en Estados Unidos, el Lunes 16 de Septiembre de 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Sulfatinib
CAS:1308672-74-3
Sulfatinib (KDR-IN-1) (HMPL-012) is a potent and highly selective tyrosine kinase inhibitor against VEGFR1/2/3, FGFR1 …
Fórmula:
C24H28N6O3S
Pureza:
100%
Forma y color:
Solid
Peso molecular:
480.58
Ref: TM-T4075
1mg | 46,00 € | ||
1ml | 83,00 € | ||
5mg | 78,00 € | ||
10mg | 94,00 € | ||
25mg | 153,00 € | ||
50mg | 224,00 € | ||
100mg | 347,00 € |
Entrega estimada en Estados Unidos, el Lunes 16 de Septiembre de 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
c-met-IN-1
CAS:2084836-84-8
c-met-IN-1 is a potent and selective c-Met inhibitor (IC50: 1.1 nM) with antitumor activity.
Fórmula:
C35H37FN6O5
Pureza:
98%
Forma y color:
Solid
Peso molecular:
640.7
Ref: TM-T10653
25mg | 1.688,00 € | ||
50mg | 2.225,00 € | ||
100mg | 2.897,00 € |
Entrega estimada en Estados Unidos, el Lunes 16 de Septiembre de 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
HKI-357
CAS:848133-17-5
HKI-357 irreversibly inhibits EGFR/ERBB2 (IC50: 34/33 nM), blocks EGFR Y1068 autophosphorylation, and AKT/MAPK phosphorylation.
Fórmula:
C31H29ClFN5O3
Pureza:
98.31%
Forma y color:
Solid
Peso molecular:
574.05
Ref: TM-T11569
1mg | 78,00 € | ||
1ml | 186,00 € | ||
5mg | 149,00 € | ||
10mg | 222,00 € | ||
25mg | 452,00 € | ||
50mg | 647,00 € | ||
100mg | 920,00 € |
Entrega estimada en Estados Unidos, el Lunes 16 de Septiembre de 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Vepafestinib
CAS:2129515-96-2
Vepafestinib is a RET inhibitor with potential antineoplastic activity[1].
Fórmula:
C26H30N6O3
Pureza:
98.54%
Forma y color:
Solid
Peso molecular:
474.55
Ref: TM-T9445
1mg | 153,00 € | ||
1ml | 400,00 € | ||
5mg | 368,00 € | ||
50mg | 1.189,00 € | ||
100mg | 1.613,00 € |
Entrega estimada en Estados Unidos, el Lunes 16 de Septiembre de 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
BMX-IN-1
CAS:1431525-23-3
BMX-IN-1 (BMX kinase inhibitor) is a selective inhibitor of bone marrow tyrosine kinase on chromosome …
Fórmula:
C29H24N4O4S
Pureza:
98%
Forma y color:
Solid
Peso molecular:
524.59
Ref: TM-T14692
1mg | 52,00 € | ||
1ml | 155,00 € | ||
5mg | 123,00 € | ||
10mg | 184,00 € | ||
25mg | 383,00 € | ||
50mg | 537,00 € | ||
100mg | 735,00 € |
Entrega estimada en Estados Unidos, el Lunes 16 de Septiembre de 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Paltimatrectinib
CAS:2353522-15-1
Paltimatrectinib (PBI-200) is a potent tyrosine kinase inhibitor with anticancer activity that inhibits myosin-related kinase …
Fórmula:
C20H15F5N6
Pureza:
99.96%
Forma y color:
Solid
Peso molecular:
434.37
Ref: TM-T62447
1mg | 185,00 € |
Entrega estimada en Estados Unidos, el Lunes 16 de Septiembre de 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
TAK-020
CAS:1627603-21-7
TAK-020 is a potent covalent inhibitor of Btk with potential antitumor activity for the study …
Fórmula:
C18H17N5O3
Pureza:
98.79%
Forma y color:
Solid
Peso molecular:
351.36
Ref: TM-T9529
1mg | 143,00 € | ||
1ml | 375,00 € | ||
5mg | 346,00 € | ||
10mg | 616,00 € | ||
25mg | 1.277,00 € | ||
50mg | 1.977,00 € | ||
100mg | 3.044,00 € |
