
Cycle cellulaire/point de contrôle
Les inhibiteurs du cycle cellulaire/des points de contrôle sont des composés qui perturbent la progression normale du cycle cellulaire, en particulier aux points de contrôle régulateurs clés. Ces inhibiteurs sont cruciaux pour étudier la division cellulaire, comprendre la prolifération des cellules cancéreuses et développer des thérapies anticancéreuses. En ciblant des phases spécifiques du cycle cellulaire, ces inhibiteurs peuvent induire un arrêt du cycle cellulaire, conduisant à l'apoptose ou à la sénescence des cellules à division rapide. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de haute qualité du cycle cellulaire/des points de contrôle pour soutenir vos recherches en biologie du cancer, biologie cellulaire et développement de médicaments.
Sous-catégories appartenant à la catégorie "Cycle cellulaire/point de contrôle"
- Aurora Kinase(114 produits)
- CDK(545 produits)
- Arrêt du cycle cellulaire(5 produits)
- Chk(48 produits)
- DYRK(47 produits)
- Dynamine(27 produits)
- Ferroptose(226 produits)
- HSP(179 produits)
- Intégrine(249 produits)
- Kinésine(87 produits)
- LIM Kinase(20 produits)
- Microtubules associés(274 produits)
- PKC(124 produits)
- PLK(25 produits)
- ROCK(62 produits)
- Rho(6 produits)
- Wee1(14 produits)
- c-Myc(76 produits)
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3859 produits trouvés pour "Cycle cellulaire/point de contrôle"
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Diaveridine
CAS :Diaveridine (AI3-23935) (DVD) is a popular antibacterial synergist that is widely used in combination with sulfonamide.Formule :C13H16N4O2Degré de pureté :99.10%Couleur et forme :White SolidMasse moléculaire :260.29Enoxacin hydrate
CAS :Enoxacin hydrate (AT-2266 hydrate) is a broad-spectrum 6-fluoronaphthyridinone antibacterial agent.Formule :C15H17FN4O3H2ODegré de pureté :99.50%Couleur et forme :SolidMasse moléculaire :347.34AZ1495
CAS :AZ1495: oral IRAK4 inhibitor (IC50: 5 nM), IRAK1 (23 nM), treats MYD88L265P DLBCL.Formule :C21H31N5O2Degré de pureté :98.81%Couleur et forme :SolidMasse moléculaire :385.5Ref: TM-T14367
1mg93,00€5mg156,00€10mg245,00€25mg349,00€50mg494,00€100mg750,00€200mg1.009,00€1mL*10mM (DMSO)170,00€Ribociclib succinate
CAS :Ribociclib succinate (LEE011 succinate) is a highly specific CDK4/6 inhibitor (IC50: 10 nM and 39 nM, respectively).Formule :C27H36N8O5Degré de pureté :99.9%Couleur et forme :SolidMasse moléculaire :552.63Ref: TM-T15732
2mg34,00€5mg49,00€10mg70,00€25mg92,00€50mg109,00€100mg165,00€200mg258,00€500mg459,00€1mL*10mM (DMSO)60,00€JH-RE-06
CAS :JH-RE-06 disrupts mutagenic translesion synthesis (TLS) by preventing the recruitment of mutagenic POLζ.Formule :C20H16Cl3N3O4Degré de pureté :99.29%Couleur et forme :SolidMasse moléculaire :468.72Ref: TM-T15611
1mg44,00€5mg93,00€10mg152,00€25mg334,00€50mg587,00€100mg1.044,00€1mL*10mM (DMSO)95,00€DHODH-IN-11
CAS :DHODH-IN-11 is a leflunomide derivative and weak dihydroorotate dehydrogenase (DHODH) inhibitor with a pKa of 5.03.Formule :C15H11N3O2Degré de pureté :98.14%Couleur et forme :SolidMasse moléculaire :265.27AZ-Dyrk1B-33
CAS :AZ-Dyrk1B-33 (3-(2-Methyl-4-pyrimidinyl)-1-(phenylmethyl)-1H-pyrrolo[2,3-c]pyridine) is a potent and selective Dyrk1B kinase inhibitor with an IC50 of 7 nM.Formule :C19H16N4Degré de pureté :99.91%Couleur et forme :SolidMasse moléculaire :300.36Ref: TM-T14364
1mg44,00€5mg92,00€10mg147,00€25mg289,00€50mg419,00€100mg583,00€200mg787,00€1mL*10mM (DMSO)100,00€Pyrimethamine
