GPCR/G-Protéine
Les inhibiteurs des GPCR/protéines G sont des composés qui ciblent les récepteurs couplés aux protéines G (GPCR) et les protéines G associées, qui jouent un rôle crucial dans la transmission des signaux de l'extérieur vers l'intérieur des cellules. Ces inhibiteurs sont essentiels pour étudier les voies de signalisation médiées par les GPCR, impliquées dans de nombreux processus physiologiques, y compris la perception sensorielle, la réponse immunitaire et la neurotransmission. Les inhibiteurs des GPCR sont également importants dans le développement de médicaments, car de nombreux agents thérapeutiques ciblent ces récepteurs. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de GPCR/protéines G de haute qualité pour soutenir vos recherches en pharmacologie, biologie cellulaire et domaines connexes.
Sous-catégories appartenant à la catégorie "GPCR/G-Protéine"
- récepteur 5-HT(1.025 produits)
- Récepteur d'adénosine(251 produits)
- Récepteur adrénergique(3.025 produits)
- Récepteur de la bombésine(35 produits)
- Récepteur de la bradykinine(61 produits)
- CXCR(158 produits)
- CaSR(34 produits)
- Récepteur cannabinoïde(218 produits)
- Cholécystokinine(1 produits)
- Récepteur de la dopamine(445 produits)
- Récepteur de l'endothéline(86 produits)
- Récepteur GNRH(84 produits)
- GPCR19(36 produits)
- GRK(33 produits)
- GTPase(23 produits)
- Récepteur du glucagon(195 produits)
- Hérisson/Smoothened(49 produits)
- Récepteur de l'histamine(385 produits)
- Récepteur LPA(21 produits)
- Récepteur de la mélatonine(26 produits)
- Récepteur OX(41 produits)
- Récepteur opioïde(327 produits)
- PAFR(14 produits)
- PKA(60 produits)
- Récepteur S1P(18 produits)
- SGLT(31 produits)
- Récepteur Sigma(46 produits)
Affichez 19 plus de sous-catégories
6011 produits trouvés pour "GPCR/G-Protéine"
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Clencyclohexerol-d10
CAS :Argipressin inhibits central corticotropin-releasing hormone. Argipressin acts as an inhibitory factor in the regulation of central CRH levels.Formule :C14H20Cl2N2O2Couleur et forme :SolidMasse moléculaire :329.29SAR247799
CAS :SAR247799 is a selective and G-protein-biased S1P1 agonist that activates downstream G-protein signaling pathways more preferentially on endothelial cells.Formule :C21H16ClN3O5Couleur et forme :SolidMasse moléculaire :425.82Asenapine
CAS :Asenapine (Org 5222) is a 5-HT receptor, adrenergic receptor, and histamine receptor antagonist with antipsychotic properties for the treatment of schizophreniaFormule :C17H16ClNODegré de pureté :99.64%Couleur et forme :CoaMasse moléculaire :285.77RU-SKI 43 Hydrochloride
CAS :RU-SKI 43 Hydrochloride is a selective Hedgehog acyltransferase inhibitor (IC50 850 nM) with reported anticancer activity in tumor biology studies.Formule :C22H31ClN2O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :423.01SLIGRL-NH2
CAS :SLIGRL-NH2 (Protease-Activated Receptor-2 Activating Peptide) is a PAR-2 agonist that induces non-histaminergic pruritus.Formule :C29H56N10O7Degré de pureté :98.29%Couleur et forme :SolidMasse moléculaire :656.821-Phenylbiguanide HCl
CAS :Compound PDK0269, as 5-HT3 receptor agonists(3–100 μM, pEC50 5.05±0.06), acutely increased XII (hypoglossal) burst frequency and regularity, and decreased bursts/episode . Phenylbiguanide produced a dose-related (10-500 microM) increase in the release of dopamine (280-2000%). When nomifensine (5 microM) was included in the Ringer solution, the effect of Compound PDK0269 on the release of dopamine was ameliorated or inhibited.Formule :C8H12ClN5Degré de pureté :99.31%Couleur et forme :SolidMasse moléculaire :213.67Sumatriptan
