Protéases/Protéasome
Les inhibiteurs de protéases et de protéasomes sont des composés qui bloquent l'activité des protéases et du protéasome, impliqués dans la dégradation et le renouvellement des protéines. Ces inhibiteurs sont essentiels pour étudier la régulation de l'homéostasie des protéines, le contrôle du cycle cellulaire et l'apoptose. Les inhibiteurs de protéases et de protéasomes sont également utilisés dans le traitement de maladies telles que le cancer, où une dégradation anormale des protéines joue un rôle dans la progression de la maladie. En inhibant les protéases ou le protéasome, ces composés peuvent induire la mort cellulaire dans les cellules cancéreuses et sont des outils essentiels tant pour la recherche fondamentale que pour le développement thérapeutique. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de protéases et de protéasomes de haute qualité pour soutenir vos recherches en biochimie, biologie cellulaire et développement de médicaments.
Sous-catégories appartenant à la catégorie "Protéases/Protéasome"
- Acétyl-CoA Carboxylase(38 produits)
- Cystéine protéase(111 produits)
- DPP-4(27 produits)
- Glutaminase(46 produits)
- Protéase du VIH(506 produits)
- PAI-1(26 produits)
- Inhibiteurs de protéase(50 produits)
- Récepteur activé par une protéase(55 produits)
- Protéasome(86 produits)
- Sérine protéase(54 produits)
- p97(15 produits)
Affichez 3 plus de sous-catégories
985 produits trouvés pour "Protéases/Protéasome"
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MDL-28170
CAS :MDL-28170 (Calpain Inhibitor III) is a Cysteine protease.Formule :C22H26N2O4Degré de pureté :95.06%Couleur et forme :SolidMasse moléculaire :382.45Ref: TM-T2470
1mg34,00€2mg49,00€5mg71,00€10mg90,00€25mg128,00€50mg167,00€100mg284,00€1mL*10mM (DMSO)75,00€Bemnifosbuvir hemisulfate
CAS :Bemnifosbuvir hemisulfate (AT-527) is a potent inhibitor of HCV virus replication.Formule :C48H68F2N14O18P2SDegré de pureté :99.98%Couleur et forme :SolidMasse moléculaire :1261.15Telaprevir
CAS :Telaprevir (Incivek) (VX-950) is an effective inhibitor of HCV NS3-4A serine protease (IC50: 0.35 μM).Formule :C36H53N7O6Degré de pureté :96.9% - 98.89%Couleur et forme :SolidMasse moléculaire :679.85NSC 405020
CAS :NSC 405020 is a noncatalytic inhibitor of MT1-MMP.Formule :C12H15Cl2NODegré de pureté :96.93% - 99.07%Couleur et forme :SolidMasse moléculaire :260.16CGS 27023A
CAS :CGS 27023A is a non-peptidic, potent, and orally active stromelysin inhibitor.Formule :C18H24ClN3O5SDegré de pureté :99.08%Couleur et forme :SolidMasse moléculaire :429.92Picolamine
CAS :Picolamine acts as a potential inhibitor of DPP-4.Formule :C6H8N2Degré de pureté :98.3%Couleur et forme :Light Yellow LiquidMasse moléculaire :108.14Bortezomib-pinanediol
CAS :Bortezomib-pinanediol is a proteasome inhibitor. is a prodrug of Bortezomib.Formule :C29H39BN4O4Degré de pureté :97.5%Couleur et forme :Yellow SolidMasse moléculaire :518.46SB-3CT
CAS :SB-3CT is a potent and specific gelatinase inhibitor for MMP-2(Ki=13.9 nM) and MMP-9(Ki=600 nM).Formule :C15H14O3S2Degré de pureté :98% - 99.38%Couleur et forme :SolidMasse moléculaire :306.4Ref: TM-T2009
1mg46,00€2mg62,00€5mg94,00€10mg150,00€25mg234,00€50mg349,00€100mg518,00€500mg1.134,00€1mL*10mM (DMSO)94,00€Tenofovir alafenamide hemifumarate
CAS :Tenofovir alafenamide hemifumarate (GS-7340 hemifumarate) is an oral phosphonoamidate prodrug of the HIV reverse transcriptase nucleotide inhibitor tenofovir.
