Apoptose
Les inhibiteurs de l'apoptose sont des composés qui empêchent ou retardent le processus de mort cellulaire programmée, connu sous le nom d'apoptose. Ces inhibiteurs sont essentiels pour étudier les mécanismes de survie cellulaire et sont utilisés pour enquêter sur les maladies où l'apoptose est dysrégulée, telles que le cancer, les troubles neurodégénératifs et les maladies auto-immunes. En modulant l'apoptose, ces inhibiteurs peuvent aider au développement de thérapies visant à contrôler la mort cellulaire. Chez CymitQuimica, nous offrons une sélection complète d'inhibiteurs de l'apoptose de haute qualité pour soutenir vos recherches en biologie cellulaire, oncologie et domaines connexes.
Sous-catégories appartenant à la catégorie "Apoptose"
- ASK(6 produits)
- BCL(11 produits)
- Caspase(125 produits)
- FOXO1(3 produits)
- IAP(66 produits)
- Mdm2(12 produits)
- PD-1/PD-L1(125 produits)
- PDK(9 produits)
- PERK(25 produits)
- Sérine/thréonine kinase(15 produits)
- Survivant(13 produits)
- TNF(92 produits)
- c-RET(51 produits)
- p53(62 produits)
Affichez 6 plus de sous-catégories
5593 produits trouvés pour "Apoptose"
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CDK1/Cyc B-IN-1
CAS :<p>CDK1/Cyc B-IN-1: Potent CDK1/Cyc B inhibitor, IC50 97 nM, induces apoptosis, arrests G2/M cycle, halts cancer growth.</p>Formule :C14H12ClN3O2S2Couleur et forme :SolidMasse moléculaire :353.85HJC0416
CAS :<p>HJC0416 is a potent orally bioavailable signal transducer and activator of transcription 3 inhibitor.</p>Formule :C18H17ClN2O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :392.86VRT-043198
CAS :<p>VRT-043198, a VX-765 metabolite, is a potent ICE/caspase-1 inhibitor, crossing the blood-brain barrier with K i of 0.8/0.6 nM.</p>Formule :C22H29ClN4O6Couleur et forme :SolidMasse moléculaire :480.94CMLD012072
CAS :<p>CMLD012072 is a potent eukaryotic initiation factor 4A (eIF4A) inhibitor with potent anti-neoplastic activity. It can induce RNA clamping of eIF4A1 and eIF4A2.</p>Formule :C32H32N2O7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :556.61AG6033
CAS :<p>AG6033, a novel CRBN modulator, degrades GSPT1/IKZF1 and inhibits various tumors.</p>Formule :C30H23N5O4Couleur et forme :SolidMasse moléculaire :517.53HDAC-IN-31
CAS :<p>HDAC-IN-31: Oral HDAC inhibitor; targets HDAC1, 2, 3; weak on HDAC8; potential in fighting lymphoma.</p>Formule :C25H24N4O2Couleur et forme :SolidMasse moléculaire :412.48RIPK1-IN-15
CAS :<p>RIPK1-IN-15 (Compound 2.5) is a potent RIPK1 inhibitor that has the potential in neurodegenerative, autoimmune, and inflammatory diseases research [1].</p>Formule :C19H19N3O2Couleur et forme :SolidMasse moléculaire :321.37ABT-100
CAS :<p>ABT-100 is a potent, highly selective, and orally active farnesyl transferase inhibitor with broad-spectrum antitumor activity.</p>Formule :C27H19F3N4O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :504.46Prexasertib mesylate
CAS :<p>Prexasertib (LY2606368), a Chk1/2 inhibitor, enhances therapy in acute lymphoblastic leukemia, causing DNA damage and antitumor effects.</p>Formule :C19H23N7O5SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :461.49Verrucarin J
CAS :<p>Verrucarin J, a Myrothecium fungus metabolite, triggers apoptosis in some cancer cells and fights Candida, Mucor, and JUNV (IC50: 1.2 ng/mL).</p>Formule :C27H32O8Couleur et forme :SolidMasse moléculaire :484.54PAK4-IN-2
