GPCR/G-Protéine
Les inhibiteurs des GPCR/protéines G sont des composés qui ciblent les récepteurs couplés aux protéines G (GPCR) et les protéines G associées, qui jouent un rôle crucial dans la transmission des signaux de l'extérieur vers l'intérieur des cellules. Ces inhibiteurs sont essentiels pour étudier les voies de signalisation médiées par les GPCR, impliquées dans de nombreux processus physiologiques, y compris la perception sensorielle, la réponse immunitaire et la neurotransmission. Les inhibiteurs des GPCR sont également importants dans le développement de médicaments, car de nombreux agents thérapeutiques ciblent ces récepteurs. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de GPCR/protéines G de haute qualité pour soutenir vos recherches en pharmacologie, biologie cellulaire et domaines connexes.
Sous-catégories appartenant à la catégorie "GPCR/G-Protéine"
- récepteur 5-HT(1.025 produits)
- Récepteur d'adénosine(249 produits)
- Récepteur adrénergique(3.023 produits)
- Récepteur de la bombésine(35 produits)
- Récepteur de la bradykinine(61 produits)
- CXCR(158 produits)
- CaSR(34 produits)
- Récepteur cannabinoïde(217 produits)
- Cholécystokinine(1 produits)
- Récepteur de la dopamine(445 produits)
- Récepteur de l'endothéline(86 produits)
- Récepteur GNRH(84 produits)
- GPCR19(33 produits)
- GRK(33 produits)
- GTPase(23 produits)
- Récepteur du glucagon(194 produits)
- Hérisson/Smoothened(49 produits)
- Récepteur de l'histamine(385 produits)
- Récepteur LPA(21 produits)
- Récepteur de la mélatonine(26 produits)
- Récepteur OX(41 produits)
- Récepteur opioïde(327 produits)
- PAFR(14 produits)
- PKA(60 produits)
- Récepteur S1P(18 produits)
- SGLT(31 produits)
- Récepteur Sigma(46 produits)
Affichez 19 plus de sous-catégories
5986 produits trouvés pour "GPCR/G-Protéine"
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ML224
CAS :ML224 (NCGC00242364) is a TSHR antagonist for the treatment of Graves' orbital disease and Graves' hyperthyroidism.Formule :C31H31N3O5Degré de pureté :99.14%Couleur et forme :SolidMasse moléculaire :525.59Granisetron
CAS :Granisetron, a serotonin receptor (5HT-3 selective) antagonist, is used as an antinauseant and antiemetic for cancer chemotherapy.
Formule :C18H24N4OCouleur et forme :SolidMasse moléculaire :312.41SANT 2
CAS :SANT 2 is a Hedgehog (Hh) signaling pathway antagonist with potential anti-inflammatory and anti-cancer activities.Formule :C26H26ClN3O4Degré de pureté :99.23%Couleur et forme :SolidMasse moléculaire :479.96Thiethylperazine
CAS :Thiethylperazine (Tietilperazina) is a D2 receptor and H1 receptor antagonist, and an ABCC1 activator with antimicrobial and antiemetic activity.Formule :C22H29N3S2Degré de pureté :98.72%Couleur et forme :SolidMasse moléculaire :399.62GPR34 receptor antagonist 3
Compound 5e, a GPR34 receptor antagonist, exhibits selective inhibition of lysophosphatidylserine-induced ERK1/2 phosphorylation in a dose-dependent manner,Couleur et forme :Odour SolidFexofenadine-d6
CAS :Fexofenadine D6 is an antihistamine pharmaceutical drug.Fexofenadine D6 is deuterium labeled is Fexofenadine.Formule :C32H39NO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :507.69Apraclonidine hydrochloride
CAS :Apraclonidine hydrochloride (ALO 2145) is an α2-adrenergic agonist and a weak α-1 adrenergic receptor agonist.Formule :C9H11Cl3N4Degré de pureté :99.74%Couleur et forme :SolidMasse moléculaire :281.57Lanreotide
CAS :Lanreotide, a somatostatin analogue, suppresses GH/IGF-I hypersecretion in acromegaly patients. It also used to manage neuroendocrine tumours.Formule :C54H69N11O10S2Couleur et forme :SolidMasse moléculaire :1096.32GLP-1R modulator L7-028
CAS :GLP-1R modulator L7-028 is a variant modulator that enhances affinity for GLP-1 and cAMP signaling.Formule :C24H28N2O3Degré de pureté :98.76% - >99.99%Couleur et forme :SolidMasse moléculaire :392.49Eticlopride hydrochloride
CAS :Eticlopride, an antipsychotic, is a Selective dopamine D2/D3 receptor antagonist (Ki: 0.5/0.16 nM).Formule :C17H25ClN2O3·HClDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :377.31Spiroxatrine
CAS :Spiroxatrine (R 5188) is a 5-HT1α and α2-adrenergic dual antagonist with sedative activity for the study of diseases related to the cardiovascular system.Formule :C22H25N3O3Degré de pureté :99.94%Couleur et forme :SolidMasse moléculaire :379.45Travoprost (Standard)
CAS :Travoprost (Standard) is the standard substance of Travoprost, and it is applicable for quantitative analysis, quality control, and related research in biochemical experiments. Travoprost (Fluprostenol isopropyl ester) is used to treat glaucoma and ocular hypertension,is a potent and selective FP prostaglandin receptor agonist.Formule :C26H35F3O6Couleur et forme :Colorless OilMasse moléculaire :500.55GLP-1R modulator C16
CAS :GLP-1R modulator C16 is a variable modulator that significantly increases the binding affinity of GLP-4.Formule :C21H26ClFN2O3Degré de pureté :99.6% - >99.99%Couleur et forme :SolidMasse moléculaire :408.89rac-Propranolol-d7
CAS :Rac-Propranolol-d7 is the deuterated form of Rac-Propranolol. Propranolol is a β-adrenergic receptor antagonist that inhibits β1AR.Formule :C16H14D7NO2Couleur et forme :SolidMasse moléculaire :266.39UCSF924
CAS :UCSF924 is a potent and specific agonist of dopamine D4 receptor (DRD4) partial (EC50: 4.2 nM, Ki: 3 nM).Formule :C20H22N2O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :322.4Fedovapagon
CAS :Fedovapagon (VA106483) is a pressin V2 receptor (V2R) agonist for the study of overactive bladder syndrome.Formule :C27H34N4O3Degré de pureté :99.46%Couleur et forme :SolidMasse moléculaire :462.58SB-200646A
CAS :SB-200646A: oral 5-HT2B/2C antagonist; higher affinity than 5-HT2A (pKi: 7.5, 6.9 vs 5.2); anxiolytic with in vivo effects.Formule :C15H15ClN4ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :302.76SAR247799
