
Apoptose
Les inhibiteurs de l'apoptose sont des composés qui empêchent ou retardent le processus de mort cellulaire programmée, connu sous le nom d'apoptose. Ces inhibiteurs sont essentiels pour étudier les mécanismes de survie cellulaire et sont utilisés pour enquêter sur les maladies où l'apoptose est dysrégulée, telles que le cancer, les troubles neurodégénératifs et les maladies auto-immunes. En modulant l'apoptose, ces inhibiteurs peuvent aider au développement de thérapies visant à contrôler la mort cellulaire. Chez CymitQuimica, nous offrons une sélection complète d'inhibiteurs de l'apoptose de haute qualité pour soutenir vos recherches en biologie cellulaire, oncologie et domaines connexes.
Sous-catégories appartenant à la catégorie "Apoptose"
- ASK(6 produits)
- BCL(11 produits)
- Caspase(125 produits)
- FOXO1(3 produits)
- IAP(66 produits)
- Mdm2(12 produits)
- PD-1/PD-L1(125 produits)
- PDK(9 produits)
- PERK(25 produits)
- Sérine/thréonine kinase(15 produits)
- Survivant(13 produits)
- TNF(92 produits)
- c-RET(51 produits)
- p53(62 produits)
Affichez 6 plus de sous-catégories
5592 produits trouvés pour "Apoptose"
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α-Lipoic Acid sodium
CAS :<p>α-Lipoic Acid (Thioctic acid) sodium, an essential cofactor for mitochondrial enzyme complexes, serves as an antioxidant.</p>Formule :C8H13NaO2S2Couleur et forme :SolidMasse moléculaire :228.31Quinidine
CAS :<p>Quinidine is a stereoisomer of the antimalarial agent quinine and a class Ia antiarrhythmic agent. for the treatment of abnormal heart rhythms and also malaria.</p>Formule :C20H24N2O2Degré de pureté :97.03% - 99.99%Couleur et forme :Crystals With 2 5 Mol Water Of Crystallization; Crystals From Dilute Alcohol Physical Description Crystals Or White Powder (Ntp 1992)Masse moléculaire :324.423-hydroxy-3-phenylpentanamide
CAS :<p>Chiral 3-hydroxy-3-phenylpentanamide: neuroprotective, may treat anxiety/depression/addiction, anticancer.</p>Formule :C11H15NO2Degré de pureté :98.42%Couleur et forme :SolidMasse moléculaire :193.24Fimepinostat
CAS :<p>Fimepinostat (CUDC 907) is an orally bioavailable inhibitor of both PI3K class I and pan-HDAC enzymes, with potential antineoplastic activity.</p>Formule :C23H24N8O4SDegré de pureté :98.27% - 99.87%Couleur et forme :SolidMasse moléculaire :508.55HX 531
CAS :<p>HX 531 is a RXR antagonist (IC50 of 18 nM).Cost-effective and quality-assured.</p>Formule :C29H29N3O4Degré de pureté :98.59% - 99.86%Couleur et forme :SolidMasse moléculaire :483.56Sodium benzoate
CAS :<p>Sodium benzoate (Benzoic acid sodium salt) is a D-Amino Acid Oxidase Inhibitor.Sodium Benzoate is a Food Preservative.</p>Formule :C7H5NaO2Degré de pureté :99.72%Couleur et forme :White Solid CrystallineMasse moléculaire :144.10Clodronic acid disodium salt
CAS :<p>Clodronic acid disodium salt (Lodronate), a bisphosphonate, is a potent antiosteolytic agent which inhibits bone resorption.</p>Formule :CH4Cl2O6P0·2NaDegré de pureté :>99.99% - ≥98%Couleur et forme :White SolidMasse moléculaire :288.86RH01687
CAS :<p>RH01687 is a potent β-cell protector , exhibits β-cell-protective activities against endoplasmic reticulum (ER) stress.</p>Formule :C12H9ClN6O2SDegré de pureté :97.93%Couleur et forme :SolidMasse moléculaire :336.76Perifosine
