Cycle cellulaire/point de contrôle
Les inhibiteurs du cycle cellulaire/des points de contrôle sont des composés qui perturbent la progression normale du cycle cellulaire, en particulier aux points de contrôle régulateurs clés. Ces inhibiteurs sont cruciaux pour étudier la division cellulaire, comprendre la prolifération des cellules cancéreuses et développer des thérapies anticancéreuses. En ciblant des phases spécifiques du cycle cellulaire, ces inhibiteurs peuvent induire un arrêt du cycle cellulaire, conduisant à l'apoptose ou à la sénescence des cellules à division rapide. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de haute qualité du cycle cellulaire/des points de contrôle pour soutenir vos recherches en biologie du cancer, biologie cellulaire et développement de médicaments.
Sous-catégories appartenant à la catégorie "Cycle cellulaire/point de contrôle"
- Aurora Kinase(94 produits)
- CDK(500 produits)
- Arrêt du cycle cellulaire(4 produits)
- Chk(42 produits)
- DYRK(48 produits)
- Dynamine(23 produits)
- Ferroptose(215 produits)
- HSP(169 produits)
- Intégrine(224 produits)
- Kinésine(66 produits)
- LIM Kinase(19 produits)
- Microtubules associés(261 produits)
- PKC(102 produits)
- PLK(28 produits)
- ROCK(70 produits)
- Rho(2 produits)
- Wee1(15 produits)
- c-Myc(69 produits)
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3477 produits trouvés pour "Cycle cellulaire/point de contrôle"
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RWJ 50271
CAS :<p>RWJ 50271 inhibits LFA-1/ICAM-1 interaction with IC50 5.0 μM in HL60 cells.</p>Formule :C18H17F3N4O2SDegré de pureté :99.09%Couleur et forme :SolidMasse moléculaire :410.41MKC9989
CAS :<p>MKC9989 is an inhibitor of Hydroxy aryl aldehydes (HAA). MKC9989 also inhibits IRE1α with an IC50 of 0.23 to 44 μM.</p>Formule :C17H20O7Degré de pureté :99.3%Couleur et forme :SolidMasse moléculaire :336.34BMS-1001 hydrochloride
CAS :<p>BMS-1001 hydrochloride is an orally active inhibitor of human PD-1/PD-L1 immune checkpoint with low-toxicity in cells.BMS-1001 alleviates the inhibitory effect</p>Formule :C35H35ClN2O7Degré de pureté :97.36%Couleur et forme :SolidMasse moléculaire :631.11Nedaplatin
CAS :<p>Nedaplatin, a cisplatin derivative, induces tumor DNA damage (IC50: 94 μM) through platinum-DNA cross-links, causing apoptosis.</p>Formule :C2H8N2O3PtDegré de pureté :99.88% - >99.99%Couleur et forme :Straw Yellow PowderMasse moléculaire :303.17Ganciclovir
CAS :<p>Ganciclovir (2'-Nor-2'-deoxyguanosine) is an ACYCLOVIR analog that is a potent inhibitor of the Herpesvirus family including cytomegalovirus.</p>Formule :C9H13N5O4Degré de pureté :99.55% - 99.58%Couleur et forme :White PowderMasse moléculaire :255.23Procaine hydrochloride
CAS :<p>Procaine HCl is a benzoic acid derivative used as a local anesthetic, blocking nerve impulses and sensation.</p>Formule :C13H20N2O2·HClDegré de pureté :99.1% - 99.22%Couleur et forme :White Crystalline PowderMasse moléculaire :272.77Teplizumab
CAS :<p>Teplizumab (MGA-031) is a humanized monoclonal antibody against CD3 that slows the loss of beta cell function.Teplizumab is used to treat type 1 diabetes.</p>Degré de pureté :SDS-PAGE:95.8%;SEC-HPLC:99.7%Couleur et forme :LiquidMasse moléculaire :145.79 kDaBMVC-8C3O