CAS :Sumatriptan (GR 43175 free base) is a 5-HT1 receptor agonist with anti-inflammatory activity used in acute migraine and acute myocardial infarction.Formule :C14H21N3O2SDegré de pureté :99.93%Couleur et forme :White To Off-White Crystalline PowderMasse moléculaire :295.4Aramisulpride
CAS :Aramisulpride is a dual antagonist of the dopamine D2 receptor and serotonin receptor, primarily utilized for investigating metabolic disorders.Formule :C17H27N3O4SCouleur et forme :SolidMasse moléculaire :369.48SANT 2
CAS :SANT 2 is a Hedgehog (Hh) signaling pathway antagonist with potential anti-inflammatory and anti-cancer activities.Formule :C26H26ClN3O4Degré de pureté :99.23%Couleur et forme :SolidMasse moléculaire :479.96Argipressin
CAS :Argipressin is a vasoconstrictive and antidiuretic hormone, binding to V1 receptors with Kd ~1.4 nM in rat heart and aortic cells.Formule :C46H65N15O12S2Degré de pureté :98%Couleur et forme :White PowderMasse moléculaire :1084.23MrgprX2 antagonist-1
CAS :MrgprX2 antagonist-1 (compound E23) is a MrgprX2 antagonist applicable to cutaneous inflammation.Formule :C15H15F5N4O2SDegré de pureté :99.80%Couleur et forme :SolidMasse moléculaire :410.36Acrivastine D7
CAS :Acrivastine D7 is a deuterium labeled Acrivastine. Acrivastine is a short acting antagonist of histamine 1 receptor.Formule :C22H24N2O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :355.48Quetiapine-d8 Hemifumarate
CAS :Quetiapine-d8 Hemifumarate is a deuterated compound of Quetiapine Hemifumarate. Quetiapine Hemifumarate has a CAS number of 111974-72-2. Quetiapine Fumarate, an atypical antipsychotic, is used in the treatment of bipolar I mania, schizophrenia, bipolar II depression, bipolar I depression.Formule :C25H21D8N3O6SCouleur et forme :SolidMasse moléculaire :507.63Lanreotide
CAS :Lanreotide, a somatostatin analogue, suppresses GH/IGF-I hypersecretion in acromegaly patients. It also used to manage neuroendocrine tumours.Formule :C54H69N11O10S2Couleur et forme :SolidMasse moléculaire :1096.32GPR34 receptor antagonist 3
Compound 5e, a GPR34 receptor antagonist, exhibits selective inhibition of lysophosphatidylserine-induced ERK1/2 phosphorylation in a dose-dependent manner,Couleur et forme :Odour SolidLysosphingomyelin (d18:1)
CAS :Sphingomyelins are phosphorylcholine, sphingosine, and fatty acid. Lysosphingomyelin, missing the fatty acid, activates diverse cellular pathways.Formule :C23H49N2O5PCouleur et forme :SolidMasse moléculaire :464.628SYL-4
CAS :SYL-4 is a potential P2Y12 receptor antagonist with a Ki value of 7.35 ± 1.72 for use in synthetic dyes.Formule :C20H15N3O5SDegré de pureté :95.76%Couleur et forme :SoildMasse moléculaire :409.42ML 00253764
CAS :melanocortin MC4 receptor antagonistFormule :C18H18BrFN2OCouleur et forme :SolidMasse moléculaire :377.25Calcitonin (salmon)
CAS :Calcitonin (salmon), a calcium regulating hormone, is used to treat osteoporosis in women who are at least 5 years past menopause.Formule :C145H240N44O48S2Degré de pureté :99.41% - 99.80%Couleur et forme :PowderMasse moléculaire :3431.85MRS-3777 hemioxalate
CAS :MRS-3777 hemioxalate, a selective adenosine A3 receptor antagonist, reverses the anti-injury perception effects of its corresponding agonist and serves as a valuable tool for studying inflammatory pain.