CAS :<p>Perifosine (KRX-0401) is an oral-active, alkyl-phosphocholine Akt inhibitor with potential antineoplastic activity.</p>Formule :C25H52NO4PDegré de pureté :99.94% - >99.99%Couleur et forme :SolidMasse moléculaire :461.66Lubiprostone
CAS :<p>Lubiprostone (RU-0211), an activator of ClC-2 chloride channels, is used in the therapy of idiopathic chronic constipation.</p>Formule :C20H32F2O5Degré de pureté :97.31% - 98.54%Couleur et forme :White Odorless Crystals Or Crystalline PowderMasse moléculaire :390.464-IBP
CAS :<p>4-IBP is a selective σ1 agonist with a high level of affinity for the σ1 receptor (Ki = 1.7 nM) and a moderate affinity for the σ2 receptor (Ki = 25.2 nM) .</p>Formule :C19H21IN2ODegré de pureté :98.99%Couleur et forme :SolidMasse moléculaire :420.29Tenilsetam
CAS :<p>Tenilsetam: an endonuclease, nootropic, AGE inhibitor potential for Alzheimer's.</p>Formule :C8H10N2OSDegré de pureté :99.52%Couleur et forme :SolidMasse moléculaire :182.24Ferrostatin-1
CAS :<p>Ferrostatin-1 (Fer-1) is a potent and selective inhibitor of iron death, potently inhibits Erastin-induced iron death in HT-1080 cells. High-Quality, Low-Cost!</p>Formule :C15H22N2O2Degré de pureté :96.1% - 99.68%Couleur et forme :SolidMasse moléculaire :262.35Rosiglitazone potassium
CAS :<p>Rosiglitazone (BRL 49653) is an oral PPARγ agonist (EC50: 60 nM), TRPC5 activator (EC50: 30 μM), and TRPM3 inhibitor, used in obesity and diabetes research.</p>Formule :C18H18KN3O3SCouleur et forme :SolidMasse moléculaire :395.52Saquinavir
CAS :<p>Saquinavir (Ro 31-8959) is a potent HIV protease inhibitor, is an antiretroviral drug used together with other medications to treat or prevent HIV/AIDS.</p>Formule :C38H50N6O5Degré de pureté :99.50% - >99.99%Couleur et forme :SolidMasse moléculaire :670.84L524-0366
CAS :<p>L524-0366 ([1-(3-chlorophenyl)triazol-4-yl]-thiomorpholino-methanone) is a TWEAK-Fn14 signaling cascade inhibitor.</p>Formule :C13H13ClN4OSDegré de pureté :98.6% - 99.13%Couleur et forme :SolidMasse moléculaire :308.79PX-12
CAS :<p>PX-12, a Trx-1 inhibitor, promotes apoptosis, reduces HIF-1α/VEGF, and inhibits tumor growth, suggesting use in advanced cancer therapy.</p>Formule :C7H12N2S2Degré de pureté :98% - 99.21%Couleur et forme :SolidMasse moléculaire :188.31Vandetanib trifluoroacetate
CAS :<p>Vandetanib trifluoroacetate: oral VEGFR2/KDR inhibitor, IC50=40nM, also blocks VEGFR3/FLT4 (110nM) and EGFR/HER1 (500nM).</p>Formule :C24H25BrF4N4O4Couleur et forme :SolidMasse moléculaire :589.386Sulindac sodium
CAS :<p>Sulindac (sodium) (MK-231) is an NSAID used for arthritis pain, swelling, gout, and as an immunomodulator in CRC therapy.</p>Formule :C20H16FNaO3SCouleur et forme :SolidMasse moléculaire :378.39PYR-41
CAS :<p>PYR-41 is the first cell-permeable inhibitor of ubiquitin-activating enzyme E1, with no activity at E2.</p>Formule :C17H13N3O7Degré de pureté :98.25%Couleur et forme :SolidMasse moléculaire :371.3Fenobam hydrate
CAS :<p>Fenobam hydrate blocks mGluR5, preventing calcium mobilization, and may reduce stress, anxiety, and pain.</p>Formule :C11H13ClN4O3Couleur et forme :SolidMasse moléculaire :284.7Romidepsin
