GPCR/G-Protéine
Les inhibiteurs des GPCR/protéines G sont des composés qui ciblent les récepteurs couplés aux protéines G (GPCR) et les protéines G associées, qui jouent un rôle crucial dans la transmission des signaux de l'extérieur vers l'intérieur des cellules. Ces inhibiteurs sont essentiels pour étudier les voies de signalisation médiées par les GPCR, impliquées dans de nombreux processus physiologiques, y compris la perception sensorielle, la réponse immunitaire et la neurotransmission. Les inhibiteurs des GPCR sont également importants dans le développement de médicaments, car de nombreux agents thérapeutiques ciblent ces récepteurs. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de GPCR/protéines G de haute qualité pour soutenir vos recherches en pharmacologie, biologie cellulaire et domaines connexes.
Sous-catégories appartenant à la catégorie "GPCR/G-Protéine"
- récepteur 5-HT(1.025 produits)
- Récepteur d'adénosine(249 produits)
- Récepteur adrénergique(3.030 produits)
- Récepteur de la bombésine(35 produits)
- Récepteur de la bradykinine(61 produits)
- CXCR(159 produits)
- CaSR(34 produits)
- Récepteur cannabinoïde(217 produits)
- Cholécystokinine(1 produits)
- Récepteur de la dopamine(444 produits)
- Récepteur de l'endothéline(86 produits)
- Récepteur GNRH(84 produits)
- GPCR19(33 produits)
- GRK(33 produits)
- GTPase(22 produits)
- Récepteur du glucagon(196 produits)
- Hérisson/Smoothened(49 produits)
- Récepteur de l'histamine(385 produits)
- Récepteur LPA(21 produits)
- Récepteur de la mélatonine(26 produits)
- Récepteur OX(42 produits)
- Récepteur opioïde(325 produits)
- PAFR(14 produits)
- PKA(55 produits)
- Récepteur S1P(17 produits)
- SGLT(31 produits)
- Récepteur Sigma(46 produits)
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5984 produits trouvés pour "GPCR/G-Protéine"
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Antidepressant agent 3
Agent 3: orally active, antidepressant, anxiolytic, boosts performance and cognition.Formule :C17H30ClN5O2SCouleur et forme :SolidMasse moléculaire :403.97PACAP (1-27), human, ovine, rat TFA
PACAP (1-27) TFA is a pacap-38 fragment and PACAP receptor antagonist with IC50s: 3nm (rat PAC1), 2nm (rat VPAC1), 5nm (human VPAC2).Formule :C144H225F3N40O41SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :3261.68IRAK inhibitor 4 trans
IRAK inhibitor 4 targets and blocks IRAK4 activity; refers to its trans molecular configuration.Formule :C33H35F3N6O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :620.66(d(CH2)51,Tyr(Me)2,Dab5,Arg8)-Vasopressin
CAS :(d(CH2)5[Tyr(Me)2, Dab5]AVP), a vasopressin V1a receptor-specific antagonist, demonstrates a pA2 value of 6.71 [1].Formule :C52H76N14O11S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1137.38Astressin
CAS :Astressin is a truncated CRF analog; binds strongly to receptor's extracellular domain, likely acting as a neutral competitive antagonist.Formule :C161H269N49O42Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :3563.16[Gly8]-GLP-1(7-37) acetate
[Gly8]-GLP-1(7-37) acetate is a derivative of GLP-1, where glycine at position 8 is replaced with alanine. [Gly8]-GLP-1(7-37) acetate is also a peptide fragment of the GLP-1 receptor (GLP-1R) agonist, Dulaglutide.Couleur et forme :Odour SolidIsrapafant
CAS :Israpafant: PAF receptor blocker, IC50 0.84nM, hinders platelet aggregation, eosinophil activation, boosts calcium transit, anti-nephrotoxic.Formule :C28H29ClN4SCouleur et forme :SolidMasse moléculaire :489.07(±)5-iPF2α-VI
CAS :Isoprostanes are prostaglandin (PG)-like products of free-radical induced lipid peroxidation.Formule :C20H34O5Couleur et forme :SolidMasse moléculaire :354.487HTR2A antagonist 1
