GPCR/G-Protéine
Les inhibiteurs des GPCR/protéines G sont des composés qui ciblent les récepteurs couplés aux protéines G (GPCR) et les protéines G associées, qui jouent un rôle crucial dans la transmission des signaux de l'extérieur vers l'intérieur des cellules. Ces inhibiteurs sont essentiels pour étudier les voies de signalisation médiées par les GPCR, impliquées dans de nombreux processus physiologiques, y compris la perception sensorielle, la réponse immunitaire et la neurotransmission. Les inhibiteurs des GPCR sont également importants dans le développement de médicaments, car de nombreux agents thérapeutiques ciblent ces récepteurs. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de GPCR/protéines G de haute qualité pour soutenir vos recherches en pharmacologie, biologie cellulaire et domaines connexes.
Sous-catégories appartenant à la catégorie "GPCR/G-Protéine"
- récepteur 5-HT(1.025 produits)
- Récepteur d'adénosine(249 produits)
- Récepteur adrénergique(3.023 produits)
- Récepteur de la bombésine(35 produits)
- Récepteur de la bradykinine(61 produits)
- CXCR(158 produits)
- CaSR(34 produits)
- Récepteur cannabinoïde(217 produits)
- Cholécystokinine(1 produits)
- Récepteur de la dopamine(445 produits)
- Récepteur de l'endothéline(86 produits)
- Récepteur GNRH(84 produits)
- GPCR19(33 produits)
- GRK(33 produits)
- GTPase(23 produits)
- Récepteur du glucagon(194 produits)
- Hérisson/Smoothened(49 produits)
- Récepteur de l'histamine(385 produits)
- Récepteur LPA(21 produits)
- Récepteur de la mélatonine(26 produits)
- Récepteur OX(41 produits)
- Récepteur opioïde(327 produits)
- PAFR(14 produits)
- PKA(60 produits)
- Récepteur S1P(18 produits)
- SGLT(31 produits)
- Récepteur Sigma(46 produits)
Affichez 19 plus de sous-catégories
5990 produits trouvés pour "GPCR/G-Protéine"
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Talinolol
CAS :(±)-Talinolol is a selective β1 adrenoceptor antagonist well known for its cardioprotective and antihypertensive activity.Formule :C20H33N3O3Degré de pureté :98.8%Couleur et forme :SolidMasse moléculaire :363.49Ref: TM-T21640
2mg34,00€5mg52,00€1mL*10mM (DMSO)52,00€10mg92,00€25mg178,00€50mg313,00€100mg535,00€200mg775,00€S1RA hydrochloride
CAS :S1RA hydrochloride (E-52862 hydrochloride) is an effective and specific sigma-1 receptor(σ1R, Ki: 17 nM) antagonist, and has good selectivity against σ2R (Ki >Formule :C20H24ClN3O2Degré de pureté :98% - 99.84%Couleur et forme :SolidMasse moléculaire :373.87Ref: TM-T4229
1mg35,00€5mg75,00€1mL*10mM (DMSO)84,00€10mg105,00€25mg205,00€50mg334,00€100mg492,00€500mg973,00€Almotriptan
CAS :Almotriptan (LAS 31416), a triptan and 5-HT1B/1D agonist, treats migraines by constricting cranial vessels and altering blood flow.Formule :C17H25N3O2SDegré de pureté :99.85%Couleur et forme :Light Yellow Or White PowerMasse moléculaire :335.46Ciproxifan maleate
CAS :Ciproxifan maleate (FUB 359)(FUB-359 maleate) is a highly potent and selective histamin H3-receptor antagonist with IC50 of 9.2 nM, with low apparent affinityFormule :C20H22N2O6Degré de pureté :99.39%Couleur et forme :SolidMasse moléculaire :386.4Ref: TM-T2004
1mg40,00€2mg52,00€5mg75,00€1mL*10mM (DMSO)82,00€10mg101,00€25mg205,00€50mg380,00€100mg565,00€Triptorelin acetate(57773-63-4 free base)
CAS :Triptorelin acetate is a GnRH agonist for hormone-responsive cancers, precocious puberty, and assisted reproduction.Formule :C66H86N18O15Degré de pureté :99.59% - 99.90%Couleur et forme :White PowderMasse moléculaire :1371.53Ref: TM-T21410
5mg52,00€10mg78,00€1mL*10mM (DMSO)116,00€25mg119,00€50mg172,00€100mg259,00€200mg388,00€Metergoline
CAS :Metergoline (Methergoline) is a dopamine agonist and serotonin antagonist.Formule :C25H29N3O2Degré de pureté :99.83% - 99.97%Couleur et forme :SolidMasse moléculaire :403.52Epinastine hydrochloride
CAS :Epinastine hydrochloride (WAL-801CL HCl) is an antihistamine and mast cell stabilizer that is used in eye drops to treat allergic conjunctivitis.Formule :C16H15N3·HClDegré de pureté :99.26% - 99.62%Couleur et forme :White SolidMasse moléculaire :285.77BD 1008 dihydrobromide
CAS :BD 1008 dihydrobromide: selective σ1 receptor antagonist (Ki=2 nM), high σ1 and moderate σ2 affinity.