CAS :<p>Romidepsin (NSC-630176), an IV histone deacetylase inhibitor, treats refractory cutaneous/peripheral T-cell lymphomas.</p>Formule :C24H36N4O6S2Degré de pureté :99.4% - 99.94%Couleur et forme :SolidMasse moléculaire :540.7Paroxetine
CAS :<p>Paroxetine is a inhibitor of serotonin uptake that is effective in the treatment of depression.</p>Formule :C19H20FNO3Degré de pureté :98.89% - 99.45%Couleur et forme :White To Off-White PowderMasse moléculaire :329.37Benidipine
CAS :<p>Benidipine: potent oral calcium blocker, boosts nitric oxide synthase, enhances coronary flow, protects heart cells post-ischemia.</p>Formule :C28H31N3O6Couleur et forme :SolidMasse moléculaire :505.56TASIN-1 Hydrochloride
CAS :<p>TASIN-1 Hydrochloride (TASIN-1 HCl) is a selective inhibitor of truncated APC that acts by selectively killing colorectal cancer cells that express truncated</p>Formule :C18H29ClN2O3SDegré de pureté :99.94%Couleur et forme :SolidMasse moléculaire :388.95Panobinostat lactate
CAS :<p>Panobinostat lactate: potent, non-selective, oral HDAC inhibitor; treats refractory multiple myeloma.</p>Formule :C24H29N3O5Couleur et forme :SolidMasse moléculaire :439.512Topotecan hydrochloride hydrate
CAS :<p>Orally active Topotecan HCl hydrate inhibits Topoisomerase I, blocks G0/G1 & S phases, and induces apoptosis.</p>Formule :C23H26ClN3O6Couleur et forme :SolidMasse moléculaire :475.93NVP-ADW742
CAS :<p>NVP-ADW742 (ADW) is an IGF-1R inhibitor with IC50 of 0.17 μM, >16-fold more potent against IGF-1R than InsR; little activity to HER2, PDGFR, VEGFR-2, Bcr-Abl</p>Formule :C28H31N5ODegré de pureté :96.14% - 98.70%Couleur et forme :SolidMasse moléculaire :453.58Oprozomib
CAS :<p>Oprozomib inhibits 20S proteasome β5/LMP7, is orally available, and may have cancer-fighting properties. IC50: β5 - 36 nM; LMP7 - 82 nM.</p>Formule :C25H32N4O7SDegré de pureté :98% - 99.87%Couleur et forme :SolidMasse moléculaire :532.61Ivachtin
CAS :<p>Ivachtin (Caspase-3 Inhibitor VII) is a nonpeptide, noncompetitive and reversibl caspase-3 inhibitor(IC50 = 23 nM) and is a modest inhibitor of the remaining</p>Formule :C20H21N3O7SDegré de pureté :99.74%Couleur et forme :SolidMasse moléculaire :447.46Afimetoran
CAS :<p>Afimetoran (BMS-986256) is a toll-like receptor antagonist. Afimetoran can be used in the research of inflammatory and autoimmune diseases.</p>Formule :C26H32N6ODegré de pureté :99.81% - 99.94%Couleur et forme :SolidMasse moléculaire :444.57Candesartan Cilexetil
CAS :<p>Candesartan Cilexetil, an angiotensin II blocker (IC50: 0.26 nM), turns to candesartan in the body, which dilates blood vessels by hindering AT1.</p>Formule :C33H34N6O6Degré de pureté :98.22% - >99.99%Couleur et forme :White Crystalline PowderMasse moléculaire :610.66AZD1208 hydrochloride
CAS :<p>AZD1208 hydrochloride is a highly selective, potent and orally active PIM inhibitor.</p>Formule :C21H22ClN3O2SCouleur et forme :SolidMasse moléculaire :415.94CCPA
CAS :<p>CCPA (2-chloro-N(6)cyclopentyladenosine) is a potent and selective agonist of adenosine A1 receptor</p>Formule :C15H20ClN5O4Degré de pureté :99.1%Couleur et forme :Off-White To Light Yellow SolidMasse moléculaire :369.8Iproniazid
CAS :<p>Iproniazid is an irreversible monoamine oxidase inhibitor. It is used as an antidepressive agent.</p>Formule :C9H13N3ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :179.22LYN-1604 hydrochloride
