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Tirosina quinasa / adaptadores

Tirosina quinasa / adaptadores

Los inhibidores de tirosina quinasa y adaptadores son compuestos que se dirigen a las tirosina quinasas y sus proteínas adaptadoras asociadas, las cuales desempeñan roles cruciales en la señalización celular, el crecimiento y la diferenciación. Estos inhibidores son herramientas esenciales en la investigación del cáncer, ya que muchas tirosina quinasas están involucradas en las vías de señalización que impulsan el crecimiento tumoral y la metástasis. Al inhibir las tirosina quinasas, estos compuestos pueden bloquear cascadas de señalización críticas, ofreciendo potenciales estrategias terapéuticas para varios tipos de cáncer y otras enfermedades que implican una señalización celular anormal. En CymitQuimica, ofrecemos una amplia gama de inhibidores de tirosina quinasa y adaptadores de alta calidad para apoyar su investigación en oncología, biología molecular y desarrollo de terapias dirigidas.

Subcategorías de "Tirosina quinasa / adaptadores"

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Se han encontrado 1342 productos de "Tirosina quinasa / adaptadores"

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  • Logo de CymitQuimica
    Targetmol
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    EGFR-IN-42

    <p>EGFR-IN-42 (17b) is a potent EGFR inhibitor with nanomolar efficacy, merging tamoxifen/endoxifen and gefitinib, exhibiting enhanced anti-cancer action.</p>
    Fórmula:C49H53ClFN5O5
    Forma y color:Solid
    Peso molecular:846.43

    Ref: TM-T74457

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    VEGFR-2-IN-55

    <p>VEGFR-2-IN-55 (Compound 30) is an effective VEGFR-2 kinase inhibitor with an IC50 of 1.24 nM and exhibits anti-tumor activity.</p>
    Forma y color:Odour Solid

    Ref: TM-T200578

  • GIP (1-30) amide,human
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    GIP (1-30) amide,human

    CAS:
    GIP (1-30) amide (Human) is a glucose-dependent insulinotropic polypeptide that stimulates insulin secretion, reducing postprandial glycemic issues.
    Fórmula:C162H240N40O47S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:3531.94

    Ref: TM-TP1584

  • Lyso-Monosialoganglioside GM3
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    Lyso-Monosialoganglioside GM3

    CAS:
    <p>Lyso-Monosialoganglioside GM3 (Lyso-GM3) is an analog of Ganglioside GM3 with antitumor properties. It inhibits the increase in EGFR kinase activity induced by EGF in A431 epithelial cancer cells.</p>
    Fórmula:C41H74N2O20
    Forma y color:Solid
    Peso molecular:915.028

    Ref: TM-T206584

  • MC-Val-Cit-PAB-Amide-TLR7 agonist 4 Conjugate
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    MC-Val-Cit-PAB-Amide-TLR7 agonist 4 Conjugate

    CAS:
    <p>MC-Val-Cit-PAB-Amide-TLR7 agonist 4 Conjugate is a conjugate formed by linking MC-Val-Cit-PAB-Amide and TLR7 agonist 4, useful for cancer research.</p>
    Fórmula:C52H72N12O11
    Pureza:97.70%
    Forma y color:Solid
    Peso molecular:1041.2

    Ref: TM-T74468

  • SJF 1528
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    SJF 1528

    CAS:
    <p>Potent EGFR &amp; HER2 degrader; DC50 of 39.2 nM in OVCAR8, 736 nM in HeLa; has lapatinib, VHL ligand; inhibits HER2+ breast cancer (IC50=102 nM for SKBr3).</p>
    Fórmula:C55H57ClFN7O8S
    Forma y color:Solid
    Peso molecular:1030.61

    Ref: TM-T36245

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    Acetyl Gastric Inhibitory Peptide (human)

    CAS:
    Acetyl Gastric Inhibitory Peptide: improved insulinotropic, antihyperglycemic, for diabetes/obesity research.
    Fórmula:C228H340N60O67S
    Forma y color:Solid
    Peso molecular:5025.6

    Ref: TM-T76310

  • MS9427
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    MS9427

    CAS:
    <p>MS9427: PROTAC EGFR degrader, 7.1 nM (WT), 4.3 nM (L858R); targets mutant via UPS and autophagy; inhibits NSCLC cell growth; anticancer research.</p>
    Fórmula:C48H58ClFN8O12
    Forma y color:Solid
    Peso molecular:993.47

    Ref: TM-T74633

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    DSPE-PEG2000-GE11

    <p>DSPE-PEG2000-GE11 is a PEG compound composed of DSPE and an EGFR-targeting peptide (GE11). GE11 is applicable for cancer cells that overexpress EGFR. DSPE-PEG2000-GE11 is utilized in drug delivery.</p>
    Forma y color:Odour Solid