Formule :C15H24Br2Cl2N2Degré de pureté :97.81%Couleur et forme :SolidMasse moléculaire :463.08SSR240612
CAS :SSR240612 is a potent, and orally active specific non-peptide bradykinin B1 receptor antagonist (Kis = 0.48-0.73 and 358-481 nM for B1 and B2 receptors,Formule :C42H53ClN4O7SDegré de pureté :98.59% - 99.16%Couleur et forme :SolidMasse moléculaire :793.41Ref: TM-T5048
1mg222,00€5mg512,00€1mL*10mM (DMSO)612,00€10mg700,00€25mg982,00€50mg1.333,00€100mg1.783,00€BWX 46 Acetate
BWX 46 Acetate is a potent, highly selective neuropeptide Y (NPY) receptor agonist with IC50 of 0.5 nM.Formule :C118H190N36O30S2Degré de pureté :96.86%Couleur et forme :SolidMasse moléculaire :2657.12LM11A-31 dihydrochloride
CAS :LM11A-31 dihydrochloride is a water-soluble, BBB-penetrating p75NTR ligand and proNGF antagonist.Formule :C12H27Cl2N3O2Degré de pureté :99.47% - 99.9%Couleur et forme :SolidMasse moléculaire :316.27Regadenoson
CAS :Regadenoson (CVT-3146) is a selective A2A receptor agonist that increases coronary blood flow with a longer half-life than adenosine.Formule :C15H18N8O5Degré de pureté :99.57% - 99.81%Couleur et forme :Off-White SolidMasse moléculaire :390.35Ref: TM-T2671
2mg44,00€5mg62,00€1mL*10mM (DMSO)69,00€10mg96,00€25mg170,00€50mg259,00€100mg394,00€500mg887,00€[Sar9,Met(O2)11]-Substance P acetate
[Sar9,Met(O2)11]-Substance P acetate is an NK1 agonist, raising MAP and HR equally to septide but with unique timing and behaviors.Formule :C66H106N18O18SDegré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :1471.75Ranitidine
CAS :Ranitidine (HSDB 3925) is a non-imidazole blocker of those histamine receptors that mediate gastric secretion (H2 receptors).Formule :C13H22N4O3SDegré de pureté :99.52%Couleur et forme :Solid SolidMasse moléculaire :314.40Raclopride tartrate
CAS :Raclopride is a selective antagonist on D2 dopamine receptor ( D2 Ki: 1.8 nm, D3 Ki: 3.5 nm, D4 Ki: 2400, D1 Ki: 18000 nM).Formule :C19H26Cl2N2O9Couleur et forme :SolidMasse moléculaire :497.32Ambrisentan sodium
CAS :Ambrosentan (BSF 208075) sodium is a selective and oral effective antagonist of ET type A receptor ( ETAR ).Formule :C22H21N2NaO4Couleur et forme :SolidMasse moléculaire :400.41F-15599
CAS :F-15599 is a highly selective G-protein biased 5-HT1A receptor agonist(Ki : 3.4 nM).Formule :C19H21ClF2N4ODegré de pureté :98.72%Couleur et forme :SolidMasse moléculaire :394.85Ref: TM-T7281
1mg49,00€5mg92,00€1mL*10mM (DMSO)104,00€10mg152,00€25mg295,00€50mg477,00€100mg715,00€200mg982,00€MF-766
CAS :MF-766: potent, selective oral EP4 antagonist, Ki=0.23 nM, IC50=1.4 nM; shifts to 1.8 nM with 10% HS. Useful in cancer, inflammation studies.Formule :C27H21F3N2O3Degré de pureté :99.54% - 99.59%Couleur et forme :SolidMasse moléculaire :478.46Tofogliflozin (hydrate)
CAS :Tofogliflozin hydrate (CSG-452 hydrate) is a potent and highly specific inhibitor of SGLT2(Ki of 2.9 nM, 14.9 nM, and 6.4 nM for human, rat, and mouse SGLT2).Formule :C22H28O7Degré de pureté :97.03% - 98.78%Couleur et forme :SolidMasse moléculaire :404.45Ref: TM-T5016
1mg35,00€2mg49,00€5mg74,00€1mL*10mM (DMSO)82,00€10mg109,00€25mg202,00€50mg324,00€100mg505,00€200mg717,00€Chlorcyclizine
CAS :CHLORCYCLIZINE is a histamine H1 antagonist and a potent hepatitis C virus (HCV) entry inhibitor.Formule :C18H21ClN2Degré de pureté :98.75%Couleur et forme :SolidMasse moléculaire :300.83Ozagrel hydrochloride