CAS :<p>LYN-1604 HCl activates ULK1 (EC50: 18.94 nM); key for studying TNBC.</p>Formule :C33H44Cl3N3O2Couleur et forme :SolidMasse moléculaire :621.08Sophocarpine
CAS :<p>Sophocarpine, a major ingredient of Sophora alopecuroides, has a wide range of pharmacological effects.</p>Formule :C15H22N2ODegré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :246.35Simazine
CAS :<p>Simazine (Tafazine), a chlorotriazine herbicide/pesticide, may cause reproductive harm, endocrine disruption, and cancer.</p>Formule :C7H12ClN5Degré de pureté :99.82%Couleur et forme :SolidMasse moléculaire :201.66Deferitrin
CAS :<p>Deferitrin (GT-56-252) is an iron chelator. It potentially for the treatment of thalassemia and iron overload.</p>Formule :C11H11NO4SDegré de pureté :98.71%Couleur et forme :SolidMasse moléculaire :253.27EF24
CAS :<p>EF24 treatment boosts caspase 3/9 activity, hinders MEK1/ERK phosphorylation, and exhibits strong anti-tumor effects in OSCC by deactivating MAPK/ERK.</p>Formule :C19H15F2NODegré de pureté :99.71%Couleur et forme :SolidMasse moléculaire :311.33WYE-354
CAS :<p>WYE-354 is a selective mTOR inhibitor (IC50=5 nM), targeting mTORC1/C2 over PI3Kα (>100x) and PI3Kγ (>500x), sparing P-AKT(T308).</p>Formule :C24H29N7O5Degré de pureté :97.86% - 99.61%Couleur et forme :SolidMasse moléculaire :495.53SEC inhibitor KL-1
CAS :<p>KL-1, a potent SEC inhibitor, disrupts the AFF4-CCNT1 interaction with a Ki of 3.48 μM, selectively targeting the SEC.</p>Formule :C18H16ClNO4Degré de pureté :97.42%Couleur et forme :SolidMasse moléculaire :345.78Moexipril hydrochloride
CAS :<p>Moexipril hydrochloride (Moexipril HCl) is a potent orally active nonsulfhydrylangiotensin converting enzyme (ACE)inhibitor, used for the treatment of</p>Formule :C27H34N2O7·HClDegré de pureté :97.8%Couleur et forme :A Fine White To Off-White PowderMasse moléculaire :535.03Dexrazoxane
CAS :<p>Dexrazoxane (ICRF-187) is a mitosis-blocking anticancer drug, iron chelator, and anthracycline cardioprotectant.</p>Formule :C11H16N4O4Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :268.27Terameprocol
CAS :<p>Terameprocol (EM-1421), a synthetic NDGA derivative, shows potent anti-HIV, antiangiogenic, and anticancer properties.</p>Formule :C22H30O4Degré de pureté :99.38%Couleur et forme :SolidMasse moléculaire :358.47PD168393
CAS :<p>PD168393 is an irreversible EGFR inhibitor (IC50: 0.70 nM), irreversibly alkylate Cys-773; inactive against PKC, FGFR, PDGFR, and insulin.</p>Formule :C17H13BrN4ODegré de pureté :99.13% - 99.83%Couleur et forme :SolidMasse moléculaire :369.22Lupeol
CAS :<p>Lupeol (Monogynol B) is a novel androgen receptor inhibitor with anti-inflammatory and antioxidant activity.</p>Formule :C30H50ODegré de pureté :98% - 99.96%Couleur et forme :Needles From Alcohol Acetone White PowderMasse moléculaire :426.72Piperazine Erastin
CAS :<p>Piperazine erastin is an analog of erastin. It causes an iron-dependent form of non-apoptotic cell death termed ferroptosis.</p>Formule :C35H41ClN6O4Degré de pureté :99.52%Couleur et forme :SolidMasse moléculaire :645.19Demethylzeylasteral