CAS :<p>BMVC-8C3O is a DNA G-quadruplex (G4) ligand.Cost-effective and quality-assured.</p>Formule :C42H53I3N4O3Degré de pureté :99.72%Couleur et forme :SolidMasse moléculaire :1042.61Trimethoprim
CAS :<p>Trimethoprim (NSC-106568) inhibits dihydrofolate reductase, CYP2C8, and OCT2 - an antibacterial agent.</p>Formule :C14H18N4O3Degré de pureté :99.80% - 99.81%Couleur et forme :White To Yellowish PowderMasse moléculaire :290.32Pefloxacin Mesylate Dihydrate
CAS :<p>Pefloxacin Mesylate Dihydrate (1589 RB) , an antibacterial agent, restrains bacterial DNA replication by inhibiting DNA gyrase (topoisomerase).</p>Formule :C17H20FN3O3·CH4O3S·2H2ODegré de pureté :99.79%Couleur et forme :SolidMasse moléculaire :465.49MYCi361
CAS :<p>MYCi361 (NUCC-0196361) is an inhibitor of MYC (binding to MYC with Kd of 3.2 μM).</p>Formule :C26H16ClF9N2O2Degré de pureté :99.52%Couleur et forme :SolidMasse moléculaire :594.86KJ Pyr 9
CAS :<p>KJ Pyr 9 is an MYC inhibitor (Kd: 6.5 nM in vitro assay).</p>Formule :C22H15N3O4Degré de pureté :99.56% - ≥98%Couleur et forme :SolidMasse moléculaire :385.37Vedolizumab
CAS :<p>Vedolizumab is a humanized monoclonal antibody that targets the α4β7 integrin for the treatment of Crohn's disease and ulcerative colitis.</p>Degré de pureté :SDS-PAGE:98.4%;SEC-HPLC:99.1%Couleur et forme :LiquidMasse moléculaire :146.80 kDadAURK-4 hydrochloride
<p>dAURK-4 hydrochloride, a derivative of Alisertib, functions as a potent and selective degrader of AURKA (Aurora A), exhibiting anticancer properties [1].</p>Formule :C52H53Cl2FN8O12Degré de pureté :99.44%Couleur et forme :SolidMasse moléculaire :1071.93Rifaximin
CAS :<p>Rifaximin: an oral semi-synthetic antibiotic from rifamycin SV; targets bacterial RNA polymerase to halt growth.</p>Formule :C43H51N3O11Degré de pureté :99.18% - 99.40%Couleur et forme :Red-Orange Crystalline PowderMasse moléculaire :785.88Levofloxacin hydrate
CAS :<p>Levofloxacin hydrate (Cravit hydrate) is a third-generation fluoroquinolone antibiotic and optically active L-isomer of ofloxacin with antibacterial activity.</p>Formule :C18H20FN3O4H2ODegré de pureté :98.26%Couleur et forme :Pale Yellow SolidMasse moléculaire :370.38Otelixizumab
CAS :<p>Otelixizumab (ChAglyCD3) is a chimeric monoclonal antibody targeting CD3, used in research on Type 1 diabetes and autoimmune diseases.</p>Degré de pureté :>95%Couleur et forme :LiquidHu7691 free base
CAS :<p>Hu7691 free base is an Akt inhibitor that inhibits Akt1, Akt2 and Akt3 and induces differentiation of neuroblastoma cells.</p>Formule :C22H21F3N4ODegré de pureté :98.89%Couleur et forme :SolidMasse moléculaire :414.423Tegafur
CAS :<p>Tegafur (FT 207) is a congener of the antimetabolite fluorouracil with antineoplastic activity.</p>Formule :C8H9FN2O3Degré de pureté :99.16% - 99.89%Couleur et forme :White Crystalline PowderMasse moléculaire :200.17SIBA
CAS :<p>SIBA, a synthetic SAH analog, inhibits SAM-dependent transmethylation and blocks HSV-1 replication.</p>Formule :C14H21N5O3SDegré de pureté :99.48%Couleur et forme :SolidMasse moléculaire :339.41BAY-524
CAS :<p>BAY-524 is an inhibitor of Bub1(IC50 = 450 nM.human Bub1 in the presence of 2 mM ATP).</p>Formule :C24H24F2N6O3Degré de pureté :98.68% - 99.57%Couleur et forme :SolidMasse moléculaire :482.48Nadifloxacin