CAS :SAR247799 is a selective and G-protein-biased S1P1 agonist that activates downstream G-protein signaling pathways more preferentially on endothelial cells.Formule :C21H16ClN3O5Couleur et forme :SolidMasse moléculaire :425.82Asenapine hydrochloride
CAS :Asenapine hydrochloride (Org 5222 hydrochloride) is an antagonist of 5-hydroxytryptamine, adrenergic, dopamine, and histamine receptors with antipsychotic effects.Formule :C17H17Cl2NOCouleur et forme :SolidMasse moléculaire :322.23Eplivanserin (mixture)
CAS :Eplivanserin mixture is a selective serotonin reuptake inhibitor and a 5-HT2A receptor antagonist,Formule :C19H21FN2O2Couleur et forme :SolidMasse moléculaire :328.387Nefazodone
CAS :Nefazodone (Nefadar) is an oral antidepressant that is an antagonist of postsynaptic 5-HT 2A receptors and 5-HT 2C receptors, and SNDRI.Formule :C25H32ClN5O2Degré de pureté :99.85%Couleur et forme :White To Off-White Crystalline PowderMasse moléculaire :470.01Ref: TM-T21451
2mg42,00€5mg60,00€10mg87,00€1mL*10mM (DMSO)95,00€25mg177,00€50mg276,00€100mg422,00€200mg604,00€Piribedil D8
CAS :Piribedil D8 is the deuterium labeled Piribedil, which is an agent of antiparkinsonian.Formule :C16H18N4O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :306.39Setiptiline maleate
CAS :Setiptiline maleate is a norepinephrine reuptake inhibitor, 2-adrenergic receptor antagonist, H1 receptor inverse agonist, 5-HT serotonin receptor antagonist.Formule :C23H23NO4Degré de pureté :99.94%Couleur et forme :SolidMasse moléculaire :377.43Trimethobenzamide
CAS :Trimethobenzamide (Ro 2-9578) is a D2 antagonist used to prevent nausea and vomiting.Formule :C21H28N2O5Couleur et forme :SolidMasse moléculaire :388.46RU-SKI 43 Hydrochloride
CAS :RU-SKI 43 Hydrochloride is a selective Hedgehog acyltransferase inhibitor (IC50 850 nM) with reported anticancer activity in tumor biology studies.Formule :C22H31ClN2O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :423.01Fenoterol-d6 Hydrobromide
CAS :Fenoterol-d6 Hydrobromide is a deuterated compound of Fenoterol Hydrobromide. Fenoterol Hydrobromide has a CAS number of 1944-12-3. Fenoterol hydrobromide, the hydrobromide salt of fenoterol, is a β2 adrenoreceptor agonist with bronchodilator activity.Formule :C17H16D6BrNO4Masse moléculaire :390.30Sulfisoxazole (Standard)
CAS :Sulfisoxazole (Standard) is the standard substance of Sulfisoxazole, and it is applicable for quantitative analysis, quality control, and related research in biochemical experiments. Sulfisoxazole (Sulfafurazole) is a short-acting sulfonamide antibacterial with activity against a wide range of gram-negative and gram-positive organisms.Sulfisoxazole inhibits breast cancer exosome release by targeting endothelin receptor A.Formule :C11H13N3O3SCouleur et forme :White To Cream PowderMasse moléculaire :267.30Tiotidine
CAS :Tiotidine is a selective histamine H2-receptor antagonist (pA2=7.3-7.8 for guinea-pig right atrium).Formule :C10H16N8S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :312.42BMS-986020 sodium
CAS :BMS-986020 sodium (AM152 sodium) is a high-affinity LPA1 antagonist for investigating idiopathic pulmonary fibrosis.Formule :C29H25N2NaO5Degré de pureté :99.83%Couleur et forme :SolidMasse moléculaire :504.51Cimetidine (Standard)
CAS :Cimetidine (Standard) is the standard substance of Cimetidine, and it is applicable for quantitative analysis, quality control, and related research in biochemical experiments. Cimetidine (SKF-92334) is a histamine congener, it competitively inhibits HISTAMINE binding to HISTAMINE H2 RECEPTORS. Cimetidine has a range of pharmacological actions. It inhibits GASTRIC ACID secretion, as well as PEPSIN and GASTRIN output.Formule :C10H16N6SCouleur et forme :Crystals Physical Description White Crystals With A Slight Sulfur-Mercaptan Odor (Ntp 1992)Masse moléculaire :252.34TFLLR-NH2(TFA)
CAS :TFLLR-NH2 (TFA) is a selective PAR1 agonist with an EC50 of 1.9 μM. EC50: 1.9 μM (PAR1)Formule :C33H54F3N9O8Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :761.83ML 00253764
CAS :melanocortin MC4 receptor antagonistFormule :C18H18BrFN2OCouleur et forme :SolidMasse moléculaire :377.25Thioridazine
CAS :Thioridazine: an antipsychotic, anti-anxiety drug, blocks dopamine D2, PI3K-Akt-mTOR; halts angiogenesis, kills cancer cells, targets CSCs.Formule :C21H26N2S2Couleur et forme :SolidMasse moléculaire :370.57Olanzapine D3
CAS :Olanzapine D3 is the deuterium labeled Olanzapine.Formule :C17H20N4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :315.45Ziprasidone amino acid
CAS :Ziprasidone Impurity C is a byproduct of Ziprasidone, an antipsychotic that blocks 5-HT and dopamine receptors.Formule :C21H23ClN4O2SCouleur et forme :SolidMasse moléculaire :430.954-Hydroxyatomoxetine D3
CAS :4-Hydroxyatomoxetine D3, a deuterium variant, is Atomoxetine's active metabolite, metabolized by CYP2D6, an adrenergic reuptake blocker.Formule :C17H21NO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :274.37GRK2 Inhibitor
CAS :GRK2 Inhibitor is an inhibitor of β-Adrenergic Receptor Kinase 1 (β ARK1).Formule :C12H9NO6Couleur et forme :SolidMasse moléculaire :263.2Cariprazine D6
CAS :Cariprazine D6 (RGH-188 D6) is a deuterium-labeled Cariprazine. Cariprazine is an antipsychotic agent (D3 receptors, Ki: 0.085 nM; D2 receptors, Ki: 0.49 nM).Formule :C21H26D6Cl2N4ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :433.45Calcium-Sensing Receptor Antagonists I
CAS :Calcium-Sensing Receptor Antagonists I functions as an antagonist to the parathyroid hormone receptors that sense calcium.Formule :C23H24N2O2Couleur et forme :SolidMasse moléculaire :360.45Lecirelin
CAS :Lecirelin is a synthetic GnRH (gonadotropin releasing hormone) analogue which shows a great efficacy in the treatment of bovine ovarian follicular cysts.Formule :C59H84N16O12Couleur et forme :SolidMasse moléculaire :1209.4Vilazodone-d8