Formule :C17H19N5OC2H2O4Degré de pureté :97.10%Couleur et forme :SolidMasse moléculaire :354.39Gizzerosine
CAS :Gizzerosine, a biogenic amine formed during feed processing, is a toxicant that induces mortality in livestock.Formule :C11H20N4O2Couleur et forme :SolidMasse moléculaire :240.3Neurotensin(8-13)
CAS :Neurotensin(8-13) is Neurotensin (NT) fragment, Neurotensin(8-13) results in a decrease in cell-surface NT1 receptors (NTR1) density.Formule :C38H64N12O8Degré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :816.99Ramelteon-d5
CAS :Ramelteon-d5 is a deuterated compound of Ramelteon.Formule :C16H16D5NO2Couleur et forme :SolidMasse moléculaire :264.37Tiapride-d3
Tiapride-d3 is a deuterated form of Tiapride, a selective dopamine D2 receptor antagonist and an antipsychotic compound.Formule :C15H21D3N2O4SCouleur et forme :SolidMasse moléculaire :331.45Quetiapine-d8 Fumarate
CAS :Quetiapine-d8 Fumarate is a deuterated compound of Quetiapine Fumarate. Quetiapine Fumarate has a CAS number of 111974-72-2. Quetiapine Fumarate, an atypical antipsychotic, is used in the treatment of bipolar I mania, schizophrenia, bipolar II depression, bipolar I depression.Formule :C25H21D8N3O6SCouleur et forme :SolidMasse moléculaire :507.63Revdofilimab
CAS :Revdofilimab (ABBV-368) is a human IgG1 monoclonal antibody targeting OX40, a receptor on certain T cells.Degré de pureté :98.80% - 98.80%Couleur et forme :LiquidMasse moléculaire :145.60 kDaTaranabant racemate
CAS :Taranabant racemate is an antagonist and/or inverse agonist of the Cannabinoid-1 (CB1) receptor.Formule :C27H25ClF3N3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :515.95Travoprost (Standard)
CAS :Travoprost (Standard) is the standard substance of Travoprost, and it is applicable for quantitative analysis, quality control, and related research in biochemical experiments. Travoprost (Fluprostenol isopropyl ester) is used to treat glaucoma and ocular hypertension,is a potent and selective FP prostaglandin receptor agonist.Formule :C26H35F3O6Couleur et forme :Colorless OilMasse moléculaire :500.55Granisetron
CAS :Granisetron, a serotonin receptor (5HT-3 selective) antagonist, is used as an antinauseant and antiemetic for cancer chemotherapy.
