
Apoptose
Les inhibiteurs de l'apoptose sont des composés qui empêchent ou retardent le processus de mort cellulaire programmée, connu sous le nom d'apoptose. Ces inhibiteurs sont essentiels pour étudier les mécanismes de survie cellulaire et sont utilisés pour enquêter sur les maladies où l'apoptose est dysrégulée, telles que le cancer, les troubles neurodégénératifs et les maladies auto-immunes. En modulant l'apoptose, ces inhibiteurs peuvent aider au développement de thérapies visant à contrôler la mort cellulaire. Chez CymitQuimica, nous offrons une sélection complète d'inhibiteurs de l'apoptose de haute qualité pour soutenir vos recherches en biologie cellulaire, oncologie et domaines connexes.
Sous-catégories appartenant à la catégorie "Apoptose"
- ASK(6 produits)
- BCL(11 produits)
- Caspase(125 produits)
- FOXO1(3 produits)
- IAP(66 produits)
- Mdm2(12 produits)
- PD-1/PD-L1(125 produits)
- PDK(9 produits)
- PERK(25 produits)
- Sérine/thréonine kinase(15 produits)
- Survivant(13 produits)
- TNF(92 produits)
- c-RET(51 produits)
- p53(62 produits)
Affichez 6 plus de sous-catégories
5592 produits trouvés pour "Apoptose"
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Nebivolol hydrochloride
CAS :<p>Nebivolol hydrochloride is a beta-1 blocker and vasodilator treating hypertension and heart failure in the elderly.</p>Formule :C22H25F2NO4·HClDegré de pureté :99.77% - >99.99%Couleur et forme :White To Off-White PowderMasse moléculaire :441.90Sunitinib
CAS :<p>Sunitinib (SU 11248) is a multi-targeted receptor tyrosine kinase (RTK) inhibitor that inhibits VEGFR2 and PDGFRβ (IC50=80/2 nM).</p>Formule :C22H27FN4O2Degré de pureté :98% - 99.67%Couleur et forme :Yellow SolidMasse moléculaire :398.47Cetrimonium bromide
CAS :<p>Cetrimonium bromide (Lauroseptol) is is a mixture of different quaternary ammonium salts, which is a known component of the broad-spectrum antiseptic cetrimide.</p>Formule :C19H42BrNDegré de pureté :≥95%Couleur et forme :SolidMasse moléculaire :364.46Tirabrutinib hydrochloride
CAS :<p>Tirabrutinib hydrochloride is a potent, highly selective, irreversible oral BTK inhibitor.Cost-effective and quality-assured.</p>Formule :C25H23ClN6O3Degré de pureté :99.04% - 99.27%Couleur et forme :SolidMasse moléculaire :490.94Polyinosinic-polycytidylic acid sodium
CAS :<p>Polyinosinic-polycytidylic acid sodium (Poly(I:C) sodium) is a synthetic analog of double-stranded RNA and an agonist of toll-like receptor 3 (TLR3) and</p>Formule :(C10H13N4O8P)x·(C9H14N3O8P)x·xNaDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :695.403Onvatilimab
CAS :<p>Onvatilimab (JNJ-61610588) is a human IgG1 κ monoclonal antibody with antitumor effects for advanced head and neck cancers.</p>Degré de pureté :98.11% (SEC-HPLC) - > 95%Couleur et forme :LiquidMasse moléculaire :144.52 kDaABT-751
CAS :Formule :C18H17N3O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :371.4103Ref: IN-DA006YB9
1gÀ demander1mg50,00€5mg52,00€10mg68,00€25mg129,00€50mg150,00€100mg163,00€250mg555,00€Metamizole sodium
CAS :<p>Metamizole sodium (Analgin) is a drug that has analgesic, anti-inflammatory, and antipyretic properties. It is the sodium sulfonate of AMINOPYRINE.</p>Formule :C13H16N3NaO4SDegré de pureté :99.52%Couleur et forme :White Or Almost White Crystal PowderMasse moléculaire :333.34Ruplizumab
