GPCR/G-Protéine
Les inhibiteurs des GPCR/protéines G sont des composés qui ciblent les récepteurs couplés aux protéines G (GPCR) et les protéines G associées, qui jouent un rôle crucial dans la transmission des signaux de l'extérieur vers l'intérieur des cellules. Ces inhibiteurs sont essentiels pour étudier les voies de signalisation médiées par les GPCR, impliquées dans de nombreux processus physiologiques, y compris la perception sensorielle, la réponse immunitaire et la neurotransmission. Les inhibiteurs des GPCR sont également importants dans le développement de médicaments, car de nombreux agents thérapeutiques ciblent ces récepteurs. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de GPCR/protéines G de haute qualité pour soutenir vos recherches en pharmacologie, biologie cellulaire et domaines connexes.
Sous-catégories appartenant à la catégorie "GPCR/G-Protéine"
- récepteur 5-HT(1.025 produits)
- Récepteur d'adénosine(249 produits)
- Récepteur adrénergique(3.030 produits)
- Récepteur de la bombésine(35 produits)
- Récepteur de la bradykinine(61 produits)
- CXCR(159 produits)
- CaSR(34 produits)
- Récepteur cannabinoïde(217 produits)
- Cholécystokinine(1 produits)
- Récepteur de la dopamine(445 produits)
- Récepteur de l'endothéline(86 produits)
- Récepteur GNRH(84 produits)
- GPCR19(33 produits)
- GRK(33 produits)
- GTPase(22 produits)
- Récepteur du glucagon(196 produits)
- Hérisson/Smoothened(49 produits)
- Récepteur de l'histamine(385 produits)
- Récepteur LPA(21 produits)
- Récepteur de la mélatonine(26 produits)
- Récepteur OX(42 produits)
- Récepteur opioïde(325 produits)
- PAFR(14 produits)
- PKA(58 produits)
- Récepteur S1P(17 produits)
- SGLT(31 produits)
- Récepteur Sigma(46 produits)
Affichez 19 plus de sous-catégories
5982 produits trouvés pour "GPCR/G-Protéine"
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Galanin-Like Peptide (porcine)
CAS :Galanin-Like Peptide (porcine) is a 60 amino acid neuropeptide originally isolated from the porcine hypothalamus.Formule :C281H443N81O78Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :6204.02L-797,591
CAS :L-797,591 is a selective agonist of somatostatin receptor subtype 1.Formule :C38H49N5O2Couleur et forme :SolidMasse moléculaire :607.83O-Desethyl Dapagliflozin
CAS :O-Desethyl Dapagliflozin (Empagliflozin-4) is a SGLT2 inhibitor, IC50=33nM.Formule :C19H21ClO6Degré de pureté :98.33%Couleur et forme :SolidMasse moléculaire :380.82Ref: TM-T67849
1mg57,00€5mg120,00€10mg187,00€25mg321,00€50mg470,00€100mg683,00€1mL*10mM (DMSO)135,00€Prostaglandin D2 methyl ester
CAS :PGD2: made in mast cells during allergic reactions, causes vasodilation and inhibits blood clots. PGD2 methyl ester is a similar, fat-soluble prodrug.Formule :C21H34O5Couleur et forme :SolidMasse moléculaire :366.498Metipranolol
CAS :Metipranolol (Betamann) is a type of β- Adrenergic receptors（ β- A potent antagonist of adrenergic receptor on guinea pig atria β 1- Adrenergic receptors and rat uterus β The 2-adrenergic receptor exhibited the beta blocking potentials (pA2) of 8.3 and 8.4, respectively. It is also a potent substituent in the 3H DHA binding assay, with a ligand concentration of 0.7 nM and a Ki of 39 ± 24 nM.Formule :C17H27NO4Degré de pureté :98.37%Couleur et forme :SolidMasse moléculaire :309.4hNTS1R agonist-1
Compound 10, an hNTS1R agonist-1, acts as a full agonist with a strong affinity for hNTS1R (K i: 6.9 nM), showing the ability to cross the blood-brain barrier (Formule :C37H62N10O9Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :790.95Nizatidine
CAS :Nizatidine (Acinon) is a competitive and reversible histamine H2-receptor antagonist with antacid activity.Formule :C12H21N5O2S2Degré de pureté :99.43%Couleur et forme :White To Off-White Crystalline PowderMasse moléculaire :331.464-Thiouridine 5′-triphosphate disodium
