
Immunologie et Inflammation
Les inhibiteurs en immunologie et inflammation sont des composés qui modulent la réponse immunitaire et les processus inflammatoires. Ces inhibiteurs sont cruciaux pour étudier les mécanismes de la régulation immunitaire, l'auto-immunité et l'inflammation chronique, ainsi que pour développer des traitements pour les maladies inflammatoires, les allergies et les troubles immunitaires. En ciblant des voies clés du système immunitaire, ces inhibiteurs peuvent aider à réduire les réponses immunitaires excessives ou inappropriées. Chez CymitQuimica, nous offrons une large sélection d'inhibiteurs de haute qualité en immunologie et inflammation pour soutenir vos recherches en immunologie, inflammation et développement thérapeutique.
Sous-catégories appartenant à la catégorie "Immunologie et Inflammation"
- RCC(136 produits)
- CXCR(147 produits)
- Paroi cellulaire(5 produits)
- Récepteur IL(113 produits)
- IκB/IKK(61 produits)
- LTR(3 produits)
- MALT(23 produits)
- MRP(6 produits)
- NADPH-oxydase(1 produits)
- NF-κB(445 produits)
- NOD(17 produits)
- NOS(63 produits)
- Nrf2(78 produits)
- PGE Synthase(31 produits)
- ROS(69 produits)
- TGF-beta/Smad(58 produits)
- TLR(66 produits)
- Thioredoxine(12 produits)
- gp120/CD4(4 produits)
Affichez 11 plus de sous-catégories
3035 produits trouvés pour "Immunologie et Inflammation"
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(E/Z)-IT-603
CAS :<p>(E/Z)-IT-603 is a cell-permeable c-Rel inhibitor. IT-603 directly and reversibly binds to c-Rel to change its conformation and blocks its DNA binding activity.</p>Formule :C11H9BrN2O3SDegré de pureté :99.35%Couleur et forme :SolidMasse moléculaire :329.17Nodakenin
CAS :<p>Nodakenin ((+)-Marmesinin) is a compound with anti-allergic and anti-inflammatory activities.</p>Formule :C20H24O9Degré de pureté :95.46% - 98.93%Couleur et forme :SolidMasse moléculaire :408.4TLR7 agonist 2
CAS :<p>TLR7 agonist 2 (TLR7-IN-1) is a specific and effective Toll-like Receptor 7 (TLR7) agonist (LEC=0.4 μM).</p>Formule :C17H16N6O2Degré de pureté :99.33%Couleur et forme :SolidMasse moléculaire :336.35sphondin
CAS :<p>Sphondin inhibits IL-1beta, reduces COX-2 and PGE(2) in A549 cells, and has anticonvulsant, anti-inflammatory, anti-proliferative properties.</p>Formule :C12H8O4Degré de pureté :99.9% - ≥95%Couleur et forme :SolidMasse moléculaire :216.19IMM-H007
CAS :<p>IMM-H007 is a novel lipid-lowering agent, increasing abca1 protein expression</p>Formule :C22H23N5O8Degré de pureté :97.73%Couleur et forme :SolidMasse moléculaire :485.45AEM1
CAS :<p>AEM1 is an inhibitor of deregulated NRF2 transcriptional activity in cancer.</p>Formule :C20H14FN3O2SDegré de pureté :98.37% - 99.88%Couleur et forme :SolidMasse moléculaire :379.41Eclitasertib
CAS :<p>Eclitasertib is a potent inhibitor of receptor-interacting protein kinase 1 (RIPK1, IC50 of <1 µΜ).</p>Formule :C19H18N6O3Degré de pureté :99.85%Couleur et forme :SolidMasse moléculaire :378.38Ginsenoside Rb3