CAS :Vilazodone D8 is a deuterium-labeled vilazodone. Vilazodone is a combined inhibitor of serotonin specific reuptake (SSRI) and agonist of 5-HT1A receptor partial.Formule :C26H27N5O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :449.57Allura Red AC (Standard)
CAS :Allura Red AC (Standard) is the standard substance of Allura Red AC, and it is applicable for quantitative analysis, quality control, and related research in biochemical experiments. Allura Red AC (CI 16035) is a very important food azo dye used in the food, pharmaceutical, paper, cosmetic and textile industries.Allura Red AC promotes susceptibility to experimental colitis via mouse intestinal serotonin.Formule :C18H14N2Na2O8S2Couleur et forme :Dark Maroon Solid PowderMasse moléculaire :496.42Brombuterol hydrochloride
CAS :Brombuterol is an agonist of the β2-adrenergic receptor (β2-AR).1It has been used as an illicit feed additive to increase the muscle-to-fat ratio of livestock.Formule :C12H19Br2ClN2OCouleur et forme :SolidMasse moléculaire :402.56Methyldopate
CAS :Methyldopate, an ethyl ester prodrug of methyldopa, inhibits dopamine decarboxylase to treat hypertension.Formule :C12H17NO4Couleur et forme :SolidMasse moléculaire :239.27Clomipramine D3 hydrochloride
CAS :Clomipramine D3 hydrochloride is the deuterium-labeled Clomipramine. Clomipramine is a serotonin transporter, norepinephrine transporter dopamine transporter blocker (Ki: 0.14, 54 and 3 nM).Formule :C19H24Cl2N2Couleur et forme :SolidMasse moléculaire :354.33(+)-Penbutolol
CAS :(+)-Penbutolol is an antagonist of β-adrenoceptor(IC50 of 0.74 μM). (+)-Penbutolol is an optical isomer of l-penbutolol with Na+ channel-blocking action.Formule :C18H29NO2Couleur et forme :SolidMasse moléculaire :291.43Quetiapine-d8 Fumarate
CAS :Quetiapine-d8 Fumarate is a deuterated compound of Quetiapine Fumarate. Quetiapine Fumarate has a CAS number of 111974-72-2. Quetiapine Fumarate, an atypical antipsychotic, is used in the treatment of bipolar I mania, schizophrenia, bipolar II depression, bipolar I depression.Formule :C25H21D8N3O6SCouleur et forme :SolidMasse moléculaire :507.634-(4-Chlorobenzyl)phthalazin-1(2H)-one
CAS :4-(4-Chlorobenzyl)phthalazin-1(2H)-one is a useful organic compound for research related to life sciences. The catalog number is T67610 and the CAS number is 53242-88-9.Formule :C15H11ClN2OCouleur et forme :SolidMasse moléculaire :270.72Dehydroaripiprazole
CAS :Dehydroaripiprazole (DM-14857), aripiprazole's active metabolite, is formed by CYP3A4 and CYP2D6, with similar antipsychotic effects.Formule :C23H25Cl2N3O2Degré de pureté :98.7%Couleur et forme :SolidMasse moléculaire :446.37Ivabradine-d6 hydrochloride
CAS :Ivabradine HCl: novel If inhibitor, IC50 2.9 μM; lowers heart rate. Ivabradine D6 HCl is its deuterium variant.Formule :C27H37ClN2O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :511.08MrgprX2 antagonist-1
CAS :MrgprX2 antagonist-1 (compound E23) is a MrgprX2 antagonist applicable to cutaneous inflammation.Formule :C15H15F5N4O2SDegré de pureté :99.80%Couleur et forme :SolidMasse moléculaire :410.361-Methyl-4-imidazoleacetic Acid (hydrochloride)
CAS :MIMA, a stable histamine byproduct from N-methylhistamine oxidation, indicates systemic mastocytosis via urinary levels.Formule :C6H9ClN2O2Couleur et forme :SolidMasse moléculaire :176.601Canagliflozin (Standard)
CAS :Canagliflozin (Standard) is the standard substance of Canagliflozin, and it is applicable for quantitative analysis, quality control, and related research in biochemical experiments. Canagliflozin (JNJ 28431754AAA) is a selective SGLT2 inhibitor that inhibits CHO cells expressing mSGLT2, rSGLT2, and hSGLT2 (IC50=2/3.7/4.4 nM). Canagliflozin can be used for the treatment of type II diabetes mellitus (T2DM).Formule :C24H25FO5SCouleur et forme :SolidMasse moléculaire :444.52Alosetron D3 Hydrochloride
CAS :Alosetron D3 (GR 68755 D3) Hydrochloride is a deuterium-labeled Alosetron. Alosetron is an antagonist of 5HT3-receptor.Formule :C17H19ClN4ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :333.83GLP-1 receptor agonist 7
CAS :GLP-1 receptor agonist 7, potential for diabetes research, from patent WO2021219019A1.Formule :C31H30ClFN4O5Couleur et forme :SolidMasse moléculaire :593.05Tetrahexyldecyl ascorbate
CAS :Tetrahexyldecyl ascorbate is a precursor of ascorbic acid, a more stable and permeable form of vitamin C. anti-hyperpigmentation antioxidant that inhibits MMP.Formule :C70H128O10Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1129.76BW 723C86
CAS :BW 723C86 is a 5-HT2B receptor agonist with anxiolytic effects, inducing overeating and reduced grooming in rats, useful in studying neurological disorders.Formule :C16H19ClN2OSDegré de pureté :99.35%Couleur et forme :SolidMasse moléculaire :322.85(Rac)-Mirabegron-d5
CAS :(Rac)-Mirabegron D5 is a deuterium labeled (Rac)-Mirabegron. Mirabegron is a selective agonist of β3-adrenoceptor.Formule :C21H24N4O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :401.54GB-88
CAS :GB-88 is an selective , oral non-peptide antagonist of PAR2, inhibits PAR2 activated Ca2+ release with an IC50 of 2 μM.Formule :C32H42N4O4Couleur et forme :SolidMasse moléculaire :546.7Doxazosin D8
CAS :Doxazosin D8, a deuterium-labeled version, is a selective AP1 adrenergic antagonist and a quinazoline derivative.Formule :C23H25N5O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :459.52Hydroxyzine dihydrochloride-d4
CAS :Hydroxyzine dihydrochloride-d4 is a deuterated compound of Hydroxyzine dihydrochloride.Formule :C21H25D4Cl3N2O2Couleur et forme :SolidMasse moléculaire :451.85Propranolol-d7 hydrochloride
CAS :Propranolol D7 HCl: deuterium-labeled, nonselective βAR antagonist.Formule :C16H22ClNO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :302.85Ziprasidone D8