CAS :Ozagrel hydrochloride (OKY-046 HCl) is a selective thromboxane A(2) synthetase inhibitor used for the improvement of postoperative cerebrovascular contractionFormule :C13H12N2O2·HClDegré de pureté :99.80%Couleur et forme :White Or Off White Crystalline PowderMasse moléculaire :264.71A2B receptor antagonist 2
CAS :A2B receptor antagonist 2 is an antagonist of adenosine receptor A2B (Ki = 2.30 μM for rA1, 6.8 μM for rA2A, 3.44 μM for hA2B).Formule :C12H15N5Degré de pureté :100%Couleur et forme :SolidMasse moléculaire :229.28Cinacalcet
CAS :Cinacalcet (AMG 073) is an orally active, allosteric Ca receptor (CaR) agonist, treatment of cardiovascular disease .Formule :C22H22F3NDegré de pureté :99.48%Couleur et forme :Yellow OilMasse moléculaire :357.41Mequitazine
CAS :Mequitazine (Virginan) is an effective, nonsedative and long-acting histamine H1 antagonist.Formule :C20H22N2SDegré de pureté :99.98%Couleur et forme :SolidMasse moléculaire :322.47BAY-545
CAS :BAY-545 is an antagonist of A2B adenosine receptor(IC50 : 59 nM).Formule :C18H22F3N3O4SDegré de pureté :98.05%Couleur et forme :SolidMasse moléculaire :433.45Ref: TM-T8512
1mg84,00€5mg161,00€1mL*10mM (DMSO)172,00€10mg235,00€25mg420,00€50mg605,00€100mg842,00€200mg1.134,00€Tripelennamine
CAS :Tripelennamine: ethylenediamine derivative, H1-receptor blocker, reduces allergic reactions, treats rhinitis and conjunctivitis.Formule :C16H21N3Couleur et forme :SolidMasse moléculaire :255.36Lixisenatide acetate (320367-13-3 free base)
CAS :Lixisenatide acetate is a receptor agonist similar to glucagon-like peptide-1 (glp-1) for the treatment of type 2 diabetes mellitus (T2DM).Formule :C215H347N61O65S·6C2H4O2Degré de pureté :98% - 99.9%Couleur et forme :SolidMasse moléculaire :5218.88GRA Ex-25
CAS :GRA Ex-25 (GRA-Ex-25) is an inhibitor of glucagon receptor.Formule :C29H36F3N3O5Degré de pureté :98.2% - 98.88%Couleur et forme :SolidMasse moléculaire :563.61Ref: TM-T3422
1mg50,00€5mg105,00€1mL*10mM (DMSO)130,00€10mg161,00€25mg314,00€50mg470,00€100mg708,00€200mg964,00€Cinaciguat
CAS :Cinaciguat (BAY 58-2667) is a pioneering sGC activator for acute heart failure treatment.Formule :C36H39NO5Degré de pureté :98% - 99.18%Couleur et forme :SolidMasse moléculaire :565.7Ref: TM-T1984
1mg46,00€5mg92,00€1mL*10mM (DMSO)103,00€10mg138,00€25mg200,00€50mg278,00€100mg394,00€200mg537,00€Brefonalol
CAS :Brefonalol is a vasodilating beta-adrenergic receptor blocker.Formule :C22H28N2O2Couleur et forme :SolidMasse moléculaire :352.47Siramesine
CAS :Siramesine (Lu 28-179)(Lu 28-179) is a selective sigma-2 receptor agonist, which has been shown to trigger cell death of cancer cells and to exhibit a potentFormule :C30H31FN2ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :454.58Ondansetron
CAS :Ondansetron (GR 38032) is a serotonin 5-HT3 receptor antagonist used mainly as an antiemetic.Formule :C18H19N3ODegré de pureté :99.92%Couleur et forme :White To Yellow CrystalsMasse moléculaire :293.36Quipazine
CAS :Quipazine: 5-HT agonist, Ki 1.4 nM at 5-HT3R, anti-SARS-CoV-2 (EC50 31.64 μM), for neurological research.Formule :C13H15N3Couleur et forme :SolidMasse moléculaire :213.28BRL-15572 hydrochloride
CAS :BRL-15572 hydrochloride: selective h5-HT1D antagonist with high affinity; useful for studying h5-HT1D responses.Formule :C25H28Cl2N2OCouleur et forme :SolidMasse moléculaire :443.41Xanthine amine congener hydrochloride
CAS :Xanthine amine congener (XAC) hydrochloride is a non-selective adenosine receptor antagonist that induces convulsions in mice.Formule :C21H29ClN6O4Couleur et forme :SolidMasse moléculaire :464.95Nonapeptide-1