CAS :<p>Ginsenoside Rb3 (Gypenoside IV) is a natural triterpenoid saponin, exhibiting inhibition effect on TNFα-induced NF-κB transcriptional activity.</p>Formule :C53H90O22Degré de pureté :98% - 99.98%Couleur et forme :SolidMasse moléculaire :1079.27RO2959 Hydrochloride
CAS :<p>RO2959 Hydrochloride (RO2959 HCl) is a potent and selective inhibitor of CRAC channel(IC50: 402 nM). It is also a potent inhibitor of human IL-2.</p>Formule :C21H20ClF2N5OSDegré de pureté :99.24%Couleur et forme :SolidMasse moléculaire :463.93Tizoxanide
CAS :<p>Tizoxanide (Desacetyl-nitazoxanide) is a metabolite of lamivudine.</p>Formule :C10H7N3O4SDegré de pureté :98.89% - 99.28%Couleur et forme :SolidMasse moléculaire :265.25Ibuprofen Lysine
CAS :<p>Ibuprofen Lysine (Neoprofen) is a non-steroidal anti-inflammatory drug.</p>Formule :C19H32N2O4Degré de pureté :99.26%Couleur et forme :CoaMasse moléculaire :352.47GSK-J4
CAS :<p>GSK-J4 (GSK J4 HCl) is a cell permeable prodrug of GSK-J1, a dual inhibitor of the H3K27me3/me2 demethylases JMJD3/KDM6B and UTX/KDM6A. Cost effective and quality assured.</p>Formule :C24H27N5O2Degré de pureté :98.24% - 99.98%Couleur et forme :SolidMasse moléculaire :417.5Cyclo(his-pro)
CAS :<p>Cyclo(his-pro) is a cyclic dipeptide that shields against oxidative damage by activating Nrf2.</p>Formule :C11H14N4O2Degré de pureté :99.87%Couleur et forme :SolidMasse moléculaire :234.25Nitroarginine
CAS :<p>Nitroarginine (N'-Nitro-L-arginine) is a competitive inhibitor of nitric oxide synthase which causes the selective reduction of blood flow to tumor cells[1].</p>Formule :C6H13N5O4Degré de pureté :99.85%Couleur et forme :SolidMasse moléculaire :219.2Suplatast (Tosilate)
CAS :<p>Suplatast Tosilate (IPD 1151T) is a novel capsular anti-asthmatic drug. It ( IC50 above 100 μM) inhibits both IgE production, IL-4 and IL-5 synthesis.</p>Formule :C23H33NO7S2Degré de pureté :99.34% - 99.65%Couleur et forme :White Or Off-White CrystalsMasse moléculaire :499.64TR-14035
CAS :<p>TR-14035 (MDK-1191) is a dual antagonist of α4β7/α4β1 integrins (IC50s: 7/87nM).</p>Formule :C24H21Cl2NO5Degré de pureté :98.98%Couleur et forme :SolidMasse moléculaire :474.33CTX-0294885
CAS :<p>CTX-0294885, a bisanilino pyrimidine, inhibits many kinases; used for Sepharose-based kinase capture.</p>Formule :C22H24ClN7ODegré de pureté :98.73% - ≥95%Couleur et forme :SolidMasse moléculaire :437.93CORM-3
CAS :<p>CORM-3 is a carbon monoxide-releasing molecule with anti-inflammatory and cardioprotective activity.</p>Formule :C5H4ClNO5RuDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :294.61AS-2444697
CAS :<p>AS-2444697, an IRAK-4 inhibitor (C50=21 nM), offers renal protection via anti-inflammatory effects on human and rat IRAK-4.</p>Formule :C19H21ClN6O4Degré de pureté :97.17%Couleur et forme :SolidMasse moléculaire :432.86CY-09
CAS :<p>CY-09 is an NLRP3 inhibitor.</p>Formule :C19H12F3NO3S2Degré de pureté :99.25% - >99.99%Couleur et forme :SolidMasse moléculaire :423.43Ginsenoside Rg6
CAS :<p>Ginsenoside Rg6 inhibits the proliferation and induces apoptosis of human lymphoma JK cells</p>Formule :C42H70O12Degré de pureté :97.34%Couleur et forme :SolidMasse moléculaire :767Berbamine