Formule :C21H29N6O5PC4H4O4Degré de pureté :99.33% - 99.96%Couleur et forme :SolidMasse moléculaire :534.51Trelagliptin succinate
CAS :Trelagliptin succinate (SYR-472 succinate) is a long-acting inhibitor of dipeptidyl peptidase-4 (DPP-4), being developed for the treatment of type 2 diabetes (Formule :C22H26FN5O6Degré de pureté :99.27% - 99.92%Couleur et forme :SolidMasse moléculaire :475.47Ilomastat
CAS :Ilomastat (GM6001) (GM6001, Galardin) is a broad spectrum matrix metalloprotease (MMP) inhibitor.Formule :C20H28N4O4Degré de pureté :97.04% - 99.51%Couleur et forme :SolidMasse moléculaire :388.46Ref: TM-T2743
1mg46,00€2mg62,00€5mg89,00€10mg145,00€25mg255,00€50mg429,00€100mg620,00€200mg880,00€1mL*10mM (DMSO)94,00€Ledipasvir (acetone)
CAS :Ledipasvir (acetone) (GS-5885 acetone) is an HCV NS5A polymerase inhibitor, used for the treatment of hepatitis C virus infection.Formule :C52H60F2N8O7Degré de pureté :99.72%Couleur et forme :SolidMasse moléculaire :947.08Ref: TM-T4203
1mg34,00€2mg46,00€5mg66,00€10mg88,00€25mg144,00€50mg222,00€100mg340,00€200mg504,00€1mL*10mM (DMSO)92,00€2-Benzylsuccinic acid
CAS :2-Benzylsuccinic acid (DL-Benzylsuccinic acid) is a bacterial xenobiotic metabolite.Formule :C11H12O4Degré de pureté :99.01% - ≥95%Couleur et forme :SolidMasse moléculaire :208.21(R)-MG-132
CAS :(R)-MG-132 (Z-Leu-D-leu-leu-al) is the enantiomer of MG-132. (R)-MG-132 stereoisomer is a more potent proteasome inhibitor than MG-132.Formule :C26H41N3O5Degré de pureté :99.90%Couleur et forme :SolidMasse moléculaire :475.62Ref: TM-T12628
2mg38,00€5mg57,00€10mg79,00€25mg120,00€50mg177,00€100mg268,00€200mg398,00€1mL*10mM (DMSO)71,00€Odanacatib
CAS :Odanacatib is an inhibitor of cathepsin K with potential anti-osteoporotic activity.Formule :C25H27F4N3O3SDegré de pureté :98.53% - 99.53%Couleur et forme :SolidMasse moléculaire :525.56Dabigatran
CAS :Dabigatran (BIBR 953ZW), a thrombin inhibitor, prevents thrombus formation, reducing stroke and embolism risk in nonvalvular atrial fibrillation patients.Formule :C25H25N7O3Degré de pureté :97.44% - 98.7%Couleur et forme :Tan SolidMasse moléculaire :471.51CTTHWGFTLC, CYCLIC acetate(244082-19-7 free base)
CTTHWGFTLC, CYCLIC acetate is an inhibitor for matrix metalloproteinases (MMP)-2 and MMP-9.Formule :C54H75N13O16S2Degré de pureté :99.71%Couleur et forme :SolidMasse moléculaire :1226.39Mericitabine
CAS :Mericitabine (R-7128) is an HCV inhibitor that terminates RNA chains, halting replication.Formule :C18H26FN3O6Degré de pureté :97.77% - 98.54%Couleur et forme :SolidMasse moléculaire :399.41Ref: TM-T16710
1mg50,00€5mg103,00€10mg142,00€25mg239,00€50mg350,00€100mg500,00€200mg682,00€1mL*10mM (DMSO)110,00€Elbasvir
CAS :Elbasvir (MK-8742) is an NS5A inhibitor developed for chronic HCV treatment.Formule :C49H55N9O7Degré de pureté :98.95% - 99.85%Couleur et forme :SolidMasse moléculaire :882.02Ref: TM-T4544
1mg42,00€2mg52,00€5mg79,00€10mg113,00€25mg200,00€50mg334,00€100mg537,00€1mL*10mM (DMSO)111,00€AF 399
CAS :AF 399 is a CCR4 antagonist. It reverses the tumor-promoting environment.Formule :C12H17N3O3SDegré de pureté :99.83%Couleur et forme :SolidMasse moléculaire :283.35Ref: TM-T23646
1mg64,00€5mg129,00€10mg188,00€25mg299,00€50mg427,00€100mg575,00€200mg750,00€1mL*10mM (DMSO)124,00€Daclatasvir dihydrochloride
CAS :Daclatasvir dihydrochloride is an oral antiviral that treats chronic hepatitis C by inhibiting HCV's NS5A; rare liver enzyme elevation, seldom causes jaundice.Formule :C40H52Cl2N8O6Degré de pureté :99.67%Couleur et forme :SolidMasse moléculaire :811.8Ref: TM-T1786
1g230,00€5mg39,00€10mg48,00€25mg57,00€50mg67,00€100mg77,00€500mg161,00€1mL*10mM (DMSO)49,00€Glecaprevir