Formule :C18H24N4OCouleur et forme :SolidMasse moléculaire :312.415-HT2B antagonist-1
CAS :Orally active 5-HT2B antagonist; IC50 = 33.4 nM; potential for hepatocellular, cardiovascular, GI disease research.Formule :C11H14BrN5Degré de pureté :99.965%Couleur et forme :SolidMasse moléculaire :296.17BW 723C86
CAS :BW 723C86 is a 5-HT2B receptor agonist with anxiolytic effects, inducing overeating and reduced grooming in rats, useful in studying neurological disorders.Formule :C16H19ClN2OSDegré de pureté :99.35%Couleur et forme :SolidMasse moléculaire :322.85Bromperidol hydrochloride
CAS :Bromperidol hydrochloride is a D2 dopamine receptor antipsychotic; enhances Spectinomycin's mycobactericidal effects.Formule :C21H24BrClFNO2Couleur et forme :SolidMasse moléculaire :456.78Zilpaterol-d7
CAS :Zilpaterol-d7 (trans-(±)-Zilpaterol-d7) is a deuterium-labeled version of Zilpaterol, a β-adrenergic receptor agonist.Formule :C14H12D7N3O2Couleur et forme :SolidMasse moléculaire :268.361-Methyl-4-imidazoleacetic Acid (hydrochloride)
CAS :MIMA, a stable histamine byproduct from N-methylhistamine oxidation, indicates systemic mastocytosis via urinary levels.Formule :C6H9ClN2O2Couleur et forme :SolidMasse moléculaire :176.601SB-200646A
CAS :SB-200646A: oral 5-HT2B/2C antagonist; higher affinity than 5-HT2A (pKi: 7.5, 6.9 vs 5.2); anxiolytic with in vivo effects.Formule :C15H15ClN4ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :302.76Zaloglanstat
CAS :Zaloglanstat (ISC-27864) is a selective, orally active mPGES-1 inhibitor with an IC50 of 5 nM, analgesic in osteoarthritis and inflammatory arthritis.Formule :C21H20ClF3N4O2Degré de pureté :99.97%Couleur et forme :SolidMasse moléculaire :452.86Ref: TM-T39000
1mg154,00€5mg371,00€1mL*10mM (DMSO)409,00€10mg620,00€25mg1.305,00€50mg1.765,00€100mg2.367,00€Eplivanserin (mixture)
CAS :Eplivanserin mixture is a selective serotonin reuptake inhibitor and a 5-HT2A receptor antagonist,Formule :C19H21FN2O2Couleur et forme :SolidMasse moléculaire :328.387Clothiapine
CAS :Clothiapine is an atypical antipsychotic of the dibenzothiazepine chemical class.Formule :C18H18ClN3SDegré de pureté :99.93%Couleur et forme :SolidMasse moléculaire :343.87Allura Red AC (Standard)
CAS :Allura Red AC (Standard) is the standard substance of Allura Red AC, and it is applicable for quantitative analysis, quality control, and related research in biochemical experiments. Allura Red AC (CI 16035) is a very important food azo dye used in the food, pharmaceutical, paper, cosmetic and textile industries.Allura Red AC promotes susceptibility to experimental colitis via mouse intestinal serotonin.Formule :C18H14N2Na2O8S2Couleur et forme :Dark Maroon Solid PowderMasse moléculaire :496.42Fedovapagon
CAS :Fedovapagon (VA106483) is a pressin V2 receptor (V2R) agonist for the study of overactive bladder syndrome.Formule :C27H34N4O3Degré de pureté :99.46%Couleur et forme :SolidMasse moléculaire :462.58Cimbuterol-d9
CAS :Cimbuterol-d9 is a deuterated compound of Cimbuterol.Formule :C13H10D9N3ODegré de pureté :99.22%Couleur et forme :SolidMasse moléculaire :242.37Furprofen
CAS :Furprofen, an NSAID, inhibits PGE synthesis, offers analgesic effects, and is orally taken for pain relief.Formule :C14H12O4Degré de pureté :98.62% - 99.25%Couleur et forme :SolidMasse moléculaire :244.24L-798106
CAS :L-798106 (CM9) is an EP3 receptor antagonist that inhibits EP4, EP1, and EP2 receptors and attenuates PGE2-induced cough.Formule :C27H22BrNO4SDegré de pureté :98.97%Couleur et forme :SolidMasse moléculaire :536.44Hydroxyzine D8