CAS :<p>Nadifloxacin (OPC7251) has been used in trials studying the treatment of Acne Vulgaris.</p>Formule :C19H21FN2O4Degré de pureté :99.03% - 99.7%Couleur et forme :Off-White Crystalline SolidMasse moléculaire :360.38Doxifluridine
CAS :<p>Doxifluridine (AMC 0101) is a fluoropyrimidine derivative and oral prodrug of the antineoplastic agent 5-fluorouracil (5-FU) with antitumor activity.</p>Formule :C9H11FN2O5Degré de pureté :99.47% - 99.86%Couleur et forme :White SolidMasse moléculaire :246.19CDK4/6-IN-2
CAS :<p>CDK4/6-IN-2 是一种CDK4和CDK6抑制剂，IC50分别为 2.7 和 16 nM。</p>Formule :C27H32F2N8Degré de pureté :99.47%Couleur et forme :SolidMasse moléculaire :506.59Folinic acid calcium
CAS :<p>Folinic acid calcium (Leucovorin Calcium) is the active metabolite of folic acid. Leucovorin is used principally as an antidote to folic acid antagonists.</p>Formule :C20H21CaN7O7Degré de pureté :98.72% - >99.99%Couleur et forme :Yellow Crystalline PowderMasse moléculaire :511.51Kira8
CAS :<p>Kira8 (AMG-18) is a mono-selective IRE1α inhibitor that allosterically attenuates IRE1α RNase activity (IC50: 5.9 nM).</p>Formule :C31H29ClN6O3SDegré de pureté :98.07%Couleur et forme :SolidMasse moléculaire :601.12MBQ-167
CAS :<p>MBQ-167 is a dual inhibitor of Rac/Cdc42 (IC50s: 103 nM for Rac 1/2/3 and 78 nM for Cdc42 in MDA-MB-231 cells, respectively).</p>Formule :C22H18N4Degré de pureté :98.07% - 99.52%Couleur et forme :SolidMasse moléculaire :338.41BOS-172722
CAS :<p>BOS-172722 is an inhibitor of monopolar spindle 1 (MPS1) checkpoint(IC50 of 2 nM).</p>Formule :C24H30N8ODegré de pureté :99.37%Couleur et forme :SolidMasse moléculaire :446.55Enoxacin
CAS :<p>Enoxacin (NSC-629661) is a broad-spectrum 6-fluoronaphthyridinone antibacterial agent (fluoroquinolones) structurally related to nalidixic acid.</p>Formule :C15H17FN4O3Degré de pureté :98.68% - 99.89%Couleur et forme :Off-White To Yellow CrystalsMasse moléculaire :320.32Folinic Acid Calcium Salt Pentahydrate
CAS :<p>Folinic Acid Calcium Salt Pentahydrate (Leucovorin Calcium Pentahydrate), a reduced folic acid, is used in combination with other chemotherapeutics.</p>Formule :C20H21CaN7O7·5H2ODegré de pureté :99.17% - >99.99%Couleur et forme :Yellowish-White To Yellow PowderMasse moléculaire :601.58Tadocizumab
CAS :<p>Tadocizumab (C4G1) is a humanized monoclonal antibody targeting integrin αIIbβ3 with antiplatelet and antithrombotic effects.</p>Degré de pureté :97.1% (SDS-PAGE); 97.2% (SEC-HPLC) - 97.1% (SDS-PAGE); 97.2% (SEC-HPLC)Couleur et forme :LiquidCibisatamab
CAS :<p>Cibisatamab, a T-cell bispecific antibody, targets CEA on cancer cells and CD3 on T-cells, inducing T-cell-mediated tumor cell killing.</p>Degré de pureté :SDS-PAGE:99.1%;SEC-HPLC:96.5%Couleur et forme :LiquidMasse moléculaire :191.1 kDaButylparaben
CAS :<p>Butylparaben (Butyl 4-hydroxybenzoate) is a standardized chemical allergen, increasing histamine release, and cell-mediated immunity.</p>Formule :C11H14O3Degré de pureté :98.15%Couleur et forme :Small Colorless Crystals Or Powder Tongue Aqueous Solutions Slightly Acidic To Litmus (Ntp 1992)Masse moléculaire :194.23HLM006474
CAS :<p>HLM006474 is a pan inhibitor of E2F. This inhibits E2F4 DNA-binding (IC50: 29.8 μM in A375 cells).</p>Formule :C25H25N3O2Degré de pureté :98.45% - 99.04%Couleur et forme :SolidMasse moléculaire :399.48Procaine