CAS :Pyrimethamine (Pirimecidan) is a competitive inhibitor of dihydrofolate reductase (DHFR), used as an antimalarial drug.Formule :C12H13ClN4Degré de pureté :99.67%Couleur et forme :CrystalsMasse moléculaire :248.71Mps1-IN-3
CAS :Mps1-IN-3 is an effective and selective inhibitor of MPS1 kinase (IC50: 50 nM).Formule :C26H31N7O4SDegré de pureté :99.25%Couleur et forme :SolidMasse moléculaire :537.63Ref: TM-T16130
2mg34,00€5mg54,00€10mg87,00€25mg149,00€50mg255,00€100mg384,00€200mg538,00€1mL*10mM (DMSO)64,00€HBX 19818
CAS :HBX 19818 is a specific ubiquitin-specific protease 7 (USP7) inhibitor (IC50: 28.1 μM).Formule :C25H28ClN3ODegré de pureté :97.71%Couleur et forme :SolidMasse moléculaire :421.96Ref: TM-T15464
1mg35,00€5mg80,00€10mg111,00€25mg177,00€50mg253,00€100mg353,00€200mg502,00€1mL*10mM (DMSO)89,00€TAME hydrochloride
CAS :TAME hydrochloride (Tos-Arg-OMe HCl) is a kind od amino acid derivatives.Formule :C14H23ClN4O4SDegré de pureté :99.11% - 99.21%Couleur et forme :White Fine Crystalline PowderMasse moléculaire :378.87Netarsudil Dihydrochloride
CAS :Netarsudil Dihydrochloride (AR-13324 Dihydrochloride) is an inhibitor of Rho-related protein kinase (ROCK) and norepinephrine transporter (NET) and is effective in reducing intraocular pressure (IOP).Cost-effective and quality-assured.Formule :C28H29Cl2N3O3Degré de pureté :99.94% - 99.98%Couleur et forme :SolidMasse moléculaire :526.45GSK-1520489A
CAS :GSK-1520489A is an active PKMYT1 inhibitor.Formule :C21H23N5O3SDegré de pureté :99.85%Couleur et forme :SolidMasse moléculaire :425.5XPW1
CAS :XPW1 is a CDK9 inhibitor with antitumor activity, inhibits DNA repair procedures, and can be used for the research of clear cell renal cell carcinoma.Formule :C36H39ClFN7O2Degré de pureté :98.08%Couleur et forme :SoildMasse moléculaire :656.19Cyclin K degrader 1
Cyclin K degrader 1 is a Cyclin K degrader.Cyclin K degrader 1 is a degrader converted from AT-7519.Cyclin K degrader 1 has weak degrading activity against Cyclin K but does not result in a sustained decrease in degradation affinity.Cyclin K degrader 1 is a degrader converted from AT-7519.Formule :C23H17Cl2N5O2Degré de pureté :99.76%Couleur et forme :SolidMasse moléculaire :466.32Cibisatamab
CAS :Cibisatamab, a T-cell bispecific antibody, targets CEA on cancer cells and CD3 on T-cells, inducing T-cell-mediated tumor cell killing.Degré de pureté :SDS-PAGE:99.1%;SEC-HPLC:96.5%Couleur et forme :LiquidMasse moléculaire :191.1 kDaCirtuvivint
CAS :Cirtuvivint (SM08502) is a potent and orally active CDC-like kinase (CLK) inhibitor that can be used to study arthritis.Formule :C24H25N7ODegré de pureté :99.95% - 99.96%Couleur et forme :SolidMasse moléculaire :427.5Butylparaben
CAS :Butylparaben (Butyl 4-hydroxybenzoate) is a standardized chemical allergen, increasing histamine release, and cell-mediated immunity.Formule :C11H14O3Degré de pureté :98.15%Couleur et forme :Small Colorless Crystals Or Powder Tongue Aqueous Solutions Slightly Acidic To Litmus (Ntp 1992)Masse moléculaire :194.23LY 345899
CAS :LY 345899 is a Folate analog and is a methylenetetrahydrofolate dehydrogenase and MTHFD2 inhibitor (IC50: 96 nM and 663 nM, respectively and a Ki: 18 nM for
Formule :C20H21N7O7Degré de pureté :99.7%Couleur et forme :SolidMasse moléculaire :471.42HLM006474
CAS :HLM006474 is a pan inhibitor of E2F. This inhibits E2F4 DNA-binding (IC50: 29.8 μM in A375 cells).Formule :C25H25N3O2Degré de pureté :99.04% - 99.20%Couleur et forme :SolidMasse moléculaire :399.48TAO Kinase inhibitor 2
CAS :TAO Kinase inhibitor 2 is a TAO kinase inhibitor with an IC50 of 50-500 nM. TAO Kinase inhibitor 2 inhibits KIAA1361 and JIK with IC50s of 50-500 nM.