CAS :Hydroxyzine D8, a deuterium-labeled version of Hydroxyzine, acts as a histamine H1-receptor antagonist.Formule :C21H27ClN2O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :382.95Spiroxatrine
CAS :Spiroxatrine (R 5188) is a 5-HT1α and α2-adrenergic dual antagonist with sedative activity for the study of diseases related to the cardiovascular system.Formule :C22H25N3O3Degré de pureté :99.94%Couleur et forme :SolidMasse moléculaire :379.45Cimetidine (Standard)
CAS :Cimetidine (Standard) is the standard substance of Cimetidine, and it is applicable for quantitative analysis, quality control, and related research in biochemical experiments. Cimetidine (SKF-92334) is a histamine congener, it competitively inhibits HISTAMINE binding to HISTAMINE H2 RECEPTORS. Cimetidine has a range of pharmacological actions. It inhibits GASTRIC ACID secretion, as well as PEPSIN and GASTRIN output.Formule :C10H16N6SCouleur et forme :Crystals Physical Description White Crystals With A Slight Sulfur-Mercaptan Odor (Ntp 1992)Masse moléculaire :252.34GLP-1 receptor agonist 7
CAS :GLP-1 receptor agonist 7, potential for diabetes research, from patent WO2021219019A1.Formule :C31H30ClFN4O5Couleur et forme :SolidMasse moléculaire :593.05WZ4141
CAS :WZ4141 is an intermediate in compound synthesis.Formule :C16H13N3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :279.29Benoxathian hydrochloride
CAS :Benoxathian hydrochloride is effective α 1 Adrenaline receptor antagonist. Benoxathian hydrochloride has value in the study of anorexia.Formule :C19H24ClNO4SCouleur et forme :SolidMasse moléculaire :397.91UCSF924
CAS :UCSF924 is a potent and specific agonist of dopamine D4 receptor (DRD4) partial (EC50: 4.2 nM, Ki: 3 nM).Formule :C20H22N2O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :322.4Fexofenadine-d6
CAS :Fexofenadine D6 is an antihistamine pharmaceutical drug.Fexofenadine D6 is deuterium labeled is Fexofenadine.Formule :C32H39NO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :507.69Tulobuterol-d9 HCl
CAS :Tulobuterol-d9 HCl is a deuterated compound of Tulobuterol HCl.Formule :C12H10D9Cl2NOCouleur et forme :SolidMasse moléculaire :273.25Antazoline phosphate
CAS :Antazoline phosphate: H1 histamine receptor antagonist with anticholinergic effects, eases allergies.Formule :C17H22N3O4PDegré de pureté :98%Couleur et forme :CoaMasse moléculaire :363.35PD176252
CAS :PD176252 is a BB1 and BB2 antagonist, GRPR inhibitor, and FPR1/FPR2 agonist that inhibits the growth and proliferation of a wide range of cancer cells.Formule :C32H36N6O5Degré de pureté :99.00%Couleur et forme :SolidMasse moléculaire :584.673-O-Methyldopa-d3
CAS :3-O-Methyldopa-d3 is a deuterated compound of 3-O-Methyldopa. 3-O-Methyldopa has a CAS number of 300-48-1.Formule :C10H10D3NO4Couleur et forme :SolidMasse moléculaire :214.23Diphenylpyraline
CAS :Diphenylpyridine is the first generation antihistamine, which has the anticholinergic effect of diphenylpiperidine.Formule :C19H23NOCouleur et forme :SolidMasse moléculaire :281.39Dapagliflozin impurity
CAS :Dapagliflozin impurity is the enantiomer of Dapagliflozin, Dapagliflozin is a sodium glucose transporter 2 inhibitor.Formule :C21H25ClO7Couleur et forme :SolidMasse moléculaire :424.87Cetirizine D4
CAS :Cetirizine D4 is a deuterium-labeled Cetirizine. Cetirizine is a second-generation antihistamine and a long-acting histamine H1-receptor antagonist.Formule :C21H25ClN2O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :392.91SHA 68