CAS :<p>Procaine (Vitamin H3) is a slow-acting ester local anesthetic with a short effect, used for infiltration, nerve, and spinal blocks.</p>Formule :C13H20N2O2Degré de pureté :99.57% - 99.73%Couleur et forme :Anhydrous Plates Tables From Ligroin Or Ether SolidMasse moléculaire :236.31Tidutamab
CAS :<p>Tidutamab (XmAb-18087) is a humanized bispecific antibody targeting the growth inhibitory receptor 2 (SSTR2) and T cell binding domain (CD3).</p>Degré de pureté :97.9% (SDS-PAGE); 97.8% (SEC-HPLC) - 97.9% (SDS-PAGE); 97.8% (SEC-HPLC)Couleur et forme :LiquidATN-161 trifluoroacetate salt
CAS :<p>ATN-161 TFA salt, a new integrin α5β1 inhibitor, curbs angiogenesis, liver metastases growth, enhances survival in mice.</p>Formule :C25H36F3N9O10SDegré de pureté :98% - 99.98%Couleur et forme :SolidMasse moléculaire :711.67Foralumab
CAS :<p>Foralumab (NI-0401) is a human anti-CD3 monoclonal antibody for the study of COVID-19 infection.</p>Degré de pureté :96.7% (SDS-PAGE); 96.4% (SEC-HPLC) - 96.7% (SDS-PAGE); 96.4% (SEC-HPLC)Couleur et forme :LiquidOrbofiban TFA
CAS :<p>Orbofiban TFA is an orally active GPIIb/IIIa platelet receptor antagonist with inhibitory effects on platelet aggregation for the study of unstable coronary</p>Formule :C19H24F3N5O6Degré de pureté :97.21% - 98.72%Couleur et forme :SolidMasse moléculaire :475.42MKC8866
CAS :<p>MKC8866, a selective IRE1 RNase inhibitor with an IC50 of 0.29 μM, curbs breast and prostate cancer cell growth.</p>Formule :C18H19NO7Degré de pureté :99.28% - 99.854%Couleur et forme :SolidMasse moléculaire :361.35Rifapentine
CAS :<p>Rifapentine (Rifapentinum) is a long-acting, cyclopentyl-substituted derivative of rifamycin used to treat mycobacterium infections.</p>Formule :C47H64N4O12Degré de pureté :95.74% - ≥98%Couleur et forme :SolidMasse moléculaire :877.03TK216
CAS :<p>TK216 is a potent inhibitor of E26 transformation-specific (ETS) with anticancer activity.</p>Formule :C19H15Cl2NO3Degré de pureté :97.22%Couleur et forme :SolidMasse moléculaire :376.23Monalizumab
CAS :<p>Monalizumab, a humanized antibody, enhances NK cell function by inhibiting NKG2A; used in HNSCC studies.</p>Degré de pureté :95% - > 95%Couleur et forme :LiquidMasse moléculaire :147 kDa (average)NMDI14
CAS :<p>NMDI14 is an inhibitor of nonsense mediated RNA decay (NMD).</p>Formule :C21H25N3O4SDegré de pureté :97.79% - 99.37%Couleur et forme :SolidMasse moléculaire :415.51DNA2 inhibitor C5
CAS :<p>DNA2 inhibitor C5 is a specific cancer sensitizer with an IC50 of 20 μM, targeting multiple DNA2 activities.</p>Formule :C10H6N2O5Degré de pureté :99.05%Couleur et forme :SolidMasse moléculaire :234.16Pazufloxacin Mesylate
CAS :<p>Pazufloxacin Mesylate (T-3762) is a fluoroquinolone antibiotic.</p>Formule :C16H15FN2O4·CH4O3SDegré de pureté :99.88% - 99.93%Couleur et forme :Crystalline SolidMasse moléculaire :414.4RG7800
CAS :<p>RG7800 (RO6885247) has the potential for spinal muscular atrophy treatment. RG7800 is an SMN2 splicing modifier.</p>Formule :C24H28N6ODegré de pureté :99.44%Couleur et forme :SolidMasse moléculaire :416.52PZL-A