CAS :4-Thiouridine 5′-triphosphate (4-Thio-UTP) tetrasodium functions as a potent agonist at P2Y 2 and P2Y 4 receptors, with half-maximal effective concentrations (Formule :C9H11N2Na2O14P3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :546.19Orexin B, rat, mouse
CAS :Orexin B, rat, mouse is an endogenous agonist at Orexin receptor with Kis of 420 and 36 nM for OX1 and OX2, respectively.Formule :C126H215N45O34SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :2936.45Dp[Tyr(methyl)2,Arg8]-Vasopressin
CAS :Dp[Tyr(Me)2,Arg8]-Vasopressin is a non-selective antagonist of the peptide arginine vasopressin V1b receptor [1].Formule :C49H70N14O12S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1111.3[Leu13]-Motilin
CAS :[Leu13]-Motilin (KW-5139) is an analogue of the gastrointestinal hormone motilin that induces concentration-dependent contractions in rabbit gastrointestinalFormule :C121H190N34O35Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :2681.01human GALP (3-32)
Human GALP (3-32) (Galanin-like peptide (3-32)) serves as a high-affinity agonist for galanin receptors GalR1 (IC50 = 33 nM) and GalR2 (IC50 = 15 nM), asFormule :C137H213N43O38SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :3102.49Imnopitant dihydrochloride
CAS :Imnopitant dihydrochloride is a neurokinin NK1 receptor antagonist [1] .Formule :C28H30Cl2F6N4OCouleur et forme :SolidMasse moléculaire :623.46SR-31747 free base
CAS :SR-31747: immunosuppressive anti-inflammatory agent, inhibits cell growth by blocking sterol isomerase.Formule :C23H34ClNCouleur et forme :SolidMasse moléculaire :359.98Fasitibant chloride hydrochloride
CAS :Fasitibant chloride( MEN16132) is an effective and selective non-peptide antagonist of kinin B2 receptor.Formule :C36H50Cl4N6O6SCouleur et forme :SolidMasse moléculaire :836.7Neuropeptide W-30 (human)
CAS :Neuropeptide W-30 (human) serves as a crucial stress mediator within the central nervous system, influencing the hypothalamus-pituitary-adrenal (HPA) axis and sympathetic outflow. It acts as an endogenous ligand for the two related orphan G-protein-coupled receptors (GPCRs), GPR7 and GPR8, binding and activating them at comparable effective doses [1] [2] [3].Formule :C165H249N49O37SCouleur et forme :SolidMasse moléculaire :3543.11CCR8 agonist 1
CCR8 agonist1 (Compound 2) is an activator of CCR8 and is applicable in studies related to autoimmune diseases.Formule :C22H29NO3Couleur et forme :SolidMasse moléculaire :355.47AR-C126313
CAS :AR-C126313 is a thiouracil derivative.
Formule :C28H23N7O3SCouleur et forme :SolidMasse moléculaire :537.59Adrenocorticotropic Hormone (ACTH) (4-10), human
CAS :Adrenocorticotropic Hormone (ACTH) (4-10) is an agonist of potent melanocortin(MC4R) receptor .Formule :C44H59N13O10SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :962.09Colulintide
CAS :Colulintide is an analog of amylin, utilized in obesity research.Couleur et forme :SolidDanshenol B
Danshenol B is a natural product that can be used as a reference standard.Formule :C22H26O4Couleur et forme :SolidMasse moléculaire :354.446Stressin I TFA
Stressin I (Cyclo(31-34)[DPhe12, Nle21, 38, Glu31, Lys34]Ac-hCRF(4-41)) TFA, with a K i of 1.7 nM, is a potent and selective agonist of the CRF1 receptor.Degré de pureté :98%Couleur et forme :Odour SolidN-Desmethyl Pimavanserin
CAS :N-Desmethyl Pimavanserin (AC-279) is the active metabolite of Pimavanserin and is used in the treatment of insomnia and other sleep disorders.Formule :C24H32FN3O2Degré de pureté :98.02%Couleur et forme :SolidMasse moléculaire :413.53MRS2500 tetraammonium
CAS :Highly potent and selective antagonist of the platelet P2Y1 receptorFormule :C13H21IN6O8P2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :578.19BAM(8-22) TFA
BAM(8-22) TFA activates Mrgprs, induces mouse scratching, and is a proenkephalin A derivative.Formule :C93H128F3N25O25SCouleur et forme :SolidMasse moléculaire :2085.22Apadenoson TFA
Apadenoson TFA is a potent adenosine A2A receptor (A2AR) agonist that can be used to improve survival in patients infected with SARS.