CAS :Nonapeptide-1 (Melanostatine™ 5) can inhibit the synthesis of melanin, which makes it of interest for treating certain skin conditions.Formule :C61H87N15O9SDegré de pureté :100%Couleur et forme :SolidMasse moléculaire :1206.5Sonepiprazole mesylate
CAS :Sonepiprazole mesylate is a selective D4 antagonistFormule :C22H31N3O6S2Couleur et forme :SolidMasse moléculaire :497.63Syk Inhibitor II dihydrochloride
CAS :Syk inhibitor II selectively blocks Syk (IC50 = 41 nM), impacting platelet function and inflammation, with lower potency against other kinases.Formule :C14H17Cl2F3N6ODegré de pureté :98.53%Couleur et forme :SolidMasse moléculaire :413.22Ref: TM-T4391
1mg130,00€2mg212,00€5mg455,00€1mL*10mM (DMSO)455,00€10mg647,00€25mg947,00€50mg1.264,00€100mg1.700,00€Cetrorelix diacetate
CAS :Cetrorelix diacetate (NS-75A) is is a gonadotropin-releasing hormone antagonist.Formule :C74H100ClN17O18Degré de pureté :98.38%Couleur et forme :SolidMasse moléculaire :1551.17Ref: TM-T5520L
1mg50,00€5mg95,00€10mg142,00€1mL*10mM (DMSO)239,00€25mg276,00€50mg414,00€100mg608,00€500mg1.288,00€Amitriptyline
CAS :Amitriptyline: a tricyclic antidepressant used for depression and neuropathic pain.Formule :C20H23NDegré de pureté :98.24% - 99.64%Couleur et forme :Crystals SolidMasse moléculaire :277.4(S)-Amisulpride
CAS :(S)-Amisulpride ((S) Amisulpride) (Esamisulpride) is a potent dopamine D2/D3 receptor antagonist.Formule :C17H27N3O4SDegré de pureté :98.38%Couleur et forme :SolidMasse moléculaire :369.48Ref: TM-T26375
1mg34,00€5mg84,00€1mL*10mM (DMSO)94,00€10mg123,00€25mg225,00€50mg358,00€100mg485,00€200mg622,00€SAX-187
CAS :SAX-187 (SAX-187) has high-affinity binding at the human 5-HT6 receptor.Formule :C15H13ClN4O2S2Degré de pureté :97.82% - 98%Couleur et forme :SolidMasse moléculaire :380.87Ref: TM-T3183
1mg79,00€5mg152,00€1mL*10mM (DMSO)166,00€10mg245,00€25mg398,00€50mg532,00€100mg735,00€200mg973,00€AHN 1-055 hydrochloride
CAS :AHN 1-055 hydrochloride (3α-Bis-(4-fluorophenyl) Methoxytropane hydrochloride) is an inhibitor of dopamine transporter (DAT) and dopamine uptake(IC50 = 71 nM).Formule :C21H24ClF2NODegré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :379.87Ref: TM-T39429
2mg34,00€5mg49,00€1mL*10mM (DMSO)50,00€10mg75,00€25mg130,00€50mg192,00€100mg295,00€200mg442,00€Ibrolipim
CAS :Ibrolipim (NO-1886) attenuates high glucose-induced endothelial dysfunction in cultured human umbilical vein endothelial cells via PI3K/Akt pathway.Formule :C19H20BrN2O4PDegré de pureté :98.04%Couleur et forme :SolidMasse moléculaire :451.25Detomidine hydrochloride
CAS :Detomidine hydrochloride (MPV-253 AII) produce dose-dependent sedative and analgesic effects, mediatated by activation of α2 catecholamine receptors.Formule :C12H14N2·HClDegré de pureté :99.97%Couleur et forme :SolidMasse moléculaire :222.71Almotriptan Malate
CAS :Almotriptan Malate (PNU180638), a selective 5-HT1B/1D receptor agonist, is used in the therapy of Migraine attacks in adults.Formule :C17H25N3O2S·C4H6O5Degré de pureté :99.95%Couleur et forme :Pale Yellow SolidMasse moléculaire :469.55HCGRP-(8-37) acetate
HCGRP-(8-37) acetate is a human calcitonin gene-related peptide (hCGRP) fragment acetate and also an antagonist of CGRP receptor.Formule :C141H234N44O40Degré de pureté :99.29%Couleur et forme :SolidMasse moléculaire :3185.64WAY-100635 Monomaleate