CAS :<p>PAK4-IN-2 inhibits PAK4 with IC50 2.7 nM, arrests MV4-11 cells at G0/G1, and induces apoptosis, promising for cancer research.</p>Formule :C18H21ClN6Couleur et forme :SolidMasse moléculaire :356.85PARP-1-IN-2
CAS :<p>PARP-1-IN-2 is a potent PARP1 inhibitor that crosses the blood-brain barrier (IC50: 149 nM).PARP-1-IN-2 showed significant antiproliferative activity against</p>Formule :C22H15Cl2N3O2Degré de pureté :98.82%Couleur et forme :SolidMasse moléculaire :424.28PD180970
CAS :<p>PD180970 is an inhibitor of Bcr-Abl with IC50s of 5 nM, 0.8 nM and 50 nM for the autophosphorylation of p210Bcr-Abl, Src and Kit.</p>Formule :C21H15Cl2FN4ODegré de pureté :98.67%Couleur et forme :SolidMasse moléculaire :429.27MSN-50
CAS :<p>MSN-50, an inhibitor of Bax and Bak oligomerization, inhibits liposome permeabilization, prevents genotoxic cell death and promotes neuroprotection.</p>Formule :C36H38BrN3O6Couleur et forme :SolidMasse moléculaire :688.61WK-298
CAS :<p>WK-298 is an effective MDM2/MDMX-p53 interaction inhibitor.</p>Formule :C35H38Cl2N6ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :629.62AP1867
CAS :<p>AP1867 is a synthetic FKBP12F36V-directed ligand.</p>Formule :C38H47NO11Couleur et forme :SolidMasse moléculaire :693.78NSC-741909
CAS :<p>NSC-741909 is an anticancer agent that acts by suppressing the growth of several cell lines.</p>Formule :C16H14ClNODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :271.74ATB-337
CAS :<p>S-Diclofenac, an NSAID with H2S-releasing moiety, protects gastric mucosa while inhibiting prostaglandins.</p>Formule :C23H15Cl2NO2S3Couleur et forme :SolidMasse moléculaire :504.47KF24345
CAS :<p>KF24345 is an inhibitor of adenosine uptake.</p>Formule :C31H38N6O5Couleur et forme :SolidMasse moléculaire :574.67LY5
CAS :<p>LY5 is an inhibitor of STAT3 that acts by inhibiting cell viability, cell migration, and angiogenesis in medulloblastoma cells.</p>Formule :C15H11N3O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :329.33NU-8165
CAS :<p>NU-8165 is an MDM2-p53 protein-protein interaction inhibitor.</p>Formule :C24H22ClNO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :407.89IHMT-TRK-284
CAS :<p>IHMT-TRK-284: Oral type II TRK inhibitor; targets TRKA, TRKB, TRKC (IC50s: 10.5, 0.7, 2.6 nM); selective and anti-tumor effective.</p>Formule :C25H27N7OSCouleur et forme :SolidMasse moléculaire :473.59D44
CAS :<p>D44 is a Plasmodium FKBPs inhibitor.</p>Formule :C16H16N4OSCouleur et forme :SolidMasse moléculaire :312.39BRD4 Inhibitor-15
CAS :<p>BRD4 Inhibitor-15 targets BRD4 with 18 nM IC50, induces apoptosis in 22RV1 cells, and lowers c-Myc, aiding prostate cancer research.</p>Formule :C22H21N3O2Couleur et forme :SolidMasse moléculaire :359.42PDGFR-IN-1
CAS :<p>PDGFR-IN-1 is a platelet-derived growth factor receptor (PDGFR) inhibitor, strongly inhibiting PDGFRα and PDGFRβ, useful for studying solid tumors.</p>Formule :C25H30N8ODegré de pureté :99.13% - 99.49%Couleur et forme :SolidMasse moléculaire :458.56Fomesafen
CAS :<p>Fomesafen (PP-021) is a diphenyl ether herbicide and an inhibitor of efficient and selective protoporphyrinogen IX oxidase (PPO).</p>Formule :C15H10ClF3N2O6SDegré de pureté :99.91% - 99.93%Couleur et forme :White Crystalline Solid Fomesafen Is A White Crystalline Solid Used As An HerbicideMasse moléculaire :438.76CRA-026440