Formule :C25H31F3N6O8Degré de pureté :98.08%Couleur et forme :SoildMasse moléculaire :600.55L 152804
CAS :L 152804: Y5 receptor antagonist, reduces food intake/boosts energy, leads to weight loss in obese mice.Formule :C23H26O4Degré de pureté :99.82%Couleur et forme :SolidMasse moléculaire :366.45Ref: TM-T15679
5mg50,00€10mg80,00€25mg117,00€50mg178,00€100mg259,00€200mg369,00€1mL*10mM (DMSO)51,00€Secretin (33-59), rat TFA
Secretin (33-59), rat (TFA), a 27-aa peptide, stimulates the secretin receptor, increasing pancreas secretion of bicarbonate, enzymes, and K+.Formule :C131H217F3N42O44Couleur et forme :SolidMasse moléculaire :3141.37TCMCB07 TFA
TCMCB07 TFA is a cyclic nonapeptide and an orally active, brain-penetrating antagonist of the melanocortin receptor 4 (MC4R), playing a significant role inFormule :C63H87N15O11·xC2HF3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1230.46 (free base)Guanylin(human)
CAS :Peptide that activates gut guanylyl cyclase, secreted by GI mucosa, regulates water and electrolytes in gut and kidneys.Formule :C58H87N15O21S4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1458.65G-Protein antagonist peptide acetate
G-Protein antagonist peptide acetate is a truncated substance P-related peptide, competes with receptor for G protein binding.Formule :C59H68N12O11SDegré de pureté :98.06%Couleur et forme :SolidMasse moléculaire :1153.33BMS-753426
CAS :BMS-753426 is a potent and orally bioavailable antagonist of CCR2 .
Formule :C25H33F3N6O2Couleur et forme :SolidMasse moléculaire :506.5748-iso-15-keto Prostaglandin F2α
CAS :8-iso-15-keto Prostaglandin F2α (8-iso-15-keto PGF2α) is a metabolite of the isoprostane 8-iso PGF2α in rabbits, monkeys, and humans.Formule :C20H32O5Couleur et forme :SolidMasse moléculaire :352.471BQ-3020 ammonium
BQ-3020 ammonium, a selective endothelin receptor (ET B receptor) agonist, demonstrates inhibition of [125 I] ET-1 binding to ET B receptors with an IC50 of 0.2Formule :C96H140N20O25S·xNH3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :2006.32 (free base)NF546 hydrate
NF546 (hydrate), a selective non-nucleotide P2Y11 agonist, exhibits a pEC50 value of 6.27 and induces interleukin-8 secretion from human monocyte-derivedFormule :C47H44N6Na4O17P4·5H2ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :1424.0115-keto Latanoprost
CAS :Latanoprost, a PG analog for ocular pressure, metabolizes into 15-keto latanoprost, a less potent variant reducing intraocular pressure and pupil size.Formule :C26H38O5Couleur et forme :SolidMasse moléculaire :430.58FXR/TGR5 agonist 1
CAS :FXR/TGR5 agonist 1 acts as an agonist on both FXR and TGR5 receptors and is utilized for treating fatty liver disease.Formule :C31H32ClN3O3Couleur et forme :SolidMasse moléculaire :530.07A3AR agonist 1
A3AR Agonist 1 (Compound 12), with a Ki of 25.8 nM, is a potent A3 adenosine receptor (A3AR) agonist that promotes β-arrestin2 recruitment with an effectiveFormule :C28H34N6O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :550.61CCR8 antagonist 1
CAS :CCR8 antagonist 1 is an antagonist of C-C Motif Chemokine Receptor 8 (CCR8) with a Ki value of 1.6 nM.Formule :C26H29N3O5SDegré de pureté :99.51%Couleur et forme :SolidMasse moléculaire :495.59PG 106 acetate