CAS :Glecaprevir (ABT-493) is an HCV NS3/4A protease inhibitor, (IC50s: 3.5-11.3 nM).Formule :C38H46F4N6O9SDegré de pureté :99.16% - 99.69%Couleur et forme :SolidMasse moléculaire :838.87Paritaprevir
CAS :Paritaprevir (ABT450) 是一种非结构蛋白 3/4A 蛋白酶抑制剂，对 HCV 1a 和 HCV 1b 的 EC50 值分别为 1 和 0.21 nM。它也是SARS-CoV 3CLpro 的抑制剂，IC50为 1.31 μM。
Formule :C40H43N7O7SDegré de pureté :99.72%Couleur et forme :SolidMasse moléculaire :765.887-benzyl-5,6-dimethyl-7H-pyrrolo[2,3-d]pyrimidin-4-amine
CAS :7-benzyl-5,6-dimethyl-7H-pyrrolo[2,3-d]pyrimidin-4-amine is a inhibitor of Hepatitis C Virus(HCV).Formule :C15H16N4Degré de pureté :99.22%Couleur et forme :SolidMasse moléculaire :252.31Avatrombopag
CAS :Avatrombopag (YM477) is a new oral thrombopoietin (TPO) receptor agonist, activating TPO receptor and increasing megakaryocytic proliferation/differentiationFormule :C29H34Cl2N6O3S2Degré de pureté :99.01% - 99.63%Couleur et forme :SolidMasse moléculaire :649.65Ref: TM-T7417
1mg57,00€5mg120,00€10mg187,00€25mg339,00€50mg540,00€100mg747,00€200mg1.035,00€1mL*10mM (DMSO)167,00€PSI-6206
CAS :PSI-6206 (RO 2433) (RO2433) is a selective HCV RNA polymerase inhibitor.Formule :C10H13FN2O5Degré de pureté :98% - 99.79%Couleur et forme :SolidMasse moléculaire :260.22S 3304
CAS :S 3304 is a novel matrix metalloproteinases inhibitor which is specific for MMP-2 and MMP-9.Formule :C24H20N2O4S2Degré de pureté :98.09%Couleur et forme :SolidMasse moléculaire :464.56Ref: TM-T16966
1mg42,00€2mg60,00€5mg105,00€10mg170,00€25mg281,00€50mg395,00€100mg537,00€200mg725,00€1mL*10mM (DMSO)108,00€Balicatib
CAS :Balicatib (AAE581) is a potent and selective inhibitor of cathepsin K, used in trials studying the treatment of osteoporosis.Formule :C23H33N5O2Degré de pureté :97.78% - 98.17%Couleur et forme :White To Off-White Solid PowderMasse moléculaire :411.54Ref: TM-T1850
2mg39,00€5mg58,00€10mg94,00€25mg212,00€50mg358,00€100mg572,00€200mg803,00€1mL*10mM (DMSO)64,00€Clemizole hydrochloride
CAS :Clemizole hydrochloride blocks H1 histamine receptors and inhibits HCV replication and NS4B RNA binding.Formule :C19H21Cl2N3Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :362.3Talabostat mesylate
CAS :Talabostat mesylate (PT100): Oral DPP4 inhibitor, IC50 0.18 nM, targets tumor-linked proteins, boosts hematopoiesis.Formule :C10H23BN2O6SDegré de pureté :98% - 99.91%Couleur et forme :SolidMasse moléculaire :310.18Darunavir Ethanolate
CAS :Darunavir Ethanolate (UIC 94017) is an HIV PROTEASE INHIBITOR that is used in the treatment of AIDS and HIV INFECTIONS.Formule :C29H43N3O8SDegré de pureté :99.84% - 99.86%Couleur et forme :SolidMasse moléculaire :593.74Ref: TM-T3335
5mg37,00€10mg52,00€25mg80,00€50mg111,00€100mg165,00€200mg236,00€500mg399,00€1mL*10mM (DMSO)48,00€Anagliptin
CAS :Anagliptin (SK-0403) is a potent Inhibitor of DPP-4(IC50 of 3.8 nM), for the treatment of type 2 diabetes mellitus.Formule :C19H25N7O2Degré de pureté :97.59% - 99.98%Couleur et forme :SolidMasse moléculaire :383.45Ref: TM-T7133
1mg44,00€5mg96,00€10mg130,00€25mg212,00€50mg314,00€100mg477,00€200mg677,00€1mL*10mM (DMSO)92,00€Samatasvir
CAS :Samatasvir (ATOLIHZIXHZSBA-BTSKBWHGSA-N) is a pan-genotypic inhibitor of the HCV non-structural protein 5A.Formule :C47H48N8O6S2Degré de pureté :98.03%Couleur et forme :SolidMasse moléculaire :885.06Ref: TM-T9567
1mg55,00€5mg116,00€10mg187,00€25mg376,00€50mg632,00€100mg1.008,00€1mL*10mM (DMSO)197,00€L-Albizziin
CAS :L-Albizziin (L-beta-Ureidoalanine) is a glutamase inhibitor and is a glutaminyl-tRNA synthetase inhibitor.Formule :C4H9N3O3Degré de pureté :99.98%Couleur et forme :White PowderMasse moléculaire :147.13NQ301