CAS :Ziprasidone D8, deuterium-labeled, is a potent antipsychotic, antagonizing 5-HT and dopamine receptors.Formule :C21H21ClN4OSDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :420.99Metipranolol hydrochloride
CAS :Metipranolol hydrochloride is a non-selective β-adrenergic receptor blocking agent.Formule :C17H28ClNO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :345.86Bombesin
CAS :Bombesin: 14-amino acid peptide from toad skin with two mammalian homologs, neuromedin B and gastrin-releasing peptide.Formule :C71H110N24O18SCouleur et forme :While Lyophilized PowderMasse moléculaire :1619.85Cetirizine D4
CAS :Cetirizine D4 is a deuterium-labeled Cetirizine. Cetirizine is a second-generation antihistamine and a long-acting histamine H1-receptor antagonist.Formule :C21H25ClN2O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :392.91Tulobuterol-d9 HCl
CAS :Tulobuterol-d9 HCl is a deuterated compound of Tulobuterol HCl.Formule :C12H10D9Cl2NOCouleur et forme :SolidMasse moléculaire :273.25Aramisulpride
CAS :Aramisulpride is a dual antagonist of the dopamine D2 receptor and serotonin receptor, primarily utilized for investigating metabolic disorders.Formule :C17H27N3O4SCouleur et forme :SolidMasse moléculaire :369.483-O-Methyldopa-d3
CAS :3-O-Methyldopa-d3 is a deuterated compound of 3-O-Methyldopa. 3-O-Methyldopa has a CAS number of 300-48-1.Formule :C10H10D3NO4Couleur et forme :SolidMasse moléculaire :214.23L 888607
CAS :L 888607 is an effective and selective CRTH2 agonist (Ki: 0.8 nM).Formule :C19H15ClFNO2SCouleur et forme :SolidMasse moléculaire :375.84β2AR/M-receptor agonist-2
CAS :β2AR/M-receptor agonist-2 is a dual-function compound acting as a muscarinic antagonist and β2 adrenoceptor agonist (MABA).Formule :C36H49ClN4O7SCouleur et forme :SolidMasse moléculaire :717.31SUN B8155
CAS :SUN B8155 is a CT receptor agonist that induces cAMP formation in cells expressing recombinant human CT receptor.Formule :C14H15N3O3Degré de pureté :99.38% - 99.99%Couleur et forme :SolidMasse moléculaire :273.29GLP-1 receptor agonist 2
CAS :GLP-1 receptor agonist 2 is a glucagon-like peptide-1 receptor (GLP-1R) agonist.Formule :C30H31ClFN5O4Couleur et forme :SolidMasse moléculaire :580.05Ceralifimod
CAS :Ceralifimod (ONO-4641) is a potent agonist for sphingosine 1-phosphate receptors 1 and 5 (EC50s: 27.3, 334 pM for human S1P receptor 1 and 5).Formule :C27H33NO4Couleur et forme :SolidMasse moléculaire :435.56Gizzerosine
CAS :Gizzerosine, a biogenic amine formed during feed processing, is a toxicant that induces mortality in livestock.Formule :C11H20N4O2Couleur et forme :SolidMasse moléculaire :240.3SB-408124 Hydrochloride
CAS :SB-408124 Hydrochloride is a non-peptide OX1 receptor antagonist(Ki of 57 nM and 27 nM in both whole cell and membrane, respectively).Formule :C19H19ClF2N4ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :392.83MK-761 TFA
MK-761 TFA is an effective, orally active β2-adrenergic receptor blocker. It exhibits antihypertensive properties and positive inotropic effects, along with vasodilatory activity.Formule :C15H20F3N3O4Couleur et forme :SolidMasse moléculaire :363.332Bradykinin (1-5)
CAS :Bradykinin (1-5), a stable metabolite of BK produced by ACE, serves as a marker for in vivo BK generation.Formule :C27H40N8O6Couleur et forme :SolidMasse moléculaire :572.66Benoxathian hydrochloride
CAS :Benoxathian hydrochloride is effective α 1 Adrenaline receptor antagonist. Benoxathian hydrochloride has value in the study of anorexia.Formule :C19H24ClNO4SCouleur et forme :SolidMasse moléculaire :397.91Hydroxyzine D8
CAS :Hydroxyzine D8, a deuterium-labeled version of Hydroxyzine, acts as a histamine H1-receptor antagonist.Formule :C21H27ClN2O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :382.95(S)-ZINC-3573
CAS :(S)-ZINC 3573 is a negative control for (R)-ZINC 3573. (S)-ZINC 3573 displays no activity at MRGPRX2 at concentrations below 100 μM.Formule :C18H21N5Couleur et forme :SolidMasse moléculaire :307.401Endothelin-3 (Rat,Human) (TFA)
Endothelin-3 (Rat, Human) (TFA) is a 21-amino acid vasoactive peptide of endothelial origi, an agonist for the endothelin receptor type B (EDNRB).Formule :C123H169F3N26O35S4·xC2HF3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :2757.07 (free base)Lysosphingomyelin (d18:1)
CAS :Sphingomyelins are phosphorylcholine, sphingosine, and fatty acid. Lysosphingomyelin, missing the fatty acid, activates diverse cellular pathways.Formule :C23H49N2O5PCouleur et forme :SolidMasse moléculaire :464.628Timapiprant sodium
CAS :Timapiprant sodium: potent DP2 antagonist; inhibits mast cell activation; displaces [3H]PGD2, Ki=3-13 nM.Formule :C21H17FN2NaO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :371.367Altanserin
CAS :Altanserin, a 5-HT2A receptor binder, is tagged with F-18 for brain PET scans.Formule :C22H22FN3O2SCouleur et forme :SolidMasse moléculaire :411.49Acrivastine D7
CAS :Acrivastine D7 is a deuterium labeled Acrivastine. Acrivastine is a short acting antagonist of histamine 1 receptor.Formule :C22H24N2O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :355.484-Hydroxypropranolol-d7 hydrochloride
CAS :Deuterium-labeled 4-Hydroxypropranolol HCl, a Propranolol metabolite that blocks β1/β2 receptors.Formule :C16H22ClNO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :318.85Doxepin D3 Hydrochloride
CAS :Doxepin D3 Hydrochloride is a deuterium-labeled doxepin hydrochloride.Doxepin hydrochloride is an oral active tricyclic antidepressant used as a sedative.Doxepin hydrochloride is also an effective CYP450 inhibitor, significantly inhibiting CYP450 2C19 andFormule :C19H22ClNODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :318.86Substance P TFA
CAS :Substance P TFA is a CNS neuropeptide, serving as a neurotransmitter and modulator, targeting NK1R.Formule :C65H99F3N18O15SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :1461.67Diphenylpyraline