CAS :<p>Demethylzeylasteral (T-96), isolated from Tripterygium wilfordii, has anti-inflammatory, immunosuppressive and anti-tumor activities.</p>Formule :C29H36O6Degré de pureté :98.74% - 99.82%Couleur et forme :SolidMasse moléculaire :480.59BTdCPU
CAS :<p>BTdCPU is a potent activator of heme-regulated eIF2α kinase (HRI) . BTdCPU promotes eIF2α phosphorylation and induced apoptosis in resistant cell.</p>Formule :C13H8Cl2N4OSDegré de pureté :98.94% - 99.59%Couleur et forme :SolidMasse moléculaire :339.2CCG-1423
CAS :<p>CCG-1423, a selective RhoA pathway inhibitor, suppresses SRF-mediated transcription.</p>Formule :C18H13ClF6N2O3Degré de pureté :99.80%Couleur et forme :SolidMasse moléculaire :454.75Purvalanol A
CAS :<p>Purvalanol A (NG-60) is an effective and cell-permeable CDK inhibitor with IC50 of 70/4/35/850 nM for cdk2-cyclin A/B/E, and cdk4-cyclin D1, respectively.</p>Formule :C19H25ClN6ODegré de pureté :98.13% - 99.68%Couleur et forme :PowderMasse moléculaire :388.89NQDI-1
CAS :<p>NQDI-1 (NQDI 1) is a selective inhibitor of apoptosis signal-regulating kinase 1 (ASK1, MAP3K5) (IC50/Ki: 3 μM/500 nM).</p>Formule :C19H13NO4Degré de pureté :97.1% - 98.10%Couleur et forme :SolidMasse moléculaire :319.31HJC0152 hydrochloride
CAS :<p>HJC0152 hydrochloride (HJC0152) is a signal transducer and activator of transcription 3 (STAT3) inhibitor.</p>Formule :C15H14Cl3N3O4Degré de pureté :99.01% - 99.06%Couleur et forme :SolidMasse moléculaire :406.64EGFR-IN-12
CAS :<p>EGFR-IN-12 (EGFR Inhibitor) is a cell permeable and selective inhibitor of EGFR kinase (IC50: 21 nM) and blocks receptor autophosphorylation in cells.</p>Formule :C21H18F3N5ODegré de pureté :98.3% - 99.76%Couleur et forme :SolidMasse moléculaire :413.4Ganoderic acid D
CAS :<p>Ganoderic acid D, a Ganoderma component, inhibits HeLa cell growth with an IC50 of 17.3µM after 48h.</p>Formule :C30H42O7Degré de pureté :98.06% - 99.98%Couleur et forme :SolidMasse moléculaire :514.65Citric acid monohydrate
CAS :<p>Citric Acid Monohydrate: tricarboxylic, from citrus, antioxidant, stabilizes drugs, preservative.</p>Formule :C6H10O8Degré de pureté :99.87%Couleur et forme :White Solid CrystallineMasse moléculaire :210.14Protosappanin B
CAS :<p>Protosappanin B enhances cell survival, growth protein 43; degrades p53 via MDM2 ubiquitination.</p>Formule :C16H16O6Degré de pureté :98% - 98.86%Couleur et forme :SolidMasse moléculaire :304.29Flavokawain A
CAS :<p>NSC-37445 shows anti-tumor properties; Flavokawain A may reduce inflammation by hindering specific signaling in macrophages.</p>Formule :C18H18O5Degré de pureté :97.1% - 99.72%Couleur et forme :SolidMasse moléculaire :314.332Degrasyn
CAS :<p>Degrasyn (WP1130) inhibits DUBs (USP5, UCH-L1, USP9x, USP14, UCH37) and Bcr/Abl without affecting the 20S proteasome.</p>Formule :C19H18BrN3ODegré de pureté :98.32% - 99.98%Couleur et forme :SolidMasse moléculaire :384.27Meisoindigo
CAS :<p>Meisoindigo (Natura-α) is a derivative of indigo natural, might induces apoptosis and myeloid differentiation of acute myeloid leukemia (AML).</p>Formule :C17H12N2O2Degré de pureté :98.03% - 98.19%Couleur et forme :SolidMasse moléculaire :276.29Cysteamine hydrochloride
CAS :<p>Cysteamine hydrochloride (Thioethanolamine Hydrochloride) is an agent for the treatment of nephropathic cystinosis and an antioxidant.</p>Formule :C2H7NS·HClDegré de pureté :99.34% - 99.87%Couleur et forme :White Crystalline Powder With A Strong And Disagreeable SmellMasse moléculaire :113.61Astaxanthin