CAS :<p>PZL-A, PZL-A, an activator of mtDNA synthesis, restored the activity of POLγ mutant variant.</p>Formule :C19H17ClN4O2Degré de pureté :99.88%Couleur et forme :SoildMasse moléculaire :368.82CMPD101
CAS :<p>CMPD101 is a membrane-permeable small-molecule inhibitor of GRK2/3 (IC50: 18 nM and 5.4 nM).</p>Formule :C24H21F3N6ODegré de pureté :99.01% - 99.04%Couleur et forme :SolidMasse moléculaire :466.46Oxolinic acid
CAS :<p>Oxolinic acid (Nidantin) is a synthetic antimicrobial related to NALIDIXIC ACID and used in URINARY TRACT INFECTIONS.</p>Formule :C13H11NO5Degré de pureté :98.39% - 99.72%Couleur et forme :Crystals From Dimethylformamide White Crystalline PowderMasse moléculaire :261.23Abituzumab
CAS :<p>Abituzumab (DI17E6) is a humanized monoclonal antibody targeting integrin alphaV, exhibiting anti-cancer activity and can be used in prostate cancer research.</p>Degré de pureté :>95%Couleur et forme :LiquidBersanlimab
CAS :<p>Bersanlimab (BI-505) is a fully human monoclonal antibody targeting Intercellular Adhesion Molecule-1 (ICAM-1).Bersanlimab has anticancer properties.</p>Degré de pureté :> 95% - > 95%Couleur et forme :LiquidMasse moléculaire :144.22 kDaCHK1-IN-4 hydrochloride
<p>CHK1-IN-4 hydrochloride is a potent inhibitor of checkpoint kinase 1 (chk1).</p>Formule :C18H19BrClN7O2Degré de pureté :99.29%Couleur et forme :SoildMasse moléculaire :480.75Ribociclib succinate
CAS :<p>Ribociclib succinate (LEE011 succinate) is a highly specific CDK4/6 inhibitor (IC50: 10 nM and 39 nM, respectively).</p>Formule :C27H36N8O5Degré de pureté :99.9%Couleur et forme :SolidMasse moléculaire :552.63JH-RE-06
CAS :<p>JH-RE-06 disrupts mutagenic translesion synthesis (TLS) by preventing the recruitment of mutagenic POLζ.</p>Formule :C20H16Cl3N3O4Degré de pureté :99.29%Couleur et forme :SolidMasse moléculaire :468.72Cinoxacin
CAS :<p>Cinoxacin (Compound 64716), an older synthetic antimicrobial, was related to the quinolone class of antibiotics.</p>Formule :C12H10N2O5Degré de pureté :99.62% - 99.98%Couleur et forme :SolidMasse moléculaire :262.22Danofloxacin mesylate
CAS :<p>Danofloxacin mesylate (CP 76136-27) is a synthetic antibacterial agent of the fluoroquinolone class, acts principally by the inhibition of bacterial DNA-gyrase.</p>Formule :C19H20FN3O3·CH4O3SDegré de pureté :99.73%Couleur et forme :Crystalline SolidMasse moléculaire :453.48Valacyclovir hydrochloride
CAS :<p>Valacyclovir hydrochloride (Valaciclovir hydrochloride) is an acyclovir prodrug that inhibits viral DNA replication after metabolization.</p>Formule :C13H20N6O4·HClDegré de pureté :98.65% - ≥95%Couleur et forme :White To Off-White Crystalline PowerMasse moléculaire :360.80Mps1-IN-3
CAS :<p>Mps1-IN-3 is an effective and selective inhibitor of MPS1 kinase (IC50: 50 nM).</p>Formule :C26H31N7O4SDegré de pureté :99.25%Couleur et forme :SolidMasse moléculaire :537.63ART558
CAS :<p>ART558 is a potent, selective, low molecular weight, allosteric DNA polymerase activity of Polθ inhibitor (IC50=7.9 nM).</p>Formule :C21H21F3N4O2Degré de pureté :99.18% - 99.67%Couleur et forme :SolidMasse moléculaire :418.41Simurosertib
CAS :<p>Simurosertib (TAK-931) is a selective and ATP-competitive cell division cycle 7 kinase inhibitor (IC50: <0.3 nM).</p>Formule :C17H19N5OSDegré de pureté :99.93% - 99.93%Couleur et forme :SolidMasse moléculaire :341.43Elarofiban TFA