PG 106 acetate: Selective hMC3 receptor antagonist, IC50=210 nM; inactive on hMC5 and hMC4, EC50=9900 nM.Formule :C53H73N13O11Degré de pureté :98.24%Couleur et forme :SolidMasse moléculaire :1068.23Drinabant
CAS :Drinabant (AVE-1625) is an orally active CB1 receptor antagonist.Formule :C23H20Cl2F2N2O2SDegré de pureté :99.8%Couleur et forme :SolidMasse moléculaire :497.38Muscarinic toxin 3
CAS :Muscarinic toxin 3 (MT3), a potent non-competitive antagonist of mAChR and adrenoceptors, exhibits pIC50 values of 6.71 for M1, 8.79 for M4, 8.86 for α1A, 7.57Formule :C319H489N89O97S8Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :7379.35(Iso)-WAY-260022
CAS :(Iso)-WAY-260022 ((Iso)-NRI-022) is a stereoisomer of WAY-260022, a norepinephrine reuptake inhibitor and selective inhibitor of 5-hydroxytryptamine and dopamine transport proteins.Formule :C21H31F3N2O2Degré de pureté :97.68% - 99.36%Couleur et forme :SoildMasse moléculaire :400.48Adenosine receptor antagonist 1
CAS :A2aR-selective antagonist with IC50 of 0.29 nM; 14x more selective over A2bR.Formule :C22H15ClFN7OCouleur et forme :SolidMasse moléculaire :447.86CCR2 antagonist 1
CAS :CCR2 antagonist 1 is a high-affinity and long-residence-time antagonist of CCR2 (Ki: 2.4 nM).Formule :C28H32BrF3N2OCouleur et forme :SolidMasse moléculaire :549.47B7-33
CAS :B7-33 is a single-chain relaxin analog and a selective agonist for relaxin receptor 1 (RXFP1). It binds to RXFP1 and preferentially activates the pERK pathway in cells expressing RXFP1, rather than cAMP. B7-33 serves as an antifibrotic agent and provides cardioprotective effects.Formule :C131H229N41O36SCouleur et forme :SolidMasse moléculaire :2986.54Prazobind
CAS :Prazobind is a prazosinoid substance that blocks insulin stimulation of IP1 (inositol phosphate) accumulation and is an effective α1 adrenoceptor blocker.Formule :C23H27N5O3Couleur et forme :SolidMasse moléculaire :421.501Donetidine
CAS :Donetidine is a histamine H2 receptor antagonist used to treat digestive disorders.Formule :C20H25N5O3SDegré de pureté :99.32%Couleur et forme :SolidMasse moléculaire :415.51GPR55 agonist 4
GPR55 agonist 4 (Compound 28), with an EC50 of 131 nM for hGPR55 and 1.41 nM for rGPR55, effectively induces β-arrestin recruitment to human GPR55 [1].Formule :C19H16FN5O2Couleur et forme :SolidMasse moléculaire :365.36Oxatomide
CAS :Oxatomide: Dual H1/P2X7 antagonist, antihistamine, anti-allergic, treats immune diseases, IC50: 0.95 μM (P2X7), 0.43 μM (5-HT).Formule :C27H30N4ODegré de pureté :99.28% - 99.72%Couleur et forme :White PowderMasse moléculaire :426.55Ref: TM-T19839
1mg35,00€5mg75,00€10mg114,00€25mg222,00€50mg356,00€100mg557,00€500mg1.153,00€1mL*10mM (DMSO)84,00€AB21 oxalate
AB21 oxalate, a potent and selective S1R antagonist, exhibits binding affinities (Kis) of 13 nM and 102 nM for S1R and S2R, respectively.
Formule :C25H30N2O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :438.52Guanylin (mouse, rat)
CAS :Guanylin (mouse, rat), a peptide consisting of 15 amino acids, acts as an activator of intestinal guanylate cyclase and is utilized in diarrhea research [1].