CAS :WAY-100635 maleate is a selective 5-hydroxytryptamine 1A receptor antagonist with an IC50 value of 0.91 nM and a Ki value of 0.39 nM.Formule :C25H34N4O2·C4H4O4Degré de pureté :98.44% - 99.46%Couleur et forme :SolidMasse moléculaire :538.64Ref: TM-T2631
2mg43,00€5mg63,00€1mL*10mM (DMSO)74,00€10mg89,00€25mg170,00€50mg315,00€100mg470,00€200mg680,00€500mg1.054,00€Ponesimod
CAS :Ponesimod (ACT-128800) is an orally available sphingosine-1-phosphate receptor 1 (S1PR1, S1P1) agonist with potential immunomodulating activity.Formule :C23H25ClN2O4SDegré de pureté :99.42% - 99.96%Couleur et forme :SolidMasse moléculaire :460.97Ref: TM-T3258
1mg43,00€2mg56,00€5mg88,00€1mL*10mM (DMSO)92,00€10mg124,00€25mg221,00€50mg383,00€100mg565,00€500mg1.215,00€[Sar9] Substance P acetate(77128-75-7 free base)
[Sar9]-Substance P acetate, an NK-1 receptor agonist, mimics SP's effect on progesterone metabolism.Formule :C66H104N18O15SDegré de pureté :96.67%Couleur et forme :SolidMasse moléculaire :1421.71Benzotript
CAS :Benzotript is an gastrin-receptor antagonist, with anti-gastrinic.Formule :C18H15ClN2O3Degré de pureté :97.82%Couleur et forme :SolidMasse moléculaire :342.776Ref: TM-T8578
1mg124,00€2mg178,00€5mg269,00€1mL*10mM (DMSO)286,00€10mg408,00€25mg672,00€50mg945,00€100mg1.279,00€Urantide acetate(669089-53-6 free base)
Urantide acetate: selective UT receptor blocker, doesn't affect other contractions or relaxations, partial agonist in Ca²⁺ assay.Formule :C53H70N10O14S2Degré de pureté :99.22%Couleur et forme :SolidMasse moléculaire :1135.31AM1241
CAS :AM-1241 is a selective cannabinoid CB2 receptor agonist with Ki of 3.4 nM, exhibits 82-fold selectivity over CB1 receptor.Formule :C22H22IN3O3Degré de pureté :98.937% - 99.1%Couleur et forme :SolidMasse moléculaire :503.33Ref: TM-T6755
2mg35,00€5mg49,00€10mg84,00€1mL*10mM (DMSO)87,00€25mg168,00€50mg275,00€100mg495,00€500mg1.071,00€MCL0020
CAS :MCL0020 is a potent and selective melanocortin MC4 receptor antagonist, reverses stress-induced anorexia but has no effect on food intake in free-feeding rats.Formule :C34H39N7O4Degré de pureté :99.18%Couleur et forme :SolidMasse moléculaire :609.725'-N-Ethylcarboxamidoadenosine
CAS :NECA, an adenosine receptor agonist, boosts brain extravasation of fluorescein and dextran without affecting the blood-brain barrier.Formule :C12H16N6O4Degré de pureté :98.95% - ≥95%Couleur et forme :PowderMasse moléculaire :308.29S1p receptor agonist 1
CAS :S1p receptor agonist 1 (S1p-receptor-agonist-1) is an S1P receptor agonist.Formule :C23H24FN3O3Degré de pureté :99.07% - 99.9%Couleur et forme :SolidMasse moléculaire :409.45Secretin (33-59), rat
CAS :Secretin (33-59), rat (Secretin (rat)) is a classical hormone in the gastrointestinal system and a neuropeptide.Formule :C129H216N42O42Degré de pureté :98.12%Couleur et forme :SolidMasse moléculaire :3027.35Fexofenadine hydrochloride
CAS :Fexofenadine hydrochloride (Terfenidine carboxylate hydrochloride) is a second generation antihistamine that is used for the treatment of allergic rhinitis,Formule :C32H39NO4·HClDegré de pureté :99.39% - ≥95%Couleur et forme :SolidMasse moléculaire :538.13Ozanimod
CAS :Ozanimod (RPC-1063) (RPC1063) is a specific oral S1P Receptor 1 modulator.Formule :C23H24N4O3Degré de pureté :98.68% - 99.58%Couleur et forme :SolidMasse moléculaire :404.46Ref: TM-T6923
1mg46,00€5mg90,00€1mL*10mM (DMSO)90,00€10mg137,00€25mg268,00€50mg430,00€100mg622,00€200mg879,00€500mg1.305,00€Indacaterol
CAS :Indacaterol (Onbrez; Arcapta) is a β2-Adrenergic Agonist. The mechanism of action of indacaterol is as an Adrenergic beta2-Agonist.Formule :C24H28N2O3Degré de pureté :99.96%Couleur et forme :SolidMasse moléculaire :392.49AC 187 Acetate
