
Cycle cellulaire/point de contrôle
Sous-catégories appartenant à la catégorie "Cycle cellulaire/point de contrôle"
- Aurora Kinase(114 produits)
- CDK(545 produits)
- Arrêt du cycle cellulaire(5 produits)
- Chk(48 produits)
- DYRK(47 produits)
- Dynamine(27 produits)
- Ferroptose(226 produits)
- HSP(179 produits)
- Intégrine(249 produits)
- Kinésine(87 produits)
- LIM Kinase(20 produits)
- Microtubules associés(274 produits)
- PKC(124 produits)
- PLK(25 produits)
- ROCK(62 produits)
- Rho(6 produits)
- Wee1(14 produits)
- c-Myc(76 produits)
3859 produits trouvés pour "Cycle cellulaire/point de contrôle"
TH1760
CAS :TH1760 inhibits NUDT15 (IC50=25nM); boosts 6-thioguanine efficacy in leukemia by raising 6-thio-(d)GTP.Formule :C20H18N4O5SDegré de pureté :97.31%Couleur et forme :SoildMasse moléculaire :426.45Sulfameter
CAS :Sulfameter (Sulfametoxydiazine) is a long-acting sulfonamide antibacterial agent used to treat urinary tract infections and leprosy.Formule :C11H12N4O3SDegré de pureté :99.46% - 99.90%Couleur et forme :Crystalline SolidMasse moléculaire :280.3Tegafur
CAS :Tegafur (FT 207) is a congener of the antimetabolite fluorouracil with antineoplastic activity.Formule :C8H9FN2O3Degré de pureté :99.16% - 99.89%Couleur et forme :White Crystalline PowderMasse moléculaire :200.17Upamostat
CAS :Upamostat is an inhibitor of a serine protease and is a urokinase plasminogen activator (uPA) inhibitor.Formule :C32H47N5O6SDegré de pureté :99.41%Couleur et forme :SolidMasse moléculaire :629.81Ref: TM-T13257
1mg64,00€2mg94,00€5mg145,00€10mg226,00€25mg379,00€50mg538,00€100mg730,00€1mL*10mM (DMSO)163,00€ATN-161 acetate
CAS :ATN-161 acetate, a pentapeptide compound derived from the synergistic region of fibronectin, is an integrin-alpha5 antagonist with antitumor activity.Formule :C25H39N9O10SDegré de pureté :98.27%Couleur et forme :SoildMasse moléculaire :657.7Ref: TM-T10398L
1mg190,00€5mg471,00€10mg663,00€25mg1.036,00€50mg1.429,00€100mg1.830,00€200mg2.498,00€Abituzumab
CAS :Abituzumab (DI17E6) is a humanized monoclonal antibody targeting integrin alphaV, exhibiting anti-cancer activity and can be used in prostate cancer research.Degré de pureté :>95%Couleur et forme :LiquidMasse moléculaire :144.58 kDaBT173
CAS :BT173 is a novel inhibitor of homeodomain interacting protein kinase 2 (HIPK2 ), attenuating renal fibrosis through suppression of the TGF-ß1/Smad3 pathway.Formule :C18H12BrN3O2Degré de pureté :98.247%Couleur et forme :SolidMasse moléculaire :382.21MKC8866
CAS :MKC8866, a selective IRE1 RNase inhibitor with an IC50 of 0.29 μM, curbs breast and prostate cancer cell growth.Formule :C18H19NO7Degré de pureté :99.28% - 99.854%Couleur et forme :SolidMasse moléculaire :361.35Ref: TM-T15594
1mg84,00€2mg109,00€5mg177,00€10mg250,00€25mg423,00€50mg557,00€100mg760,00€200mg1.018,00€1mL*10mM (DMSO)192,00€N-Dodecyl-β-D-maltoside
CAS :N-Dodecyl-β-D-maltoside (Lauryl Maltoside) has also been employed in applications such as in the purification and stabilization of RNA polymerase and theFormule :C24H46O11Degré de pureté :99.18% - >99.99%Couleur et forme :White PowderMasse moléculaire :510.62Tinengotinib