CAS :<p>Berbamine is a natural product extracted from Phellodendron amurense.</p>Formule :C37H40N2O6Degré de pureté :98.92% - 99.67%Couleur et forme :White Crystal PowderMasse moléculaire :608.72Dehydroevodiamine
CAS :<p>Dehydroevodiamine (DHED), a constituent of Evodia rutaecarpa, has various biological effects such as hypotensive, negative chronotropic, ion channel depressant</p>Formule :C19H15N3ODegré de pureté :99.54%Couleur et forme :SolidMasse moléculaire :301.34Galloylpaeoniflorin
CAS :<p>Galloylpaeoniflorin (6'-O-Galloyl paeoniflorin) may be developed as a cytoprotector against ROS-mediated oxidative stress.</p>Formule :C30H32O15Degré de pureté :99.82%Couleur et forme :SolidMasse moléculaire :632.57BX795
CAS :<p>BX795 selectively inhibits PDK1 (IC50: 6 nM), 140x over PKA, 1600x over PKC, 100x over GSK3β in cell-free assays.</p>Formule :C23H26IN7O2SDegré de pureté :98% - 99.57%Couleur et forme :SolidMasse moléculaire :591.47Demethyleneberberine
CAS :<p>Demethyleneberberine, which is composed of a potential antioxidant structure, could penetrate the membrane of mitochondria and accumulate in mitochondria either</p>Formule :C19H18NO4Degré de pureté :98.08% - 99.18%Couleur et forme :SolidMasse moléculaire :324.35Danicopan
CAS :<p>Danicopan (ACH-4471), an oral factor D inhibitor, binds strongly (Kd 0.54 nM) and may treat PNH and aHUS.</p>Formule :C26H23BrFN7O3Degré de pureté :99.94%Couleur et forme :SolidMasse moléculaire :580.41BI-69A11
CAS :<p>BI-69A11 is a dual AKT/NFkB inhibitor, increasing colon cancer cell sensitivity to mda-7/IL-24.</p>Formule :C25H16ClN3O2Degré de pureté :96.97%Couleur et forme :SolidMasse moléculaire :425.871-Caffeoylquinic acid
CAS :<p>1-Caffeoylquinic acid: a lignin precursor with anti-influenza, antioxidant properties, and moderates post-meal glucose release.</p>Formule :C16H18O9Degré de pureté :99.15% - 99.16%Couleur et forme :SolidMasse moléculaire :354.31Stachydrine
CAS :<p>Stachydrine, found in leonurus herb, aids blood flow, blocks NF-κB pathway, and indicates citrus intake.</p>Formule :C7H13NO2Degré de pureté :99.94% - ≥95%Couleur et forme :SolidMasse moléculaire :143.18Metyrosine
CAS :<p>Metyrosine: antihypertensive, tyrosine hydroxylase inhibitor, controls COX-2, lowers blood pressure.</p>Formule :C10H13NO3Degré de pureté :98.68% - 99.72%Couleur et forme :SolidMasse moléculaire :195.22FICZ
CAS :<p>FICZ (6-Formylindolo[3,2-b]carbazole) is a potent aryl agonist for the hydrocarbon receptor (AhR, Kd: 70 pM).</p>Formule :C19H12N2ODegré de pureté :98.97%Couleur et forme :SolidMasse moléculaire :284.31anemarsaponin B
CAS :<p>Anemarsaponin B has anti-inflammatory effect in LPS-treated RAW 264.7macrophages, the effect is associated with the inhibition of NF-κB transcriptional activity</p>Formule :C45H74O18Degré de pureté :99.06% - 99.81%Couleur et forme :SolidMasse moléculaire :903.062-AMINO-5-PHENYL-THIOPHENE-3-CARBOXYLIC
CAS :<p>2-AMINO-5-PHENYL-THIOPHENE-3-CARBOXYLIC is Inhibitior of IKKβ.</p>Formule :C11H10N2OSDegré de pureté :99.48%Couleur et forme :SolidMasse moléculaire :218.27Vanillic Acid