AC 187 Acetate is a potent antagonist of amylin receptor .AC 187 shows more selective for amylin receptor than calcitonin and CGRP receptors.Formule :C129H209N37O42Degré de pureté :99.71%Couleur et forme :SolidMasse moléculaire :2950.262-Methoxyidazoxan monohydrochloride
CAS :L-Albizziin (2-Methoxyidazoxan monohydrochloride) is a highly potent selective antagonist of the alpha 2r adrenergic receptor.Formule :C12H14N2O3·HClDegré de pureté :98.99%Couleur et forme :SolidMasse moléculaire :270.725-Benzyloxygramine
CAS :5-Benzyloxygramine blocks the Dopamin receptors and antagonizes the effects of 5-HT on the rat uterus and the rabbit ear.Formule :C18H20N2ODegré de pureté :99.13%Couleur et forme :SolidMasse moléculaire :280.36Preladenant
CAS :Preladenant (SCH-420814) is an orally bioavailable antagonist of the adenosine A2A receptor (Ki: 1.1 nM) and has >1000-fold selectivity over all other adenosineFormule :C25H29N9O3Degré de pureté :98.02% - 99.68%Couleur et forme :SolidMasse moléculaire :503.56Bromodiphenhydramine hydrochloride
CAS :Bromodiphenhydramine hydrochloride is a new antihistaminic in the control of cutaneous.Formule :C17H21BrClNODegré de pureté :97.29%Couleur et forme :SolidMasse moléculaire :370.71BMS 182874 hydrochloride
CAS :BMS 182874 hydrochloride is a nonpeptide endothelin (El) receptor antagonist.Formule :C17H20ClN3O3SDegré de pureté :97.01%Couleur et forme :SolidMasse moléculaire :381.88Ref: TM-T21790
1mg77,00€2mg92,00€5mg140,00€1mL*10mM (DMSO)146,00€10mg205,00€25mg343,00€50mg477,00€100mg665,00€200mg897,00€Bavisant dihydrochloride hydrate
CAS :Bavisant dihydrochloride (JNJ31001074AAC) is an oral H3 receptor antagonist for ADHD treatment. Phase 2 trials show no significant benefits at 10 mg/day.Formule :C19H31Cl2N3O3Couleur et forme :SolidMasse moléculaire :420.38Sar-[D-Phe8]-des-Arg9-Bradykinin acetate
Sar-[D-Phe8]-des-Arg9-Bradykinin acetate is a potent and selective bradykinin B1 receptor agonist (EC50 = 9.02 nM in rabbit aorta) that is resistant toFormule :C49H70N12O13Degré de pureté :99.93%Couleur et forme :SolidMasse moléculaire :1035.159-FLUORENOL
CAS :9-FLUORENOL is a dopamine reuptake inhibitor with IC50 of 9 μM, and a major metabolite of a compound developed as a wakefulness-promoting agent.Formule :C13H10ODegré de pureté :99.98%Couleur et forme :Off-White Crystalline PowderMasse moléculaire :182.22BMY 7378 dihydrochloride
CAS :BMY 7378 dihydrochloride (BMY7378 HCl) , α1D-adrenergic receptor antagonist, is a weak partial agonist/antagonist of 5-HT1A receptor.Formule :C22H33Cl2N3O3Degré de pureté :97.32% - 99.08%Couleur et forme :SolidMasse moléculaire :458.42BGC-20-1531 hydrochloride(1186532-61-5 free base)
CAS :BGC-20-1531 hydrochloride(1186532-61-5 free base) (GTPL3380 hydrochloride) is a EP4 antagonist for the treatment of acute migraine.Formule :C26H25ClN2O6SDegré de pureté :98.94% - 99.85%Couleur et forme :SolidMasse moléculaire :529FK962
CAS :FK962 is an somatostatin release enhancer , exerts cognitive-enhancing actions.Formule :C14H17FN2O2Degré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :264.3Ref: TM-T7829
2mg34,00€5mg52,00€1mL*10mM (DMSO)57,00€10mg82,00€25mg144,00€50mg200,00€100mg278,00€200mg389,00€Ursodeoxycholic acid sodium
CAS :Ursodeoxycholic acid sodium (Sodium Ursodeoxycholate) is a naturally occurring secondary bile acid with anti-inflammatory and cytoprotective activities.Formule :C24H40NaO4Degré de pureté :99.66% - 99.96%Couleur et forme :SolidMasse moléculaire :415.56Arformoterol Tartrate