CAS :SHA 68 is a potent and selective non-peptide antagonist of neuropeptide S receptor (NPSR) with IC50 values of 22.0 nM for NPSR Asn107 and 23.8 nM for NPSR Ile107.Formule :C26H24FN3O3Degré de pureté :99.44%Couleur et forme :SolidMasse moléculaire :445.49Methyldopate
CAS :Methyldopate, an ethyl ester prodrug of methyldopa, inhibits dopamine decarboxylase to treat hypertension.Formule :C12H17NO4Couleur et forme :SolidMasse moléculaire :239.27Nefazodone
CAS :Nefazodone (Nefadar) is an oral antidepressant that is an antagonist of postsynaptic 5-HT 2A receptors and 5-HT 2C receptors, and SNDRI.Formule :C25H32ClN5O2Degré de pureté :99.85%Couleur et forme :White To Off-White Crystalline PowderMasse moléculaire :470.01Ref: TM-T21451
2mg42,00€5mg60,00€10mg87,00€1mL*10mM (DMSO)95,00€25mg177,00€50mg276,00€100mg422,00€200mg604,00€MK-761 TFA
MK-761 TFA is an effective, orally active β2-adrenergic receptor blocker. It exhibits antihypertensive properties and positive inotropic effects, along with vasodilatory activity.Formule :C15H20F3N3O4Couleur et forme :SolidMasse moléculaire :363.332Altanserin
CAS :Altanserin, a 5-HT2A receptor binder, is tagged with F-18 for brain PET scans.Formule :C22H22FN3O2SCouleur et forme :SolidMasse moléculaire :411.49Emedastine Difumarate
CAS :Emedastine Difumarate, an H1 receptor blocker for allergic conjunctivitis, reduces histamine-induced eye inflammation.Formule :C25H34N4O9Couleur et forme :SolidMasse moléculaire :534.56Paliperidone Palmitate
CAS :Paliperidone: atypical antipsychotic, dopamine & serotonin antagonist, affects α1/α2 adrenergic and H1 histamine receptors.Formule :C39H57FN4O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :664.893-Hydroxy agomelatine
CAS :3-Hydroxy agomelatine (3-Hydroxyagomelatine) is a 5-HT2C receptor antagonist used in the study of neurological disorders.Formule :C15H17NO3Couleur et forme :SolidMasse moléculaire :259.3Omidenepag
CAS :Omidenepag (UR-7276) is an EP2 agonist and a novel topical ocular hypotensive agent.Omidenepag can be used to study glaucoma and hypertension.Formule :C23H22N6O4SDegré de pureté :99.67% - 99.77%Couleur et forme :SolidMasse moléculaire :478.52Diacetolol D7
CAS :Diacetolol D7 is deuterium-labeled diacetone Roller. Diacetol is the main metabolite of Acetolol. Diacetololβ-adrenoceptor shielding and anti-arrhythmic agent.Formule :C16H24N2O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :315.42Endothelin-3 (Rat,Human) (TFA)
Endothelin-3 (Rat, Human) (TFA) is a 21-amino acid vasoactive peptide of endothelial origi, an agonist for the endothelin receptor type B (EDNRB).Formule :C123H169F3N26O35S4·xC2HF3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :2757.07 (free base)Flibanserin-d4
CAS :Flibanserin: Serotonin 5-HT1A agonist (Ki=1 nM), 5-HT2A antagonist (49 nM). Flibanserin D4 is deuterium-labeled.Formule :C20H21F3N4ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :394.43Terlipressin
CAS :Terlipressin is a potent vasoconstrictor that acts via V1 receptors on arteriolar smooth muscle cells.Formule :C52H74N16O15S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1227.37Triamterene (Standard)
CAS :Triamterene (Standard) is the standard substance of Triamterene, and it is applicable for quantitative analysis, quality control, and related research in biochemical experiments. Triamterene is a barosensitive epithelial sodium channel (ENaC) blocker with a diuretic effect. It can also act as an inhibitor of the TGR5 receptor, reducing GLP-1 secretion and cAMP level increases induced by TGR5 activation in a dose-dependent manner.Formule :C12H11N7Couleur et forme :Yellow Yellow SolidMasse moléculaire :253.263-Hydroxy agomelatine D3