HTR2A antagonist 1 (Compound 15f) is an HTR2A antagonist with an IC50 of 42.79 nM. It induces sub-G1 cell cycle arrest and apoptosis in colorectal cancer cells by activating the p53/p21/caspase 3 signaling pathway. HTR2A antagonist 1 exhibits good liver microsomal stability and is useful for colorectal cancer research.Formule :C35H43Cl2F2N5O4Couleur et forme :SolidMasse moléculaire :706.65A3AR agonist 1
A3AR Agonist 1 (Compound 12), with a Ki of 25.8 nM, is a potent A3 adenosine receptor (A3AR) agonist that promotes β-arrestin2 recruitment with an effectiveFormule :C28H34N6O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :550.61CMKLR1 antagonist 1
CMKLR1 antagonist 1 (compound S-26d) is a potent, orally active antagonist of the chemokine-like receptor 1 (CMKLR1), exhibiting a pIC50 of 7.44 in hCMKLR1-Couleur et forme :Odour SolidLys-(Des-Arg9,Leu8)-Bradykinin
CAS :Lys-(Des-Arg9,Leu8)-Bradykinin is a selective antagonist of the bradykinin B1 receptor [1].Formule :C47H75N13O11Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :998.18Prostaglandin F2α 1,11-lactone
CAS :Prostaglandin F2α 1,11-lactone (PGF2α 1,11-lactone) is a lipid-soluble prodrug of Prostaglandin F2α and can be used in studies about treating glaucoma.Formule :C20H32O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :336.47Spns2-IN-1
Spns2-IN-1 is a potent Spns2 inhibitor, effectively impeding Spns2-dependent S1P transport with an IC50 value of 1.4±0.3 μM, crucial for modulating the immuneDegré de pureté :98%Couleur et forme :Odour Solid9-deoxy-9-methylene-16,16-dimethyl Prostaglandin E2
CAS :Meteneprost is a strong, long-lasting Prostaglandin E2 analog effective in ending early monkey pregnancies without causing fever or GI issues.Formule :C23H38O4Couleur et forme :SolidMasse moléculaire :378.553[Deamino-Pen1,Val4,D-Arg8]-vasopressin
CAS :[Deamino-Pen1,Val4,D-Arg8]-vasopressin (AVP-A) is an antagonist of arginine-vasopressin (AVP).Formule :C48H69N13O11S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1068.27Prolactin Releasing Peptide (1-31), human acetate
Prolactin Releasing Peptide (1-31), human (acetate), is a potent GPR10 ligand with high affinity, eliciting prolactin secretion.Formule :C162H26N56O44SCouleur et forme :SolidMasse moléculaire :3724.17Palonosetron N-oxide
CAS :Palonosetron N-oxide: metabolite and potential impurity of 5-HT3 antagonist palonosetron; forms under oxidative stress.Formule :C19H24N2O2Couleur et forme :SolidMasse moléculaire :312.413Urocortin II, human acetate
Urocortin II, human acetate, is a selective endogenous peptide agonist of type 2 corticotropin-releasing factor (CRF2) receptors, used to study the role of CRF2 receptors in feeding behavior.Couleur et forme :Odour SolidCannabinol methyl ether
CAS :Cannabinol methyl ether, a phytocannabinoid, serves as an analytical reference standard. This compound can be obtained through isolation from Cannabis plants, derived from cannabinol, or synthesized. The physiological and toxicological properties of cannabinol methyl ether remain unknown. It is designed exclusively for research and forensic applications.Formule :C22H28O2Couleur et forme :SolidMasse moléculaire :324.5Prostaglandin F2α methyl ester
CAS :Prostaglandin F2α methyl ester is a highly lipid-soluble PGF2α analog used to maintain low intraocular pressure.Formule :C21H36O5Couleur et forme :SolidMasse moléculaire :368.51Msh (11-13)
CAS :Msh (11-13) is a bioactive chemical.Formule :C16H30N4O4Couleur et forme :SolidMasse moléculaire :342.43Zenagamtide sodium
Zenagamtide is an agonist for both glucagon-like peptide-1 (GLP-1) and amylin receptors.Couleur et forme :Odour SolidNeurokinin A(4-10)
CAS :Neurokinin A(4-10)(TFA) is an agonist of tachykinin NK2 receptor .Formule :C34H54N8O10SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :766.91(D-Arg8)-Inotocin