Formule :C25H24N2O3Degré de pureté :98.58%Couleur et forme :SoildMasse moléculaire :400.47MYCi975
CAS :MYCi975 (NUCC-0200975) is an orally active inhibitor of MYC.Formule :C25H16Cl2F6N2O2Degré de pureté :99.3% - 99.82%Couleur et forme :SolidMasse moléculaire :561.3Otelixizumab
CAS :Otelixizumab (ChAglyCD3) is a chimeric monoclonal antibody targeting CD3, used in research on Type 1 diabetes and autoimmune diseases.Degré de pureté :>95%Couleur et forme :LiquidLerociclib dihydrochloride
CAS :Lerociclib dihydrochloride (G1T38 dihydrochloride) is a potent and selective inhibitor of CDK4/CDK6, with IC50s of 2 nM and 1 nM for CDK6/CyclinD3 and CDK4/Formule :C26H36Cl2N8ODegré de pureté :97.4%Couleur et forme :SolidMasse moléculaire :547.52TAK-901
CAS :TAK-901 has been used in trials studying the treatment of Lymphoma, Myelofibrosis, Multiple Myeloma, Myeloid Metaplasia, and Advanced Solid Tumors, among othersFormule :C28H32N4O3SDegré de pureté :99.02% - 99.59%Couleur et forme :SolidMasse moléculaire :504.64Ref: TM-T2709
1mg35,00€5mg70,00€10mg104,00€25mg202,00€50mg329,00€100mg525,00€200mg748,00€1mL*10mM (DMSO)79,00€Trilaciclib hydrochloride
CAS :Trilaciclib hydrochloride (G1T28 hydrochloride) is an inhibitor of CDK4/6 (IC50s: 1 nM and 4 nM for CDK4 and CDK6).Formule :C24H32Cl2N8ODegré de pureté :99.69% - 99.89%Couleur et forme :SolidMasse moléculaire :519.47Hycanthone
CAS :Hycanthone (Etrenol(mesylate)) is a potent drug of antischistosomal.Formule :C20H24N2O2SDegré de pureté :98.78%Couleur et forme :Yellow-Orange Powder (Ntp 1992)Masse moléculaire :356.48NU6140
CAS :NU6140 is a selective inhibitor of CDK2-cyclin A (IC50, 0.41 μM).Formule :C23H30N6O2Degré de pureté :98.33%Couleur et forme :SolidMasse moléculaire :422.52Ref: TM-T16359
2mg39,00€5mg60,00€10mg92,00€25mg177,00€50mg285,00€100mg414,00€200mg580,00€1mL*10mM (DMSO)67,00€Rifapentine
CAS :Rifapentine (Rifapentinum) is a long-acting, cyclopentyl-substituted derivative of rifamycin used to treat mycobacterium infections.Formule :C47H64N4O12Degré de pureté :95.74% - ≥98%Couleur et forme :SolidMasse moléculaire :877.03Vitamin D2
CAS :Ergocaliferol (Vitamin D2), derived from ergosterol by UV, inhibits bladder tumor promotion and leukemia, and blocks DNA Polymerase.Formule :C28H44ODegré de pureté :98.73% - 99.89%Couleur et forme :Prisms From Acetone 1998)Masse moléculaire :396.65R-10015