Entrega estimada en Estados Unidos, el Lunes 16 de Septiembre de 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
EGFR-IN-1 hydrochloride
CAS:2227455-78-7
EGFR-IN-1 HCl targets L858R/T790M EGFR mutants over wild-type; IC50: 4 nM in H1975, 28 nM …
Fórmula:
C28H31ClN6O4
Pureza:
99.8%
Forma y color:
Solid
Peso molecular:
551.04
Ref: TM-T11157L
1mg | 95,00 € | ||
1ml | 335,00 € | ||
5mg | 238,00 € | ||
10mg | 352,00 € | ||
25mg | 550,00 € | ||
50mg | 737,00 € | ||
100mg | 1.012,00 € | ||
500mg | 2.033,00 € |
Entrega estimada en Estados Unidos, el Lunes 16 de Septiembre de 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
AZ-23
CAS:915720-21-7
AZ-23 is an inhibitor of ATP-competitive and Trk kinase A/B/C. For TrkA, TrkB, FGFR1, Flt3, …
Fórmula:
C17H19ClFN7O
Pureza:
99.4%
Forma y color:
Solid
Peso molecular:
391.83
Ref: TM-T14363
1mg | 96,00 € |
Entrega estimada en Estados Unidos, el Lunes 30 de Septiembre de 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
HM43239
CAS:2294874-49-8
HM43239: oral FLT3 inhibitor; IC50: FLT3 WT 1.1nM, ITD 1.8nM, D835Y 1.0nM; blocks p-STAT5/p-ERK; affects …
Fórmula:
C29H33ClN6
Pureza:
98.56%
Forma y color:
Solid
Peso molecular:
501.07
Ref: TM-T9428
1mg | 69,00 € | ||
1ml | 186,00 € | ||
5mg | 150,00 € | ||
10mg | 221,00 € | ||
25mg | 434,00 € | ||
50mg | 620,00 € | ||
100mg | 862,00 € |
Entrega estimada en Estados Unidos, el Lunes 30 de Septiembre de 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Vecabrutinib
CAS:1510829-06-7
Vecabrutinib (SNS-062) is a potent and noncovalent BTK and ITK inhibitor (Kd: 0.3 nM and …
Fórmula:
C22H24ClF4N7O2
Pureza:
100%
Forma y color:
Solid
Peso molecular:
529.92
Ref: TM-T17220
1mg | 85,00 € | ||
1ml | 218,00 € | ||
5mg | 183,00 € | ||
10mg | 300,00 € | ||
25mg | 487,00 € | ||
50mg | 646,00 € | ||
100mg | 905,00 € |
Entrega estimada en Estados Unidos, el Martes 15 de Octubre de 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Tyk2-IN-3
CAS:1779493-12-7
Tyk2-IN-3 is an inhibitor of Tyk2 pseudokinase (IC50: 485 nM).
Fórmula:
C25H24N6O3S2
Pureza:
98%
Forma y color:
Solid
Peso molecular:
520.63
Ref: TM-T13233
25mg | 2.384,00 € | ||
50mg | 3.159,00 € | ||
100mg | 4.299,00 € |
Entrega estimada en Estados Unidos, el Martes 15 de Octubre de 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
PLX5622 hemifumarate
PLX5622 hemifumarate: selective CSF1R inhibitor (IC50: 0.016 μM, Ki: 5.9 nM), brain-penetrant, oral, clears microglia …
Fórmula:
C25H23F2N5O5
Pureza:
98%
Forma y color:
Solid
Peso molecular:
453.45
Ref: TM-T12505
200mg | 1.092,00 € |
Entrega estimada en Estados Unidos, el Martes 15 de Octubre de 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
GENZ-882706
CAS:2070864-35-4
GENZ-882706 is a potent colony stimulating factor-1 receptor (CSF-1R) Inhibitor.
Fórmula:
C26H25N5O3
Pureza:
98%
Forma y color:
Solid
Peso molecular:
455.51
Ref: TM-T11390
25mg | 1.976,00 € | ||
50mg | 2.588,00 € | ||
100mg | 4.152,00 € |
Entrega estimada en Estados Unidos, el Martes 15 de Octubre de 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
c-Met-IN-2
CAS:1635406-73-3
c-Met-IN-2 is a selective and orally available c-Met inhibitor (IC50: 0.6 nM) with antitumor activity.