CAS :'(D-Arg8)-Inotocin is a potent, selective, and competitive antagonist of the vasopressin receptor (V 1a R), exhibiting a binding affinity (K i) of 1.3 nM.Formule :C39H68N14O11S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :973.17MLS1082
CAS :MLS1082 is a D1-like dopamine receptor (D1R) orthosteric modulatothat stimulates G-protein signaling upon dopamine activation for neurodegenerative disorders.Formule :C24H23N3O2Degré de pureté :99.53%Couleur et forme :SolidMasse moléculaire :385.46ZM 253270
CAS :ZM 253270 is an nonpeptide neurokinin A antagonist.Formule :C22H26ClN7O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :471.95Norisoboldine hydrochloride
CAS :Norisoboldine hydrochloride: an oral AhR agonist from Radix Linderae, for Rheumatoid arthritis and Ulcerative colitis research.Formule :C18H20ClNO4Couleur et forme :SolidMasse moléculaire :349.81SR 142948 TFA
SR 142948 TFA is an orally active, selective non-peptide neurotensin receptor (NT) antagonist, displaying IC50 values of 1.19 nM in h-NTR1-CHO cells, 0.32 nM in HT-29 cells, and 3.96 nM in adult rat brain. In HT-29 cells, it counteracts NT-induced inositol monophosphate formation with an IC50 of 3.9 nM. It blocks NT-induced hypothermia, analgesia, and turning behavior in vivo and can cross the blood-brain barrier, making it useful for research in psychiatric disorders.Couleur et forme :Odour Solid2,3-dinor Thromboxane B1
CAS :TXB2 released from platelets becomes 11-dehydro and 2,3-dinor TXB2. Rats excrete 2,3-dinor TXB1, a reliable thromboxane biosynthesis marker.Formule :C18H32O6Couleur et forme :SolidMasse moléculaire :344.448Eledoisin
CAS :Eledoisin (Eledone peptide) is a specific agonist of NK2 and NK3 receptors.Eledoisin is an undecapeptide of mollusk origin, belonging to the tachykinin familyFormule :C54H85N13O15SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :1188.4GEP44
GEP44 is a peptide-biased triple agonist targeting the glucagon-like peptide-1 receptor (GLP-1R), neuropeptide Y1 receptor (Y1-R), and neuropeptide Y2 receptor (Y2-R). It induces GLP-1R-dependent insulin secretion in rat and human islets by offsetting the actions of Y1-R and GLP-1R agonism, controlled by Y1-R antagonists. Additionally, GEP44 enhances glucose uptake in muscle tissue through Y1-R mediation independent of insulin and significantly reduces food intake and body weight in diet-induced obese rat models. GEP44 is utilized in studies related to obesity and type 2 diabetes.Couleur et forme :Odour SolidMaridebart
CAS :Maridebart is a humanized IgG1-kappa monoclonal antibody that targets the GIPR (gastric inhibitory polypeptide receptor) [1].Couleur et forme :LiquidProstaglandin K1
CAS :Prostaglandin K1 (compound 46) is a structurally modified prostanoid analog with an EC50 and Ki of 2800 nM for the EP1 receptor.Formule :C20H32O5Couleur et forme :SolidMasse moléculaire :352.47γ3-MSH
CAS :γ3-MSH, originating from the N-terminal segment of pro-opiomelanocortin (POMC), induces aldosterone secretion in cultured human adrenal tumor cells [1].Formule :C126H188N44O37SCouleur et forme :SolidMasse moléculaire :2943.18Eloralintide
CAS :Eloralintide (LY 3841136) is an AMYR agonist, anticipated for research in type 2 diabetes and obesity.Formule :C201H319N49O65S2Couleur et forme :SolidMasse moléculaire :4526.1PG 106 acetate
PG 106 acetate: Selective hMC3 receptor antagonist, IC50=210 nM; inactive on hMC5 and hMC4, EC50=9900 nM.Formule :C53H73N13O11Degré de pureté :98.24%Couleur et forme :SolidMasse moléculaire :1068.2317-TFM-PGF1α
CAS :17-TFM-PGF1α (Compound 8) is a saturated prostaglandin analog. It exhibits a high affinity and receptor selectivity for the human prostaglandin F receptor (hFP receptor), with an EC50 of 85 nM.Formule :C24H35F3O5Couleur et forme :SolidMasse moléculaire :460.53[Ala11,D-Leu15]-Orexin B acetate