CAS :<p>PF-03732010 is a humanized antibody targeting P-calmodulin with antitumor and antimetastatic activity.</p>Degré de pureté :98.5% (SDS-PAGE); 98.7% (SEC-HPLC) - 98.5% (SDS-PAGE); 98.7% (SEC-HPLC)Couleur et forme :LiquidCiprofloxacin
CAS :<p>Ciprofloxacin (Bay-09867) mainly targets bacterial DNA Gyrase (IC50=0.22-0.31 µM) and topoisomerase IV (IC50=0.3-1.9 µM). antibiotic. High-Quality, Low-Cost!</p>Formule :C17H18FN3O3Degré de pureté :98.77% - 99.91%Couleur et forme :White PowderMasse moléculaire :331.34Luteolin
CAS :<p>Luteolin (Luteolol) belongs to the flavonoid group of natural products and is a Nrf2 inhibitor, PDE inhibitor.</p>Formule :C15H10O6Degré de pureté :96.61% - 99.71%Couleur et forme :SolidMasse moléculaire :286.24Novobiocin Sodium
CAS :<p>Novobiocin Sodium (Albamycinsodium) binds to DNA gyrase and blocks adenosine triphosphatase (ATPase) activity. Novobiocin sodium is an antibiotic compound.</p>Formule :C31H35N2NaO11Degré de pureté :99% - 99.28%Couleur et forme :SolidMasse moléculaire :634.61AZD4320
CAS :<p>AZD4320 inhibits BCL2/BCLxL; IC50: KPUM-MS3=26nM, KPUM-UH1=17nM, STR-428=170nM.</p>Formule :C45H48ClF3N4O7S3Degré de pureté :98.13% - 99.71%Couleur et forme :SolidMasse moléculaire :945.53Sonrotoclax TFA
<p>Sonrotoclax TFA is an orally available and highly potent and selective Bcl-2 inhibitor of WT and G101V mutants with antitumor activity for the study of hematologic malignancies.</p>Formule :C51H60F3N7O9SDegré de pureté :99.63%Couleur et forme :SolidMasse moléculaire :1004.12Terfenadine
CAS :<p>Terfenadine, metabolized to fexofenadine by CYP3A4, is a non-sedative antihistamine targeting H1 receptors.</p>Formule :C32H41NO2Degré de pureté :98.76% - 99.75%Couleur et forme :SolidMasse moléculaire :471.67Conatumumab
CAS :<p>Conatumumab (AMG 655) targets DR5 to induce apoptosis in tumors, with Kd of 1 nM (long DR5) and 0.8 nM (short DR5).</p>Degré de pureté :> 95% - > 95%Couleur et forme :LiquidMasse moléculaire :145 kDa (average)Sodium diatrizoate
CAS :<p>Sodium diatrizoate is an X-ray contrast medium for angiography, urography; may cause oxidative stress and apoptosis.</p>Formule :C11H8I3N2NaO4Degré de pureté :99.29% - 99.96%Couleur et forme :SolidMasse moléculaire :635.9Thiamine hydrochloride
CAS :<p>Thiamine hydrochloride (Vitamin B1) is an essential micronutrient and a cofactor for many central metabolic enzymes. High-Quality, Low-Cost!</p>Formule :C12H18Cl2N4OSDegré de pureté :99.63% - 99.96%Couleur et forme :White Crystal PowderMasse moléculaire :337.27Clofilium tosylate
CAS :<p>Clofilium tosylate is a potassium channel blocker, induces apoptosis on human promyelocytic leukemia (HL-60) cells.</p>Formule :C28H44ClNO3SDegré de pureté :99.68%Couleur et forme :SolidMasse moléculaire :510.17Certolizumab pegol
CAS :<p>Certolizumab pegol (Certolizumab) is a polyethylene glycolized and humanized anti-TNF-α monoclonal antibody.</p>Degré de pureté :95% - 98.2% (SDS-PAGE); 99.1% (SEC-HPLC)Couleur et forme :LiquidBenralizumab