CAS :<p>Elarofiban TFA (RWJ-53308 TFA) is a novel and orally active and selective GPIIb/IIIa antagonist for the study of cardiovascular disease.</p>Formule :C26H34F6N4O8Degré de pureté :99.08%Couleur et forme :SoildMasse moléculaire :644.56GSK-1520489A
CAS :<p>GSK-1520489A is an active PKMYT1 inhibitor.</p>Formule :C21H23N5O3SDegré de pureté :99.85%Couleur et forme :SolidMasse moléculaire :425.5Abrilumab
CAS :<p>Abrilumab (MEDI-7183) is a fully human monoclonal antibody against α4β7 that inhibits the α4β7 integrin.</p>Degré de pureté :98.5% (SDS-PAGE); 99% (SEC-HPLC) - 98.5% (SDS-PAGE); 99% (SEC-HPLC)Couleur et forme :LiquidCeftriaxone sodium hydrate
CAS :<p>Ceftriaxone sodium hydrate is a broad-spectrum cephalosporin antibiotic with a very long half-life and high penetrability to meninges, eyes and inner ears.</p>Formule :C18H16N8Na2O7S3·5H2ODegré de pureté :99.77% - 99.78%Couleur et forme :White Or Almost White Crystalline Powder OdorlessMasse moléculaire :661.6Cyclin K degrader 1
<p>Cyclin K degrader 1 is a Cyclin K degrader.Cyclin K degrader 1 is a degrader converted from AT-7519.Cyclin K degrader 1 has weak degrading activity against Cyclin K but does not result in a sustained decrease in degradation affinity.Cyclin K degrader 1 is a degrader converted from AT-7519.</p>Formule :C23H17Cl2N5O2Degré de pureté :99.76%Couleur et forme :SolidMasse moléculaire :466.32NU6140
CAS :<p>NU6140 is a selective inhibitor of CDK2-cyclin A (IC50, 0.41 μM).</p>Formule :C23H30N6O2Degré de pureté :98.33%Couleur et forme :SolidMasse moléculaire :422.52Gemifloxacin mesylate
CAS :<p>Gemifloxacin mesylate (Gemifloxacin mesylate) inhibits activities of DNA gyrase and topoisomerase IV, thereby inhibiting DNA replication and eventually</p>Formule :C19H24FN5O7SDegré de pureté :97.24% - ≥95%Couleur et forme :Beige SolidMasse moléculaire :485.49hSMG-1 inhibitor 11j
CAS :<p>hSMG-1 inhibitor 11j: pyrimidine, IC50=0.11 nM, >455x selective vs. mTOR/PI3Kα/γ/CDK1/CDK2; cancer research use.</p>Formule :C27H28ClN7O3SDegré de pureté :99.22% - 99.65%Couleur et forme :SolidMasse moléculaire :566.07LY 345899
CAS :<p>LY 345899 is a Folate analog and is a methylenetetrahydrofolate dehydrogenase and MTHFD2 inhibitor (IC50: 96 nM and 663 nM, respectively and a Ki: 18 nM for</p>Formule :C20H21N7O7Degré de pureté :99.7%Couleur et forme :SolidMasse moléculaire :471.42BT173
CAS :<p>BT173 is a novel inhibitor of homeodomain interacting protein kinase 2 (HIPK2 ), attenuating renal fibrosis through suppression of the TGF-ß1/Smad3 pathway.</p>Formule :C18H12BrN3O2Degré de pureté :98.247%Couleur et forme :SolidMasse moléculaire :382.21TAO Kinase inhibitor 2
CAS :<p>TAO Kinase inhibitor 2 is a TAO kinase inhibitor with an IC50 of 50-500 nM. TAO Kinase inhibitor 2 inhibits KIAA1361 and JIK with IC50s of 50-500 nM.</p>Formule :C25H24N2O3Degré de pureté :98.58%Couleur et forme :SoildMasse moléculaire :400.47Avotaciclib
CAS :<p>Avotaciclib (BEY1107) is a potent and orally active cyclin dependent kinase 1 (CDK1) inhibitor.Avotaciclib can be used to study locally advanced or metastatic</p>Formule :C13H11N7ODegré de pureté :98.02%Couleur et forme :SolidMasse moléculaire :281.27Enrofloxacin