CAS :<p>Vanillic Acid (Acide vanillique) is used as a condiment in food, which used in wine. It is an intermediate in the production of vanillin from ferulic acid.</p>Formule :C8H8O4Degré de pureté :99.82%Couleur et forme :White Odourless Crystals Or PowderMasse moléculaire :168.15L-Alanyl-L-glutamine
CAS :<p>L-Alanyl-L-glutamine (Ala-Gln), a dipeptide composed of alanine and Gln, is an alternative supplement to L-glutamine in the production of biopharmaceuticals.</p>Formule :C8H15N3O4Degré de pureté :99.71% - 99.97%Couleur et forme :SolidMasse moléculaire :217.22Berbamine dihydrochloride
CAS :<p>Berbamine dihydrochloride (Berbamine), a natural compound derived from the Berberis amurensis plant, has been shown to exhibit antitumor activity in several Ys.</p>Formule :C37H42Cl2N2O6Degré de pureté :95% - 99.99%Couleur et forme :SolidMasse moléculaire :681.65Asperulosidic acid
CAS :<p>Asperulosidic acid (ASPA) has anti-tumor, anti-oxidant, and anti-inflammatory activities. ASPA is related to the inhibition of inflammatory cytokines.</p>Formule :C18H24O12Degré de pureté :99.47%Couleur et forme :SolidMasse moléculaire :432.38YYA-021
CAS :<p>YYA-021 inhibits HIV entry, with high anti-HIV activity and low cytotoxicity.</p>Formule :C18H27N3O2Degré de pureté :97.17% - 99.87%Couleur et forme :SolidMasse moléculaire :317.43AF 12198 Acetate
<p>AF 12198 Acetate is a novel low molecular weight antagonist of IL-1</p>Formule :C98H127N19O24Degré de pureté :95.27%Couleur et forme :SolidMasse moléculaire :1955.17IL-17A inhibitor 1
CAS :<p>IL-17A inhibitor 1 is a IL-17A inhibitor with IC50 of <9.45 nM in alphalisa assay. IL-17A inhibitor 1 inhibits HT-29 cells with IC50 of 9.3 nM.</p>Formule :C24H27F5N8O4Degré de pureté :99.37% - 99.37%Couleur et forme :SolidMasse moléculaire :586.51TLR7/8 agonist 1
CAS :<p>TLR7/8 agonist 1 is a toll-like receptor TLR7/TLR8 agonist with anticancer and antiviral activities and can be used to study immune-related diseases.</p>Formule :C22H25N5Degré de pureté :99.4%Couleur et forme :SolidMasse moléculaire :359.47SB-265610
CAS :<p>SB-265610 (GSK-CXCR2) is a nonpeptide and allosteric CXCR2 antagonist.</p>Formule :C14H9BrN6ODegré de pureté :99.5%Couleur et forme :SolidMasse moléculaire :357.16Gypenoside L
CAS :<p>Gypenoside L inhibits autophagic flux and induces cell death in human esophageal cancer cells through endoplasm reticulum stress-mediated Ca2+ release.</p>Formule :C42H72O14Degré de pureté :99.42% - 99.65%Couleur et forme :SolidMasse moléculaire :801.014-IPP
CAS :<p>4-IPP (4-Iodo-6-phenylpyrimidine) is an irreversible inhibitor of macrophage migration inhibitory factor (MIF)</p>Formule :C10H7IN2Degré de pureté :99.63%Couleur et forme :SolidMasse moléculaire :282.08Siponimod
CAS :<p>Siponimod (BAF312) modulates S1P1/S1P5 with EC50s of 0.39/0.98 nM; >1000x selectivity over S1P2-4.</p>Formule :C29H35F3N2O3Degré de pureté :97.08% - 99.40%Couleur et forme :SolidMasse moléculaire :516.59Homo-PROTAC cereblon degrader 1
CAS :<p>Homo-PROTAC cereblon degrader 1 is a highly potent and efficient cereblon (CRBN) degrader with only minimal effects on IKZF1 and IKZF3.</p>Formule :C32H32N6O10Degré de pureté :98.3%Couleur et forme :SolidMasse moléculaire :660.63Chlorthenoxazine