CAS :<p>CRA-026440(PCI-34051) is a highly potent HDAC inhibitor with inhibitory effects on HDAC1, HDAC2, HDAC3, HDAC6, HDAC8 and HDAC10 with Ki values of 4,14,11,15,7</p>Formule :C23H24N4O4Degré de pureté :96.42%Couleur et forme :SolidMasse moléculaire :420.46GSK962
CAS :<p>GSK962 is a GSK963 inactive enantiomer. It can be used to confirm the on-target effects.</p>Formule :C14H18N2ODegré de pureté :99.75%Couleur et forme :SolidMasse moléculaire :230.31Dimethoate
CAS :<p>Dimethoate (L-395) is a systemic and contact insecticide for control of cattle grubs and certain other insect pests of farm animals.</p>Formule :C5H12NO3PS2Degré de pureté :99.74% - 99.91%Couleur et forme :White Crystalline SolidMasse moléculaire :229.26Mcl1-IN-4
CAS :Mcl1-IN-4 is an inhibitor of Mcl1 ( IC50:0.2 μM).Formule :C28H26N2O5SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :502.58MG-262
CAS :<p>MG-262 is a reversible proteasome inhibitor with multiple biological activities [1] [2] [3].</p>Formule :C25H42BN3O6Couleur et forme :SolidMasse moléculaire :491.43M199
CAS :<p>M199, a novel inhibitor of TLR3/9 activation, induces secretion of IL-6, IL-8 and TNFalpha in human PBMCs.</p>Formule :C17H17N3ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :279.34Didesmethylrocaglamide
CAS :<p>Didesmethylrocaglamide, a Rocaglamide derivative, is a potent eukaryotic initiation factor 4A (eIF4A) inhibitor that exhibits strong growth-inhibitory effects,</p>Formule :C27H27NO7Couleur et forme :SolidMasse moléculaire :477.51Mitochonic Acid 35
CAS :<p>Mitochonic Acid 35 is a dual TNF-α and TGF-β1 inhibitor that acts by inhibiting IκB kinase phosphorylation and Smad3 phosphorylation.</p>Formule :C19H19NO5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :341.36Semapimod
CAS :<p>Semapimod is an inhibitor of proinflammatory cytokine production, capable of suppressing TNF-α, IL-1β, and IL-6.</p>Formule :C34H52N18O2Couleur et forme :SolidMasse moléculaire :744.9DC-CPin711
CAS :<p>DC-CPin711: Potent, selective CBP bromodomain inhibitor, IC50=0.0626 μM; arrests G1 cell cycle, induces apoptosis.</p>Formule :C23H22N4O2Couleur et forme :SolidMasse moléculaire :386.45PI3K/AKT-IN-2
CAS :<p>PI3K/AKT-IN-2 inhibits PI3K/AKT, EMT, induces apoptosis, and blocks tubulin polymerization.</p>Formule :C32H27BrO10Couleur et forme :SolidMasse moléculaire :651.45VMY-1-103
CAS :<p>VMY-1-103: a strong CDK inhibitor better than purvalanol B; halts prostate/breast cancer cell growth, induces apoptosis, may treat medulloblastoma.</p>Formule :C34H42ClN9O4SCouleur et forme :SolidMasse moléculaire :708.27PDK4-IN-1
CAS :<p>PDK4-IN-1 is an anthraquinone derivative and a potent and orally active inhibitor of pyruvate dehydrogenase kinase 4 (PDK4)(IC50 value of 84 nM).</p>Formule :C22H19N3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :357.41LLL3
CAS :<p>LLL3 is a small molecule STAT3 inhibitor.</p>Formule :C16H10O4Couleur et forme :SolidMasse moléculaire :266.25W1131
CAS :<p>W1131 is a potent STAT3 inhibitor and ferroptosis trigger, reducing cancer progression and 5-FU resistance.</p>Formule :C23H19N5O4Couleur et forme :SolidMasse moléculaire :429.43AD-2646
CAS :<p>AD-2646 has antidepressant activity and inhibits 2-deoxy-D-glucose (2-DG)-induced gastric acid secretion.</p>Formule :C23H40N2O4Couleur et forme :SolidMasse moléculaire :408.57ABD56