[Ala11,D-Leu15]-Orexin B acetate is a selective agonist of orexin-2 receptor (OX2) with an EC50 of 0.13 nM, showing 400-fold selectivity over OX1 (52 nM).Formule :C122H210N44O37SDegré de pureté :98.18%Couleur et forme :SolidMasse moléculaire :2917.31Met-RANTES,human,acetate
Met-RANTES (human) acetate is the acetate salt form of Met-RANTES (human). It acts as an antagonist for CCR1 and CCR5 receptors. This compound inhibits the human chemokines MIP-1α and MIP-1β, with respective IC50 values of 5 and 2 nM. Additionally, Met-RANTES (human) acetate reduces bone destruction and alleviates adjuvant-induced arthritis (AIA) in rats.Couleur et forme :Odour SolidPACAP-38 (31-38), human, mouse, rat acetate
PACAP-38 (31-38) acetate stimulates PAC1 receptor and boosts NPY and catecholamine in sympathetic neurons.Formule :C49H87N17O13Degré de pureté :99.92%Couleur et forme :SolidMasse moléculaire :1122.32GLP-1R agonist 27
<p>GLP-1R agonist 27 (compound 21) is a potent and orally active GLP-1R agonist. It enhances the accumulation of cyclic adenosine monophosphate (cAMP), reduces blood glucose levels, and decreases food intake. GLP-1R agonist 27 shows potential for research in obesity and type 2 diabetes mellitus (T2DM).</p>Formule :C32H33N5O4SeCouleur et forme :SolidMasse moléculaire :630.6Triamterene
CAS :Triamterene is a barosensitive epithelial sodium channel (ENaC) blocker with a diuretic effect. It can also act as an inhibitor of the TGR5 receptor, reducing GLP-1 secretion and cAMP level increases induced by TGR5 activation in a dose-dependent manner.Formule :C12H11N7Degré de pureté :99.77%Couleur et forme :Yellow Yellow SolidMasse moléculaire :253.26Metipranolol
CAS :Metipranolol (Betamann) is a type of β- Adrenergic receptors（ β- A potent antagonist of adrenergic receptor on guinea pig atria β 1- Adrenergic receptors and rat uterus β The 2-adrenergic receptor exhibited the beta blocking potentials (pA2) of 8.3 and 8.4, respectively. It is also a potent substituent in the 3H DHA binding assay, with a ligand concentration of 0.7 nM and a Ki of 39 ± 24 nM.Formule :C17H27NO4Degré de pureté :98.37%Couleur et forme :SolidMasse moléculaire :309.4γ1-MSH
CAS :Endogenous melanocortin MC3 receptor agonist (pKi = 7.46) that displays ~ 40-fold selectivity over MC4.Formule :C72H97N21O14SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :1512.768β-Hydroxy-exo-THC
CAS :8β-Hydroxy-exo-THC, a cannabinoid ether analog, exhibits weak affinity for receptor sites with an IC50 of 1.2 μM.Formule :C21H30O3Couleur et forme :SolidMasse moléculaire :330.46CCR6 antagonist 1
CAS :<p>CCR6 antagonist 1 blocks CCL20/CCR6, aiding autoimmune and IBD research.</p>Formule :C17H12F3NO2Degré de pureté :99.83%Couleur et forme :SoildMasse moléculaire :319.28Adrenocorticotropic Hormone (ACTH) (4-10), human
CAS :Adrenocorticotropic Hormone (ACTH) (4-10) is an agonist of potent melanocortin(MC4R) receptor .Formule :C44H59N13O10SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :962.09CUR61414 hydrochloride
CUR61414 hydrochloride: potent cell-permeable Hedgehog pathway inhibitor, IC50=100-200 nM, selectively targets Smo (Ki=44 nM), induces cancer cell apoptosis.Formule :C31H43ClN4O5Degré de pureté :94.05%Couleur et forme :SolidMasse moléculaire :587.15Spantide II
CAS :Spantide II is an antagonist of tachykinin.Formule :C86H104Cl2N18O13Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1668.77Cisapride hydrate
CAS :Cisapride acts directly as a selective agonist of serotonin 5-HT4 receptor with IC50 value of 0.483 μM. And It also acts indirectly as a parasympathomimetic.Formule :C23H31ClFN3O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :483.96Oxatomide