Formule :C60H90N16O22S4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1515.71Xenin-8 TFA
Xenin-8 TFA, a C-terminal octapeptide derived from the 25-amino acid peptide Xenin belonging to the neurotensin/xenopsin family, is biologically active.Substance P(1-7) TFA
CAS :Substance P(1-7) TFA is a fragment of neuropeptide P (SP), with anti-harmful effects, used in neurological disease research.Formule :C43H66F3N13O12Degré de pureté :98.23%Couleur et forme :SolidMasse moléculaire :1014.063-Deoxyglucosone
CAS :3-Deoxyglucosone(3-Deoxy-D-glucosone) is synthesized by the intermediate pathway of the melad and polyol reactions.3-Deoxyglucosone reacts rapidly with proteinFormule :C6H10O5Degré de pureté :95%Couleur et forme :SolidMasse moléculaire :162.14Fezolamine
CAS :Fezolamine: a new, non-tricyclic, oral antidepressant, selectively inhibits norepinephrine uptake over serotonin or dopamine.Formule :C20H23N3Degré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :305.42GLP-1(7-37)
CAS :GLP-1 (7-37) is a truncated, bioactive form of GLP-1 that is the product of proglucagon processing in intestinal endocrine L cells.Formule :C151H228N40O47Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :3355.67Acetyl-Amylin (8-37) (human)
CAS :Acetyl-Amylin (8-37) (human) is a specific amylin antagonist [1] .Formule :C140H218N42O46Couleur et forme :SolidMasse moléculaire :3225.48Emoghrelin
CAS :Emoghrelin, extracted from Heshouwu (Polygonum multiflorum), promotes the secretion of growth hormone by activating the ghrelin receptor [1].Formule :C24H22O13Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :518.42L-796,778 acetate
L-796,778 acetate is a slective somatostatin receptor agonist with IC50 of 24nM for sst3, for sst1, sst2, sst4 and sst5, IC50 is >1000nM.Formule :C31H44N6O9Degré de pureté :98%Couleur et forme :SoildMasse moléculaire :644.72Moxonidine hydrochloride
CAS :Moxonidine Hydrochloride: selective I1 imidazoline receptor agonist, stronger than α2-AR; lowers blood pressure; central action.Formule :C9H13Cl2N5OCouleur et forme :SolidMasse moléculaire :278.14Arotinolol hydrochloride
CAS :Arotinolol HCl is a non-selective α/β-blocker, anti-hypertensive, anti-obesity, and improves aortic stiffness.
Formule :C15H22ClN3O2S3Degré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :408Velmupressin
CAS :Peptidic V2R agonist, c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-d-Arg-NEt2, with EC50: 0.07 nM (hV2R), 0.02 nM (rV2R); selective, short-acting.Formule :C42H60ClN11O8S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :946.58TAK-683 acetate
TAK-683 acetate: potent KISS1R agonist (IC50=170 pM), stable, nonapeptide. Affects GnRH, FSH, LH, testosterone; potential in prostate cancer research.Formule :C66H87N17O15Couleur et forme :SolidMasse moléculaire :1358.5Carbocyclic Thromboxane A2
CAS :Carbocyclic Thromboxane A2 can be used in related research in the field of life sciences. Its product number is T36548 and CAS number is 74034-56-3.Formule :C22H36O3Couleur et forme :SolidMasse moléculaire :348.527FFN246
CAS :FFN246, a fluorescent probe, concurrently targets the serotonin transporter (SERT) and vesicular monoamine transporter 2 (VMAT2), exhibiting excitation andFormule :C15H13FN2ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :256.27α-CGRP (mouse, rat) TFA
α-CGRP (mouse, rat) TFA, a neuropeptide belonging to the calcitonin gene-related peptide (CGRP) family, is predominantly located at neuromuscular junctions andFormule :C162H262N50O52S2·C2HF3O2Degré de pureté :98%Couleur et forme :Solidβ-Corticotropin (swine)
CAS :β-Corticotropin (swine), a synthetic analog of the peptide hormone corticotropin (ACTH), induces steroid release [1] [2].Couleur et forme :SolidObestatin(rat)