CAS :Tinengotinib is a multikinase inhibitor that targets a series of kinases , including Aurora kinases A/B, JAK1/2, FGFR1/2/3, VEGFRs, and many other kinases.Formule :C20H19ClN6ODegré de pureté :99.05%Couleur et forme :SolidMasse moléculaire :394.86Osalmid
CAS :Osalmid (Oxaphenamide) is a choleretic drug, inhibits ribonucleotide reductase activity by targeting ribonucleotide reductase small subunit M2 (RRM2).Formule :C13H11NO3Degré de pureté :99.08% - 99.6%Couleur et forme :White CrystalMasse moléculaire :229.23Foscarnet sodium
CAS :Foscarnet sodium (Phosphonoformate) is an antiviral agent used in the treatment of cytomegalovirus retinitis.Formule :CNa3O5PDegré de pureté :98.52%Couleur et forme :White Or Almost White Crystalline PowderMasse moléculaire :191.95Doxifluridine
CAS :Doxifluridine (AMC 0101) is a fluoropyrimidine derivative and oral prodrug of the antineoplastic agent 5-fluorouracil (5-FU) with antitumor activity.Formule :C9H11FN2O5Degré de pureté :99.47% - 99.86%Couleur et forme :White SolidMasse moléculaire :246.19Foralumab
CAS :Foralumab (NI-0401) is a human anti-CD3 monoclonal antibody for the study of COVID-19 infection.Degré de pureté :96.7% (SDS-PAGE); 96.4% (SEC-HPLC) - 96.7% (SDS-PAGE); 96.4% (SEC-HPLC)Couleur et forme :LiquidMasse moléculaire :146.59 kDaGemifloxacin mesylate
CAS :Gemifloxacin mesylate (Gemifloxacin mesylate) inhibits activities of DNA gyrase and topoisomerase IV, thereby inhibiting DNA replication and eventuallyFormule :C19H24FN5O7SDegré de pureté :97.24% - ≥95%Couleur et forme :Beige SolidMasse moléculaire :485.49Teplizumab
CAS :Teplizumab (MGA-031) is a humanized monoclonal antibody against CD3 that slows the loss of beta cell function.Teplizumab is used to treat type 1 diabetes.Degré de pureté :SDS-PAGE:95.8%;SEC-HPLC:99.7%Couleur et forme :LiquidMasse moléculaire :145.79 kDaCarmofur
CAS :Carmofur (HCFU) is a highly potent acid ceramidase inhibitor, used in the treatment of breast and colorectal cancer.Formule :C11H16FN3O3Degré de pureté :98.53% - 99.98%Couleur et forme :SolidMasse moléculaire :257.26Orbofiban TFA
CAS :Orbofiban TFA is an orally active GPIIb/IIIa platelet receptor antagonist with inhibitory effects on platelet aggregation for the study of unstable coronaryFormule :C19H24F3N5O6Degré de pureté :97.21% - 98.72%Couleur et forme :SolidMasse moléculaire :475.42Centrinone
CAS :Centrinone (LCR-263) (LCR-263) is a reversible inhibitor of polo-like kinase 4 (PLK4; Ki:0.16 nM).Formule :C26H25F2N7O6S2Degré de pureté :98.76%Couleur et forme :SolidMasse moléculaire :633.65DNA2 inhibitor C5
CAS :DNA2 inhibitor C5 is a specific cancer sensitizer with an IC50 of 20 μM, targeting multiple DNA2 activities.Formule :C10H6N2O5Degré de pureté :99.05%Couleur et forme :SolidMasse moléculaire :234.16Ref: TM-T15146
1mg57,00€2mg80,00€5mg113,00€10mg178,00€25mg409,00€50mg605,00€100mg860,00€500mg1.728,00€1mL*10mM (DMSO)112,00€RWJ 50271
CAS :RWJ 50271 inhibits LFA-1/ICAM-1 interaction with IC50 5.0 μM in HL60 cells.Formule :C18H17F3N4O2SDegré de pureté :99.09%Couleur et forme :SolidMasse moléculaire :410.41Ref: TM-T12783
1mg120,00€5mg295,00€10mg447,00€25mg707,00€50mg964,00€100mg1.243,00€200mg1.693,00€1mL*10mM (DMSO)326,00€Ledoxantrone trihydrochloride
CAS :Ledoxantrone trihydrochloride is a Top II inhibitor with anticancer activity and is used in the study of digestive disorders and urologic disorders.Formule :C21H30Cl3N5OSDegré de pureté :98.13%Couleur et forme :SoildMasse moléculaire :506.92Arg-Gly-Asp-Ser acetate