CAS :Arformoterol Tartrate ((R,R)-Formoterol tartrate) is the tartrate salt of arformoterol.Formule :C23H30N2O10Degré de pureté :99.98%Couleur et forme :SolidMasse moléculaire :494.49Ref: TM-T22245
5mg60,00€1mL*10mM (DMSO)85,00€10mg87,00€25mg150,00€50mg221,00€100mg329,00€200mg487,00€Pitolisant hydrochloride
CAS :Pitolisant hydrochloride (Ciproxidine) is a potent and selective inverse agonist of the histamine H3 receptor(Ki : 0.16 nM).Formule :C17H27Cl2NODegré de pureté :99.72% - 99.91%Couleur et forme :SolidMasse moléculaire :332.31Ref: TM-T7176
5mg48,00€1mL*10mM (DMSO)50,00€10mg71,00€25mg117,00€50mg187,00€100mg295,00€200mg442,00€500mg708,00€Clozapine HCl
CAS :Clozapine HCl, an atypical antipsychotic, binds CNS receptors, targets 5-HT2A/2C, has weaker D2 antagonism. Risk: Agranulocytosis.Formule :C18H20Cl2N4Couleur et forme :SolidMasse moléculaire :363.29ELA-14(human) acetate
ELA-14(human) acetate, a fragment of ELA, targets APJ, activates Gαi1 and β-arrestin-2, and prompts receptor internalization like its parent peptide.Formule :C77H123N25O19S2Degré de pureté :97.2%Couleur et forme :SolidMasse moléculaire :1767.09ML-191
CAS :ML-191 is an inhibitor of LPI-induced phosphorylation of ERK1/2.Formule :C24H25N3O3Degré de pureté :99.58%Couleur et forme :SolidMasse moléculaire :403.47Vilanterol trifenatate
CAS :Vilanterol trifenatate is a long-acting agonist of β2-adrenoceptor (β2-AR) with inherent 24-hour activity(β2-AR, β1-AR and β3-AR pEC50s of 10.37, 6.98 and 7.36, respectively)Formule :C44H49Cl2NO7Degré de pureté :99.51% - >99.99%Couleur et forme :SolidMasse moléculaire :774.77Fluparoxan HCl
CAS :Fluparoxan is a potent α2-adrenergic receptor antagonist (pKB = 7.9) with excellent α2/α1 selectivity (2630 fold).Formule :C10H11ClFNO2Couleur et forme :SolidMasse moléculaire :231.65GW842166X
CAS :GW842166X: Potent CB2 agonist, EC50=63 nM, inactive at CB1, in Phase 2 trials.Formule :C18H17Cl2F3N4O2Degré de pureté :99.47%Couleur et forme :SolidMasse moléculaire :449.25Opaganib
CAS :Opaganib (ABC294640) is an orally active and specific sphingosine kinase-2 (SphK2) inhibitor (IC50: 60 μM).Formule :C23H25ClN2ODegré de pureté :98.86% - 99.85%Couleur et forme :SolidMasse moléculaire :380.91Ref: TM-T6750
1mg38,00€2mg50,00€5mg80,00€1mL*10mM (DMSO)82,00€10mg117,00€25mg227,00€50mg394,00€100mg583,00€GSK2018682 HCl
CAS :GSK2018682 is a novel sphingosine-1-phosphate receptor 1 (s1p1) and 5 (s1p5) agonist.Formule :C22H22Cl2N4O4Couleur et forme :SolidMasse moléculaire :477.34Rotundine
CAS :Rotundine (Gindarine) (L-tetrahydropalmatine, L-THP) is a selective dopamine D1 receptor antagonist with IC50 of 166 nM.Formule :C21H25NO4Degré de pureté :99.8% - 99.91%Couleur et forme :Off-White SolidMasse moléculaire :355.43Dimethocaine
CAS :Dimethocaine (Larocaine) is a local anesthetic which also effects on the central nervous system acting as dopamine-reuptake-inhibitor.Formule :C16H26N2O2Degré de pureté :99.52%Couleur et forme :SolidMasse moléculaire :278.39Phentolamine
CAS :Phentolamine mesylate is an alpha-1 and alpha-2 selective adrenergic receptor antagonistFormule :C17H19N3ODegré de pureté :99.86% - 99.94%Couleur et forme :Crystals SolidMasse moléculaire :281.35Ataciguat
CAS :Ataciguat (HMR-1766) (HMR-1766) is a potent and specific soluble guanylate cyclase (sGC) activator.Formule :C21H19Cl2N3O6S3Degré de pureté :99.09%Couleur et forme :SolidMasse moléculaire :576.49Pipamperone HCl