CAS :Diphenylpyridine is the first generation antihistamine, which has the anticholinergic effect of diphenylpiperidine.Formule :C19H23NOCouleur et forme :SolidMasse moléculaire :281.39Diacetolol D7
CAS :Diacetolol D7 is deuterium-labeled diacetone Roller. Diacetol is the main metabolite of Acetolol. Diacetololβ-adrenoceptor shielding and anti-arrhythmic agent.Formule :C16H24N2O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :315.42R121919
CAS :R121919 (NBI30775) is an adrenocorticotropin-releasing factor receptor 1 (CRF1) receptor antagonist with antidepressant and anxiolytic activity.Formule :C22H32N6Degré de pureté :99.75%Couleur et forme :SolidMasse moléculaire :380.53Flibanserin-d4
CAS :Flibanserin: Serotonin 5-HT1A agonist (Ki=1 nM), 5-HT2A antagonist (49 nM). Flibanserin D4 is deuterium-labeled.Formule :C20H21F3N4ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :394.43Dapagliflozin impurity
CAS :Dapagliflozin impurity is the enantiomer of Dapagliflozin, Dapagliflozin is a sodium glucose transporter 2 inhibitor.Formule :C21H25ClO7Couleur et forme :SolidMasse moléculaire :424.87Rebamipide-d4
CAS :Rebamipide D4 is deuterium labeled Rebamipide.Formule :C19H15ClN2O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :374.81Terlipressin
CAS :Terlipressin is a potent vasoconstrictor that acts via V1 receptors on arteriolar smooth muscle cells.Formule :C52H74N16O15S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1227.37Fipexide hydrochloride
CAS :Fipexide (hydrochloride) is a kind of psychoactive drug of the piperazine class.Formule :C20H22Cl2N2O4Couleur et forme :SolidMasse moléculaire :425.31Cefaclor
CAS :Cefaclor (Panoral) is a cephalosporin antibiotic.Formule :C15H14ClN3O4SDegré de pureté :99.03% - 99.98%Couleur et forme :SolidMasse moléculaire :367.81Antazoline phosphate
CAS :Antazoline phosphate: H1 histamine receptor antagonist with anticholinergic effects, eases allergies.Formule :C17H22N3O4PDegré de pureté :98%Couleur et forme :CoaMasse moléculaire :363.35NBI-27914
CAS :NBI-27914 is a selective and non-peptide CRFR1 (corticotropin-releasing factor receptor 1) antagonist with analgesic effects, capable of blocking CRF-induced anxiety.Formule :C18H20Cl4N4Degré de pureté :99.47% - 99.64%Couleur et forme :SolidMasse moléculaire :434.19SKF-82958 hydrobromide
CAS :SKF-82958 hydrobromide is a D1/D5 receptor full agonist.Formule :C19H21BrClNO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :410.73Nadolol-d9
CAS :Nadolol D9 is the deuterium labeled Nadolol is a blocker of non-selective beta.
Formule :C17H27NO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :318.46Fluvoxamine
CAS :Fluvoxamine (DU-23000) is a selective, orally available 5-HT and serotonin reuptake inhibitor (SSRI) exhibiting antidepressant effects.Formule :C15H21F3N2O2Degré de pureté :99.91%Couleur et forme :SolidMasse moléculaire :318.33(R)-Praziquantel-d11
CAS :(R)-Praziquantel D11 is the deuterium labeled (R)-Praziquantel.Formule :C19H24N2O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :323.47SB-674042
CAS :SB-674042 is a nonpeptide dual antagonist of the appetite peptides OX1 and OX2 receptors.SB-674042 is used in the treatment of depression.Formule :C24H21FN4O2SDegré de pureté :99.87% - 99.9%Couleur et forme :SolidMasse moléculaire :448.51JNJ-10397049
CAS :OX2 receptor antagonistFormule :C19H20Br2N2O3Couleur et forme :SolidMasse moléculaire :484.18Clorprenaline
CAS :Clorprenaline is a β-adrenergic receptor agonist that activates adenylate cyclase, relaxation of bronchial smooth muscle cells. anti-inflammatory.Formule :C11H16ClNODegré de pureté :98.9%Couleur et forme :SolidMasse moléculaire :213.74,4-Diphenylbutylamine hydrochloride
CAS :4,4-Diphenylbutylamine shows affinity for the 5-HT2A and H1 receptors with Kis of 2589 and 1670 nM, respectively[1].Formule :C16H20ClNCouleur et forme :SolidMasse moléculaire :261.79Dexloxiglumide
CAS :Dexloxiglumide is the active enantiomer of Loxiglumide; it inhibits CCK-8-induced contractions and is a selective CCKA receptor antagonist.Formule :C21H30Cl2N2O5Couleur et forme :SolidMasse moléculaire :461.38Aripiprazole (D8)
CAS :Aripiprazole D8 (OPC-14597 D8) is the deuterium-labeled Aripiprazole. Aripiprazole is a human 5-HT1A receptor partial agonist (Ki: 4.2 nM).Formule :C23H27Cl2N3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :456.44Alimemazine D6
CAS :Alimemazine D6 is a deuterium-labeled Alimemazine. Alimemazine is an antihistamine.Formule :C18H22N2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :304.48Docosahexaenoic acid ethyl ester
CAS :Docosahexaenoic acid ethyl ester (Ethyl docosahexaenoate) enhances 6-hydroxydopamine-induced neuronal damage by inducing lipid peroxidation in the mouse striatum, and can be used to study oxidative diseases of the retina or neurons.Formule :C24H36O2Degré de pureté :98.35%Couleur et forme :SolidMasse moléculaire :356.54Virodhamine
CAS :Virodhamine (O-arachidonoyl ethanolamine), an endocannabinoid, is an antagonist of CB1 receptor and an agonist of CB2 receptor.Formule :C22H37NO2Degré de pureté :98%Couleur et forme :SoildMasse moléculaire :347.53MRGPRX4 modulator-2
CAS :MRGPRX4 modulator-2 (compound 1-55) is a highly potent antagonist of MRGPRX4 with an IC50 value of less than 100 nM. Its notable applications include research on autoimmune diseases such as psoriasis, multiple sclerosis, Steven Johnson's Syndrome, and various chronic itch conditions [1].Formule :C15H9ClF4O3Degré de pureté :99.24%Couleur et forme :SolidMasse moléculaire :348.68MRS-3777 hemioxalate
CAS :MRS-3777 hemioxalate, a selective adenosine A3 receptor antagonist, reverses the anti-injury perception effects of its corresponding agonist and serves as a valuable tool for studying inflammatory pain.