CAS :Oxatomide: Dual H1/P2X7 antagonist, antihistamine, anti-allergic, treats immune diseases, IC50: 0.95 μM (P2X7), 0.43 μM (5-HT).Formule :C27H30N4ODegré de pureté :99.28% - 99.72%Couleur et forme :White PowderMasse moléculaire :426.55Ref: TM-T19839
1mg35,00€5mg75,00€10mg114,00€25mg222,00€50mg356,00€100mg557,00€500mg1.153,00€1mL*10mM (DMSO)84,00€Bertilimumab
CAS :<p>Bertilimumab (CAT 213; iCo-008), a human monoclonal antibody that targets eotaxin-1 (CCL11), shows promise in the research of allergic disorders [1].</p>Couleur et forme :Liquid17-trifluoromethylphenyl trinor Prostaglandin F2α
CAS :A number of 17-phenyl trinor prostaglandin F2α (17-phenyl trinor PGF2α) derivatives have been approved for the treatment of glaucoma.Formule :C24H31F3O5Couleur et forme :SolidMasse moléculaire :456.5022,6-DMA hydrochloride
CAS :2,6-DMA hydrochloride is a phenethylamine and acts as an agonist of the serotonin 5-HT2 receptor, with a pA2 value of 5.09.Formule :C11H18ClNO2Couleur et forme :SolidMasse moléculaire :231.72[D-Trp8]-γ-MSH
CAS :<p>[D-Trp8]-γ-MSH is a selective melanocortin 3 (MC3) receptor agonist (IC50 values are 6.7, 340 and 600 nM for human MC3, MC5 and MC4 receptors respectively).</p>Formule :C74H99N21O16SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :1570.79Neuropeptide Y5 receptor ligand-1
CAS :Neuropeptide Y5 receptor ligand-1 (Compound 54), a carbazole derivative, acts as a powerful antagonist to the neuropeptide Y5 (NPY-5) receptor [1].Formule :C19H17N3O2Couleur et forme :SolidMasse moléculaire :319.36GB-110 hydrochloride
GB-110 HCl: potent, nonpeptidic oral PAR2 agonist; triggers Ca2+ release in HT29 cells; EC50 0.28 μM.Formule :C33H49ClN6O5Couleur et forme :SolidMasse moléculaire :645.23Neuropeptide FF
CAS :Endogenous antiopioid peptide and agonist at NPFF1 and NPFF2 receptors (Ki values are 2.82 and 0.21 nM respectively).Formule :C54H76N14O10Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1081.27d[Leu4,Lys8]-VP
CAS :Vasopressin V1B agonist; Ki: 0.16nM V1B, 64nM oxytocin; weak antidiuretic/vasopressor; minimal oxytocic action.Formule :C47H67N11O11S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1026.2Neuropeptide S(Rat)
CAS :Potent endogenous neuropeptide S receptor (NSPR) agonist (EC50 = 3.2 nM).Formule :C95H160N34O27Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :2210.52Pancreatic Polypeptide, rat
CAS :Rat Pancreatic Polypeptide: 36-amino acid peptide, NPYR4 agonist, secreted by islet PP cells.Formule :C195H298N58O57SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :4398.87Bremelanotide
CAS :Bremelanotide is a synthetic peptide analog of alpha-MSH and is an agonist at melanocortin receptors including the MC3R and MC4R.Formule :C50H68N14O10Degré de pureté :98%Couleur et forme :White PowderMasse moléculaire :1025.16Pentagastrin meglumine
CAS :Pentagastrin meglumine is a synthetic pentapeptide that has effects like gastrin when given parenterally.Formule :C44H66N8O14SCouleur et forme :SolidMasse moléculaire :963.11(S)-V-0219 hydrochloride
(S)-V-0219 hydrochloride, a GLP-1R PAM, triggers calcium in hGLP-1R HEK cells, lowers glucose in mice, and reduces fasting hunger.Formule :C20H26ClF3N4O2Couleur et forme :SolidMasse moléculaire :446.89GLI1-IN-3
GLI1-IN-3 (Compound 11a) is a triterpenoid-like compound that inhibits Hedgehog signaling in cancer cells with GLI1 overexpression. It suppresses the proliferation of non-small cell lung cancer and prostate cancer cell lines with excessive Hh signaling activation. Additionally, GLI1-IN-3 reduces the expression of GLI1 protein and its target genes associated with tumor progression and proliferation in A549 and DU-145 cancer cells.Couleur et forme :Odour SolidGLP-1R agonist 29