CAS :Endogenous peptide that suppresses food intake and body weight-gainFormule :C114H174N34O31Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :2516.81GLP-1R agonist 26
CAS :Compound 1, also known as GLP-1R agonist 26, is an agonist of the glucagon-like peptide-1 receptor (GLP-1R) with an EC50 of <10 nM.Formule :C32H29FN6O4SCouleur et forme :SolidMasse moléculaire :612.67Adrenocorticotropic Hormone (ACTH) (1-10), human
CAS :ACTH (1-10), human: a weak α-MSH mimic at high doses (100-1000 nM), derived from adrenocorticotropin.Formule :C59H78N16O16SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :1299.41Atriopeptin III (rat)
CAS :Atriopeptin III (rat) (ANP 127-150), a 24-amino acid atrial peptide, functions as a powerful vasodilator and natriuretic/diuretic agent, enhancing renalFormule :C107H165N35O34S2Masse moléculaire :2549.8S1R agonist 2
CAS :S1R agonist 2 is a selective S1R agonist with a Ki of 88 nM for S2R and 1.1 nM for S1R and is protective against ROS and NMDA-induced neurotoxicity.Formule :C21H27NODegré de pureté :99.66%Couleur et forme :SolidMasse moléculaire :309.45Pafenolol
CAS :Pafenolol is a P-glycoprotein modulator with a Ki value of 5.5 µM. pafenolol is an orally available and selective beta-adrenergic receptor antagonist.Formule :C18H31N3O3Degré de pureté :98.33%Couleur et forme :SolidMasse moléculaire :337.46Liraglutide acetate
CAS :Liraglutide acetate is the acetate salt form of Liraglutide, which is a glucagon-like peptide-1 (GLP-1) receptor agonist, utilized in the study of type 2 diabetes.Formule :C172H265N43O51·xC2H4O2Couleur et forme :SolidMasse moléculaire :3751.20 (free base)Neurokinin A TFA
CAS :Neurokinin A TFA (NKA TFA) is a neuropeptide within the neurokinin family, serving as the endogenous ligand and agonist for the NK-2 (Neurokinin 2) receptor.Formule :C52H81F3N14O16SDegré de pureté :98.704%Couleur et forme :SolidMasse moléculaire :1247.34ACTH (1-14) (TFA)
ACTH (1-14) (TFA) is a regulatory fragment of adrenocorticotropin, specifically involved in the control of cortisol and androgen synthesis [1].Formule :C79H110F3N21O22SMasse moléculaire :1794.9Gastrin I (1-14), human TFA
Gastrin I (1-14), human TFA is 1-14 fragment of human gastrin I peptide.Formule :C81H101N16F3O29Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1819.75PACAP (1-38) free acid
CAS :PACAP (1-38) free acid, an endogenous neuropeptide, potently modulates gastrointestinal and neuroendocrine functions.Couleur et forme :SolidBosentan-d4
CAS :Bosentan-d4: deuterium version of Bosentan, competitive ET A/B antagonist, Ki: 4.7nM (ET A), 95nM (ET B) in human SMC.Formule :C27H25D4N5O6SCouleur et forme :SolidMasse moléculaire :555.64[D-Arg25]-Neuropeptide Y (human)
[D-Arg25] NPY: human Y1 receptor agonist; linked to AD; shields rat neurons from β-Amyloid.Formule :C189H285N55O57SMasse moléculaire :4271.68Kadsurenin C
CAS :Kadsurenin C (compound 1), a neolignan isolated from the aerial parts of Piper kadsura, exhibits anti-inflammatory properties and significant PAF (Platelet Activating Factor) antagonistic activity, with an IC50 value of 5.1 μM [1].Formule :C21H26O5Masse moléculaire :358.43PSB-1114 triethylamine
PSB-1114 triethylamine is a potent, enzymatically stable, P2Y2 receptor agonist with a 134 nM EC50, exhibiting greater than 50-fold selectivity over P2Y4 (EC50Formule :C10H15F2N3O13P3S·xC6H15NDegré de pureté :98%Couleur et forme :Solid[D-Phe2,6, Pro3]-LH-RH
CAS :[D-Phe2,6, Pro3]-LH-RH is a potent antagonist of luteinizing hormone-releasing hormone (LHRH).Formule :C59H80N14O13Couleur et forme :SolidMasse moléculaire :1193.35(Leu31,Pro34)-Peptide YY (human)
CAS :(Leu31,Pro34)-Peptide YY (human) is a derivative of Peptide YY, acting as a potent and selective Y1 receptor agonist with a dissociation constant (KD) of 1.0 nMFormule :C195H296N54O56Couleur et forme :SolidMasse moléculaire :4292.75Cannabidivarinic acid