CAS :3-Hydroxy agomelatine D3 is a deuterated metabolite of Agomelatine and a 5-HT2C antagonist (IC50: 3.2 μM, Ki: 1.8 μM).Formule :C15H17NO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :262.32Alosetron D3 Hydrochloride
CAS :Alosetron D3 (GR 68755 D3) Hydrochloride is a deuterium-labeled Alosetron. Alosetron is an antagonist of 5HT3-receptor.Formule :C17H19ClN4ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :333.83Clorprenaline
CAS :Clorprenaline is a β-adrenergic receptor agonist that activates adenylate cyclase, relaxation of bronchial smooth muscle cells. anti-inflammatory.Formule :C11H16ClNODegré de pureté :98.9%Couleur et forme :SolidMasse moléculaire :213.7Tetrahexyldecyl ascorbate
CAS :Tetrahexyldecyl ascorbate is a precursor of ascorbic acid, a more stable and permeable form of vitamin C. anti-hyperpigmentation antioxidant that inhibits MMP.Formule :C70H128O10Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1129.76L 888607
CAS :L 888607 is an effective and selective CRTH2 agonist (Ki: 0.8 nM).Formule :C19H15ClFNO2SCouleur et forme :SolidMasse moléculaire :375.84SBI-810 hydrochloride
CAS :SBI-810 hydrochloride is a β-arrestin-2 (βarr2)-biased allosteric modulator of NTSR1 (neurotensin receptor 1), exerting analgesic effects.Formule :C27H35ClN4O2Degré de pureté :99.42%Couleur et forme :SolidMasse moléculaire :483.05Alimemazine D6
CAS :Alimemazine D6 is a deuterium-labeled Alimemazine. Alimemazine is an antihistamine.Formule :C18H22N2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :304.48Rebamipide-d4
CAS :Rebamipide D4 is deuterium labeled Rebamipide.Formule :C19H15ClN2O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :374.81Substance P TFA
CAS :Substance P TFA is a CNS neuropeptide, serving as a neurotransmitter and modulator, targeting NK1R.Formule :C65H99F3N18O15SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :1461.67SB-277011 hydrochloride
CAS :SB-277011 hydrochloride (SB-277011A hydrochloride) is a D3R antagonist, which induces delayed ejaculation in rats.Formule :C28H31ClN4ODegré de pureté :98.54%Couleur et forme :SolidMasse moléculaire :475.03Timapiprant sodium
CAS :Timapiprant sodium: potent DP2 antagonist; inhibits mast cell activation; displaces [3H]PGD2, Ki=3-13 nM.Formule :C21H17FN2NaO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :371.367Virodhamine
CAS :Virodhamine (O-arachidonoyl ethanolamine), an endocannabinoid, is an antagonist of CB1 receptor and an agonist of CB2 receptor.Formule :C22H37NO2Degré de pureté :98%Couleur et forme :SoildMasse moléculaire :347.534,4-Diphenylbutylamine hydrochloride
CAS :4,4-Diphenylbutylamine shows affinity for the 5-HT2A and H1 receptors with Kis of 2589 and 1670 nM, respectively[1].Formule :C16H20ClNCouleur et forme :SolidMasse moléculaire :261.79Ceralifimod
CAS :Ceralifimod (ONO-4641) is a potent agonist for sphingosine 1-phosphate receptors 1 and 5 (EC50s: 27.3, 334 pM for human S1P receptor 1 and 5).Formule :C27H33NO4Couleur et forme :SolidMasse moléculaire :435.56Asenapine hydrochloride
CAS :Asenapine hydrochloride (Org 5222 hydrochloride) is an antagonist of 5-hydroxytryptamine, adrenergic, dopamine, and histamine receptors with antipsychotic effects.Formule :C17H17Cl2NOCouleur et forme :SolidMasse moléculaire :322.23BMS-986224
CAS :BMS-986224 is an orally active, potent and selective APJ receptor agonist.BMS-986224 is a candidate compound for the treatment of heart failure.