GLP-1R agonist 29 (Compound 20) is a GLP-1R agonist that induces hGLP-1R-mediated cAMP stimulation with an EC50 of 0.018 nM. It exhibits favorable pharmacokinetic properties and shows good in vivo exposure, with an AUC0-∞,sc of 77688 ng·h/mL.Couleur et forme :Odour SolidSB-408124
CAS :SB408124: Non-peptide, OX1 receptor antagonist, Ki 57 nM (whole cell) and 27 nM (membrane), 50x more selective than OX2.Formule :C19H18F2N4ODegré de pureté :99.81%Couleur et forme :SolidMasse moléculaire :356.37Cetirizine methyl ester
CAS :Cetirizine methyl ester is a Cetirizine impurity, a long-acting, oral H1-antihistamine and hydroxyzine metabolite.Formule :C22H27ClN2O3Couleur et forme :SolidMasse moléculaire :402.91NF 340
CAS :P2Y11 antagonistFormule :C37H30N4Na4O15S4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :990.87Vortioxetine D8
CAS :Vortioxetine D8 is a deuterium-labeled antidepressant inhibiting 5-HT1A/B, 5-HT3A, 5-HT7 receptors & SERT (Ki: 15-1.6 nM).Formule :C18H22N2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :306.5Ontazolast
CAS :Ontazolast: a small-molecule LTB4R antagonist targeting asthma and immune disorders.Formule :C21H25N3ODegré de pureté :99.94%Couleur et forme :SoildMasse moléculaire :335.44Dipentylone hydrochloride
CAS :Dipentylone hydrochloride (Bk-dmbdp HCl) is a psychoactive synthetic cathinone and sympathomimetic stimulant. Its inhibitory activity towards the dopamine transporter (IC50=0.233µM) is tenfold higher than that towards NET and SERT, inhibiting dopamine uptake and stimulating locomotor activity in mice.Formule :C14H20ClNO3Degré de pureté :99.94%Couleur et forme :SolidMasse moléculaire :285.77SB656104
CAS :SB656104 is a bioactive chemical.Formule :C25H30ClN3O3SCouleur et forme :SolidMasse moléculaire :488.04Brexpiprazole S-oxide D8
CAS :Brexpiprazole S-oxide D8 (DM-3411 D8) is a deuterium-labeled metabolite of Brexpiprazole, a partial agonist at 5-HT1A and dopamine receptors.Formule :C25H19D8N3O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :457.61LY 344864 racemate
CAS :LY 344864 racemate is a 5-HT1F receptor agonist.Formule :C21H22FN3ODegré de pureté :99.75%Couleur et forme :SoildMasse moléculaire :351.42Tafluprost acid
CAS :Tafluprost acid is a selective agonist at the prostaglandin F receptor.Formule :C22H28F2O5Couleur et forme :SolidMasse moléculaire :410.46Leukotriene B4 Ethanolamide
CAS :<p>LTB4 binds to BLT1 (high affinity) and BLT2. LTB4-EA, a metabolite, is a stronger BLT1 antagonist, suggesting anti-inflammatory properties.</p>Formule :C22H37NO4Couleur et forme :SolidMasse moléculaire :379.541Zicronapine fumarate
CAS :Zicronapine fumarate, an antipsychotic, targets D1/D2 & 5-HT2A receptors; may treat neuropsychiatric conditions.Formule :C26H31ClN2O4Couleur et forme :SolidMasse moléculaire :470.9913,14-dihydro-15-keto Prostaglandin F1α
CAS :<p>13,14-dihydro-15-keto Prostaglandin F1α (13,14-dihydro-15-keto PGF1α) is a metabolite of PGF1α that has been reported in the rat stomach.</p>Formule :C20H36O5Couleur et forme :SolidMasse moléculaire :356.5Urocortin III, mouse
CAS :Mouse UcnIII, linked to stress behaviors, mainly occurs in the brain and rises in the hypothalamus post-restraint.Formule :C186H312N52O52S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :4172.97Ghrelin receptor full agonist-2
CAS :Ghrelin receptor full agonist-2 is a highly potent Ghrelin receptor full agonist.Formule :C26H28ClN5O5SCouleur et forme :SolidMasse moléculaire :558.05BQ-123 TFA
BQ-123 TFA: Potent ETA antagonist, IC50 = 7.3 nM, Ki = 25 nM, inhibits ET-1 cell proliferation, lowers rat BP.Formule :C33H43F3N6O9Couleur et forme :SolidMasse moléculaire :724.72(Ala13)-Apelin-13 TFA
'(Ala13)-Apelin-13 TFA acts as a potent antagonist of the apelin receptors (APJ) and impedes gastric motility via the vagal cholinergic pathway [1].'Formule :C63H107N23O16S·xC2HF3O2Couleur et forme :SolidMasse moléculaire :1474.73 (free acid)MEN 11270