CAS :<p>Chlorthenoxazine (Chlorethylbenzmethoxazone) has anti-inflammatory activity.</p>Formule :C10H10ClNO2Degré de pureté :99.64%Couleur et forme :SolidMasse moléculaire :211.64Iguratimod
CAS :<p>Iguratimod (T614) is a COX-2 inhibitor (IC50: 20 μM), does not affect COX-1, and inhibits MIF (IC50: 6.81 μM).</p>Formule :C17H14N2O6SDegré de pureté :99.93%Couleur et forme :White PowderMasse moléculaire :374.37OPHIOPOGONIN D
CAS :<p>Ophiopogonin D is a natural product,and is a CYP2J3 inducer that significantly inhibits Ang II induced NF-κB nuclear translocation.</p>Formule :C44H70O16Degré de pureté :99.46% - ≥95%Couleur et forme :SolidMasse moléculaire :855.02Flavanomarein
CAS :<p>Flavanomarein: Antioxidant with radical scavenging, lipid peroxidation inhibition, and lipid-lowering in HepG2 cells.</p>Formule :C21H22O11Degré de pureté :98.63% - 99.54%Couleur et forme :SolidMasse moléculaire :450.39GSK2981278
CAS :<p>GSK2981278 (ROR gama modulator 1) is a highly potent and selective inverse agonist of retinoic acid receptor-related orphan receptor gamma (ROR gamma).</p>Formule :C25H35NO5SDegré de pureté :99.31% - 99.67%Couleur et forme :SolidMasse moléculaire :461.61Esonarimod
CAS :<p>Esonarimod (KE-298) is an antirheumatic drug.</p>Formule :C14H16O4SDegré de pureté :97.44%Couleur et forme :SolidMasse moléculaire :280.34Brincidofovir
CAS :<p>Brincidofovir (HDP-CDV) is an orally active, lipophilic form of cidofovir.</p>Formule :C27H52N3O7PDegré de pureté :98% - 99.62%Couleur et forme :SolidMasse moléculaire :561.69Micheliolide
CAS :<p>Micheliolide(MCL) is a sesquiterpene lactone which inhibits various inflammatory response.</p>Formule :C15H20O3Degré de pureté :98% - 99.37%Couleur et forme :SolidMasse moléculaire :248.32Licochalcone D
CAS :<p>Licochalcone D may treat melanoma and heart injury, halt cell spread, and reduce inflammation and allergies.</p>Formule :C21H22O5Degré de pureté :99.03% - 99.9%Couleur et forme :SolidMasse moléculaire :354.4TOMATIDINE HYDROCHLORIDE
CAS :<p>Tomatidine hydrochloride (Tomatidine HCl) is a steriodal alkaloid structurally similar to Cyclopamine but does not inhibit hedgehog pathway.</p>Formule :C27H46ClNO2Degré de pureté :99.75% - ≥95%Couleur et forme :SolidMasse moléculaire :452.11GKT136901
CAS :<p>GKT136901 (AK120765) is an inhibitor of NOX1/4.It acts as Selective and Direct Scavenger of Peroxynitrite</p>Formule :C19H15ClN4O2Degré de pureté :99.16%Couleur et forme :SolidMasse moléculaire :366.8cangrelor tetrasodium
CAS :<p>Cangrelor tetrasodium is a reversible and selective antagonist of platelet P2Y12, with prompt and potent antiplatelet effects.</p>Formule :C17H21Cl2F3N5Na4O12P3S2Degré de pureté :98.51% - 98.6%Couleur et forme :SolidMasse moléculaire :864.294-Octyl itaconate
CAS :<p>4-Octyl Itaconate is a cell-permeable derivative of Itaconate, an anti-inflammatory metabolite.</p>Formule :C13H22O4Degré de pureté :99.3% - 99.94%Couleur et forme :SolidMasse moléculaire :242.31Rhoifolin