CAS :NQ301, an antithrombotic agent, inhibits collagen-challenged rabbit platelet aggregation (IC50: 10 mg/mL).Formule :C18H12ClNO3Degré de pureté :99.74% - 99.76%Couleur et forme :SolidMasse moléculaire :325.75Glutaminase C-IN-1
CAS :Glutaminase C-IN-1 (Compound 968) is a Glutaminase C allosteric inhibitor.Formule :C27H27BrN2ODegré de pureté :99.68% - >99.99%Couleur et forme :SolidMasse moléculaire :475.42Ref: TM-T3964
2mg42,00€5mg60,00€10mg87,00€25mg162,00€50mg273,00€100mg378,00€200mg557,00€1mL*10mM (DMSO)67,00€2,4-Dioxaspiro(5.5)undec-8-ene, 3-(2-furanyl)-
CAS :2,4-Dioxaspiro(5.5)undec-8-ene, 3-(2-furanyl)- (Ulinastatin) ,as an urinary trypsin inhibitor (UTI), is a glycoprotein that is isolated from healthy human urineFormule :C13H16O3Degré de pureté :99.53% - 99.81%Couleur et forme :SolidMasse moléculaire :220.26Ref: TM-T8802
1mg82,00€5mg168,00€10mg244,00€25mg404,00€50mg567,00€100mg767,00€500mg1.521,00€1mL*10mM (DMSO)146,00€Ximelagatran
CAS :Ximelagatran, oral direct thrombin inhibitor, transforms to active melagatran in body.Formule :C24H35N5O5Degré de pureté :95.48% - 99.60%Couleur et forme :SolidMasse moléculaire :473.57Sofosbuvir
CAS :Sofosbuvir (GS 7977) is a uridine monophosphate analog inhibitor of hepatitis C virus (HCV) polymerase NS5B that is used as an antiviral agent in the treatmentFormule :C22H29FN3O9PDegré de pureté :99.77% - 99.82%Couleur et forme :SolidMasse moléculaire :529.45Proteinase K
CAS :Proteinase K (Protease K) is a non-specific serine protease. Proteinase K hydrolyzes peptide bonds and is used for protein digestion. Cost-effective and quality-assured.Formule :C29H27N2O12PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :626.511Histatin 5 acetate
Histatin 5 acetate inhibits the activity of the host matrix metalloproteinases MMP-2 and MMP-9 with IC50s of 0.57 and 0.25 μM, respectively.Formule :C135H199N51O35Degré de pureté :98.72%Couleur et forme :SolidMasse moléculaire :3096.35MUN57694
CAS :MUN57694 is an inhibitor of 26S proteasome.Formule :C23H25N3O4Degré de pureté :99%Couleur et forme :SolidMasse moléculaire :407.46Ref: TM-T9090
2mg35,00€5mg52,00€10mg86,00€25mg145,00€50mg210,00€100mg296,00€200mg414,00€1mL*10mM (DMSO)64,00€Lersivirine
CAS :Lersivirine (UK-453061)(UK 453061) is a second-generation non-nucleoside reverse transcriptase inhibitor (NNRTI) under development for HIV infection therapy.Formule :C17H18N4O2Degré de pureté :98.01%Couleur et forme :SolidMasse moléculaire :310.35Clemizole
CAS :Clemizole is an H1 histamine receptor antagonist, can inhibit NS4B's RNA binding and hepatitis C virus (HCV) replication.Formule :C19H20ClN3Degré de pureté :98% - 99.65%Couleur et forme :SolidMasse moléculaire :325.84Ref: TM-T1822
1mg42,00€5mg82,00€10mg101,00€25mg152,00€50mg256,00€100mg460,00€500mg973,00€1mL*10mM (DMSO)93,00€VCH-916 free acid(1200133-34-1 free base)
CAS :VCH-916 is a novel nonnucleoside HCV NS5B polymerase inhibitor.Formule :C26H37NO4SDegré de pureté :98.45%Couleur et forme :SolidMasse moléculaire :459.64Boceprevir
CAS :Boceprevir (SCH 503034), an oral HCV NS3 protease inhibitor, has a Ki of 14 nM and EC90 of 350 nM.Formule :C27H45N5O5Degré de pureté :95% - 99.16%Couleur et forme :SolidMasse moléculaire :519.68Ref: TM-T4988
1mg34,00€5mg66,00€10mg90,00€25mg137,00€50mg177,00€100mg260,00€200mg358,00€1mL*10mM (DMSO)75,00€Voxilaprevir
CAS :Voxilaprevir is an inhibitor of hepatitis C virus (HCV) nonstructural (NS) protein 3/4A protease.Formule :C40H52F4N6O9SDegré de pureté :99.83% - 99.98%Couleur et forme :SolidMasse moléculaire :868.93Ref: TM-T19862