CAS :<p>Enrofloxacin (BAY-Vp2674) is a veterinary antibacterial agent, used in poultry.</p>Formule :C19H22FN3O3Degré de pureté :99.43% - >99.99%Couleur et forme :Pale Yellow CrystalsMasse moléculaire :359.39Trilaciclib hydrochloride
CAS :<p>Trilaciclib hydrochloride (G1T28 hydrochloride) is an inhibitor of CDK4/6 (IC50s: 1 nM and 4 nM for CDK4 and CDK6).</p>Formule :C24H32Cl2N8ODegré de pureté :99.69% - 99.89%Couleur et forme :SolidMasse moléculaire :519.47Lerociclib dihydrochloride
CAS :<p>Lerociclib dihydrochloride (G1T38 dihydrochloride) is a potent and selective inhibitor of CDK4/CDK6, with IC50s of 2 nM and 1 nM for CDK6/CyclinD3 and CDK4/</p>Formule :C26H36Cl2N8ODegré de pureté :97.4%Couleur et forme :SolidMasse moléculaire :547.52Hycanthone
CAS :<p>Hycanthone (Etrenol(mesylate)) is a potent drug of antischistosomal.</p>Formule :C20H24N2O2SDegré de pureté :98.78%Couleur et forme :Yellow-Orange Powder (Ntp 1992)Masse moléculaire :356.48Carmofur
CAS :<p>Carmofur (HCFU) is a highly potent acid ceramidase inhibitor, used in the treatment of breast and colorectal cancer.</p>Formule :C11H16FN3O3Degré de pureté :98.53% - 99.98%Couleur et forme :SolidMasse moléculaire :257.26TAK-901
CAS :<p>TAK-901 has been used in trials studying the treatment of Lymphoma, Myelofibrosis, Multiple Myeloma, Myeloid Metaplasia, and Advanced Solid Tumors, among others</p>Formule :C28H32N4O3SDegré de pureté :99.02% - 99.59%Couleur et forme :SolidMasse moléculaire :504.64SU056
CAS :<p>SU056 is a YB-1 inhibitor that induces cell-cycle arrest, apoptosis, and inhibits ovarian cancer cell migration.</p>Formule :C20H16FNO5Degré de pureté :99.89%Couleur et forme :SoildMasse moléculaire :369.34MYCi975
CAS :<p>MYCi975 (NUCC-0200975) is an orally active inhibitor of MYC.</p>Formule :C25H16Cl2F6N2O2Degré de pureté :99.3% - 99.82%Couleur et forme :SolidMasse moléculaire :561.3Vitamin D2
CAS :<p>Ergocaliferol (Vitamin D2), derived from ergosterol by UV, inhibits bladder tumor promotion and leukemia, and blocks DNA Polymerase.</p>Formule :C28H44ODegré de pureté :98.73% - 99.89%Couleur et forme :Prisms From Acetone 1998)Masse moléculaire :396.65R-10015
CAS :<p>R-10015, potent LIMK inhibitor with 38 nM IC50 for LIMK1, targets ATP pocket, and serves as a broad-spectrum HIV antiviral.</p>Formule :C20H19ClN6O2Degré de pureté :98.68%Couleur et forme :SolidMasse moléculaire :410.86Abciximab
CAS :<p>Abciximab: chimeric antibody, anti-platelet, blocks glycoprotein IIb/IIIa, vitronectin, Mac-1.</p>Degré de pureté :SDS-PAGE:95.2%;SEC-HPLC:95.9%Couleur et forme :LiquidMasse moléculaire :95.18 kDaEfalizumab
CAS :<p>Efalizumab: humanized monoclonal antibody CD11a; modulates T cell activation/adhesion; for plaque psoriasis, psoriatic arthritis research.</p>Degré de pureté :SDS-PAGE:95% SEC-HPLC:98.77%Couleur et forme :LiquidMasse moléculaire :146.14 kDaCirtuvivint
CAS :<p>Cirtuvivint (SM08502) is a potent and orally active CDC-like kinase (CLK) inhibitor that can be used to study arthritis.</p>Formule :C24H25N7ODegré de pureté :99.46% - >99.99%Couleur et forme :SolidMasse moléculaire :427.5Centrinone
CAS :<p>Centrinone (LCR-263) (LCR-263) is a reversible inhibitor of polo-like kinase 4 (PLK4; Ki:0.16 nM).</p>Formule :C26H25F2N7O6S2Degré de pureté :98.76%Couleur et forme :SolidMasse moléculaire :633.65Paprotrain