CAS :<p>Rhoifolin (Apigenin 7-O-neohesperidoside) is extracted from Turpinia arguya Seem dried leaves.</p>Formule :C27H30O14Degré de pureté :98.11% - 98.58%Couleur et forme :SolidMasse moléculaire :578.52C-178
CAS :<p>C-178 inhibits STING by binding Cys91, blocking palmitoylation and TBK1 activation in HEK293T cells.</p>Formule :C17H10N2O5Degré de pureté :97.69%Couleur et forme :SolidMasse moléculaire :322.27TLR3-IN-1
CAS :<p>TLR3-IN-1 (CU CPT 4a) is a selective TLR3 inhibitor. It can inhibit TLR3/dsRNA complex-mediated downstream signaling pathways and inhibit the TNF-α and IL-1β.</p>Formule :C18H13ClFNO3SDegré de pureté :98.56%Couleur et forme :SolidMasse moléculaire :377.82MLT-943
CAS :<p>MLT-943 is a potent, selective and orally active MALT1 protease inhibitor. [1].</p>Formule :C16H14ClF3N6O2Degré de pureté :99.72% - 99.82%Couleur et forme :SolidMasse moléculaire :414.77E6446
CAS :<p>E6446 inhibits Toll-like receptor (TLR)7 and 9 signaling.</p>Formule :C27H35N3O3Degré de pureté :98.72%Couleur et forme :SolidMasse moléculaire :449.59Bay 11-7085
CAS :<p>Bay 11-7085 can irreversibly inhibit the IκBα phosphorylation induced by TNFα (IC50: 10 μM).</p>Formule :C13H15NO2SDegré de pureté :99.76% - 99.94%Couleur et forme :White SolidMasse moléculaire :249.33Glu-urea-Lys TFA(1025796-69-3 free base)
<p>Glu-urea-Lys TFA (1025796-69-3 free base) is a PSMA inhibitor.</p>Formule :C14H22F3N3O9Degré de pureté :99.91%Couleur et forme :SolidMasse moléculaire :433.34Fas C-Terminal Tripeptide Acetate
<p>Fas C-Terminal Tripeptide Acetate shows inhibitory activity of Fas/FAP-1 binding.</p>Formule :C18H33N3O8Degré de pureté :99.12%Couleur et forme :SolidMasse moléculaire :419.47CU-CPT-9a
CAS :<p>CU-CPT-9a is a potent TLR8 inhibitor (IC50 : 0.5 nM), that suppresses TLR8-mediated proinflammatory signaling in various cell lines and human primary cells-</p>Formule :C17H15NO2Degré de pureté :99.01%Couleur et forme :SolidMasse moléculaire :265.31Ginsenoside Rg2
CAS :<p>Ginsenoside Rg2 (Chikusetsusaponin I) is one of the major active components of ginseng, act as an NF-κB inhibitor.</p>Formule :C42H72O13Degré de pureté :99.77% - 99.78%Couleur et forme :SolidMasse moléculaire :785.01Convallatoxin
CAS :<p>Convallatoxin is a natural product.</p>Formule :C29H42O10Degré de pureté :99.27% - 99.53%Couleur et forme :Prisms From Methanol + Ether SolidMasse moléculaire :550.64GSK717
CAS :<p>GSK717: potent, selective NOD2 inhibitor; disrupts NOD2/TLR2 synergy; no effect on NOD1, TNFR1, TLR2.</p>Formule :C28H28N4O2Degré de pureté :97.34% - 99.01%Couleur et forme :SolidMasse moléculaire :452.55NG,NG-dimethyl-L-Arginine dihydrochloride
CAS :<p>NG,NG-dimethyl-L-Arginine dihydrochloride is an endogenous nitric oxide synthase inhibitor.</p>Formule :C8H20Cl2N4O2Degré de pureté :97.83% - 99.18%Couleur et forme :SolidMasse moléculaire :275.18Bortezomib
CAS :<p>Bortezomib (LDP 341) is a 20S proteasome inhibitor (Ki=0.6 nM) that is reversible and selective.</p>Formule :C19H25BN4O4Degré de pureté :97.79% - >99.99%Couleur et forme :Yellow SolidMasse moléculaire :384.24Dehydrodiisoeugenol