1mg75,00€5mg295,00€10mg423,00€25mg708,00€50mg954,00€100mg1.288,00€200mg1.738,00€1mL*10mM (DMSO)394,00€PythiDC
CAS :PythiDC is a selective collagen prolyl 4-hydroxylase inhibitor, neither causing general toxicity nor disrupting iron homeostasis.Formule :C10H6N2O4SDegré de pureté :98.13%Couleur et forme :SolidMasse moléculaire :250.23FT011
CAS :FT011, a direct anti-fibrotic agent,attenuates cardiac remodelling and dysfunction in experimental diabetic cardiomyopathy.Formule :C20H17NO5Degré de pureté :98.98%Couleur et forme :SolidMasse moléculaire :351.35HCV-IN-31
CAS :HCV-IN-31 is a HCV inhibitor with an EC50/EC95 of 15.7 μM.Formule :C12H17FN6O3Degré de pureté :99.83%Couleur et forme :SolidMasse moléculaire :312.3GK921
CAS :GK921 is a transglutaminase 2 (TGase) inhibitor.Formule :C21H20N4ODegré de pureté :97.44% - 99.49%Couleur et forme :SolidMasse moléculaire :344.41Grazoprevir hydrate
CAS :Grazoprevir: Hepatitis C protease inhibitor effective against various genotypes, including drug-resistant strains.Formule :C38H52N6O10SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :784.92Proteasome inhibitor IX
CAS :Proteasome inhibitor IX (PS-IX) is an inhibitor of chymotrypsin-like activity of the 20S proteasome (IC50 ~1 μM).Formule :C20H21B2NO5Degré de pureté :99.77%Couleur et forme :SolidMasse moléculaire :377.01Ombitasvir
CAS :Ombitasvir (ABT-267) inhibits HCV protein NS5A, effective orally, EC50: 0.82-19.3 pM (genotypes 1-5), 366 pM (genotype 6a).Formule :C50H67N7O8Degré de pureté :97.27% - 99.56%Couleur et forme :SolidMasse moléculaire :894.11Ref: TM-T7158
2mg40,00€5mg75,00€10mg105,00€25mg215,00€50mg313,00€100mg462,00€500mg973,00€1mL*10mM (DMSO)105,00€2-(2-bromophenyl)-5-chloro-4H-3,1-benzoxazin-4-one
CAS :2-(2-bromophenyl)-5-chloro-4H-3,1-benzoxazin-4-one is an human neutrophil elastase inhibitor.Formule :C14H7BrClNO2Degré de pureté :97.36%Couleur et forme :SolidMasse moléculaire :336.57Coblopasvir
CAS :Coblopasvir is a pan-genotypic non-structural protein 5A (NS5A) inhibitor. It can be used to study chronic hepatitis C virus infection.Formule :C41H50N8O8Degré de pureté :99.33%Couleur et forme :SolidMasse moléculaire :782.88GW280264X
CAS :GW280264X (Carbamic acid) is an inhibitor of ADAM17 .Formule :C28H41N5O6SDegré de pureté :99.51%Couleur et forme :SolidMasse moléculaire :575.72Ref: TM-T8961
1mg156,00€5mg319,00€10mg477,00€25mg773,00€50mg1.063,00€100mg1.431,00€1mL*10mM (DMSO)404,00€Ivachtin
CAS :Ivachtin (Caspase-3 Inhibitor VII) is a nonpeptide, noncompetitive and reversibl caspase-3 inhibitor(IC50 = 23 nM) and is a modest inhibitor of the remaining
Formule :C20H21N3O7SDegré de pureté :99.74%Couleur et forme :SolidMasse moléculaire :447.46VCH-916
CAS :VCH-916 is a new nonnucleoside inhibitor of HCV NS5B polymerase.Formule :C26H36KNO4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :497.732-PMPA
CAS :2-PMPA (2-(Phosphonomethyl)pentanedioic acid) is a potent and selective inhibitor of glutamate carboxypeptidase II (GCPII) (IC50=300 pM).Formule :C6H11O7PDegré de pureté :97.4% - 99.5%Couleur et forme :SolidMasse moléculaire :226.12Omarigliptin
CAS :Omarigliptin is a potent and selective oral dipeptidyl peptidase 4 (DPP4) inhibitor with IC50 value of 1.6 nM. Cost-effective and quality-assured.Formule :C17H20F2N4O3SDegré de pureté :99.68% - 99.77%Couleur et forme :SolidMasse moléculaire :398.43Ref: TM-T2316
1mg38,00€2mg50,00€5mg80,00€10mg117,00€25mg200,00€50mg333,00€100mg477,00€500mg1.063,00€1mL*10mM (DMSO)131,00€7-Amino-4-methylcoumarin-3-acetic acid
CAS :7-Amino-4-methylcoumarin-3-acetic acid (7-Amino-4-methylcoumarin) is more suitable as a substrate for enteropeptidase than GD(4)K-NA.Formule :C12H11NO4Degré de pureté :98.38%Couleur et forme :SolidMasse moléculaire :233.22Tegobuvir