Arg-Gly-Asp-Ser acetate targets integrin, binding pro-caspase-8, -9, -3, but not -1; inhibits receptor function.Formule :C17H31N7O10Degré de pureté :98.14%Couleur et forme :SolidMasse moléculaire :493.47GRL0617
CAS :GRL0617 is a selective and competitive SARS-CoVPLpro and deubiquitinase noncovalent inhibitor(IC50 : 0.6 μM, Ki : 0.49 μM).Formule :C20H20N2ODegré de pureté :99.31%Couleur et forme :SolidMasse moléculaire :304.39Ref: TM-T11464
1mg34,00€5mg74,00€10mg105,00€25mg178,00€50mg313,00€100mg500,00€500mg1.063,00€1mL*10mM (DMSO)82,00€P 218
CAS :P 218 is a novel DHFR inhibitor with antimalarial activity and antifolate effects and can be used to study Buruli ulcer.Formule :C18H25ClN4O4Degré de pureté :98.83%Couleur et forme :SoildMasse moléculaire :396.87Procarbazine hydrochloride
CAS :Procarbazine hydrochloride (NSC-77213 HCl) is the hydrochloride salt of a methylhydrazine derivative with antineoplastic and mutagenic activities.Formule :C12H19N3O·HClDegré de pureté :96.99% - ≥98%Couleur et forme :(Ntp 1992)Masse moléculaire :257.76Rifabutin
CAS :Rifabutin (LM-427), a semisynthetic ansamycin, blocks bacterial RNA synthesis by inhibiting RNA polymerase.Formule :C46H62N4O11Degré de pureté :98.87% - 99.7%Couleur et forme :Red-Violet Crystalline PowderMasse moléculaire :847.00C527
CAS :C527 is a is a pan DUB enzyme inhibitor. Which has a high potency for the USP1/UAF1 complex (IC50=0.88 μM).Formule :C17H8FNO3Degré de pureté :97.22%Couleur et forme :SolidMasse moléculaire :293.25Monalizumab
CAS :Monalizumab, a humanized antibody, enhances NK cell function by inhibiting NKG2A; used in HNSCC studies.Degré de pureté :95% - >95.0% (SDS-PAGE); 100% (SEC-HPLC)Couleur et forme :LiquidMasse moléculaire :147 kDaAbrilumab
CAS :Abrilumab (MEDI-7183) is a fully human monoclonal antibody against α4β7 that inhibits the α4β7 integrin.Degré de pureté :98.5% (SDS-PAGE); 99% (SEC-HPLC) - 98.5% (SDS-PAGE); 99% (SEC-HPLC)Couleur et forme :LiquidMasse moléculaire :143.80 kDaEnrofloxacin
CAS :Enrofloxacin (BAY-Vp2674) is a veterinary antibacterial agent, used in poultry.
Formule :C19H22FN3O3Degré de pureté :99.43% - >99.99%Couleur et forme :Pale Yellow CrystalsMasse moléculaire :359.39Rifaximin
CAS :Rifaximin: an oral semi-synthetic antibiotic from rifamycin SV; targets bacterial RNA polymerase to halt growth.Formule :C43H51N3O11Degré de pureté :99.18% - 99.40%Couleur et forme :Red-Orange Crystalline PowderMasse moléculaire :785.88hSMG-1 inhibitor 11j
CAS :hSMG-1 inhibitor 11j: pyrimidine, IC50=0.11 nM, >455x selective vs. mTOR/PI3Kα/γ/CDK1/CDK2; cancer research use.
Formule :C27H28ClN7O3SDegré de pureté :99.22% - 99.65%Couleur et forme :SolidMasse moléculaire :566.07Levofloxacin hydrate
CAS :Levofloxacin hydrate (Cravit hydrate) is a third-generation fluoroquinolone antibiotic and optically active L-isomer of ofloxacin with antibacterial activity.Formule :C18H20FN3O4H2ODegré de pureté :98.26%Couleur et forme :Pale Yellow SolidMasse moléculaire :370.38Procaine
CAS :Procaine (Vitamin H3) is a slow-acting ester local anesthetic with a short effect, used for infiltration, nerve, and spinal blocks.