CAS :<p>Benralizumab (MEDI-563) is a monoclonal antibody targeting the interleukin-5 receptor alpha (IL-5Rα).</p>Degré de pureté :> 95%Couleur et forme :LiquidMasse moléculaire :146.06 kDaMatrine
CAS :<p>Matrine (Vegard), an alkaloid isolated from the Sophora genus, acts as a kappa opioid receptor agonist.</p>Formule :C15H24N2ODegré de pureté :97.16% - >99.99%Couleur et forme :SolidMasse moléculaire :248.36BT-13
CAS :<p>BT-13 activates RET receptor without GFLs, fostering sensory neuron neurite growth in vitro.</p>Formule :C23H27F4N3O4SDegré de pureté :99.23%Couleur et forme :SolidMasse moléculaire :517.54Pranlukast
CAS :<p>Pranlukast (ONO-1078) is a cysteinyl leukotriene receptor-1 antagonist.</p>Formule :C27H23N5O4Degré de pureté :99.41%Couleur et forme :Off-White SolidMasse moléculaire :481.5Benzbromarone
CAS :<p>Benzbromarone (Desuric) is a CYP2C9 inhibitor with Ki value of 19.3 nM.</p>Formule :C17H12Br2O3Degré de pureté :99.37% - 99.73%Couleur et forme :SolidMasse moléculaire :424.08Hydralazine hydrochloride
CAS :<p>Hydralazine hydrochloride, an antihypertensive phthalazine, induces vasodilation and may inhibit tumor DNA methylation.</p>Formule :C8H9ClN4Degré de pureté :99.85% - 99.86%Couleur et forme :Yellow Crystals White Crystalline SolidMasse moléculaire :196.64Triclabendazole
CAS :<p>Triclabendazole (CGA89317) has been used in trials studying Parasitic Disease.</p>Formule :C14H9Cl3N2OSDegré de pureté :99.11%Couleur et forme :White To Brown Crystalline PowderMasse moléculaire :359.66Tiratricol
CAS :<p>Tiratricol, a thyroid hormone metabolite for hyperlipidemia and obesity, studied in Allan-Herndon-Dudley Syndrome treatment.</p>Formule :C14H9I3O4Degré de pureté :98.77% - 99.16%Couleur et forme :SolidMasse moléculaire :621.93CITCO
CAS :<p>CITCO, an imidazothiazole, selectively inhibits BTSCs growth with 49 nM EC50 on PXR and is a CAR agonist.</p>Formule :C19H12Cl3N3OSDegré de pureté :99.24%Couleur et forme :SolidMasse moléculaire :436.74NVP-2
CAS :<p>NVP-2 selectively inhibits CDK9 (IC50: 0.514 nM), prompts apoptosis, and affects other CDKs (IC50: 0.584-0.706 μM).</p>Formule :C27H37ClN6O2Degré de pureté :99.13%Couleur et forme :SolidMasse moléculaire :513.07Perphenazine
CAS :<p>Perphenazine (Trilafon) is a phenothiazine derivative and a dopamine antagonist with antiemetic and antipsychotic properties.</p>Formule :C21H26ClN3OSDegré de pureté :99.3% - 99.99%Couleur et forme :SolidMasse moléculaire :403.97Dihydroartemisinin
CAS :<p>Dihydroartemisinin (Artenimol) is an antimalarial drug. High-Quality, Low-Cost!</p>Formule :C15H24O5Degré de pureté :98% - 99.41%Couleur et forme :White SolidMasse moléculaire :284.35(20S)-Protopanaxadiol
CAS :<p>(20S)-Protopanaxadiol (20-Epiprotopanaxadiol) (20-Epiprotopanaxadiol), an apoptosis inducer, is an aglycon metabolic derivative of the protopanaxadiol-type</p>Formule :C30H52O3Degré de pureté :97.07% - 98.91%Couleur et forme :SolidMasse moléculaire :460.73Triclosan
CAS :<p>Triclosan (Irgasan) is an antibacterial and antifungal agent.</p>Formule :C12H7Cl3O2Degré de pureté :99.63%Couleur et forme :White Solid CrystallineMasse moléculaire :289.54Citicoline sodium