CAS :Cannabidivarinic acid (CBDVA), the carboxylic acid precursor to cannabidivarin (CBDV), is a non-psychoactive cannabinoid found in Cannabis and known for its anti-inflammatory properties.Formule :C20H26O4Couleur et forme :SolidMasse moléculaire :330.42CCK (27-33) (non-sulfated)
CAS :CCK (27-33), a non-sulfated peptide, inhibits [3H]naloxone binding (IC50=4uM) and guinea pig ileum contractions (IC50=17uM), reversed by naloxone.Formule :C45H57N9O10S2Couleur et forme :SolidMasse moléculaire :948.12Biotinyl-neuropeptide W-23 (human)
CAS :Biotinyl-neuropeptide W-23 (human) is a biotinylated form of neuropeptide W-23 (human), which functions as an agonist for the NPBW1 (GPR7) and NPBW2 (GPR8)Formule :C129H197N37O30S2Couleur et forme :SolidMasse moléculaire :2810.3Esmolol acid hydrochloride
CAS :Esmolol acid (ASL-8123) hydrochloride is a mild antagonist of β-adrenergic receptors. It inhibits the heart rate and diastolic pressure responses induced by Isoproterenol in a dose-dependent manner and is applicable for renal failure research.Formule :C15H24ClNO4Couleur et forme :SolidMasse moléculaire :317.81CACPD2011a-0001278239
CAS :CACPD2011a-0001278239 is a β2AR hybrid agonist with high affinity binding to both the wild-type and T164I β2AR variants. It exhibits neither cytotoxicity nor mutagenicity, making it suitable for asthma research.Formule :C21H22N4O4Couleur et forme :SolidMasse moléculaire :394.4216,16-dimethyl Prostaglandin E1
CAS :16,16-dimethyl Prostaglandin E1 is a PGE1 (T1626) analog that induces bronchoconstriction and vascular smooth muscle contraction and inhibits indomethacin-Formule :C22H38O5Couleur et forme :SolidMasse moléculaire :382.541PAMP-12(human, porcine) TFA
PAMP-12(human, porcine) TFA, a significant constituent of immunoreactive (ir)-PAMP, derives from the adrenomedullin precursor and functions as a potentCouleur et forme :Odour SolidNeuropeptide W-23 (human) (TFA)
Neuropeptide W-23 (human) (NPW-23) TFA, representing the active form of Neuropeptide W, functions as an endogenous agonist for both NPBW1 (GPR7) and NPBW2 (GPR8Couleur et forme :Odour SolidTecastemizole
CAS :Tecastemizole (R 43512) is a selective antagonist of H1 receptor and a major metabolite of astemizole with anti-inflammatory effects.Formule :C19H21FN4Degré de pureté :99.70%Couleur et forme :SolidMasse moléculaire :324.4Ref: TM-T26253
1mg57,00€5mg125,00€10mg177,00€25mg304,00€50mg437,00€100mg615,00€500mg1.225,00€1mL*10mM (DMSO)138,00€Plecanatide acetate
CAS :Plecanatide acetate: GC-C receptor agonist, EC50=190 nM (T84 cells), anti-inflammatory in murine colitis.Formule :C67H108N18O28S4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1741.94Acetyl-(D-Arg2)-GRF (1-29) amide (human)
CAS :Acetyl-(D-Arg2)-GRF (1-29) amide (human) serves as an antagonist to growth hormone-releasing factor (GRF) and inhibits growth hormone (GH) secretion, withFormule :C154H255N47O43SMasse moléculaire :3485.03Oxopurpureine
CAS :Oxopurpureine, classified as an oxoaporphine compound, functions to inhibit plant pathogens.Formule :C21H19NO6Couleur et forme :SolidMasse moléculaire :381.38Sulfatroxazole
CAS :Sulfatroxazole (Isosulfafurazole) (compound 12) is a selective antagonist of the ETA receptor with an IC50 of 0.26 μM.Formule :C11H13N3O3SCouleur et forme :SolidMasse moléculaire :267.3[D-p-Cl-Phe6,Leu17]-VIP
CAS :Selective vasoactive intestinal peptide (VIP) receptor antagonist (IC50 = 125.8 nM). Displays no activity on glucagon, secretin or GRF receptors.Formule :C148H239ClN44O42Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :3342.24Phendioxan
CAS :Phendioxan is a biochemcial.Formule :C25H27NO5Couleur et forme :SolidMasse moléculaire :421.49
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