Formule :C13H20N2O2Degré de pureté :99.57% - 99.73%Couleur et forme :Anhydrous Plates Tables From Ligroin Or Ether SolidMasse moléculaire :236.31ATN-161 trifluoroacetate salt
CAS :ATN-161 TFA salt, a new integrin α5β1 inhibitor, curbs angiogenesis, liver metastases growth, enhances survival in mice.Formule :C25H36F3N9O10SDegré de pureté :98% - 99.98%Couleur et forme :SolidMasse moléculaire :711.67Hu7691 free base
CAS :Hu7691 free base is an Akt inhibitor that inhibits Akt1, Akt2 and Akt3 and induces differentiation of neuroblastoma cells.Formule :C22H21F3N4ODegré de pureté :98.89%Couleur et forme :SolidMasse moléculaire :414.423BMVC-8C3O
CAS :BMVC-8C3O is a DNA G-quadruplex (G4) ligand.Cost-effective and quality-assured.Formule :C42H53I3N4O3Degré de pureté :99.72%Couleur et forme :SolidMasse moléculaire :1042.61Ref: TM-T13584
1mg101,00€5mg192,00€10mg285,00€25mg462,00€50mg623,00€100mg858,00€200mg1.153,00€1mL*10mM (DMSO)371,00€TK216
CAS :TK216 is a potent inhibitor of E26 transformation-specific (ETS) with anticancer activity.Formule :C19H15Cl2NO3Degré de pureté :97.22%Couleur et forme :SolidMasse moléculaire :376.23Trimethoprim
CAS :Trimethoprim (NSC-106568) inhibits dihydrofolate reductase, CYP2C8, and OCT2 - an antibacterial agent.Formule :C14H18N4O3Degré de pureté :99.80% - 99.81%Couleur et forme :White To Yellowish PowderMasse moléculaire :290.32NMDI14
CAS :NMDI14 is an inhibitor of nonsense mediated RNA decay (NMD).Formule :C21H25N3O4SDegré de pureté :97.79% - 99.37%Couleur et forme :SolidMasse moléculaire :415.51Ref: TM-T12235
1mg35,00€5mg74,00€10mg119,00€25mg236,00€50mg356,00€100mg537,00€200mg762,00€1mL*10mM (DMSO)84,00€BAY-524
CAS :BAY-524 is an inhibitor of Bub1(IC50 = 450 nM.human Bub1 in the presence of 2 mM ATP).Formule :C24H24F2N6O3Degré de pureté :98.68% - 99.57%Couleur et forme :SolidMasse moléculaire :482.48Ref: TM-T14505
1mg96,00€5mg177,00€10mg298,00€25mg482,00€50mg658,00€100mg892,00€1mL*10mM (DMSO)178,00€Pazufloxacin Mesylate
CAS :Pazufloxacin Mesylate (T-3762) is a fluoroquinolone antibiotic.Formule :C16H15FN2O4·CH4O3SDegré de pureté :99.88% - 99.93%Couleur et forme :Crystalline SolidMasse moléculaire :414.4Nedaplatin
CAS :Nedaplatin, a cisplatin derivative, induces tumor DNA damage (IC50: 94 μM) through platinum-DNA cross-links, causing apoptosis.Formule :C2H8N2O3PtDegré de pureté :99.88% - >99.99%Couleur et forme :Straw Yellow PowderMasse moléculaire :303.17GSK-3 inhibitor 4
CAS :Orally active GSK-3 inhibitor 4 targets GSK-3α/β, CDK2/5 (IC50: 0.45-0.68 μM) and may aid in Alzheimer's research by lowering Tau protein.Formule :C22H15F2N5ODegré de pureté :99.82%Couleur et forme :SoildMasse moléculaire :403.38Ref: TM-T77341
1mg315,00€5mg873,00€10mg1.080,00€25mg1.431,00€50mg1.783,00€100mg2.250,00€500mg3.537,00€Tenofovir diphosphate TEA
CAS :Tenofovir diphosphate TEA (TFV-DP TEA) is an ATP-competitive DNA polymerase inhibitor that inhibits HIV-1 reverse transcriptase that\has anti-HIV/HBV potential.Formule :C9H16N5O10P3·C6H15NDegré de pureté :93.45% - 98.51%Couleur et forme :SolidMasse moléculaire :548.36RG7800
CAS :RG7800 (RO6885247) has the potential for spinal muscular atrophy treatment. RG7800 is an SMN2 splicing modifier.Formule :C24H28N6ODegré de pureté :99.44%Couleur et forme :SolidMasse moléculaire :416.52Y-33075 dihydrochloride
CAS :Y-33075 dihydrochloride is a selective inhibitor of ROCK(IC50 of 3.6 nM).Formule :C16H18Cl2N4ODegré de pureté :98.88% - 99.89%Couleur et forme :SolidMasse moléculaire :353.25Ref: TM-T13384L
1mg34,00€5mg66,00€10mg102,00€25mg192,00€50mg341,00€100mg510,00€200mg732,00€1mL*10mM (DMSO)78,00€GSK-626616