CAS :<p>ABD56 inhibits osteoclast formation and activity in vitro and in vivo.</p>Formule :C17H18O3Couleur et forme :SolidMasse moléculaire :270.32Trehalose 6-behenate
CAS :<p>Trehalose 6-behenate is a Th1/Th17 skewing vaccine adjuvant.</p>Formule :C34H64O12Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :664.86N1,N11-Diethylnorspermine
CAS :<p>DENSPM: potent anticancer, spurs polyamine breakdown, triggers cytochrome c release and caspase 3, kills GBM via SSAT & H2O2.</p>Formule :C13H32N4Couleur et forme :SolidMasse moléculaire :244.42MBC-11
CAS :<p>MBC-11: First bone-targeting bisphosphonate-etidronate conjugate with araC, may treat TIBD.</p>Formule :C11H20N3O14P3Degré de pureté :>99.99% - >99.99%Couleur et forme :SolidMasse moléculaire :511.21GRI977143
CAS :<p>GRI977143: selective LPA2 agonist (EC50=3.3μM), blocks caspases 3/7/8/9, limits DNA fragmentation.</p>Formule :C22H17NO4SDegré de pureté :98.07%Couleur et forme :SolidMasse moléculaire :391.44A-385358
CAS :<p>A-385358 is a selective Bcl-xL inhibitor with Kis of 0.80 nM for Bcl-xL and 67 nM for Bcl-2, respectively.</p>Formule :C32H41N5O5S2Degré de pureté :99.97%Couleur et forme :SolidMasse moléculaire :639.83NKP-1339
CAS :<p>NKP-1339 (IT-139) induces G2/M cell cycle arrest, blockage of DNA synthesis, and induction of apoptosis via the mitochondrial pathway.</p>Formule :C14H12Cl4N4NaRuDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :502.14Flonoltinib
CAS :<p>Flonoltinib (JAK2/FLT3-IN-1) is an orally active and efficient JAK2/FLT3 inhibitor with anti-cancer properties.</p>Formule :C25H34FN7ODegré de pureté :99.52%Couleur et forme :SolidMasse moléculaire :467.58BR102375
CAS :<p>BR102375 is a non-TZD PPAR γ full agonist (EC50: 0.28 μM) for the treatment of type 2 diabetes.</p>Formule :C31H34N6O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :554.64Antitumor agent-44
CAS :<p>Antitumor agent-44 (Compound 5n) elicits potent antitumor effects by inducing disruption of mitochondrial homeostasis, cell cycle arrest, and apoptosis in human</p>Formule :C24H15N3O3Couleur et forme :SolidMasse moléculaire :393.39PIK-C98
CAS :<p>PIK-C98 is an inhibitor of PI3K that acts by displaying potent preclinical activity against multiple myeloma.</p>Formule :C16H10Cl2N2OSDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :349.23RET-IN-12
CAS :<p>RET-IN-12 is a RET inhibitor capable of acting on RET(WT) (IC50: 0.3 nM) and RET(V804M) (IC50: 1 nM).</p>Formule :C30H30F3N5O4Couleur et forme :SolidMasse moléculaire :581.59PDE5/HDAC-IN-1
CAS :<p>PDE5/HDAC-IN-1 is a potent inhibitor of phosphodiesterase 5 (PDE5) and HDAC, with IC50 values of 46.3 nM and 14.5 nM, respectively.</p>Formule :C27H29BrN4O4Couleur et forme :SolidMasse moléculaire :553.45Cinnabarinic acid
CAS :<p>mGlu4 receptor agonist</p>Formule :C14H8N2O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :300.22A-802715
CAS :<p>A-802715 is a novel methylxanthine derivative that decreases the endogenous formation and blood levels of pro-inflammatory substances and increases the</p>Formule :C16H26N4O3Degré de pureté :96.29%Couleur et forme :SolidMasse moléculaire :322.4Tezacitabine
CAS :<p>Tezacitabine, a nucleoside analogue, inhibits ribonucleotide reductase, disrupts DNA replication, and induces apoptosis in tumor cells.</p>Formule :C10H12FN3O4Couleur et forme :SolidMasse moléculaire :257.22Apoptotic agent-2