CAS :<p>Citicoline sodium aids in making phosphatidylcholine and acetylcholine, protects the brain from trauma, and improves memory.</p>Formule :C14H25N4NaO11P2Degré de pureté :99.26% - 99.37%Couleur et forme :White SolidMasse moléculaire :510.31Ecabet Sodium
CAS :<p>Ecabet Sodium (TA-2711) is a potential new agent in the management of distal colitis.</p>Formule :C20H27NaO5SDegré de pureté :99.90%Couleur et forme :SolidMasse moléculaire :402.48GPNA hydrochloride
CAS :<p>GPNA hydrochloride inhibits Gln transporter ASCT2, induces apoptosis in A549 cells, blocks SNAT1/2/4/5 & LAT1/2 transporters, and is a GGT substrate.</p>Formule :C11H14ClN3O5Degré de pureté :99.13%Couleur et forme :SolidMasse moléculaire :303.7Dasatinib
CAS :<p>Dasatinib (BMS-354825) is a tyrosine kinase inhibitor that inhibits Src and Bcr-Abl (Ki=16/30 pM) and is orally active and ATP-competitive.</p>Formule :C22H26ClN7O2SDegré de pureté :99.59% - 99.86%Couleur et forme :Pale-Yellow SolidMasse moléculaire :488.01Lercanidipine
CAS :<p>Lercanidipine (Masnidipine) is a calcium channel blocker of the dihydropyridine class.</p>Formule :C36H41N3O6Degré de pureté :99.92%Couleur et forme :White To Light Yellow SolidMasse moléculaire :611.73Abacavir
CAS :<p>Abacavir (Ziagen) is a nucleoside reverse transcriptase inhibitor analog of guanosine.</p>Formule :C14H18N6ODegré de pureté :99.36% - 99.81%Couleur et forme :White PowderMasse moléculaire :286.33Xanthone
CAS :<p>Xanthone (Xanthenone) is currently used as ovicide for codling moth eggs and as a larvicide.</p>Formule :C13H8O2Degré de pureté :99.44% - 99.86%Couleur et forme :Off-White PowderMasse moléculaire :196.2Enavatuzumab
CAS :<p>Enavatuzumab (PDL192) is a humanized monoclonal antibody targeting TWEAK receptor with anti-tumor activity.</p>Degré de pureté :>95%Couleur et forme :LiquidMyricetin
CAS :<p>Myricetin (Cannabiscetin) is a natural flavonoid and MEK1 inhibitor. Myricetin has hypoglycemic and antioxidant activities. Cost-effective and quality-assured.</p>Formule :C15H10O8Degré de pureté :97.92% - 99.85%Couleur et forme :Yellow Needles From Dilute Alcohol SolidMasse moléculaire :318.24NSC-87877
CAS :<p>NSC-87877 inhibits Shp2 (IC50=0.318μM), Shp1 (IC50=0.355μM), and DUSP26 phosphatases.</p>Formule :C19H13N3O7S2Degré de pureté :97.35%Couleur et forme :SolidMasse moléculaire :459.45Imidazole ketone erastin
CAS :<p>View and buy Imidazole ketone erastin from TargetMol.Imidazole ketone erastin (IKE) is an inducer of ferroptosis. It has inhibition of the system Xc- cystine/glutamate transporter.Cited in 22 publications.</p>Formule :C35H35ClN6O5Degré de pureté :98.48% - 99.87%Couleur et forme :SolidMasse moléculaire :655.14Adapalene
CAS :<p>Adapalene (CD271) is a dual RAR and RXR agonist, utilized in the treatment of skin conditions.</p>Formule :C28H28O3Degré de pureté :99.53% - 99.76%Couleur et forme :White To Off-White Crystalline PowderMasse moléculaire :412.52Benzenebutanoic acid, sodium salt (1:1)
CAS :Formule :C10H12NaO2Degré de pureté :%Couleur et forme :SolidMasse moléculaire :187.1909PF-4878691
CAS :<p>PF-4878691 (3M-852A) is an effective and selective Toll-like receptor 7 agonists modelled. It is used to dissociate its antiviral and inflammatory activities.</p>Formule :C17H23N5O2SDegré de pureté :98.43%Couleur et forme :SolidMasse moléculaire :361.46Escin