CAS :GSK-626616: strong, oral DYRK3 inhibitor (IC50: 0.7 nM), affects DYRK family, may treat anemia.Formule :C18H10Cl2N4OSDegré de pureté :98.27%Couleur et forme :SolidMasse moléculaire :401.27BAY-2402234
CAS :BAY-2402234: a selective DHODH inhibitor targeting myeloid cancers with low-nanomolar potency.Formule :C21H18ClF5N4O4Degré de pureté :98.9%Couleur et forme :SolidMasse moléculaire :520.84Ref: TM-T14501
1mg170,00€2mg234,00€5mg349,00€10mg537,00€25mg858,00€50mg1.161,00€100mg1.558,00€1mL*10mM (DMSO)401,00€Diaveridine
CAS :Diaveridine (AI3-23935) (DVD) is a popular antibacterial synergist that is widely used in combination with sulfonamide.Formule :C13H16N4O2Degré de pureté :99.10%Couleur et forme :White SolidMasse moléculaire :260.29Enoxacin hydrate
CAS :Enoxacin hydrate (AT-2266 hydrate) is a broad-spectrum 6-fluoronaphthyridinone antibacterial agent.Formule :C15H17FN4O3H2ODegré de pureté :99.50%Couleur et forme :SolidMasse moléculaire :347.34AZ1495
CAS :AZ1495: oral IRAK4 inhibitor (IC50: 5 nM), IRAK1 (23 nM), treats MYD88L265P DLBCL.Formule :C21H31N5O2Degré de pureté :98.81%Couleur et forme :SolidMasse moléculaire :385.5Ref: TM-T14367
1mg93,00€5mg156,00€10mg245,00€25mg349,00€50mg494,00€100mg750,00€200mg1.009,00€1mL*10mM (DMSO)170,00€Ribociclib succinate
CAS :Ribociclib succinate (LEE011 succinate) is a highly specific CDK4/6 inhibitor (IC50: 10 nM and 39 nM, respectively).Formule :C27H36N8O5Degré de pureté :99.9%Couleur et forme :SolidMasse moléculaire :552.63Ref: TM-T15732
2mg34,00€5mg49,00€10mg70,00€25mg92,00€50mg109,00€100mg165,00€200mg258,00€500mg459,00€1mL*10mM (DMSO)60,00€JH-RE-06
CAS :JH-RE-06 disrupts mutagenic translesion synthesis (TLS) by preventing the recruitment of mutagenic POLζ.Formule :C20H16Cl3N3O4Degré de pureté :99.29%Couleur et forme :SolidMasse moléculaire :468.72Ref: TM-T15611
1mg44,00€5mg93,00€10mg152,00€25mg334,00€50mg587,00€100mg1.044,00€1mL*10mM (DMSO)95,00€DHODH-IN-11
CAS :DHODH-IN-11 is a leflunomide derivative and weak dihydroorotate dehydrogenase (DHODH) inhibitor with a pKa of 5.03.Formule :C15H11N3O2Degré de pureté :98.14%Couleur et forme :SolidMasse moléculaire :265.27AZ-Dyrk1B-33
CAS :AZ-Dyrk1B-33 (3-(2-Methyl-4-pyrimidinyl)-1-(phenylmethyl)-1H-pyrrolo[2,3-c]pyridine) is a potent and selective Dyrk1B kinase inhibitor with an IC50 of 7 nM.Formule :C19H16N4Degré de pureté :99.91%Couleur et forme :SolidMasse moléculaire :300.36Ref: TM-T14364
1mg44,00€5mg92,00€10mg147,00€25mg289,00€50mg419,00€100mg583,00€200mg787,00€1mL*10mM (DMSO)100,00€Pyrimethamine
CAS :Pyrimethamine (Pirimecidan) is a competitive inhibitor of dihydrofolate reductase (DHFR), used as an antimalarial drug.Formule :C12H13ClN4Degré de pureté :99.67%Couleur et forme :CrystalsMasse moléculaire :248.71Mps1-IN-3
CAS :Mps1-IN-3 is an effective and selective inhibitor of MPS1 kinase (IC50: 50 nM).Formule :C26H31N7O4SDegré de pureté :99.25%Couleur et forme :SolidMasse moléculaire :537.63Ref: TM-T16130
2mg34,00€5mg54,00€10mg87,00€25mg149,00€50mg255,00€100mg384,00€200mg538,00€1mL*10mM (DMSO)64,00€HBX 19818
CAS :HBX 19818 is a specific ubiquitin-specific protease 7 (USP7) inhibitor (IC50: 28.1 μM).Formule :C25H28ClN3ODegré de pureté :97.71%Couleur et forme :SolidMasse moléculaire :421.96Ref: TM-T15464
1mg35,00€5mg80,00€10mg111,00€25mg177,00€50mg253,00€100mg353,00€200mg502,00€1mL*10mM (DMSO)89,00€TAME hydrochloride
CAS :TAME hydrochloride (Tos-Arg-OMe HCl) is a kind od amino acid derivatives.Formule :C14H23ClN4O4SDegré de pureté :99.11% - 99.21%Couleur et forme :White Fine Crystalline PowderMasse moléculaire :378.87Netarsudil Dihydrochloride