Formule :C17H19N5OC2H2O4Degré de pureté :97.10%Couleur et forme :SolidMasse moléculaire :354.39TP-16
CAS :TP-16 is a novel potent and selective EP4 antagonist that blocks the function of IMCs and enhances cytotoxic T cell-mediated tumor elimination in vivo.Formule :C24H22FNO4SDegré de pureté :98.53% - 99.15%Couleur et forme :SolidMasse moléculaire :439.5Tegaserod
CAS :Tegaserod is a 5-HT4R agonist and 5-HT2B receptor antagonist with antitumor activity used in the treatment of irritable bowel syndrome (IBS).Formule :C16H23N5ODegré de pureté :99.20% - 99.89%Couleur et forme :SolidMasse moléculaire :301.39Asenapine
CAS :Asenapine (Org 5222) is a 5-HT receptor, adrenergic receptor, and histamine receptor antagonist with antipsychotic properties for the treatment of schizophreniaFormule :C17H16ClNODegré de pureté :99.64%Couleur et forme :CoaMasse moléculaire :285.77Clothiapine
CAS :Clothiapine is an atypical antipsychotic of the dibenzothiazepine chemical class.Formule :C18H18ClN3SDegré de pureté :99.93%Couleur et forme :SolidMasse moléculaire :343.87Emedastine Difumarate
CAS :Emedastine Difumarate, an H1 receptor blocker for allergic conjunctivitis, reduces histamine-induced eye inflammation.Formule :C25H34N4O9Couleur et forme :SolidMasse moléculaire :534.56SB-269970 hydrochloride
CAS :SB-269970 hydrochloride (SB-269970A) , a hydrochloride salt form of SB-269970, is a 5-HT7 receptor antagonist (pKi of 8.3) and exhibits >50-fold selectivityFormule :C18H28N2O3S·HClDegré de pureté :99.8%Couleur et forme :SolidMasse moléculaire :388.95Ipragliflozin (L-Proline)
CAS :Ipragliflozin is a highly potent and selective SGLT2 inhibitor with an IC50 of 2.8 nM; little and NO potency for SGLT1/3/4/5/6.Formule :C26H30FNO7SCouleur et forme :SolidMasse moléculaire :519.58Bromperidol hydrochloride
CAS :Bromperidol hydrochloride is a D2 dopamine receptor antipsychotic; enhances Spectinomycin's mycobactericidal effects.Formule :C21H24BrClFNO2Couleur et forme :SolidMasse moléculaire :456.78Glucagon (1-29), bovine, human, porcine
CAS :Corynoxine B (Cory B) is a naturally occurring alkaloid isolated from Uncaria rhynchophylla (Miq. ) and is an autophagy inducer.Formule :C153H225N43O49SDegré de pureté :99.56% - 99.91%Couleur et forme :SolidMasse moléculaire :3482.75Clozapine-d8
CAS :Clozapine-d8 is a deuterium-labeled analog of Clozapine, used as an internal standard for mass spectrometric analysis of this atypical antipsychotic.Formule :C18H19ClN4Couleur et forme :SolidMasse moléculaire :334.87Agomelatine-d6
CAS :Agomelatine D6 (S-20098 D6) is a deuterium-labeled Agomelatine. Agomelatine is a specific agonist of MT1 and MT2 receptors.Formule :C15H17NO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :249.345-HT3 antagonist 5
CAS :5-HT3 antagonist 5, a quinoxalin-2-carboxamide, blocks 5-HT3 receptors and has antidepressant effects in mice.Formule :C16H13N3O2Degré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :279.29Quetiapine-d4 hemifumarate
CAS :Quetiapine D4 hemifumarate is the deuterium labeled Quetiapine hemifumarate. Quetiapine hemifumarate is a agonist of 5-HT receptors and a antagonist of dopamine receptor,with ntidepressant and anxiolytic.Formule :C25H29N3O6SDegré de pureté :98%Couleur et forme :White SolidMasse moléculaire :503.61SYL-4
CAS :SYL-4 is a potential P2Y12 receptor antagonist with a Ki value of 7.35 ± 1.72 for use in synthetic dyes.Formule :C20H15N3O5SDegré de pureté :95.76%Couleur et forme :SoildMasse moléculaire :409.42Agomelatine (L(+)-Tartaric acid)
CAS :Agomelatine (L(+)-Tartaric acid) is an MT1/MT2 agonist and selective 5-HT2C antagonist, supporting melatonergic and serotonergic signaling studies in neuroscience.Formule :C19H23NO8Degré de pureté :99.79%Couleur et forme :SolidMasse moléculaire :393.39BMS-986224
CAS :BMS-986224 is an orally active, potent and selective APJ receptor agonist.BMS-986224 is a candidate compound for the treatment of heart failure.