CAS :<p>Dehydrodiisoeugenol suppresses COX-2 expression and NF-κB activity, reducing inflammation in LPS-stimulated murine macrophages.</p>Formule :C20H22O4Degré de pureté :99.97%Couleur et forme :SolidMasse moléculaire :326.39SP-13786
CAS :<p>SP-13786 is an inhibitor of fibroblast activation protein (FAP) and prolyl oligopeptidase (PREP).Cost-effective and quality-assured.</p>Formule :C17H14F2N4O2Degré de pureté :99.52% - 99.96%Couleur et forme :SolidMasse moléculaire :344.32TLR7/8/9-IN-1
CAS :<p>TLR7/8/9-IN-1 is a potent inhibitor of Toll-like receptors 7/8/9 (TLR7/8/9) with an IC50 of 43 nM.</p>Formule :C27H37N3O2Degré de pureté :99.56%Couleur et forme :SolidMasse moléculaire :435.6Stachydrine Hydrochloride
CAS :<p>Stachydrine Hydrochloride is an effective component that mainly extracted from the leaf of Leonurussibiricus.</p>Formule :C7H14ClNO2Degré de pureté :99.53% - 99.71%Couleur et forme :Light Yellow PasteMasse moléculaire :179.64Ginsenoside Rg1
CAS :<p>Ginsenoside Rg1 (Panaxoside Rg1) is a class of steroid glycosides, and triterpene saponins found exclusively in the plant genus Panax (ginseng).</p>Formule :C42H72O14Degré de pureté :99% - 99.74%Couleur et forme :White Crystalline PowderMasse moléculaire :801.01GSK963
CAS :<p>GSK963 (Racemate), a structurally distinct, potent and selective inhibitor of RIP1 kinase(IC50=29 nM).</p>Formule :C14H18N2ODegré de pureté :98.00%Couleur et forme :SolidMasse moléculaire :230.31Kaempferol-3-O-glucorhamnoside
CAS :<p>Kaempferol-3-O-glucorhamnoside (Kaempferol 3-glucorhamnoside), a flavonoid derived from plant Thesium chinense Turcz, inhibits inflammatory responses via MAPK</p>Formule :C27H30O15Degré de pureté :96.96% - 98.17%Couleur et forme :SolidMasse moléculaire :594.5Saikosaponin D
CAS :<p>Saikosaponin D is a novel SERCA inhibitor by inhibiting NF-κB and STAT3 signaling to protect against acetaminophen-induced hepatotoxicity.</p>Formule :C42H68O13Degré de pureté :98.34% - 99.73%Couleur et forme :White PowderMasse moléculaire :780.98TLR4-IN-C34
CAS :<p>TLR4-IN-C34 is an inhibitor of TLR4, and reduces systemic inflammation in models of endotoxemia and necrotizing enterocolitis</p>Formule :C17H27NO9Degré de pureté :99.69%Couleur et forme :SolidMasse moléculaire :389.4RCGD423
CAS :<p>RCGD423, a small molecule gp130 modulator, prevents articular cartilage degeneration and promotes repair.</p>Formule :C15H11BrN2SDegré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :331.23Bropirimine
CAS :<p>Bropirimine (U-54461) (U-54461) is a biological response modifier that is thought to act through the induction of lymphokines.</p>Formule :C10H8BrN3ODegré de pureté :99.01%Couleur et forme :SolidMasse moléculaire :266.09GP130 receptor agonist-1
CAS :<p>GP130 receptor agonist-1 (N-(4-Fluorophenyl)-4-phenyl-2-thiazolami) is a potent, brain-penetrant and orally active GP130 receptor agonist.</p>Formule :C15H11FN2SDegré de pureté :99.62%Couleur et forme :SolidMasse moléculaire :270.32IMD-0354
CAS :<p>IMD-0354 (IKK2 Inhibitor V) is an IKKβ inhibitor and inhibits IκBα phosphorylation in NF-κB pathway.</p>Formule :C15H8ClF6NO2Degré de pureté :99.65% - 99.98%Couleur et forme :SolidMasse moléculaire :383.67HPGDS inhibitor 1