Formule :C24H23ClN4O6Degré de pureté :98.61% - 99.67%Couleur et forme :SolidMasse moléculaire :498.92Agomelatine-d6
CAS :Agomelatine D6 (S-20098 D6) is a deuterium-labeled Agomelatine. Agomelatine is a specific agonist of MT1 and MT2 receptors.Formule :C15H17NO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :249.34Cefaclor
CAS :Cefaclor (Panoral) is a cephalosporin antibiotic.Formule :C15H14ClN3O4SDegré de pureté :99.03% - 99.98%Couleur et forme :SolidMasse moléculaire :367.81Etofylline clofibrate
CAS :Etofylline clofibrate has a hypolipidemic and antithrombotic effect and it also has an agonistic interaction with intimal PGI2.Formule :C19H21ClN4O5Couleur et forme :SolidMasse moléculaire :420.85Telcagepant
CAS :Telcagepant (MK-0974) is an oral calcitonin gene-related peptide receptor (CGRP) antagonist that blocks CGRP receptors, migraines and for pain relief.Formule :C26H27F5N6O3Degré de pureté :98.98% - 98.98%Couleur et forme :SolidMasse moléculaire :566.52Canagliflozin (Standard)
CAS :Canagliflozin (Standard) is the standard substance of Canagliflozin, and it is applicable for quantitative analysis, quality control, and related research in biochemical experiments. Canagliflozin (JNJ 28431754AAA) is a selective SGLT2 inhibitor that inhibits CHO cells expressing mSGLT2, rSGLT2, and hSGLT2 (IC50=2/3.7/4.4 nM). Canagliflozin can be used for the treatment of type II diabetes mellitus (T2DM).Formule :C24H25FO5SCouleur et forme :SolidMasse moléculaire :444.52Agomelatine (L(+)-Tartaric acid)
CAS :Agomelatine (L(+)-Tartaric acid) is an MT1/MT2 agonist and selective 5-HT2C antagonist, supporting melatonergic and serotonergic signaling studies in neuroscience.Formule :C19H23NO8Degré de pureté :99.79%Couleur et forme :SolidMasse moléculaire :393.39SKF-82958 hydrobromide
CAS :SKF-82958 hydrobromide is a D1/D5 receptor full agonist.Formule :C19H21BrClNO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :410.73Fenoterol-d6 Hydrobromide
CAS :Fenoterol-d6 Hydrobromide is a deuterated compound of Fenoterol Hydrobromide. Fenoterol Hydrobromide has a CAS number of 1944-12-3. Fenoterol hydrobromide, the hydrobromide salt of fenoterol, is a β2 adrenoreceptor agonist with bronchodilator activity.Formule :C17H16D6BrNO4Masse moléculaire :390.30Docosahexaenoic acid ethyl ester
CAS :Docosahexaenoic acid ethyl ester (Ethyl docosahexaenoate) enhances 6-hydroxydopamine-induced neuronal damage by inducing lipid peroxidation in the mouse striatum, and can be used to study oxidative diseases of the retina or neurons.Formule :C24H36O2Degré de pureté :98.35%Couleur et forme :SolidMasse moléculaire :356.54Sumanirole maleate
CAS :Sumanirole maleate (PNU-95666E) is a D2 receptor full agonist with high selectivity that plays a vital role in Parkinson's disease and restless leg syndrome.Formule :C15H17N3O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :319.31Pimozide-d4
CAS :Pimozide D4 is a deuterium labeled Pimozide.Formule :C28H29F2N3ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :465.57Bradykinin (1-5)
CAS :Bradykinin (1-5), a stable metabolite of BK produced by ACE, serves as a marker for in vivo BK generation.Formule :C27H40N8O6Couleur et forme :SolidMasse moléculaire :572.66