CAS :Tegobuvir (GS 333126) is a specific and covalent HCV NS5B polymerase inhibitor.Formule :C25H14F7N5Degré de pureté :99.21%Couleur et forme :SolidMasse moléculaire :517.4Ref: TM-T17029
1mg84,00€5mg177,00€10mg295,00€25mg504,00€50mg712,00€100mg982,00€1mL*10mM (DMSO)202,00€2-Cyanopyrimidine
CAS :2-Cyanopyrimidine (m-Hydroxyphenylpropionic acid) is inhibitor of cathepsin K(IC50 : 170 nM)Formule :C5H3N3Degré de pureté :99.27%Couleur et forme :Crystalline SolidMasse moléculaire :105.1Ledipasvir hydrochloride
CAS :Ledipasvir hydrochloride, a hepatitis C NS5A inhibitor, has EC50 of 34 pM (1a) and 4 pM (1b), also inhibits SARS-CoV 3CL pro (IC50 1.62 µM).Formule :C49H55ClF2N8O6Couleur et forme :SolidMasse moléculaire :925.46Anagliptin hydrochloride
CAS :Anagliptin (SK-0403) hydrochloride: potent, selective oral DPP-4 inhibitor; IC50: DPP-4 3.8 nM, DPP-8 68 nM, DPP-9 60 nM.Formule :C19H26ClN7O2Couleur et forme :SolidMasse moléculaire :419.91Bz-RS-ISer(3-Ph)-Ome
CAS :Bz-RS-ISer(3-Ph)-Ome (Methyl (2R,3S)-3-(benzoylamino)-2-hydroxy-3-phenylpropanoate) is a paclitaxel derivative that inhibits the HSV replication cycle.
Formule :C17H17NO4Degré de pureté :99.36% - 99.89%Couleur et forme :White CrystalMasse moléculaire :299.32L-006235
CAS :L-006235 is a potent and reversible inhibitor of cathepsin K with IC50 of 0.25 nM.Formule :C24H30N6O2SDegré de pureté :99.37%Couleur et forme :SolidMasse moléculaire :466.6Ref: TM-T21616
2mg39,00€5mg60,00€10mg92,00€25mg177,00€50mg299,00€100mg432,00€200mg602,00€1mL*10mM (DMSO)62,00€NM107
CAS :NM107, a ribonucleoside, inhibits HCV NS5B polymerase. It has broad antiviral properties with EC50 of 1.85 μM in wild-type cells.Formule :C10H15N3O5Degré de pureté :97.85%Couleur et forme :White To Off-White PowderMasse moléculaire :257.24Simeprevir
CAS :Simeprevir (TMC435) is a potent HCV NS3/4A protease inhibitor, and inhibits HCV replication with EC50 of 8 nM.Formule :C38H47N5O7S2Degré de pureté :99.45% - 99.92%Couleur et forme :SolidMasse moléculaire :749.94Efegatran
CAS :Efegatran is a hematologic agent and platelet aggregation inhibitor.
Formule :C21H32N6O3Couleur et forme :SolidMasse moléculaire :416.52T-26c
CAS :T-26c is highly potent and selective matrix metalloproteinase-13 (MMP-13) inhibitor (IC50: 6.75 pM).Formule :C24H21N3O6SDegré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :479.51Ref: TM-T5361
1mg46,00€2mg60,00€5mg90,00€10mg144,00€25mg236,00€50mg403,00€100mg582,00€1mL*10mM (DMSO)92,00€JNJ0966
CAS :JNJ0966 is a highly selective MMP-9 zymogen inhibitor (IC50: 440 nM).Formule :C16H16N4O2S2Degré de pureté :99.46% - 99.62%Couleur et forme :SolidMasse moléculaire :360.45Ref: TM-T4783
2mg34,00€5mg46,00€10mg64,00€25mg126,00€50mg219,00€100mg315,00€200mg434,00€1mL*10mM (DMSO)35,00€Tris(4-aminophenyl)methane
CAS :Tris(4-aminophenyl)methane (Leucopararosaniline), a triphenylmethane dye, is a weak HCV helicase inhibitor.Formule :C19H19N3Degré de pureté :95.73%Couleur et forme :Beige Solid CrystallineMasse moléculaire :289.37Saxagliptin
CAS :Saxagliptin (BMS-477118) is a selective and reversible DPP4 inhibitor with IC50 of 26 nM.Formule :C18H25N3O2Degré de pureté :99.17% - 99.95%Couleur et forme :SolidMasse moléculaire :315.41KKI-5 acetate(97145-43-2 free base)
KKI-5 acetate: Serine protease inhibitor, targets kallikrein/plasmin, potential anticancer and angioedema therapy.Formule :C37H59N11O11Degré de pureté :99.44%Couleur et forme :SolidMasse moléculaire :833.95Asunaprevir