CAS :R-10015, potent LIMK inhibitor with 38 nM IC50 for LIMK1, targets ATP pocket, and serves as a broad-spectrum HIV antiviral.Formule :C20H19ClN6O2Degré de pureté :98.68%Couleur et forme :SolidMasse moléculaire :410.86Ref: TM-T12609
1mg50,00€5mg112,00€10mg170,00€25mg280,00€50mg371,00€100mg525,00€200mg712,00€1mL*10mM (DMSO)124,00€SIBA
CAS :SIBA, a synthetic SAH analog, inhibits SAM-dependent transmethylation and blocks HSV-1 replication.Formule :C14H21N5O3SDegré de pureté :99.48%Couleur et forme :SolidMasse moléculaire :339.41Ref: TM-T12908
1mg52,00€5mg94,00€10mg117,00€25mg220,00€50mg329,00€100mg469,00€200mg652,00€1mL*10mM (DMSO)104,00€Abciximab
CAS :Abciximab: chimeric antibody, anti-platelet, blocks glycoprotein IIb/IIIa, vitronectin, Mac-1.Degré de pureté :SDS-PAGE:95.2%;SEC-HPLC:95.9%Couleur et forme :LiquidMasse moléculaire :95.18 kDaPaprotrain
CAS :Paprotrain ((alphaZ)-alpha-(3-Pyridinylmethylene)-1H-indole-3-acetonitrile) inhibits the ATPase activity of MKLP-2 with an IC50 of 1.35 μM and a Ki of 3.36 μM.Formule :C16H11N3Degré de pureté :99.91%Couleur et forme :SolidMasse moléculaire :245.28Ref: TM-T12359
5mg46,00€10mg58,00€25mg92,00€50mg160,00€100mg236,00€200mg353,00€500mg580,00€1mL*10mM (DMSO)49,00€SU056
CAS :SU056 is a YB-1 inhibitor that induces cell-cycle arrest, apoptosis, and inhibits ovarian cancer cell migration.
Formule :C20H16FNO5Degré de pureté :99.89%Couleur et forme :SoildMasse moléculaire :369.34DI-87
CAS :DI-87 (TRE-515) is a novel and orally available dCK (deoxycytidine kinase) inhibitor. DI-87 binds to dCK reduces the production of dNTP inhibits tumor growth.Formule :C23H30N6O3S2Degré de pureté :99.76%Couleur et forme :SolidMasse moléculaire :502.65MALAT1-IN-1
CAS :MALAT1-IN-1 is an effective dose-dependent Malat1 inhibitor, not altering Neat1 expression.Formule :C19H21N3O2Degré de pureté :99.58%Couleur et forme :SolidMasse moléculaire :323.39Ref: TM-T16007
5mg39,00€10mg63,00€25mg120,00€50mg224,00€100mg432,00€200mg623,00€1mL*10mM (DMSO)44,00€Metarrestin
CAS :Metarrestin (ML246) is a first-in-class perinucleolar compartment inhibitor with a favorable PK profile, which effectively suppresses metastasis.