CAS :Pipamperone blocks 5-HT2A/B/C, D2/D3/D4, α1/α2 receptors; favors 5-HT2A/D4 over D2; negligible affinity for H1, mACh. Highly selective at low doses.Formule :C21H31ClFN3O2Couleur et forme :SolidMasse moléculaire :411.95Dynamin inhibitory peptide Acetate
Dynamin inhibitory peptide Acetate is a peptide with the sequence Gln-Val-Pro-Ser-Arg-Pro-Asn-Arg-Ala-Pro that inhibit the GTPase dynamin.Formule :C49H84N18O16Degré de pureté :97.28%Couleur et forme :SolidMasse moléculaire :1181.3Ref: TM-T21798L
1mg73,00€5mg198,00€10mg294,00€25mg467,00€1mL*10mM (DMSO)474,00€50mg642,00€100mg853,00€AZD1283
CAS :AZD1283 is an effective P2Y12 receptor antagonist (EC50: 3.0 ug/kg/min, binding IC50: 11 nM).Formule :C23H26N4O5SDegré de pureté :98.37% - 99.63%Couleur et forme :SolidMasse moléculaire :470.54Methiothepin mesylate
CAS :Methiothepin mesylate (Metitepine mesylate) is a potent and non-selective 5-HT2 receptor antagonist, used as an antipsychotic.Formule :C21H28N2O3S3Degré de pureté :98% - 99.92%Couleur et forme :SolidMasse moléculaire :452.65Pentagastrin
CAS :Pentagastrin (ICI-50123) is a synthetic polypeptide that has effects like gastrin when given parenterally, which can cause the secretion and synthesis ofFormule :C37H49N7O9SDegré de pureté :96.98% - 99.49%Couleur et forme :Fine Colorless Needle-Shaped Crystals From 2-Ethoxyethanol + Water SolidMasse moléculaire :767.89(E)-3,4,5-Trimethoxycinnamic acid
CAS :(E)-3,4,5-Trimethoxycinnamic acid (O-Methylsinapic acid) is a natural product from the roots and rhizomes of Notopterygium incisum.Formule :C12H14O5Degré de pureté :99.83%Couleur et forme :SolidMasse moléculaire :238.24L-DOPA methyl ester (hydrochloride)
CAS :L-DOPA methyl ester (LDME) is an agonist of dopamine D1 receptor.
Formule :C10H14ClNO4Degré de pureté :98.69% - 99.81%Couleur et forme :White SolidMasse moléculaire :247.675Eformoterol Hemifumarate
CAS :Formoterol fumarate (Eformoterol Hemifumarate), an effective, specific and long-acting β2-adrenoceptor agonist, is utilized in the treatment of COPD and asthmaFormule :C19H24N2O4C4H4O4Degré de pureté :99.86% - >99.99%Couleur et forme :White PowderMasse moléculaire :402.4Praliciguat
CAS :Praliciguat (IW-1973) is an orally active sGC stimulator with a 197 nM EC50 in HEK-293 cells, enhances NO signaling, and is a vasodilator.Formule :C21H14F8N6O2Degré de pureté :98.82%Couleur et forme :SolidMasse moléculaire :534.36Ref: TM-T16569
1mg142,00€2mg207,00€5mg349,00€1mL*10mM (DMSO)409,00€10mg537,00€25mg858,00€50mg1.161,00€100mg1.558,00€Tecadenoson
CAS :Tecadenoson (CVT-510) is a selective agonist of A1 adenosine receptor.
Formule :C14H19N5O5Degré de pureté :98.83%Couleur et forme :SolidMasse moléculaire :337.33Paltusotine
CAS :Paltusotine: nonpeptide SST2 agonist, orally bioavailable, regulates GH/IGF-1 in acromegaly.Formule :C27H22F2N4ODegré de pureté :99.91%Couleur et forme :SolidMasse moléculaire :456.49Aprepitant
CAS :Aprepitant (Aprepitant`) is a Substance P/Neurokinin-1 Receptor Antagonist.Formule :C23H21F7N4O3Degré de pureté :98% - 99.68%Couleur et forme :Off-White To Light Yellow Cyrstalline SolidMasse moléculaire :534.43Thonzylamine
CAS :Thonzylamine is an antihistamine/anticholinergic, combined with Clofedanol or Phenylephrine for cold, hay fever, or allergy relief.Formule :C16H22N4ODegré de pureté :99.45%Couleur et forme :SolidMasse moléculaire :286.37
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