CAS :Netarsudil Dihydrochloride (AR-13324 Dihydrochloride) is an inhibitor of Rho-related protein kinase (ROCK) and norepinephrine transporter (NET) and is effective in reducing intraocular pressure (IOP).Cost-effective and quality-assured.Formule :C28H29Cl2N3O3Degré de pureté :99.94% - 99.98%Couleur et forme :SolidMasse moléculaire :526.45GSK-1520489A
CAS :GSK-1520489A is an active PKMYT1 inhibitor.Formule :C21H23N5O3SDegré de pureté :99.85%Couleur et forme :SolidMasse moléculaire :425.5XPW1
CAS :XPW1 is a CDK9 inhibitor with antitumor activity, inhibits DNA repair procedures, and can be used for the research of clear cell renal cell carcinoma.Formule :C36H39ClFN7O2Degré de pureté :98.08%Couleur et forme :SoildMasse moléculaire :656.19Cyclin K degrader 1
Cyclin K degrader 1 is a Cyclin K degrader.Cyclin K degrader 1 is a degrader converted from AT-7519.Cyclin K degrader 1 has weak degrading activity against Cyclin K but does not result in a sustained decrease in degradation affinity.Cyclin K degrader 1 is a degrader converted from AT-7519.Formule :C23H17Cl2N5O2Degré de pureté :99.76%Couleur et forme :SolidMasse moléculaire :466.32Cibisatamab
CAS :Cibisatamab, a T-cell bispecific antibody, targets CEA on cancer cells and CD3 on T-cells, inducing T-cell-mediated tumor cell killing.Degré de pureté :SDS-PAGE:99.1%;SEC-HPLC:96.5%Couleur et forme :LiquidMasse moléculaire :191.1 kDaCirtuvivint
CAS :Cirtuvivint (SM08502) is a potent and orally active CDC-like kinase (CLK) inhibitor that can be used to study arthritis.Formule :C24H25N7ODegré de pureté :99.95% - 99.96%Couleur et forme :SolidMasse moléculaire :427.5Butylparaben
CAS :Butylparaben (Butyl 4-hydroxybenzoate) is a standardized chemical allergen, increasing histamine release, and cell-mediated immunity.Formule :C11H14O3Degré de pureté :98.15%Couleur et forme :Small Colorless Crystals Or Powder Tongue Aqueous Solutions Slightly Acidic To Litmus (Ntp 1992)Masse moléculaire :194.23LY 345899
CAS :LY 345899 is a Folate analog and is a methylenetetrahydrofolate dehydrogenase and MTHFD2 inhibitor (IC50: 96 nM and 663 nM, respectively and a Ki: 18 nM for
Formule :C20H21N7O7Degré de pureté :99.7%Couleur et forme :SolidMasse moléculaire :471.42HLM006474
CAS :HLM006474 is a pan inhibitor of E2F. This inhibits E2F4 DNA-binding (IC50: 29.8 μM in A375 cells).Formule :C25H25N3O2Degré de pureté :99.04% - 99.20%Couleur et forme :SolidMasse moléculaire :399.48TAO Kinase inhibitor 2
CAS :TAO Kinase inhibitor 2 is a TAO kinase inhibitor with an IC50 of 50-500 nM. TAO Kinase inhibitor 2 inhibits KIAA1361 and JIK with IC50s of 50-500 nM.
Formule :C25H24N2O3Degré de pureté :98.58%Couleur et forme :SoildMasse moléculaire :400.47MYCi975
CAS :MYCi975 (NUCC-0200975) is an orally active inhibitor of MYC.Formule :C25H16Cl2F6N2O2Degré de pureté :99.3% - 99.82%Couleur et forme :SolidMasse moléculaire :561.3Otelixizumab
CAS :Otelixizumab (ChAglyCD3) is a chimeric monoclonal antibody targeting CD3, used in research on Type 1 diabetes and autoimmune diseases.Degré de pureté :>95%Couleur et forme :LiquidLerociclib dihydrochloride
CAS :Lerociclib dihydrochloride (G1T38 dihydrochloride) is a potent and selective inhibitor of CDK4/CDK6, with IC50s of 2 nM and 1 nM for CDK6/CyclinD3 and CDK4/Formule :C26H36Cl2N8ODegré de pureté :97.4%Couleur et forme :SolidMasse moléculaire :547.52TAK-901
CAS :TAK-901 has been used in trials studying the treatment of Lymphoma, Myelofibrosis, Multiple Myeloma, Myeloid Metaplasia, and Advanced Solid Tumors, among othersFormule :C28H32N4O3SDegré de pureté :99.02% - 99.59%Couleur et forme :SolidMasse moléculaire :504.64Ref: TM-T2709