CAS :<p>Astaxanthin, a keto-carotenoid and xanthophyll, offers antioxidant benefits, present in red aquatic species, and used as a colorant in animal feed.</p>Formule :C40H52O4Degré de pureté :95.1% - 99.79%Couleur et forme :Needles From Acetone/Light Petroleum SolidMasse moléculaire :596.84W-7 hydrochloride
CAS :<p>W-7 hydrochloride (W-7 HCl), a calmodulin antagonist, inhibits Ca2+-calmodulin-dependent myosin light chain kinase and phosphodiesterase, W-7 hydrochloride</p>Formule :C16H22Cl2N2O2SDegré de pureté :99.63%Couleur et forme :White Crystalline SolidMasse moléculaire :377.32Voreloxin hydrochloride
CAS :<p>Voreloxin hydrochloride (SNS-595 hydrochloride) is a potent inhibitor of Topoisomerase II with broad-spectrum anti-tumor activity.</p>Formule :C18H20ClN5O4SDegré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :437.9Deoxypodophyllotoxin
CAS :<p>Deoxypodophyllotoxin is cytotoxic, antineoplastic, anti-tumor, anti-angiogenic, antiviral, and anti-inflammatory.</p>Formule :C22H22O7Degré de pureté :99.65% - 99.84%Couleur et forme :SolidMasse moléculaire :398.41Pioglitazone potassium
CAS :<p>Pioglitazone potassium is an oral PPARγ agonist with EC50 of 0.93 μM (human) and 0.99 μM (mouse), used in diabetes research.</p>Formule :C19H19KN2O3SCouleur et forme :SolidMasse moléculaire :394.53Atezolizumab
CAS :<p>Atezolizumab is an antibody inhibitor, a humanized monoclonal antibody, IgG1, which targets PD-L1. Atezolizumab has antitumor effect. Cost-effective and quality-assured.</p>Degré de pureté :95.10% - 99.3% (SEC-HPLC)Couleur et forme :LiquidMasse moléculaire :145 kDaStaurosporine
CAS :<p>Staurosporine (AM-2282) is a protein kinase inhibitor with ATP-competitive and non-selective inhibitory activity (IC50=6/15/2/3/3000 nM) against PKC, PKA, c-Fgr</p>Formule :C28H26N4O3Degré de pureté :99.24% - 99.82%Couleur et forme :Off-White PowderMasse moléculaire :466.53Mirodenafil dihydrochloride
CAS :<p>Mirodenafil dihydrochloride is a PDE-5 inhibitor developed for the treatment of erectile dysfunction.</p>Formule :C26H39Cl2N5O5SDegré de pureté :99.64% - 99.78%Couleur et forme :SolidMasse moléculaire :604.59Eriocitrin
CAS :<p>Eriocitrin: an antioxidative flavonoid; reduces exercise-induced oxidative damage and lipids; fights fatty liver and inhibits carbonic anhydrase VA.</p>Formule :C27H32O15Degré de pureté :98.41% - 99.11%Couleur et forme :SolidMasse moléculaire :596.53NSC 15364
CAS :<p>NSC 15364 (1,3-Bis(4-aminophenyl)urea) can be used for screening of ALR inhibitors by detection of hydrogen peroxide production Measured in Biochemical System.</p>Formule :C13H14N4ODegré de pureté :98.67%Couleur et forme :SolidMasse moléculaire :242.28Licofelone
CAS :<p>Licofelone (ML-3000) is a dual COX/LOX inhibitor potentially for the treatment of osteoarthritis.</p>Formule :C23H22ClNO2Degré de pureté :99.25%Couleur et forme :Yellowish SolidMasse moléculaire :379.88Y-27632 dihydrochloride
CAS :<p>View and buy Y-27632 dihydrochloride from TargetMol.Y-27632 is a selective inhibitor of ROCKs.Cited in 10 publications.</p>Formule :C14H21N3O·2HClDegré de pureté :97.96% - 99.98%Couleur et forme :SolidMasse moléculaire :320.26NVP 231