Formule :C31H30N4ODegré de pureté :99.45%Couleur et forme :SolidMasse moléculaire :474.6Ref: TM-T12006
1mg40,00€2mg52,00€5mg88,00€10mg144,00€25mg298,00€50mg512,00€100mg740,00€500mg1.539,00€Nadifloxacin
CAS :Nadifloxacin (OPC7251) has been used in trials studying the treatment of Acne Vulgaris.Formule :C19H21FN2O4Degré de pureté :99.03% - 99.7%Couleur et forme :Off-White Crystalline SolidMasse moléculaire :360.38Pefloxacin Mesylate Dihydrate
CAS :Pefloxacin Mesylate Dihydrate (1589 RB) , an antibacterial agent, restrains bacterial DNA replication by inhibiting DNA gyrase (topoisomerase).Formule :C17H20FN3O3·CH4O3S·2H2ODegré de pureté :99.79%Couleur et forme :SolidMasse moléculaire :465.49Ceftriaxone sodium hydrate
CAS :Ceftriaxone sodium hydrate is a broad-spectrum cephalosporin antibiotic with a very long half-life and high penetrability to meninges, eyes and inner ears.Formule :C18H16N8Na2O7S3·5H2ODegré de pureté :99.77% - 99.78%Couleur et forme :White Or Almost White Crystalline Powder OdorlessMasse moléculaire :661.6Ribavirin
CAS :Ribavirin (Tribavirin) is a synthetic nucleoside analog of ribofuranose with activity against hepatitis C virus and other RNA viruses.Formule :C8H12N4O5Degré de pureté :99.09% - 99.83%Couleur et forme :Less Solid Colourless SolidMasse moléculaire :244.20PTBP1-RNA-binding inhibitor P6 TFA
PTBP1-RNA-binding inhibitor P6 TFA is a stapled peptide inhibitor of PTBP1, used to inhibit RNA alternative splicing events regulated by PTBP1.Couleur et forme :Odour SolidCa2+ channel agonist 1
CAS :Ca2+ channel agonist 1 activates N-type Ca2+ channels and inhibits Cdk2 (EC50: 14.23 μM/3.34 μM) for motor nerve issues.Formule :C19H26N6ODegré de pureté :97.71%Couleur et forme :SolidMasse moléculaire :354.45Ref: TM-T10659
1mg97,00€5mg188,00€10mg284,00€25mg452,00€50mg645,00€100mg867,00€200mg1.130,00€1mL*10mM (DMSO)217,00€CDK2-IN-4
CAS :CDK2-IN-4 is a potent and selective inhibitor of CDK2 with an IC50 of 44 nM for CDK2/cyclin A.Formule :C23H18N6O2SDegré de pureté :97.24% - 99.10%Couleur et forme :SolidMasse moléculaire :442.49Ref: TM-T14916
1mg82,00€5mg192,00€10mg304,00€25mg522,00€50mg713,00€100mg1.018,00€1mL*10mM (DMSO)212,00€Cinoxacin
CAS :Cinoxacin (Compound 64716), an older synthetic antimicrobial, was related to the quinolone class of antibiotics.Formule :C12H10N2O5Degré de pureté :99.62% - 99.98%Couleur et forme :SolidMasse moléculaire :262.22Famciclovir
CAS :Famciclovir (BRL 42810) inhibits Herpes virus DNA polymerase by mimicking nucleosides.Formule :C14H19N5O4Degré de pureté :99.85% - 99.99%Couleur et forme :Off-White PowderMasse moléculaire :321.33MKC9989
CAS :MKC9989 is an inhibitor of Hydroxy aryl aldehydes (HAA). MKC9989 also inhibits IRE1α with an IC50 of 0.23 to 44 μM.Formule :C17H20O7Degré de pureté :99.3%Couleur et forme :SolidMasse moléculaire :336.34Ref: TM-T12071
1mg51,00€5mg156,00€10mg226,00€25mg376,00€50mg543,00€100mg730,00€1mL*10mM (DMSO)140,00€BRD6989
CAS :BRD6989, a cortistatin A analog, inhibits CDK8/19, enhances IL-10, and binds CDK8 with a 200 nM IC50.Formule :C16H16N4Degré de pureté :99.43%Couleur et forme :SolidMasse moléculaire :264.33Ref: TM-T14778
1mg34,00€5mg66,00€10mg92,00€25mg177,00€50mg268,00€100mg398,00€200mg575,00€1mL*10mM (DMSO)73,00€Procaine hydrochloride
CAS :Procaine HCl is a benzoic acid derivative used as a local anesthetic, blocking nerve impulses and sensation.Formule :C13H20N2O2·HClDegré de pureté :99.1% - 99.22%Couleur et forme :White Crystalline PowderMasse moléculaire :272.77