Formule :C24H23ClN4O6Degré de pureté :98.61% - 99.67%Couleur et forme :SolidMasse moléculaire :498.92cis-(Z)-Flupentixol dihydrochloride
CAS :cis-(Z)-Flupentixol dihydrochloride (Emergil) is a dopamine receptor antagonist.Formule :C23H27Cl2F3N2OSDegré de pureté :98.07%Couleur et forme :SolidMasse moléculaire :507.44Pramipexole dihydrochloride
CAS :Pramipexole dihydrochloride could be used to treat Parkinson disease.Formule :C10H18ClN3SDegré de pureté :98%Couleur et forme :White Crystalline PowderMasse moléculaire :247.79L-798106
CAS :L-798106 (CM9) is an EP3 receptor antagonist that inhibits EP4, EP1, and EP2 receptors and attenuates PGE2-induced cough.Formule :C27H22BrNO4SDegré de pureté :98.97%Couleur et forme :SolidMasse moléculaire :536.44Omidenepag
CAS :Omidenepag (UR-7276) is an EP2 agonist and a novel topical ocular hypotensive agent.Omidenepag can be used to study glaucoma and hypertension.Formule :C23H22N6O4SDegré de pureté :99.67% - 99.77%Couleur et forme :SolidMasse moléculaire :478.52LAS101057
CAS :LAS101057 is a novel orally available and potent and selective A2B receptor antagonist for the study of asthma.Formule :C18H14FN5ODegré de pureté :99.03% - >99.99%Couleur et forme :SolidMasse moléculaire :335.34(Rac)-Rotigotine hydrochloride
CAS :(Rac)-Rotigotine hydrochloride is a racemate of Rotigotine. Rotigotine is a full agonist of dopamine receptor, a partial the 5-HT1A receptor agonist.Formule :C19H26ClNOSCouleur et forme :SolidMasse moléculaire :351.93PD176252
CAS :PD176252 is a BB1 and BB2 antagonist, GRPR inhibitor, and FPR1/FPR2 agonist that inhibits the growth and proliferation of a wide range of cancer cells.Formule :C32H36N6O5Degré de pureté :99.00%Couleur et forme :SolidMasse moléculaire :584.67V-0219
CAS :V-0219 is a positive allosteric modulator of GLP-1 and can be used in studies about obesity-associated diabetes.Formule :C20H25F3N4O2Degré de pureté :99.91%Couleur et forme :SoildMasse moléculaire :410.43WAY-100635
CAS :WAY-100635 is a potent 5-HT 1A receptor antagonist pyramidal neuron firing frequency during conditioned reflexes; a dopamine D4 receptor agonist .Formule :C25H34N4O2Degré de pureté :98.972%Couleur et forme :SolidMasse moléculaire :422.563-Hydroxy agomelatine
CAS :3-Hydroxy agomelatine (3-Hydroxyagomelatine) is a 5-HT2C receptor antagonist used in the study of neurological disorders.Formule :C15H17NO3Couleur et forme :SolidMasse moléculaire :259.3Sumanirole maleate
CAS :Sumanirole maleate (PNU-95666E) is a D2 receptor full agonist with high selectivity that plays a vital role in Parkinson's disease and restless leg syndrome.Formule :C15H17N3O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :319.31Telcagepant
CAS :Telcagepant (MK-0974) is an oral calcitonin gene-related peptide receptor (CGRP) antagonist that blocks CGRP receptors, migraines and for pain relief.Formule :C26H27F5N6O3Degré de pureté :98.98% - 98.98%Couleur et forme :SolidMasse moléculaire :566.52PSB-0739
CAS :PSB-0739 Selective platelet P2Y12 receptor antagonist characterized by competitive binding with antithrombotic and platelet aggregation modulating effects.Formule :C26H17N3Na2O8S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :609.54Mozavaptan hydrochloride
CAS :Mozavaptan is a vasopressin receptor antagonist.Formule :C27H30ClN3O2Couleur et forme :SolidMasse moléculaire :464Paliperidone Palmitate
CAS :Paliperidone: atypical antipsychotic, dopamine & serotonin antagonist, affects α1/α2 adrenergic and H1 histamine receptors.Formule :C39H57FN4O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :664.89Cetirizine D8
CAS :Cetirizine D8 is a deuterium-labeled Cetirizine. Cetirizine is a second-generation antihistamine and a long-acting histamine H1-receptor antagonist.Formule :C21H25ClN2O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :396.943-Hydroxy agomelatine D3
CAS :3-Hydroxy agomelatine D3 is a deuterated metabolite of Agomelatine and a 5-HT2C antagonist (IC50: 3.2 μM, Ki: 1.8 μM).Formule :C15H17NO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :262.32Levomepromazine
CAS :Levomepromazine (Methotrimeprazine) is a Ca2+ release inducer with antiviral, anti-inflammatory, neuroprotective, sedative, and anti-nociceptive activities.Formule :C19H24N2OSDegré de pureté :99.15%Couleur et forme :SolidMasse moléculaire :328.47Pimozide-d4
CAS :Pimozide D4 is a deuterium labeled Pimozide.Formule :C28H29F2N3ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :465.57ST-836 hydrochloride
CAS :ST-836 hydrochloride is a dopamine receptor ligand; Antiparkinsonian agent .Formule :C23H35ClN4OSDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :451.07(S)-(+)-Dimethindene maleate
CAS :(S)-(+)-Dimethindene maleate is an orally available, selective muscarinic M2 receptor and histamine H1 receptor antagonist that inhibits muscarinic M1 receptorsFormule :C24H28N2O4Degré de pureté :99.94%Couleur et forme :SolidMasse moléculaire :408.49Levosalbutamol Hydrochloride
CAS :Levosalbutamol Hydrochloride is a β2-adrenergic receptor agonist. It is used to treat asthma and chronic obstructive pulmonary disease.Formule :C13H22ClNO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :275.77Haloperidol (D4')
CAS :Haloperidol D4' is deuterium-labeled haloperidol. Haloperidol is a dopamine D2 receptor antagonist.Formule :C21H23ClFNO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :379.89Ramelteon-d5
CAS :Ramelteon-d5 is a deuterated compound of Ramelteon.Formule :C16H16D5NO2Couleur et forme :SolidMasse moléculaire :264.37Cimbuterol-d9
CAS :Cimbuterol-d9 is a deuterated compound of Cimbuterol.Formule :C13H10D9N3ODegré de pureté :99.22%Couleur et forme :SolidMasse moléculaire :242.37YNT-185 dihydrochloride
CAS :Potent OX2 agonist (EC50=28nM); 100x selective over OX1; prompts wakefulness, counters cataplexy in mice.Formule :C33H39Cl2N5O5SCouleur et forme :SolidMasse moléculaire :688.67Tiapride-d3
Tiapride-d3 is a deuterated form of Tiapride, a selective dopamine D2 receptor antagonist and an antipsychotic compound.Formule :C15H21D3N2O4SCouleur et forme :SolidMasse moléculaire :331.45Zilpaterol-d7