CAS :<p>HPGDS inhibitor 1 is a novel and selective inhibitor for Hematopoietic Prostaglandin D Synthase (HPGDS) with an IC50 Value of 0.7 nM.</p>Formule :C19H19F4N3ODegré de pureté :98% - 99.18%Couleur et forme :SolidMasse moléculaire :381.37Muscone
CAS :<p>Muscone (3-Methylcyclopentadecanone) is an organic compound that is the primary contributor to the odor of musk.</p>Formule :C16H30ODegré de pureté :98.97% - ≥98%Couleur et forme :Colourless Liquid LiquidMasse moléculaire :238.41CID1231538
CAS :<p>CID1231538 is a potent GPR35 antagonist.</p>Formule :C26H22ClN3O3S2Degré de pureté :98.79%Couleur et forme :SolidMasse moléculaire :524.05Camstatin acetate
<p>Camstatin acetate, a 25-residue fragment, inhibits neuronal NOS by binding calmodulin.</p>Formule :C124H207N39O36Degré de pureté :98.3%Couleur et forme :SolidMasse moléculaire :2820.21IRAK4-IN-7
CAS :<p>IRAK4-IN-7 (CA-4948) is a selective and potent IRAK4 kinase inhibitor with in vivo activity in a TLR4-induced cytokine release model.</p>Formule :C21H19N7O3Degré de pureté :99.5%Couleur et forme :SolidMasse moléculaire :417.42BC-1382
CAS :<p>BC-1382 is a potent ubiquitin E3 ligase HECTD2 inhibitor that specificly disrupts the HECTD2/PIAS1 interaction(IC50 of 5 nM).</p>Formule :C23H29N3O5SDegré de pureté :99.15% - 99.94%Couleur et forme :SolidMasse moléculaire :459.56PFI-2 hydrochloride
CAS :<p>PFI-2 hydrochloride ((R)-PFI-2 hydrochloride) is a potent, highly selective, and cell-active inhibitor of the methyltransferase activity of SETD7 (IC50: 2 nM),</p>Formule :C23H26ClF4N3O3SDegré de pureté :99.31% - 99.91%Couleur et forme :SolidMasse moléculaire :535.98Adrenic Acid
CAS :<p>Adrenic Acid (cis-7,10,13,16-Docosatetraenoic acid) is a member of the class of compounds known as very-long-chain fatty acids.</p>Formule :C22H36O2Degré de pureté :95.63% - 98.42%Couleur et forme :SolidMasse moléculaire :332.52S-(2-aminoethyl) Isothiourea (dihydrobromide)
CAS :<p>S-(2-aminoethyl) isothiourea inhibits all NOS types: Ki for nNOS 1.8μM, eNOS 2.1μM, iNOS 0.59μM.</p>Formule :C3H11Br2N3SDegré de pureté :99.77%Couleur et forme :SolidMasse moléculaire :281.02Adenosine N1-oxide
CAS :<p>Adenosine N1-oxide (1-Oxoadenosine), which is found in royal jelly, inhibited the secretion of inflammatory mediators by activated macrophages and reduced</p>Formule :C10H13N5O5Degré de pureté :99.9%Couleur et forme :SolidMasse moléculaire :283.24BOT-64
CAS :<p>BOT-64 is an IKK-2 inhibitor which targets the Ser177 and/or Ser181 residues in the kinase's activation loop domain.BOT-64 is a cell-permeable benzoxathiole</p>Formule :C15H15NO2SDegré de pureté :99.73%Couleur et forme :SolidMasse moléculaire :273.35Flaconitine
CAS :<p>Flaconitine (Acetylaconitine) is an NF-κB inhibitor and an alkaloid.</p>Formule :C36H49NO12Degré de pureté :98% - 99.84%Couleur et forme :SolidMasse moléculaire :687.77Ipilimumab
CAS :<p>Ipilimumab (anti-CTLA-4) is an immunomodulatory monoclonal antibody directed against the cell surface antigen CTLA-4 and also a type of immune checkpoint</p>Degré de pureté :98.50% - 99.60%Couleur et forme :LiquidMasse moléculaire :148 kDa