CAS :<p>Apoptotic agent-2 reduces Bcl-2, boosts Bax & caspase-3, inducing apoptosis for cancer research.</p>Formule :C25H16ClN7SCouleur et forme :SolidMasse moléculaire :481.96MMP-9-IN-4
CAS :<p>MMP-9-IN-4 inhibits MMP-9 (IC50=7.46nM) and AKT (IC50=8.82nM), induces apoptosis and is used in cancer research.</p>Formule :C28H19F3N4O6Couleur et forme :SolidMasse moléculaire :564.47Topoisomerase II inhibitor 3
CAS :<p>Acridone-based Topoisomerase II inhibitor 3 targets topo IIα/β (IC50: 0.17μM α, 0.23μM β), causes DNA damage, and induces apoptosis.</p>Formule :C18H20N4O4Couleur et forme :SolidMasse moléculaire :356.382'-Deoxyadenosine
CAS :<p>2'-Deoxyadenosine (NSC-141848) is the DNA nucleoside A. It pairs with deoxythymidine (T) in double-stranded DNA.</p>Formule :C10H13N5O3Degré de pureté :99.71%Couleur et forme :SolidMasse moléculaire :251.24CEP-40125
CAS :<p>CEP-40125 (RXDX-107) is a DNA alkylating agent for the study of advanced solid tumors.</p>Formule :C28H45Cl2N3O2Degré de pureté :98.28%Couleur et forme :SolidMasse moléculaire :526.58CCT373567
CAS :<p>CCT373567 is a potent degrader of the transcriptional repressor BCL6 (IC50: 2.9 nM) and exhibits anti-proliferative effects.</p>Formule :C26H29ClF2N6O3Couleur et forme :SolidMasse moléculaire :547Nampt-IN-3
CAS :<p>Nampt-IN-3 simultaneously inhibit nicotinamide phosphoribosyltransferase (NAMPT) and HDAC (IC50s of 31 nM and 55 nM, respectively).</p>Formule :C29H25N7O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :503.55ARP 101
CAS :<p>ARP 101 is a selective matrix metalloproteinase-2 (MMP-2) inhibitor with anticancer activity.</p>Formule :C20H26N2O5SDegré de pureté :98.26%Couleur et forme :SolidMasse moléculaire :406.5Methylisothiazolinone
CAS :<p>Methylisothiazolinone (MI) is a powerful synthetic biocide and preservative within the group of isothiazolinones.</p>Formule :C4H5NOSDegré de pureté :99.78%Couleur et forme :Colorless Prisms LiquidMasse moléculaire :115.15CMLD010509
CAS :<p>CMLD010509 (SDS-1-021) inhibits oncogenic proteins MDM2, CCND1, MYC, MAF, MCL-1 in multiple myeloma.</p>Formule :C27H26BrNO7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :556.4Topoisomerase I inhibitor 5
CAS :<p>Topoisomerase I inhibitor 5 halts DNA replication, induces MCF-7 cell apoptosis, and overcomes drug resistance. IC50 value is noted.</p>Formule :C24H24N2O2Couleur et forme :SolidMasse moléculaire :372.46Selicrelumab
CAS :<p>Selicrelumab (RG-7876) is an antibody targeting CD40 with potential anti-tumor activity for the study of pancreatic cancer.</p>Degré de pureté :98.7% (SDS-PAGE); 95.2% (SEC-HPLC) - 98.7% (SDS-PAGE); 95.2% (SEC-HPLC)Couleur et forme :LiquidCMLD012073
CAS :<p>CMLD012073: Potent eIF4A inhibitor, halts eukaryotic translation; IC50 10 nM in NIH/3T3 cells.</p>Formule :C30H30N2O7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :530.57RET-IN-22
CAS :<p>RET-IN-22 (compound 17b) is a potent, selective, and orally active inhibitor of RET, exhibiting IC50 values of 20.9 nM for wild-type RET and 18.3 nM for RET-</p>Formule :C29H31F3N6O4Couleur et forme :SolidMasse moléculaire :584.59KRAS G12D inhibitor 14
CAS :<p>KRAS G12D inhibitor 14 is a potent inhibitor of KRAS G12D that binds KRAS G12D protein (Kd: 33 nM).</p>Formule :C20H19F3N4OSDegré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :420.45Z-LEVD-FMK