CAS :<p>NVP-231 is a potent, specific and reversible CerK inhibitor(IC50=12±2 nM) that competitively inhibits ceramide binding to CerK.</p>Formule :C25H25N3O2SDegré de pureté :99.16% - ≥95%Couleur et forme :SolidMasse moléculaire :431.55Ixabepilone
CAS :<p>Ixabepilone (Azaepothilone B) is an orally bioavailable microtubule inhibitor.</p>Formule :C27H42N2O5SDegré de pureté :98% - 99.50%Couleur et forme :SolidMasse moléculaire :506.7Tubeimoside I
CAS :<p>Tubeimoside I (Tubeimoside-1)(Lobatoside-H) is an extract from Chinese herbal medicine Bolbostemma paniculatum (MAXIM).</p>Formule :C63H98O29Degré de pureté :98.89% - 99.94%Couleur et forme :SolidMasse moléculaire :1319.43Vanillyl Alcohol
CAS :<p>Vanillyl Alcohol (3-Methoxy-4-hydroxybenzyl alcohol) possesses anti-angiogenic, anticonvulsive, anti-inflammatory, anti-oxidant and anti-nociceptive activities.</p>Formule :C8H10O3Degré de pureté :97.02% - 98.42%Couleur et forme :Crystalline White To Off-White PowderMasse moléculaire :154.16Millepachine
CAS :<p>Millepachine is a natural product found in the Chinese herbal medicine with strong antitumor effects against numerous human cancer cells.</p>Formule :C22H22O4Degré de pureté :99.73%Couleur et forme :SolidMasse moléculaire :350.41SRS11-92
CAS :<p>SRS11-92 (AA9) is a ferroptosis inhibitor and a derivative of ferrostatin-1</p>Formule :C22H28N2O2Degré de pureté :98.58%Couleur et forme :SolidMasse moléculaire :352.478-Prenylnaringenin
CAS :<p>8-Prenylnaringenin is a phytoestrogen with high estrogenic activity,</p>Formule :C20H20O5Degré de pureté :98.26% - 99.46%Couleur et forme :SolidMasse moléculaire :340.37Alantolactone
CAS :<p>Alantolactone is a selective inhibitor of STAT3 that induces cancer-associated apoptosis and has antitumor activity.Cost-effective and quality-assured.</p>Formule :C15H20O2Degré de pureté :99.02% - 99.66%Couleur et forme :Crystalline PowderMasse moléculaire :232.32Rosmarinic acid
CAS :<p>Rosmarinic acid (Labiatenic acid) is widely found in plants and has antioxidant, anti-inflammatory, and antibacterial activities.</p>Formule :C18H16O8Degré de pureté :98.88% - 99.73%Couleur et forme :Brown Fine PowderMasse moléculaire :360.31DD1
CAS :<p>DD1 (HUN85111) is a proteasome inhibitor that induces human myeloid tumor-selective apoptosis.</p>Formule :C16H14N2O3Degré de pureté :99.57%Couleur et forme :SolidMasse moléculaire :282.29Y-27632 HCl hydrate
CAS :<p>Y-27632 HCl hydrate is an orally effective, ATP-competitive ROCK1/ROCK2 inhibitor (Ki=220 nM/300 nM) that inhibits caspase-3 and suppresses stem cell apoptosis.</p>Formule :C14H25Cl2N3O2Degré de pureté :99.98%Couleur et forme :SolidMasse moléculaire :338.27SB 202190
CAS :<p>SB 202190 (FHPI) is a p38 MAPK inhibitor that inhibits p38α and p38β2 (IC50=50/100 nM) selectively and cell-permeably.</p>Formule :C20H14FN3ODegré de pureté :98% - 99.84%Couleur et forme :Pale YellowMasse moléculaire :331.34TCS7010
CAS :<p>TCS7010 (Aurora A Inhibitor I) is a novel, potent, and selective inhibitor of Aurora A with IC50 of 3.4 nM in a cell-free assay.</p>Formule :C31H31ClFN7O2Degré de pureté :98.49% - 99.62%Couleur et forme :SolidMasse moléculaire :588.07PRLX-93936