Fórmula:
C24H21FN10O
Pureza:
98%
Forma y color:
Solid
Peso molecular:
484.49
Ref: TM-T10654
25mg | 2.106,00 € | ||
50mg | 2.785,00 € | ||
100mg | 3.739,00 € |
Entrega estimada en Estados Unidos, el Martes 15 de Octubre de 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
c-Kit-IN-5-1
CAS:1003311-62-3
c-Kit-IN-5-1 (AMG-25) is a novel selective and potent c-Kit inhibitor.
Fórmula:
C23H17N5O2
Pureza:
98%
Forma y color:
Solid
Peso molecular:
395.41
Ref: TM-T22256
25mg | 1.373,00 € | ||
50mg | 1.786,00 € | ||
100mg | 2.713,00 € |
Entrega estimada en Estados Unidos, el Martes 15 de Octubre de 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
(-)-Cevimeline hydrochloride hemihydrate
(-)-Cevimeline HCl hemihydrate, a muscarinic agonist, treats Sjogren's xerostomia. Quick absorption, species-dependent metabolism.
Fórmula:
C10H19ClNO1·5S
Pureza:
98%
Forma y color:
Solid
Peso molecular:
244.78
Ref: TM-T13421
25mg | 3.673,00 € |
Entrega estimada en Estados Unidos, el Martes 15 de Octubre de 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
VEGFR2-IN-1
CAS:2765224-55-1
VEGFR2-IN-1 is a VEGFR2 inhibitor with antitumor activity used in the study of breast cancer.
Fórmula:
C22H18N6S
Pureza:
98.06%
Forma y color:
Solid
Peso molecular:
398.48
Ref: TM-T61899
1mg | 277,00 € | ||
5mg | 683,00 € | ||
10mg | 933,00 € | ||
25mg | 1.442,00 € | ||
50mg | 1.878,00 € | ||
100mg | 2.371,00 € |
Entrega estimada en Estados Unidos, el Martes 15 de Octubre de 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
BMS-066
CAS:914946-88-6
BMS-066 is an IKKβ/Tyk2 pseudokinase inhibitor. With IC50s of 9 nM and 72 nM, respectively.
Fórmula:
C19H21N7O2
Pureza:
98%
Forma y color:
Solid
Peso molecular:
379.42
Ref: TM-T14669
25mg | 2.245,00 € | ||
50mg | 2.972,00 € | ||
100mg | 4.019,00 € |
Entrega estimada en Estados Unidos, el Martes 15 de Octubre de 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
TAS05567
CAS:1429038-15-2
TAS05567 is a potent, highly selective, and ATP-competitive Syk inhibitor (IC50: 0.37 nM).
Fórmula:
C21H29N9O2
Pureza:
98%
Forma y color:
Solid
Peso molecular:
439.51
Ref: TM-T16995
25mg | 2.106,00 € | ||
50mg | 2.785,00 € | ||
100mg | 3.739,00 € |
Entrega estimada en Estados Unidos, el Martes 15 de Octubre de 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
G-744
CAS:1346669-54-2
G-744 is a selective and orally active inhibitor of Btk (IC50: 2 nM).
Fórmula:
C29H29N5O3S
Pureza:
98%
Forma y color:
Solid
Peso molecular:
527.64
Ref: TM-T15365
25mg | 2.662,00 € | ||
50mg | 3.533,00 € | ||
100mg | 4.860,00 € |
Entrega estimada en Estados Unidos, el Martes 15 de Octubre de 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
DYRKs-IN-1
CAS:1387090-01-8
DYRKs-IN-1 has antitumor activity.
Fórmula:
C30H30ClN7O4
Pureza:
98%
Forma y color:
Solid
Peso molecular:
588.06
Ref: TM-T11132
25mg | 2.662,00 € | ||
50mg | 3.533,00 € | ||
100mg | 4.860,00 € |
Entrega estimada en Estados Unidos, el Martes 15 de Octubre de 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
AZ12601011
CAS:2748337-86-0
AZ12601011 is a highly potent and selective inhibitor of the TGFBR1 kinase, administered orally. It …
Fórmula:
C19H15N5
Pureza:
98%
Forma y color:
Solid
Peso molecular:
313.36
Ref: TM-T10426
25mg | 914,00 € | ||
50mg | 1.197,00 € | ||
100mg | 1.665,00 € |
Entrega estimada en Estados Unidos, el Martes 15 de Octubre de 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
FGFR4-IN-4
CAS:2230973-67-6
FGFR4-IN-4 is a FGFR4 inhibitor with anti-tumor activity.