CAS :<p>Z-LEVD-FMK is a caspase-4 inhibitor with anti-cancer activity, capable of eliminating LPS-induced GCLC protein degradation.</p>Formule :C31H45FN4O10Couleur et forme :SolidMasse moléculaire :652.71S130
CAS :<p>S130 is a high affinity, selectiveATG4B (a major cysteine protease) inhibitor (IC50 of 3.24 μM).It suppresses autophagy flux.</p>Formule :C24H25N3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :387.47Topoisomerase II inhibitor 9
CAS :<p>Topoisomerase II inhibitor 9: Topo II blocker (IC50: 0.97 μM), DNA intercalator (IC50: 43.51 μM), arrests G2/M in Hep G-2 cells and triggers apoptosis.</p>Formule :C22H17N7O3S2Couleur et forme :SolidMasse moléculaire :491.55PARP-2-IN-3
CAS :<p>PARP-2-IN-3 is used in the study of breast cancer as a PARP-2 inhibitor with antitumor activity that induces apoptosis (apoptosis) and necrosis in cancer cells.</p>Formule :C20H20ClN3O3Degré de pureté :99.33%Couleur et forme :SolidMasse moléculaire :385.84IM-54
CAS :<p>IM-54 is a cell-permeable, effective, and selective necrosis inhibitor.</p>Formule :C19H23N3O2Degré de pureté :99.24%Couleur et forme :SolidMasse moléculaire :325.4AMG-548
CAS :<p>AMG-548, oral p38α inhibitor (Ki=0.5 nM), >1000x selectivity over p38γ/δ, blocks TNFα (IC50=3 nM), also inhibits Wnt/Casein kinase 1δ/ε.</p>Formule :C29H27N5ODegré de pureté :99.91%Couleur et forme :SolidMasse moléculaire :461.56NSC260594
CAS :<p>NSC260594 is a chemical compound that promotes apoptosis by binding to the shallow groove of the Mcl-1 protein and suppressing its expression through down-</p>Formule :C29H24N6O3Couleur et forme :SolidMasse moléculaire :504.54SMIP004
CAS :<p>SMIP004 is an SKP2 E3 ligase inhibitor. SMIP004 is a cancer cell-selective apoptosis inducer of human prostate cancer cells.</p>Formule :C13H19NODegré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :205.3Rhosin
CAS :<p>Rhosin is a specific inhibitor of RhoA GTPases (Kd: ~0.4 uM), blocking RhoA-GEF interaction, not affecting Cdc42/Rac1/LARG, and induces apoptosis.</p>Formule :C20H18N6ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :358.4SCH529074
CAS :<p>SCH529074 is a selective activator of p53 (Ki = 1 μM) and can be used in studies about non-small-cell lung carcinoma.</p>Formule :C31H36Cl2N6Degré de pureté :99.57%Couleur et forme :SolidMasse moléculaire :563.56KS106
CAS :<p>KS106 inhibits ALDH (1A1: 334 nM, 2: 2137 nM, 3A1: 360 nM), has anti-cancer properties, raises ROS, and promotes aldehyde build-up.</p>Formule :C18H15BrF3N3O2SDegré de pureté :99.31%Couleur et forme :SolidMasse moléculaire :474.3AK301
CAS :<p>AK301 is a potent and selective inhibitor of tubulin polymerization and an effective sensitizer of cancer cells to apoptotic ligands (EC50 < 200 nM).</p>Formule :C19H21ClN2O2Degré de pureté :99.27%Couleur et forme :SolidMasse moléculaire :344.84GDP366
CAS :<p>GDP366, induces cell growth inhibition, cellular senescence and mitotic catastrophe in human cancer cells. a dual inhibitor of survivin and Op18.</p>Formule :C20H17N5OSDegré de pureté :98.78% - 99.84%Couleur et forme :SolidMasse moléculaire :375.45Mcl1-IN-9
CAS :<p>Mcl1-IN-9 is a potent myeloid cell leukemia-1 (Mcl-1) Inhibitor with an IC50 of 446 nM in reengineered BCR-ABL+ B-ALL cells and a Ki of 0.03 nM.</p>Formule :C37H39ClN4O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :639.18Docetaxel trihydrate