    Ref: TM-TCL-01177

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    Cixutumumab

    CAS:
    <p>Cixutumumab (IMC-A12), a humanized monoclonal antibody targeting IGF-1R, exhibits high affinity and inhibits ligand-dependent receptor activation, impeding</p>
    Pureza:98.5% (SDS-PAGE); 97.5% (SEC-HPLC) - 98.5% (SDS-PAGE); 97.5% (SEC-HPLC)
    Forma y color:Liquid

    Ref: TM-T78279

  • HER2/neu (654-662) GP2
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    HER2/neu (654-662) GP2

    CAS:
    <p>Phage display selected Affibody ligands for HER2/neu from a protein library based on a 58-residue Staphylococcal protein A Z domain.</p>
    Fórmula:C42H77N9O11
    Pureza:98%
    Forma y color:Solid
    Peso molecular:884.11

    Ref: TM-TP1583

  • PKG inhibitor peptide
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    PKG inhibitor peptide

    CAS:
    <p>PKG inhibitor; mimics H2B phosphorylation site; Ki=86mM; blocks synthetic substrates, not histone phosphorylation; stops PKA activity on histones.</p>
    Fórmula:C38H74N18O10
    Pureza:98%
    Forma y color:Solid
    Peso molecular:943.12

    Ref: TM-TP1903

  • Tyrosine Kinase Inhibitor Library
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    Tyrosine Kinase Inhibitor Library

    <p>A unique collection of 1016 tyrosine kinase inhibitors for high throughput screening and high content screening for drug discovery in tyrosine kinase related</p>
    Forma y color:Odour Solid

    Ref: TM-L2200

  • CLK1-IN-3
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    CLK1-IN-3

    CAS:
    <p>Clk1-in-3 is a + selective and highly potent sexual Clk1 inhibitor with an IC50 of 5 nM and 300 pairs higher affinity than Dyrk1A.</p>
    Fórmula:C24H23FN6O
    Pureza:98.46% - 99.76%
    Forma y color:Soild
    Peso molecular:430.48

    Ref: TM-T72039

  • BMS-599626
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    BMS-599626

    CAS:
    <p>BMS-599626 (AC480) has been used in trials studying the treatment of Cancer, Metastases, and HER2 or EGFR Expressing Advanced Solid Malignancies.</p>
    Fórmula:C27H27FN8O3
    Pureza:98.73%
    Forma y color:Solid
    Peso molecular:530.55

    Ref: TM-T2610

  • ALKBH5-IN-5
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    ALKBH5-IN-5

    CAS:
    <p>ALKBH5-IN-5 is a highly selective, potent and covalently binding ALKBH5 inhibitor that alters m6A levels on mRNA, induces apoptosis, antitumo.</p>
    Fórmula:C13H13NO3
    Pureza:99.54%
    Forma y color:Soild
    Peso molecular:231.25

    Ref: TM-T203011

  • Varlitinib
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    Varlitinib

    CAS:
    Varlitinib (ASLAN001) is a potent, reversible, small molecule pan-EGFR inhibitor with IC50s of 7, 2, 4 nM for HER1, HER2 and HER4, respectively.
    Fórmula:C22H19ClN6O2S
    Pureza:99.7%
    Forma y color:Solid
    Peso molecular:466.94

    Ref: TM-T6719

  • IGF-I (24-41)
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    IGF-I (24-41)

    CAS:
    <p>IGF-I (24-41) is a fragment of IGF-I, affecting GH activities with anabolic, antioxidant, anti-inflammatory, and cytoprotective properties.</p>
    Fórmula:C88H133N27O28
    Pureza:98%
    Forma y color:Solid
    Peso molecular:2017.16

    Ref: TM-TP1124

  • JAK 3 inhibitor IV
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    JAK 3 inhibitor IV

    CAS:
    <p>JAK 3 inhibitor IV (ZM 39923 hydrochloride) is a JAK1/3 inhibitor with pIC50 of 4.4/7.1, almost no activity to JAK2 and modestly potent to EGFR; also found to</p>
    Fórmula:C16H19NO
    Pureza:98%
    Forma y color:Solid
    Peso molecular:241.33

    Ref: TM-T2460

  • KYL peptide
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    KYL peptide

    CAS:
    EphA4 inhibitor, Kd 0.8 μM, blocks EphA4-EphrinA5; avoids AβO damage, preserves spines & LTP; long half-life (8-12h), neuroprotective.
    Fórmula:C74H108N14O17
    Pureza:98%
    Forma y color:Solid
    Peso molecular:1465.75

    Ref: TM-TP1895