CAS :Asunaprevir (BMS-650032) is an effective hepatitis C virus (HCV) NS3 protease inhibitor.Formule :C35H46ClN5O9SDegré de pureté :99.34% - 99.8%Couleur et forme :SolidMasse moléculaire :748.29Ref: TM-T4474
1mg49,00€5mg105,00€10mg170,00€25mg335,00€50mg512,00€100mg737,00€500mg1.521,00€1mL*10mM (DMSO)170,00€PSI-6130
CAS :PSI-6130 (R 1656) is a potent and selective HCV NS5B polymerase inhibitor. PSI-6130 inhibits HCV replication with a mean IC50 of 0.6 μM.Formule :C10H14FN3O4Degré de pureté :98.63% - 99.79%Couleur et forme :SolidMasse moléculaire :259.23Ref: TM-T7607
1mg38,00€5mg94,00€10mg122,00€25mg212,00€50mg313,00€100mg457,00€200mg618,00€1mL*10mM (DMSO)73,00€Z-Gly-Gly-Arg-AMC TFA (66216-78-2 free base)
CAS :Z-Gly-Gly-Arg-AMC TFA (66216-78-2 free base) is a thrombin-specific fluorogenic substrate for testing thrombin generation in PRP and platelet-poor plasma (PPP).Formule :C30H34F3N7O9Degré de pureté :99.77%Couleur et forme :SolidMasse moléculaire :693.63Ref: TM-T8556
1mg84,00€5mg167,00€10mg245,00€25mg404,00€50mg567,00€100mg767,00€200mg1.018,00€1mL*10mM (DMSO)239,00€UAMC00039 dihydrochloride
CAS :UAMC00039 dihydrochloride is a potent, reversible and competitive dipeptidyl peptidase II inhibitor with an IC50 of 0.48 nM.Formule :C16H26Cl3N3ODegré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :382.763-O-Ethyl-L-ascorbic acid
CAS :3-O-Ethyl-L-ascorbic acid is a cosmetic tyrosinase inhibitor with whitening ability and is a stabilized vitamin C derivative.Formule :C8H12O6Degré de pureté :97.35% - 99.99%Couleur et forme :White To Very Pale Yellow Crystalline Powder Solid PowderMasse moléculaire :204.18Coblopasvir dihydrochloride
CAS :Coblopasvir dihydrochloride can be used to study chronic HCV infection and is a pan-genotypic nonstructural protein 5A (NS5A) inhibitor.Formule :C41H52Cl2N8O8Degré de pureté :99.33%Couleur et forme :SolidMasse moléculaire :855.81Ref: TM-T25268L
1mg87,00€5mg187,00€10mg305,00€25mg518,00€50mg742,00€100mg1.017,00€1mL*10mM (DMSO)298,00€Camostat free base
CAS :Camostat (FOY 305) inhibits serine protease, treats cancer, viral infections, fibrosis, and blocks SARS-CoV, Coronavirus, and SARS-CoV-2 in studies.Formule :C20H22N4O5Couleur et forme :SolidMasse moléculaire :398.41Dolutegravir sodium
CAS :Dolutegravir sodium (GSK-1349572A) salt(DTG; GSK1349572) is an HIV integrase inhibitor(IC50: 2.7 nM), modest activity against raltegravir-resistant signature
Formule :C20H18F2N3NaO5Degré de pureté :98% - 99.46%Couleur et forme :SolidMasse moléculaire :441.36Fulacimstat
CAS :Fulacimstat (BAY1142524) (BAY1142524) is a chymase inhibitor, with IC50s of 3, 4 nM for hamster and human chymase enzyme, respectively.Formule :C23H16F3N3O6Degré de pureté :99.77%Couleur et forme :SolidMasse moléculaire :487.38Ref: TM-TQ0035
1mg101,00€5mg215,00€10mg313,00€25mg512,00€50mg737,00€100mg973,00€1mL*10mM (DMSO)230,00€(S,S)-TAPI-1
CAS :"(S,S)-TAPI-1, an isomer of TAPI-1, inhibits MMPs and TACE (ADAM17), reducing cell surface protein shedding."Formule :C26H37N5O5Couleur et forme :SolidMasse moléculaire :499.6Daclatasvir
CAS :Daclatasvir (EBP 883/BMS-790052) is a potent HCV NS5A inhibitor with EC50 9-50 pM across various genotypes. Phase 3.Formule :C40H50N8O6Degré de pureté :99.81% - 99.99%Couleur et forme :SolidMasse moléculaire :738.88Patamostat
CAS :Patamostat (E-3123) inhibits trypsin, plasmin, and thrombin; may reduce acute pancreatitis progression. IC50: trypsin 39 nM, plasmin 950 nM, thrombin 1.9 μM.Formule :C20H20N4O4SCouleur et forme :SolidMasse moléculaire :412.46EIDD-1931
CAS :EIDD-1931 (Beta-d-N4-hydroxycytidine) is a ribonucleoside analog with antiviral activity. It inhibits replication of SARS-CoV, MERS-CoV, and SARS-CoV-2.