Fórmula:
C28H32Cl2N6O5
Pureza:
98%
Forma y color:
Solid
Peso molecular:
603.5
Ref: TM-T11280
25mg | 2.801,00 € | ||
50mg | 3.720,00 € | ||
100mg | 5.140,00 € |
Entrega estimada en Estados Unidos, el Martes 15 de Octubre de 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
PF-06273340
CAS:1402438-74-7
PF-06273340: selective pan-Trk inhibitor (IC50: Trk-A 6 nM, B 4 nM, C 3 nM), low …
Fórmula:
C23H22ClN7O3
Pureza:
98.00%
Forma y color:
Solid
Peso molecular:
479.92
Ref: TM-T19649
1mg | 53,00 € | ||
25mg | A consultar | ||
50mg | A consultar |
Entrega estimada en Estados Unidos, el Martes 15 de Octubre de 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Protopine hydrochloride
CAS:6164-47-2
Protopine inhibits thromboxane, lowers intracellular calcium, and reduces cell adhesion by altering adhesive factors.
Fórmula:
C20H20ClNO5
Pureza:
98%
Forma y color:
Prisms From Alc Solid
Peso molecular:
389.83
Ref: TM-TMA1944
1mg | 394,00 € | ||
500µg | 221,00 € |
Entrega estimada en Estados Unidos, el Martes 15 de Octubre de 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Ref: AN-AG007LZB
5mg | Descatalogado | Solicitar información | |
25mg | Descatalogado | Solicitar información | |
100mg | Descatalogado | Solicitar información |
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Unii-33Y9anm545
CAS:635702-64-6
Fórmula:
C21H24ClN7O2S
Pureza:
99%
Forma y color:
Solid
Peso molecular:
473.9790
Ref: AN-AG00E9EW
1g | Descatalogado | Solicitar información | |
5g | Descatalogado | Solicitar información | |
10g | Descatalogado | Solicitar información | |
100mg | Descatalogado | Solicitar información | |
250mg | Descatalogado | Solicitar información |
![discount label](https://static.cymitquimica.com/public/img/discount.png)
2-Propenethioamide, 3-[3,5-bis(1,1-dimethylethyl)-4-hydroxyphenyl]-2-cyano-, (2E)-
CAS:148741-30-4
Fórmula:
C18H24N2OS
Pureza:
95%
Forma y color:
Solid
Peso molecular:
316.4610
Ref: AN-AG001L5Z
100mg | Descatalogado | Solicitar información | |
250mg | Descatalogado | Solicitar información |
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Ref: AN-AG007R3D
1g | Descatalogado | Solicitar información | |
10mg | Descatalogado | Solicitar información | |
100mg | Descatalogado | Solicitar información | |
250mg | Descatalogado | Solicitar información |
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Ref: AN-AG00AP0L
1g | Descatalogado | Solicitar información | |
5mg | Descatalogado | Solicitar información | |
10mg | Descatalogado | Solicitar información | |
25mg | Descatalogado | Solicitar información | |
50mg | Descatalogado | Solicitar información | |
100mg | Descatalogado | Solicitar información | |
250mg | Descatalogado | Solicitar información |
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Ref: AN-AG01DU9U
1mg | Descatalogado | Solicitar información | |
2mg | Descatalogado | Solicitar información | |
5mg | Descatalogado | Solicitar información | |
10mg | Descatalogado | Solicitar información | |
25mg | Descatalogado | Solicitar información | |
50mg | Descatalogado | Solicitar información | |
100mg | Descatalogado | Solicitar información | |
250mg | Descatalogado | Solicitar información |
![discount label](https://static.cymitquimica.com/public/img/discount.png)
4-Quinazolinamine, N-(3-bromophenyl)-6,7-dimethoxy-, hydrochloride (1:1)
CAS:183322-45-4
Fórmula:
C16H15BrClN3O2
Pureza:
98%
Forma y color:
Solid
Peso molecular:
396.6662
Ref: AN-AG0027IO
10mg | Descatalogado | Solicitar información | |
50mg | Descatalogado | Solicitar información | |
250mg | Descatalogado | Solicitar información |
![discount label](https://static.cymitquimica.com/public/img/discount.png)