CAS :<p>PRLX-93936 is a selective Ras pathway protein inhibitor that modulates RAS/JNK pathway-associated protein phosphorylation, anticancer activity.</p>Formule :C21H24N4O2Couleur et forme :SolidMasse moléculaire :364.44Brassinolide
CAS :<p>Brassinolide (Brassin lactone) is a plant hormone isolated from rapeseed (Brassica napus) promoting stem elongation and cell division.</p>Formule :C28H48O6Degré de pureté :98% - 99.189%Couleur et forme :Off-White SolidMasse moléculaire :480.68Valproic Acid
CAS :<p>Valproic Acid (2-Propylpentanoic Acid) is a branched chain fatty acid which potentially enhances central GABAergic neurotransmission and inhibits Na+ channels.</p>Formule :C8H16O2Degré de pureté :97.78% - 99%Couleur et forme :Colourless To Pale Yellow Liquid ViscousMasse moléculaire :144.21Ginkgetin
CAS :<p>Ginkgetin: antiviral, antifungal, anti-inflammatory; COX-2 reducer; STAT3 inhibitor; pro-apoptotic in cancer; neuroprotective in Parkinson's.</p>Formule :C32H22O10Degré de pureté :98.63% - 99.94%Couleur et forme :SolidMasse moléculaire :566.51Nodinitib-1
CAS :<p>Nodinitib-1 (CID-1088438) is a potent and selective NOD1 inhibitor with an IC50 of 0.56 μM.</p>Formule :C14H13N3O2SDegré de pureté :99.97% - >99.99%Couleur et forme :SolidMasse moléculaire :287.34PUMA BH3 Free base
<p>PUMA BH3 acetate (PUMA BH3 Free base) is a p53 positive regulator of apoptosis (PUMA) BH3 domain polypeptide that acts as a direct activator of Bak with a Kd of</p>Formule :C130H206N42O45SDegré de pureté :96.64%Couleur et forme :SolidMasse moléculaire :3109.35Sclareol
CAS :<p>Sclareol from clary sage inhibits growth and is cytotoxic to many human Y cell lines.</p>Formule :C20H36O2Degré de pureté :99.58% - 99.97%Couleur et forme :White Fine PowderMasse moléculaire :308.5Orantinib
CAS :<p>Orantinib (NSC 702827) , a excellent effective against PDGFR autophosphorylation with Ki of 8 nM, also highly inhibits Flk-1 and FGFR1 trans-phosphorylation.</p>Formule :C18H18N2O3Degré de pureté :98.92% - 99.52%Couleur et forme :SolidMasse moléculaire :310.35DL-Buthionine-(S,R)-sulfoximine
CAS :<p>DL-Buthionine-(S,R)-sulfoximine (Butionine sulfoximine) is an inhibitor of γ-glutamylcysteine synthetase for the treatment of solid tumors.</p>Formule :C8H18N2O3SDegré de pureté :98% - 99.64%Couleur et forme :White Fine PowderMasse moléculaire :222.31K-Ras(G12C) inhibitor 12
CAS :<p>K-Ras(G12C) inhibitor 12 is an allosteric inhibitor of oncogenic K-Ras(G12C).</p>Formule :C15H17ClIN3O3Degré de pureté :97.16%Couleur et forme :SolidMasse moléculaire :449.67(Rac)-Idroxioleic acid
CAS :<p>(Rac)-Idroxioleic acid (2-Hydroxyoleic acid) is a fatty acid amide hydrolase inhibitor with anti-tumor effect.</p>Formule :C18H34O3Degré de pureté :≥98%Couleur et forme :SolidMasse moléculaire :298.46(20S)-Protopanaxatriol
CAS :<p>(20S)-Protopanaxatriol (g-PPT)(g-PPT), a metabolite of ginsenoside, could regulate endothelial cell functions through the estrogen receptor and glucocorticoid</p>Formule :C30H52O4Degré de pureté :95% - 99%Couleur et forme :SolidMasse moléculaire :476.73DMU-212
CAS :<p>DMU-212, a Resveratrol derivative, has antimitotic, antiproliferative, antioxidant properties; induces apoptosis via ERK1/2.</p>Formule :C18H20O4Degré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :300.35