CAS :<p>Escin (Aescin) is biosynthesized from protoaescigenin and barringtogenol, occurring in the seeds of Aesculus.</p>Formule :C55H86O24Degré de pureté :88.51%Couleur et forme :White PowderMasse moléculaire :1131.27Vitamin K4
CAS :<p>Vitamin K4 (Menadiol Diacetate) is a vitamin medicine for the treatment of blood coagulation disorders that caused by the lack of VK4.</p>Formule :C15H14O4Degré de pureté :99.84%Couleur et forme :White Crystalline PowderMasse moléculaire :258.27Pranoprofen
CAS :<p>Pranoprofen (Pyranoprofen) (INN) is a non-steroidal anti-inflammatory drug used in ophthalmology.</p>Formule :C15H13NO3Degré de pureté :97.98% - 99.85%Couleur et forme :SolidMasse moléculaire :255.27Tadalafil
CAS :<p>Tadalafil (IC-351) is a carboline-based compound with vasodilatory activity.</p>Formule :C22H19N3O4Degré de pureté :97.03%Couleur et forme :Off-White Cyrstalline SolidMasse moléculaire :389.40Bendamustine hydrochloride
CAS :<p>Bendamustine hydrochloride (EP-3101) (IC50 of 50 μM) is an alkylating agent associated with DNA damage.</p>Formule :C16H21Cl2N3O2·HClDegré de pureté :97.71%Couleur et forme :SolidMasse moléculaire :394.72Tetrahydroxyquinone
CAS :<p>Tetrahydroxyquinone (Tetroquinone) is a primitive anticataract drug, is also a highly redox active molecule that can take part in a redox cycle.</p>Formule :C6H4O6Degré de pureté :98.15%Couleur et forme :Penetrating Odor Black SolidMasse moléculaire :172.09Daunorubicin hydrochloride
CAS :<p>Daunorubicin hydrochloride (Rubidomycin hydrochloride), an anthracycline aminoglycoside antineoplastic, inhibits DNA replication and repair and RNA and protein</p>Formule :C27H29NO10·HClDegré de pureté :96.21% - 99.53%Couleur et forme :Cancer DrugMasse moléculaire :563.99BAY 2965501
CAS :<p>BAY 2965501 is a potent and selective diacylglycerol kinase zeta (DGKζ) inhibitor that induces pERK activation.BAY 2965501 can be used in the study of cancer.</p>Formule :C20H19FN4O3SDegré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :414.45Decitabine
CAS :<p>Decitabine (Deoxycytidine) is a deoxycytidine analog, a DNA methyltransferase inhibitor with oral activity.</p>Formule :C8H12N4O4Degré de pureté :98.06% - 99.87%Couleur et forme :Physical Description Fine White Crystalline Powder Used As A DrugMasse moléculaire :228.21Mangiferin
CAS :<p>Mangiferin (Hedysarid) is used for antidiabetes. Extracted from Mangifera indica L.</p>Formule :C19H18O11Degré de pureté :99.78% - 99.86%Couleur et forme :Light Yellow PowderMasse moléculaire :422.34Catechin
CAS :<p>Catechin (Cianidanol) is a flavan-3-ol, a type of natural phenol and antioxidant.</p>Formule :C15H14O6Degré de pureté :97.34% - 99.82%Couleur et forme :SolidMasse moléculaire :290.275-Fluorouridine
CAS :<p>5-fluorouridine is also known as FUrd, 5-Fluorouracil 1-beta-D-ribofuranoside, 5-Fur, or 5-Fluoro-uridine.</p>Formule :C9H11FN2O6Degré de pureté :99.76% - 99.85%Couleur et forme :White PowderMasse moléculaire :262.19Sildenafil citrate
CAS :<p>Sildenafil citrate, a PDE5 inhibitor for erectile dysfunction and occasionally pulmonary hypertension.</p>Formule :C28H38N6O11SDegré de pureté :99.59% - 99.97%Couleur et forme :White SolidMasse moléculaire :666.70Amrinone