N-[3-Chloro-4-[(3-fluorophenyl)methoxy]phenyl]-6-[5-[[[2-(methylsulfonyl)ethyl]amino]methyl]-2-furanyl]-4-quinazolinamine
CAS:231277-92-2
Fórmula:
C29H26ClFN4O4S
Pureza:
99%
Forma y color:
Solid
Peso molecular:
581.0575
Ref: AN-AG0039KT
1g | Descatalogado | Solicitar información | |
5g | Descatalogado | Solicitar información | |
25g | Descatalogado | Solicitar información | |
25mg | Descatalogado | Solicitar información | |
250mg | Descatalogado | Solicitar información |
![discount label](https://static.cymitquimica.com/public/img/discount.png)
4-[4-[[[[4-Chloro-3-(trifluoromethyl)phenyl]amino]carbonyl]amino]phenoxy]-N-methyl-2-pyridinecarboxamide
CAS:284461-73-0
Fórmula:
C21H16ClF3N4O3
Pureza:
99%
Forma y color:
Solid
Peso molecular:
464.8249
Ref: AN-AG0039KS
1g | Descatalogado | Solicitar información | |
5g | Descatalogado | Solicitar información | |
25g | Descatalogado | Solicitar información |
![discount label](https://static.cymitquimica.com/public/img/discount.png)
1,3-Benzodioxole, 5-(2-nitroethenyl)-
CAS:1485-00-3
Fórmula:
C9H7NO4
Pureza:
98%
Forma y color:
Solid
Peso molecular:
193.1562
Ref: AN-AG001KYU
1g | Descatalogado | Solicitar información | |
5g | Descatalogado | Solicitar información | |
25g | Descatalogado | Solicitar información | |
250mg | Descatalogado | Solicitar información |
![discount label](https://static.cymitquimica.com/public/img/discount.png)
(2E)-N-[4-[[3-Chloro-4-(2-pyridinylmethoxy)phenyl]amino]-3-cyano-7-ethoxy-6-quinolinyl]-4-(dimethylamino)-2-butenamide
CAS:698387-09-6
Fórmula:
C30H29ClN6O3
Pureza:
98%
Forma y color:
Solid
Peso molecular:
557.0427
Ref: AN-AG0035DM
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Tamaño no definido | Descatalogado | Solicitar información | |
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Ref: AN-AG00GU50
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Ref: AN-AG003MZ1
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Propanedinitrile,2-[(3,4-dihydroxyphenyl)methylene]-
CAS:118409-57-7
Fórmula:
C10H6N2O2
Pureza:
98%
Forma y color:
Solid
Peso molecular:
186.1668
Ref: AN-AG007QB5
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CHMFL-ABL-121
CAS:2270879-07-5
CHMFL-ABL-121 is a highly potent inhibitor of type II ABL kinase (IC50s: 2 nM and …
Fórmula:
C30H31F3N6OS
Pureza:
99.86%
Forma y color:
Solid
Peso molecular:
580.67
Ref: TM-T10800
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Teprotumumab
CAS:1036734-93-6
Teprotumumab is a human monoclonal antibody that blocks the IGF-1 receptor (IGF-1R). Teprotumumab binds to …
Forma y color:
Solid
Ref: TM-T76727
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CHMFL-ABL-039
CAS:2304344-56-5
CHMFL-ABL-039 is a type II native ABL kinase and drug-resistant V299L mutant BCR-ABL inhibitor (IC50s: …
Fórmula:
C31H33F3N6O3
Pureza:
98.63%
Forma y color:
Solid
Peso molecular:
594.63
Ref: TM-T10799
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CHMFL-FLT3-122
CAS:1839150-56-9
CHMFL-FLT3-122 is a potent and orally available FLT3 kinase inhibitor used to treat FLT3-ITD positive …
Fórmula:
C26H29N7O2
Pureza:
99.56%
Forma y color:
Solid
Peso molecular:
471.55
Ref: TM-T27011
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CHMFL-KIT-033
CAS:2351801-41-5
CHMFL-KIT-033 is an effective and selective c-KIT inhibitor with an IC50 value of 45 nM …
Fórmula:
C23H18FN5O2
Pureza:
97.26%
Forma y color:
Solid
Peso molecular:
415.42
Ref: TM-T10803
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Bosutinib D8
Bosutinib D8 is a deuterium-labeled Bosutinib. Bosutinib (SKI-606) is a dual Src/Abl inhibitor (IC50s: 1.2 …
Fórmula:
C26H21D8Cl2N5O3
Pureza:
98%
Forma y color:
Solid
Peso molecular:
538.5
Ref: TM-T10583
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