1mg35,00€5mg70,00€10mg104,00€25mg202,00€50mg329,00€100mg525,00€200mg748,00€1mL*10mM (DMSO)79,00€Trilaciclib hydrochloride
CAS :Trilaciclib hydrochloride (G1T28 hydrochloride) is an inhibitor of CDK4/6 (IC50s: 1 nM and 4 nM for CDK4 and CDK6).Formule :C24H32Cl2N8ODegré de pureté :99.69% - 99.89%Couleur et forme :SolidMasse moléculaire :519.47Hycanthone
CAS :Hycanthone (Etrenol(mesylate)) is a potent drug of antischistosomal.Formule :C20H24N2O2SDegré de pureté :98.78%Couleur et forme :Yellow-Orange Powder (Ntp 1992)Masse moléculaire :356.48NU6140
CAS :NU6140 is a selective inhibitor of CDK2-cyclin A (IC50, 0.41 μM).Formule :C23H30N6O2Degré de pureté :98.33%Couleur et forme :SolidMasse moléculaire :422.52Ref: TM-T16359
2mg39,00€5mg60,00€10mg92,00€25mg177,00€50mg285,00€100mg414,00€200mg580,00€1mL*10mM (DMSO)67,00€Rifapentine
CAS :Rifapentine (Rifapentinum) is a long-acting, cyclopentyl-substituted derivative of rifamycin used to treat mycobacterium infections.Formule :C47H64N4O12Degré de pureté :95.74% - ≥98%Couleur et forme :SolidMasse moléculaire :877.03Vitamin D2
CAS :Ergocaliferol (Vitamin D2), derived from ergosterol by UV, inhibits bladder tumor promotion and leukemia, and blocks DNA Polymerase.Formule :C28H44ODegré de pureté :98.73% - 99.89%Couleur et forme :Prisms From Acetone 1998)Masse moléculaire :396.65R-10015
CAS :R-10015, potent LIMK inhibitor with 38 nM IC50 for LIMK1, targets ATP pocket, and serves as a broad-spectrum HIV antiviral.Formule :C20H19ClN6O2Degré de pureté :98.68%Couleur et forme :SolidMasse moléculaire :410.86Ref: TM-T12609
1mg50,00€5mg112,00€10mg170,00€25mg280,00€50mg371,00€100mg525,00€200mg712,00€1mL*10mM (DMSO)124,00€SIBA
CAS :SIBA, a synthetic SAH analog, inhibits SAM-dependent transmethylation and blocks HSV-1 replication.Formule :C14H21N5O3SDegré de pureté :99.48%Couleur et forme :SolidMasse moléculaire :339.41Ref: TM-T12908
1mg52,00€5mg94,00€10mg117,00€25mg220,00€50mg329,00€100mg469,00€200mg652,00€1mL*10mM (DMSO)104,00€Abciximab
CAS :Abciximab: chimeric antibody, anti-platelet, blocks glycoprotein IIb/IIIa, vitronectin, Mac-1.Degré de pureté :SDS-PAGE:95.2%;SEC-HPLC:95.9%Couleur et forme :LiquidMasse moléculaire :95.18 kDaPaprotrain
CAS :Paprotrain ((alphaZ)-alpha-(3-Pyridinylmethylene)-1H-indole-3-acetonitrile) inhibits the ATPase activity of MKLP-2 with an IC50 of 1.35 μM and a Ki of 3.36 μM.Formule :C16H11N3Degré de pureté :99.91%Couleur et forme :SolidMasse moléculaire :245.28Ref: TM-T12359
5mg46,00€10mg58,00€25mg92,00€50mg160,00€100mg236,00€200mg353,00€500mg580,00€1mL*10mM (DMSO)49,00€SU056
CAS :SU056 is a YB-1 inhibitor that induces cell-cycle arrest, apoptosis, and inhibits ovarian cancer cell migration.
Formule :C20H16FNO5Degré de pureté :99.89%Couleur et forme :SoildMasse moléculaire :369.34DI-87
CAS :DI-87 (TRE-515) is a novel and orally available dCK (deoxycytidine kinase) inhibitor. DI-87 binds to dCK reduces the production of dNTP inhibits tumor growth.Formule :C23H30N6O3S2Degré de pureté :99.76%Couleur et forme :SolidMasse moléculaire :502.65MALAT1-IN-1
CAS :MALAT1-IN-1 is an effective dose-dependent Malat1 inhibitor, not altering Neat1 expression.Formule :C19H21N3O2Degré de pureté :99.58%Couleur et forme :SolidMasse moléculaire :323.39Ref: TM-T16007
5mg39,00€10mg63,00€25mg120,00€50mg224,00€100mg432,00€200mg623,00€1mL*10mM (DMSO)44,00€Metarrestin
CAS :Metarrestin (ML246) is a first-in-class perinucleolar compartment inhibitor with a favorable PK profile, which effectively suppresses metastasis.