CAS :B2 bradykinin receptor peptide antagonist, pKi 10.3; improves hypotension, bronchoconstriction; B2-selective over 29 receptors/ion channels.Formule :C60H90N20O11SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :1299.56Methicillin sodium hydrate
CAS :Methicillin sodium hydrate, a narrow-spectrum antibiotic, combats methicillin-resistant Staphylococcus strains and treats various infections.Formule :C17H21N2NaO7SCouleur et forme :SolidMasse moléculaire :420.41GLP-1 receptor agonist 9 citrate
<p>GLP-1 receptor agonist 9 citrate is an agonist of GLP-1.</p>Formule :C38H39ClFN3O12Degré de pureté :98.76%Couleur et forme :SolidMasse moléculaire :784.18Stressin I
Potent CRF1 agonist; Ki: 1.5 nM (CRF1), 224 nM (CRF2). Boosts ACTH, enhances stool frequency after i.p. administration.Formule :C203H337N57O56Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :4472.24SR 142948 dihydrochloride
SR 142948 dihydrochloride is a selective oral non-peptide NT antagonist, IC50 <4 nM, with brain penetration and potential for psychiatric research.Formule :C39H53Cl2N5O6Couleur et forme :SolidMasse moléculaire :758.77TGR5 agonist 2
TGR5 agonist 2 (compound 19) serves as a highly potent agonist of TGR5, demonstrating an EC50 value of 0.27 µM [1].Formule :C29H50NNaO6SCouleur et forme :SolidMasse moléculaire :563.77YM 09538
CAS :YM 09538 is a biochemical.Formule :C18H25ClN2O5SCouleur et forme :SolidMasse moléculaire :416.92HPP-9
HPP-9, a Proteolysis-Targeting Chimera (PROTAC) derived from Hedgehog Pathway Inhibitor-1 (HPI-1) with a pIC50 value of 6.71, is designed to degrade BETFormule :C49H52N6O11Couleur et forme :SolidMasse moléculaire :900.97GLP-1R agonist 14
CAS :GLP-1R agonist 14, also known as Compound 14, is a potent agonist of the GLP-1 receptor, demonstrating an EC50 range of 0-20 nM against human GLP-1 [1].Formule :C45H42F2N10O5Couleur et forme :SolidMasse moléculaire :840.88MrgprX2 antagonist-5
CAS :MrgprX2 antagonist-5 from patent WO2020223255A1 inhibits MrgprX2, useful for inflammatory skin disorder studies.Formule :C19H13ClF2N4O2SCouleur et forme :SolidMasse moléculaire :434.85O-Desethyl Dapagliflozin
CAS :O-Desethyl Dapagliflozin (Empagliflozin-4) is a SGLT2 inhibitor, IC50=33nM.Formule :C19H21ClO6Degré de pureté :98.33%Couleur et forme :SolidMasse moléculaire :380.82Ref: TM-T67849
1mg57,00€5mg120,00€10mg187,00€25mg321,00€50mg470,00€100mg683,00€1mL*10mM (DMSO)135,00€Antibiotic Sch 60057
CAS :Antibiotic Sch 60057 is a useful organic compound for research related to life sciences. The catalog number is T125403 and the CAS number is 203061-35-2.Formule :C45H84O6Couleur et forme :SolidMasse moléculaire :721.161Pancreatic Polypeptide, human
CAS :Endogenous high affinity agonist for human NPY Y4 receptor (Ki = 0.056 nM). Believed to play an important role in the function of the gastrointestinal tract.Formule :C185H287N53O54S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :4181.71ELA-11(human)
CAS :Apelin receptor agonist with high affinity (Ki = 14 nM). Blocks cAMP production and promotes β-arrestin activation; derived from ELA-32.Formule :C58H90N16O13S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1283.57Sufotidine
CAS :Sufotidine (AH 25352X) is a highly selective competitive H2 receptor antagonist.Formule :C20H31N5O3SDegré de pureté :99.03% - 99.92%Couleur et forme :SolidMasse moléculaire :421.56Mini Gastrin I, human
CAS :Mini Gastrin I, human, is a truncated form of the human gastrin peptide, encompassing amino acids 5-17 of the original sequence.Formule :C74H99N15O26SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :1646.73
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