CAS :<p>Amrinone (Inocor) is a positive inotropic cardiotonic (cardiotonic agent) with vasodilator properties, phosphodiesterase 3 inhibitory activity.</p>Formule :C10H9N3ODegré de pureté :98.88% - 99.45%Couleur et forme :SolidMasse moléculaire :187.2Hesperetin
CAS :<p>Hesperetin belongs to the flavanone class of flavonoids.</p>Formule :C16H14O6Degré de pureté :98.45% - 99.27%Couleur et forme :SolidMasse moléculaire :302.28Acetylcysteine
CAS :<p>Acetylcysteine (NAC) is an N-acetyl derivative of cysteine, a ROS inhibitor and mucolytic agent.</p>Formule :C5H9NO3SDegré de pureté :98.01% - >99.99%Couleur et forme :Crystals From Water SolidMasse moléculaire :163.19DCZ0415
CAS :<p>DCZ0415: Potent TRIP13 inhibitor; combats myeloma in vitro, in vivo, and in drug-resistant patients; hinders DNA repair and NF-κB activity.</p>Formule :C23H20N2O2Degré de pureté :99.34% - 99.95%Couleur et forme :SolidMasse moléculaire :356.42Nortriptyline hydrochloride
CAS :<p>Nortriptyline HCl, a metabolite of amitriptyline, treats major and atypical depression, dysthymia.</p>Formule :C19H22ClNDegré de pureté :99.85% - ≥95%Couleur et forme :SolidMasse moléculaire :299.84Avobenzone
CAS :<p>Avobenzone (Butyl methoxydibenzoylmethane), an oil-soluble ingredient, is a dibenzoylmethane derivative used in sunscreen products to absorb the full spectrum</p>Formule :C20H22O3Degré de pureté :97.93%Couleur et forme :White To Pale Yellow SolidMasse moléculaire :310.39Sanguinarine chloride
CAS :<p>Sanguinarine chloride (Pseudochelerythrine chloride), a benzophenanthridine alkaloid, stimulates apoptosis by activating the production of reactive oxygen</p>Formule :C20H14ClNO4Degré de pureté :98% - 99.41%Couleur et forme :SolidMasse moléculaire :367.78Oxcarbazepine
CAS :<p>Oxcarbazepine (GP 47680), an anti-epileptic, reduces CNS disorganized electrical activity.</p>Formule :C15H12N2O2Degré de pureté :98.46%Couleur et forme :Crystals From Ethanol SolidMasse moléculaire :252.27Unesbulin
CAS :<p>Unesbulin (PTC596) is an orally active and selective inhibitor of B-cell-specific Moloney murine leukemia virus integration site 1 (BMI-1).</p>Formule :C19H13F5N6Degré de pureté :98.71%Couleur et forme :SolidMasse moléculaire :420.34Oxaprozin
CAS :<p>Oxaprozin (Oxaprozinum) is a Nonsteroidal Anti-inflammatory Drug.</p>Formule :C18H15NO3Degré de pureté :98.53%Couleur et forme :SolidMasse moléculaire :293.32Capecitabine
CAS :<p>Capecitabine is a prodrug in the antimetabolite class, transformed into cytotoxic 5-FU by tumor cells, inhibiting DNA and RNA synthesis.</p>Formule :C15H22FN3O6Degré de pureté :99.81% - >99.99%Couleur et forme :Less Solid Colourless SolidMasse moléculaire :359.355-Fluorouracil
CAS :<p>5-Fluorouracil (5-FU) is a uracil analog, an inhibitor of DNA synthesis.</p>Formule :C4H3FN2O2Degré de pureté :98% - >99.99%Couleur et forme :White To Practically White Crystalline Powder Neoplastic Drug Chemosterilant For Insects (Epa 1998)Masse moléculaire :130.08Dutasteride
CAS :<p>Dutasteride (GI 198745) is a 5-alpha-reductase inhibitor that inhibits both type-1 and type2 isoforms of the enzyme and is used to treat benign prostatic</p>Formule :C27H30F6N2O2Degré de pureté :99.58%Couleur et forme :White Crystalline SolidMasse moléculaire :528.53Eragidomide