CAS :<p>Paprotrain ((alphaZ)-alpha-(3-Pyridinylmethylene)-1H-indole-3-acetonitrile) inhibits the ATPase activity of MKLP-2 with an IC50 of 1.35 μM and a Ki of 3.36 μM.</p>Formule :C16H11N3Degré de pureté :99.91%Couleur et forme :SolidMasse moléculaire :245.28XPW1
CAS :<p>XPW1 is a CDK9 inhibitor with antitumor activity, inhibits DNA repair procedures, and can be used for the research of clear cell renal cell carcinoma.</p>Formule :C36H39ClFN7O2Degré de pureté :98.08%Couleur et forme :SoildMasse moléculaire :656.19DI-87
CAS :<p>DI-87 (TRE-515) is a novel and orally available dCK (deoxycytidine kinase) inhibitor. DI-87 binds to dCK reduces the production of dNTP inhibits tumor growth.</p>Formule :C23H30N6O3S2Degré de pureté :99.76%Couleur et forme :SolidMasse moléculaire :502.656-Mercaptopurine
CAS :<p>6-Mercaptopurine (6-MP) is an antimetabolite antineoplastic agent with immunosuppressant properties.</p>Formule :C5H4N4SDegré de pureté :99.53% - 99.63%Couleur et forme :Yellow Crystalline Powder SolidMasse moléculaire :152.18Metarrestin
CAS :<p>Metarrestin (ML246) is a first-in-class perinucleolar compartment inhibitor with a favorable PK profile, which effectively suppresses metastasis.</p>Formule :C31H30N4ODegré de pureté :99.45%Couleur et forme :SolidMasse moléculaire :474.6N-Dodecyl-β-D-maltoside
CAS :<p>N-Dodecyl-β-D-maltoside (Lauryl Maltoside) has also been employed in applications such as in the purification and stabilization of RNA polymerase and the</p>Formule :C24H46O11Degré de pureté :99.7% - >99.99%Couleur et forme :White PowderMasse moléculaire :510.62MALAT1-IN-1
CAS :<p>MALAT1-IN-1 is an effective dose-dependent Malat1 inhibitor, not altering Neat1 expression.</p>Formule :C19H21N3O2Degré de pureté :99.58%Couleur et forme :SolidMasse moléculaire :323.39CDK2-IN-4
CAS :<p>CDK2-IN-4 is a potent and selective inhibitor of CDK2 with an IC50 of 44 nM for CDK2/cyclin A.</p>Formule :C23H18N6O2SDegré de pureté :97.24% - 99.10%Couleur et forme :SolidMasse moléculaire :442.49Ribavirin
CAS :<p>Ribavirin (Tribavirin) is a synthetic nucleoside analog of ribofuranose with activity against hepatitis C virus and other RNA viruses.</p>Formule :C8H12N4O5Degré de pureté :99.09% - 99.83%Couleur et forme :Less Solid Colourless SolidMasse moléculaire :244.20Famciclovir
CAS :<p>Famciclovir (BRL 42810) inhibits Herpes virus DNA polymerase by mimicking nucleosides.</p>Formule :C14H19N5O4Degré de pureté :99.85%Couleur et forme :Off-White PowderMasse moléculaire :321.33N4-Benzoyl-3'-O-DMT-2'-O-(2-methoxyethyl)-5-methylcytidine
<p>N4-Benzoyl-3'-O-DMT cytidine analog inhibits DNA methyltransferases like Zebularine.</p>Formule :C41H43N3O9Couleur et forme :SolidMasse moléculaire :721.79Clofarabine-5'-triphosphate
CAS :<p>Clofarabine-5'-triphosphate is a metabolite of Clofarabine, produced via phosphorylation by deoxycytidine kinase (dCK). It exhibits cytotoxicity in cancer cells by inhibiting DNA synthesis and DNA repair.</p>Formule :C10H14ClFN5O12P3Couleur et forme :SolidMasse moléculaire :543.62Erythromycin thiocyanate
CAS :<p>Erythromycin thiocyanate, a macrolide from Streptomyces erythreus, binds 50S ribosomes, halting protein synthesis in bacteria.</p>Formule :C38H68N2O13SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :793.02