Formule :C31H30N4ODegré de pureté :99.45%Couleur et forme :SolidMasse moléculaire :474.6Ref: TM-T12006
1mg40,00€2mg52,00€5mg88,00€10mg144,00€25mg298,00€50mg512,00€100mg740,00€500mg1.539,00€Nadifloxacin
CAS :Nadifloxacin (OPC7251) has been used in trials studying the treatment of Acne Vulgaris.Formule :C19H21FN2O4Degré de pureté :99.03% - 99.7%Couleur et forme :Off-White Crystalline SolidMasse moléculaire :360.38Pefloxacin Mesylate Dihydrate
CAS :Pefloxacin Mesylate Dihydrate (1589 RB) , an antibacterial agent, restrains bacterial DNA replication by inhibiting DNA gyrase (topoisomerase).Formule :C17H20FN3O3·CH4O3S·2H2ODegré de pureté :99.79%Couleur et forme :SolidMasse moléculaire :465.49Ceftriaxone sodium hydrate
CAS :Ceftriaxone sodium hydrate is a broad-spectrum cephalosporin antibiotic with a very long half-life and high penetrability to meninges, eyes and inner ears.Formule :C18H16N8Na2O7S3·5H2ODegré de pureté :99.77% - 99.78%Couleur et forme :White Or Almost White Crystalline Powder OdorlessMasse moléculaire :661.6Ribavirin
CAS :Ribavirin (Tribavirin) is a synthetic nucleoside analog of ribofuranose with activity against hepatitis C virus and other RNA viruses.Formule :C8H12N4O5Degré de pureté :99.09% - 99.83%Couleur et forme :Less Solid Colourless SolidMasse moléculaire :244.20PTBP1-RNA-binding inhibitor P6 TFA
PTBP1-RNA-binding inhibitor P6 TFA is a stapled peptide inhibitor of PTBP1, used to inhibit RNA alternative splicing events regulated by PTBP1.Couleur et forme :Odour SolidCa2+ channel agonist 1
CAS :Ca2+ channel agonist 1 activates N-type Ca2+ channels and inhibits Cdk2 (EC50: 14.23 μM/3.34 μM) for motor nerve issues.Formule :C19H26N6ODegré de pureté :97.71%Couleur et forme :SolidMasse moléculaire :354.45Ref: TM-T10659
1mg97,00€5mg188,00€10mg284,00€25mg452,00€50mg645,00€100mg867,00€200mg1.130,00€1mL*10mM (DMSO)217,00€CDK2-IN-4
CAS :CDK2-IN-4 is a potent and selective inhibitor of CDK2 with an IC50 of 44 nM for CDK2/cyclin A.Formule :C23H18N6O2SDegré de pureté :97.24% - 99.10%Couleur et forme :SolidMasse moléculaire :442.49Ref: TM-T14916
1mg82,00€5mg192,00€10mg304,00€25mg522,00€50mg713,00€100mg1.018,00€1mL*10mM (DMSO)212,00€Cinoxacin
CAS :Cinoxacin (Compound 64716), an older synthetic antimicrobial, was related to the quinolone class of antibiotics.Formule :C12H10N2O5Degré de pureté :99.62% - 99.98%Couleur et forme :SolidMasse moléculaire :262.22Famciclovir
CAS :Famciclovir (BRL 42810) inhibits Herpes virus DNA polymerase by mimicking nucleosides.Formule :C14H19N5O4Degré de pureté :99.85% - 99.99%Couleur et forme :Off-White PowderMasse moléculaire :321.33MKC9989
CAS :MKC9989 is an inhibitor of Hydroxy aryl aldehydes (HAA). MKC9989 also inhibits IRE1α with an IC50 of 0.23 to 44 μM.Formule :C17H20O7Degré de pureté :99.3%Couleur et forme :SolidMasse moléculaire :336.34Ref: TM-T12071
1mg51,00€5mg156,00€10mg226,00€25mg376,00€50mg543,00€100mg730,00€1mL*10mM (DMSO)140,00€BRD6989
CAS :BRD6989, a cortistatin A analog, inhibits CDK8/19, enhances IL-10, and binds CDK8 with a 200 nM IC50.Formule :C16H16N4Degré de pureté :99.43%Couleur et forme :SolidMasse moléculaire :264.33Ref: TM-T14778
1mg34,00€5mg66,00€10mg92,00€25mg177,00€50mg268,00€100mg398,00€200mg575,00€1mL*10mM (DMSO)73,00€Procaine hydrochloride
CAS :Procaine HCl is a benzoic acid derivative used as a local anesthetic, blocking nerve impulses and sensation.Formule :C13H20N2O2·HClDegré de pureté :99.1% - 99.22%Couleur et forme :White Crystalline PowderMasse moléculaire :272.77