CAS :<p>Eragidomide (Cereblon modulator 1) is a CRBN E3 ligase modulator, specifically binds to CRBN, thereby affecting the activity of the ubiquitin E3 ligase complex.</p>Formule :C22H18ClF2N3O4Degré de pureté :97.51% - 99.63%Couleur et forme :SolidMasse moléculaire :461.85Alexidine dihydrochloride
CAS :<p>Alexidine dihydrochloride: antifungal, antibiofilm, targets PTPMT1 for mitochondrial apoptosis, potential cancer treatment.</p>Formule :C26H58Cl2N10Degré de pureté :99.32% - 99.81%Couleur et forme :SolidMasse moléculaire :581.71Colchicine
CAS :<p>Colchicine (Colcin) is a natural product that is an inhibitor of microtubule polymerization (IC50=3 nM) and blocks microtubule polymerization by binding to</p>Formule :C22H25NO6Degré de pureté :98% - 99.96%Couleur et forme :Pale Yellow Scales Or Powder; Pale Yellow Needles When Crystallized From Ethyl Acetate To Light Used To Treat Gouty Arthritis Pseudogout Sarcoidal Arthritis And Calcific Tendinitis (EpaMasse moléculaire :399.44Belimumab
CAS :<p>Belimumab, a human IgG1λ monoclonal antibody, blocks BAFF, treating lupus and related fatigue.</p>Degré de pureté :SDS-PAGE:98.4%;SEC-HPLC:98.4%Couleur et forme :LiquidMasse moléculaire :144.07 kDaFSEN1
CAS :<p>FSEN1 is a novel and highly effective non-competitive FSP1 inhibitor with an IC50 value of 313 nM.</p>Formule :C22H22BrN5OSDegré de pureté :98.56% - 99.54%Couleur et forme :SolidMasse moléculaire :484.41MYCMI-6
CAS :<p>MYCMI-6 inhibits MYC:MAX, reduces tumor growth, triggers apoptosis, minimal side effects.</p>Formule :C20H19N7ODegré de pureté :99.23%Couleur et forme :SolidMasse moléculaire :373.41Perhexiline maleate
CAS :<p>Perhexiline maleate is an orally active inhibitor of CPT1 and CPT2 that reduces fatty acid metabolism.</p>Formule :C23H39NO4Degré de pureté :99.77% - ≥98%Couleur et forme :SolidMasse moléculaire :393.56MY-1076
CAS :<p>MY-1076 is a YAP inhibitor with antigastric cancer activity.MY-1076 induces G2/M phase block and apoptosis and inhibits polymerisation of microtubule proteins.</p>Formule :C29H33NO9Degré de pureté :99.57%Couleur et forme :SolidMasse moléculaire :539.57(11β)-17-(Acetyloxy)-11-[4-(dimethylamino)phenyl]-19-norpregna-4,9-diene-3,20-dione
CAS :Formule :C30H37NO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :475.6191A-1211212
CAS :<p>A-1211212 (BCL2-IN-1) is a potent and selective Bcl-2 inhibitor. It promotes lymphocyte apoptosis, alters colonic mucosa in mice, and improves inflammation.</p>Formule :C47H54ClN7O7SDegré de pureté :97.52% - 99.75%Couleur et forme :SolidMasse moléculaire :896.492-Butenamide, 2-cyano-N-(2,5-dibromophenyl)-3-hydroxy-
CAS :Formule :C11H8Br2N2O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :360.0014DT2216
CAS :<p>DT2216 inhibits various Bcl-XL-dependent leukemias and cancer cells, but is significantly less toxic to platelets.DT2216 is a selective B-cell lymphoma, extremely large (BCL-XL), proteolytic targeting chimera (PROTAC).DT2216 targets bcl-XL to the Von Hipp</p>Formule :C77H96ClF3N10O10S4Degré de pureté :99.63% - 99.78%Couleur et forme :SolidMasse moléculaire :1542.36JTE-013