CAS :<p>Docetaxel trihydrate (RP-56976 Trihydrate) is an antineoplastic agent that has a unique mechanism of action as an inhibitor of cellular mitosis.</p>Formule :C43H59NO17Degré de pureté :98.68% - >99.99%Couleur et forme :White Crystalline PowderMasse moléculaire :861.95Allethrin
CAS :<p>Allethrin induces oxidative stress, apoptosis and calcium release. Allethrin, a pyrethroid insecticide is a major mosquito repellent agent.</p>Formule :C19H26O3Degré de pureté :99.52%Masse moléculaire :302.41Polyphyllin II
CAS :<p>Polyphyllin II (Chonglou Saponin II) has hemostasis, expectorant, bacteriostasis, anticytotoxic, anti-pregnancy kill sperm effects.</p>Formule :C44H70O16Degré de pureté :99.92%Couleur et forme :SolidMasse moléculaire :855.02Misetionamide
CAS :<p>Misetionamide: Oral oxathiazin-like, GAPDH inhibitor with anticancer properties for research use.</p>Formule :C3H7NO3SCouleur et forme :SolidMasse moléculaire :137.16BN201
CAS :<p>BN201 (OCS-05) is a neuroprotective drug by activating SGK2 and FOXO3 pathway. BN201 is able to regulate multiple kinases in the IGF1 pathway and cross BBB.</p>Formule :C25H38FN5O4Degré de pureté :99.42% - 99.42%Couleur et forme :SolidMasse moléculaire :491.6STAT5-IN-2
CAS :<p>STAT5-IN-2 is an inhibitor of STAT5 with antileukemic effects (EC50s: 9 μM and 5 μM in K562 and KU812 cells, respectively).</p>Formule :C26H27N3ODegré de pureté :99.55%Couleur et forme :SolidMasse moléculaire :397.51Erasin
<p>Erasin is a STAT3 inhibitor induces apoptosis in various cancer cell lines (e.g., MDA-MB-231, HCC-827) and against Erlotinib-resistant cancer cells.</p>Formule :C20H19N3O3Couleur et forme :SolidMasse moléculaire :349.38Sparfosic acid trisodium
CAS :<p>Sparfosic acid trisodium is a CAD (carbamoyl-phosphate synthetase 2) inhibitor and also an aspartate transcarbamoyl transferase inhibitor with antitumour</p>Formule :C6H9NNaO8PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :277.1RLX
CAS :<p>RLX (PD 139530) is a PI3K/Akt/FoxO3a signal inhibitor with anticancer,antitussive and anti-asthmatic activity,colon cancer，toxicity toward A549 cells..</p>Formule :C13H14N2ODegré de pureté :99.81%Couleur et forme :SolidMasse moléculaire :214.26Declopramide
CAS :<p>Declopramide (OXI-104) is a chemosensitizer with antitumor activity that can be used to study colorectal cancer and inflammatory bowel disease.</p>Formule :C13H20ClN3ODegré de pureté :98.53%Couleur et forme :SolidMasse moléculaire :269.77AZD-5991 Racemate
CAS :<p>AZD-5991 Racemate is the racemate of AZD-5991. (Rac)-AZD-5991 is a novel Mcl-1 inhibitor induces upregulation of BCL2,BCL-XL, CMYC and MCL1 in AML cell lines.</p>Formule :C35H34ClN5O3S2Couleur et forme :SolidMasse moléculaire :672.26LOM612
CAS :<p>LOM612 is a potent and specific FOXO relocator FOXO3a reporter protein endogenous FOXO3a and FOXO1 , down-regulates c-Myc and cyclin D1, anti-proliferative.</p>Formule :C13H10N2O2SCouleur et forme :SolidMasse moléculaire :258.3(5Z,2E)-CU-3
CAS :<p>(5Z,2E)-CU-3 is a potent and selective inhibitor of DGKα isozyme with an IC50 value of 0.6 μM and inhibition of DGKα by competing ATP with a Km value of 0.48 mM</p>Formule :C16H12N2O4S3Degré de pureté :99.02%Couleur et forme :SolidMasse moléculaire :392.47