Formule :C9H13N3O6Degré de pureté :99.14% - 99.73%Couleur et forme :SolidMasse moléculaire :259.22Denagliptin tosylate
CAS :Denagliptin (GW823093 or GSK-823093) is a dipeptidyl peptidase IV (DPP-IV) inhibitor.Formule :C27H26F3N3O4SCouleur et forme :SolidMasse moléculaire :545.57CA-074 methyl ester
CAS :CA-074 methyl ester (Cathepsin B Inhibitor IV) is a selective inhibitor of Cathepsin B (IC50=36.3 nM). neuroprotective effect. High-Quality, Low-Cost!Formule :C19H31N3O6Degré de pureté :97.26% - 99.58%Couleur et forme :SolidMasse moléculaire :397.47Efegatran HCl
CAS :Efegatran (GYKI-14166, RGH-2958, LY294468) is a thrombin inhibitor in development by IVAX for thromboembolic disorders.Formule :C21H34Cl2N6O3Couleur et forme :SolidMasse moléculaire :489.442Brensocatib
CAS :Brensocatib (AZD7986) is a Dipeptidyl peptidase 1 (DPP1) inhibitor (pIC50s: 6.85, 7.7, 7.6, 7.8, and 7.8 in human, rat, mouse, rabbit, and dog, respectively).Formule :C23H24N4O4Degré de pureté :97.55%Couleur et forme :SolidMasse moléculaire :420.46Letermovir
CAS :Letermovir (AIC246) (AIC246) is a novel anti-CMV compound (EC50: about 5 nM in fibroblast cells). It targets the pUL56 subunit of the viral terminase complex.Formule :C29H28F4N4O4Degré de pureté :99.85% - 99.87%Couleur et forme :SolidMasse moléculaire :572.55Ref: TM-T5396
1mg84,00€5mg167,00€10mg268,00€25mg470,00€50mg670,00€100mg954,00€200mg1.288,00€1mL*10mM (DMSO)205,00€TMC647055 Choline Hydroxide Salt
TMC647055 is a potent HCV NS5B inhibitor with low toxicity and good pharmacokinetics, under clinical evaluation.Formule :C37H53N5O8SDegré de pureté :99.44%Couleur et forme :SolidMasse moléculaire :727.91Ref: TM-T21537L
1mg95,00€5mg200,00€10mg289,00€25mg520,00€50mg742,00€100mg1.018,00€1mL*10mM (DMSO)286,00€Bemnifosbuvir
CAS :Bemnifosbuvir (AT-511) is a novel phosphoramidate prodrug of 2'-fluoro-2'-C-methylguanosine-5'-monophosphate that has potent in vitro activity against HCV.Formule :C24H33FN7O7PDegré de pureté :99.35% - 99.54%Couleur et forme :SolidMasse moléculaire :581.53ABT530
CAS :ABT530 (Pibrentasvir) is an HCV NS5A inhibitor with EC50s ranging from 1.4-5.0 pM against HCV replicons containing NS5A from genotypes 1-6.Formule :C57H65F5N10O8Degré de pureté :99.15% - 99.93%Couleur et forme :SolidMasse moléculaire :1113.18LY 3000328
CAS :LY 3000328 (Cathepsin S inhibitor) is a selective inhibitor of cathepsin S.Cost-effective and quality-assured.Formule :C25H29FN4O5Degré de pureté :97.83% - 99.54%Couleur et forme :SolidMasse moléculaire :484.52Ref: TM-TQ0116
1mg90,00€2mg130,00€5mg198,00€10mg263,00€25mg462,00€50mg672,00€100mg945,00€1mL*10mM (DMSO)207,00€Paritaprevir free base
CAS :Paritaprevir (ABT-450) is an oral HCV NS3/NS4A protease inhibitor with potential against genotype 1, disrupting viral replication.Formule :C40H43N7O7SDegré de pureté :95% - 99.26%Couleur et forme :SolidMasse moléculaire :765.89Diprotin A
CAS :Diprotin A (Ile-Pro-Ile) (Ile-Pro-Ile) is a dipeptidyl peptidase IV (DPP-IV) inhibitor.Formule :C17H31N3O4Degré de pureté :99.29%Couleur et forme :White PowderMasse moléculaire :341.45
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