CAS :<p>JTE-013 is an effective and specific antagonist of S1P2.</p>Formule :C17H19Cl2N7ODegré de pureté :97.69%Couleur et forme :SolidMasse moléculaire :408.29Adarotene
CAS :<p>Adarotene (ST1926) induces apoptosis, causes DNA damage, and has strong antiproliferative effects on human tumors.</p>Formule :C25H26O3Degré de pureté :99.26%Couleur et forme :SolidMasse moléculaire :374.47Mirodenafil
CAS :<p>Mirodenafil is a PDE-5 inhibitor developed for the treatment of erectile dysfunction.</p>Formule :C26H37N5O5SDegré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :531.671,2-dimethoxy-12-methyl[1,3]benzodioxolo[5,6-c]phenanthridiniumchloride
CAS :Formule :C21H18ClNO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :383.8249Noscapine
CAS :Formule :C22H23NO7Degré de pureté :97%Couleur et forme :SolidMasse moléculaire :413.4205Nortriptyline
CAS :<p>Nortriptyline is an antidepressant compound used for smoking cessation.</p>Formule :C19H21NDegré de pureté :99.8%Couleur et forme :SolidMasse moléculaire :263.38Butanedioic acid,mono[(2R)-3,4-dihydro-2,5,7,8-tetramethyl-2-[(4R,8R)-4,8,12-trimethyltridecyl]-2H-1-benzopyran-6-yl] ester
CAS :Formule :C33H54O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :530.7789Roxadustat
CAS :<p>Roxadustat (FG-4592) is an orally bioavailable, hypoxia-inducible factor prolyl hydroxylase inhibitor (HIF-PHI), with potential anti-anemic activity.</p>Formule :C19H16N2O5Degré de pureté :99% - 99.88%Couleur et forme :SolidMasse moléculaire :352.34AP20187
CAS :<p>AP20187: Cell-permeable ligand dimerizing FKBP fusion proteins for signaling and gene expression control.</p>Formule :C82H107N5O20Degré de pureté :99.05% - 99.80%Couleur et forme :SolidMasse moléculaire :1482.75Lirentelimab
CAS :<p>Lirentelimab (AK002) is a humanized anti-Siglec-8 antibody that induces IL-5-activated apoptosis in eosinophils and inhibits IL-5-mediated mast cell activation.</p>Degré de pureté :97.7% (SDS-PAGE); 99.7% (SEC-HPLC) - 97.7% (SDS-PAGE); 99.7% (SEC-HPLC)Couleur et forme :LiquidHydroxyurea
CAS :<p>Hydroxyurea (Hydroxycarbamide), an antineoplastic agent, inhibits DNA synthesis through the inhibition of ribonucleoside diphosphate reductase.</p>Formule :CH4N2O2Degré de pureté :99.85% - 99.92%Couleur et forme :SolidMasse moléculaire :76.05(2E)-3-[(4-Methylbenzene)sulfonyl]prop-2-enenitrile
CAS :Formule :C10H9NO2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :207.2490Tamoxifen Citrate
CAS :<p>Tamoxifen Citrate is an orally active selective estrogen receptor modulator (SERM) that blocks estrogen activity in breast cells while activating estrogen signaling in cells such as those of the bone, liver, and uterus. As an Hsp90 activator, it enhances the ATPase activity of the Hsp90 chaperone complex, induces autophagy and apoptosis, and can be used to generate gene knockout models in CreER(T2) transgenic mice as well as liver injury models.</p>Formule :C32H37NO8Degré de pureté :99.19%Couleur et forme :White To Off-White White To Off-White PowderMasse moléculaire :563.65L-Selenocystine monohydrate
CAS :Formule :C6H12N2O4Se2Degré de pureté :97%Couleur et forme :SolidMasse moléculaire :334.0905