CAS :Zilpaterol-d7 (trans-(±)-Zilpaterol-d7) is a deuterium-labeled version of Zilpaterol, a β-adrenergic receptor agonist.Formule :C14H12D7N3O2Couleur et forme :SolidMasse moléculaire :268.36GSK682753A
CAS :GSK682753A is a selective and highly potent inverse agonist of the epstein-barr virus-induced receptor 2 (EBI2; IC50: 53.6 nM).Formule :C23H21Cl3N2O3Couleur et forme :SolidMasse moléculaire :479.78Cudarolimab
CAS :Cudarolimab (IBI-101) is a fully human anti-OX40 antibody with potential immune checkpoint inhibitory and anti-tumor activity for the study of cancer.Degré de pureté :97.5% (SDS-PAGE); 98.2% (SEC-HPLC) - 97.5% (SDS-PAGE); 98.2% (SEC-HPLC)Couleur et forme :LiquidMasse moléculaire :145.67 kDa5-HT2B antagonist-1
CAS :Orally active 5-HT2B antagonist; IC50 = 33.4 nM; potential for hepatocellular, cardiovascular, GI disease research.Formule :C11H14BrN5Degré de pureté :99.965%Couleur et forme :SolidMasse moléculaire :296.17LY223982
CAS :LY223982 is an effective and specific inhibitor of the leukotriene B4 receptor (IC50: 13.2 nM). It also can against [3H]LTB4 binding to LTB4 receptor.Formule :C30H30O7Degré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :502.56Ozagrel Sodium
CAS :Ozagrel Sodium is a thromboxane A2 synthase inhibitor. It is used to treat cerebrovascular diseases.Formule :C13H12N2NaO2Degré de pureté :98%Couleur et forme :White Or Off-White Crystalline PowderMasse moléculaire :251.24LUF5771
CAS :LUF5771: potent allosteric recLH & Org 43553 inhibitor, partial LH receptor activator with low efficacy.Formule :C24H23NO2Couleur et forme :SolidMasse moléculaire :357.44NAV-2729
CAS :NAV-2729 inhibits six ArfGEFs (human ARNO, EFA6, BIG1, and BRAG2 and Legionella and Rickettsia RalF), the strongest effects being against BRAG2, Arf1 and Arf6.Formule :C25H17ClN4O3Degré de pureté :98.83% - 98.91%Couleur et forme :SolidMasse moléculaire :456.88Ref: TM-T5142
2mg43,00€5mg63,00€1mL*10mM (DMSO)71,00€10mg90,00€25mg193,00€50mg286,00€100mg429,00€500mg888,00€Escitalopram Oxalate
CAS :Escitalopram Oxalate ((S)-(+)Citalopram oxalate) is a selective serotonin (5-HT) reuptake inhibitor (SSRI) with Ki of 0.89 nM.Formule :C22H23FN2O5Degré de pureté :97.39% - 99.73%Couleur et forme :White SolidMasse moléculaire :414.43Ref: TM-T6493
10mg37,00€1mL*10mM (DMSO)42,00€25mg52,00€50mg63,00€100mg86,00€200mg118,00€500mg187,00€1g268,00€Terazosin
CAS :Terazosin: oral α1-blocker, relaxes blood vessels, treats BPH and hypertension.Formule :C19H25N5O4Couleur et forme :SolidMasse moléculaire :387.43S26131
CAS :S26131 (N-[2-[7-[3-[8-(2-acetamidoethyl)naphthalen-2-yl]oxypropoxy]naphthalen-1-yl]ethyl]acetamide) behaves as an antagonist on MT1 and MT2 receptors with Ki ofFormule :C31H34N2O4Degré de pureté :99.77%Couleur et forme :SolidMasse moléculaire :498.61MK-2894 sodium salt
CAS :MK-2894 sodium salt is a highly potent and selective antagonist of second generation EP4.Formule :C25H22F3NNaO3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :496.5Icatibant Acetate
CAS :Icatibant Acetate, an antagonist of the bradykinin B2 receptor, is used in the treatment of hereditary angioedema.Formule :C61H93N19O15SDegré de pureté :99.68% - 99.90%Couleur et forme :SolidMasse moléculaire :1364.57Ref: TM-T22344
1mg66,00€2mg92,00€5mg177,00€10mg281,00€1mL*10mM (DMSO)355,00€25mg475,00€50mg677,00€100mg888,00€[Sar9,Met(O2)11]-Substance P
CAS :[Sar9,Met(O2)11]-Substance P (NA) is an agonist of NK1 receptor.Formule :C64H100N18O15SDegré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :1393.66Triprolidine
CAS :Triprolidine: oral H1 receptor blocker with motor/sensory spinal effects, for allergy research.Formule :C19H22N2Couleur et forme :SolidMasse moléculaire :278.39GR 94800 acetate
GR 94800 acetate is a potent and selective neurokinin 2(NK-2) antagonist.
Formule :C51H65N9O10Degré de pureté :97.86%Couleur et forme :SolidMasse moléculaire :964.12Zuclopenthixol dihydrochloride
CAS :Zuclopenthixol dihydrochloride is an D1 and D2 dopamine receptors antagonist.Formule :C22H27Cl3N2OSDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :473.89Buclizine dihydrochloride
CAS :Buclizine dihydrochloride (Buclina) is the hydrochloride salt form of buclizine, a piperazine histamine H1 receptor antagonist with primarily antiemetic andFormule :C28H33ClN2·2HClDegré de pureté :98.05%Couleur et forme :Off-White PowderMasse moléculaire :505.95CID 1375606
CAS :CID 1375606: Surrogate agonist for GPR27, conserved in vertebrates, mainly in CNS.Formule :C20H14Cl2N2O2Degré de pureté :99.41%Couleur et forme :SolidMasse moléculaire :385.24TFLLR-NH2 2TFA(197794-83-5(free base))
TFLLR-NH2 2TFA(197794-83-5(free base)) is an agonist of PAR1 (EC50 :1.9 μM).Formule :C35H55F6N9O10Degré de pureté :99.56%Couleur et forme :SolidMasse moléculaire :875.87Neuropeptide S (Mouse) acetate
Neuropeptide S (Mouse) acetate is a bioactive peptide.Formule :C95H160N34O29Degré de pureté :98.25%Couleur et forme :SolidMasse moléculaire :2242.5Mizagliflozin
CAS :Mizagliflozin is an orally active, selective SGLT1 inhibitor with a Ki value of 27 nM for human SGLT1.Cost-effective and quality-assured.Formule :C28H44N4O8Degré de pureté :98.66% - 99.67%Couleur et forme :SolidMasse moléculaire :564.67Ref: TM-T16083
1mg66,00€2mg96,00€5mg144,00€1mL*10mM (DMSO)173,00€10mg227,00€25mg455,00€50mg645,00€100mg938,00€200mg1.264,00€Diclofensine hydrochloride
CAS :Diclofensine hydrochloride (Ro 8-4650 hydrochloride) 是一种高效单胺再摄取抑制剂，在大鼠脑突触体中能够阻断多巴胺 (IC50=0.74 nM)、去甲肾上腺素 (IC50=2.3 nM) 和 5-羟色胺 (IC50=3.7 nM)。Formule :C17H18Cl3NODegré de pureté :98.86% - 99.93%Couleur et forme :SolidMasse moléculaire :358.69Chlorpheniramine
CAS :Chlorpheniramine is an H1 anti-histamine agent for IgE-mediated inflammation that is commonly used for allergic diseases.Formule :C16H19ClN2Couleur et forme :SolidMasse moléculaire :274.79Betahistine EP Impurity C
CAS :Betahistine EP Impurity C (NSC19005) is structurally related to Betahistine. Betahistine EP Impurity C is a dimer of Betahistine.Formule :C15H19N3Degré de pureté :99.93% - ≥95%Couleur et forme :SolidMasse moléculaire :241.33Tetracosactide
CAS :Tetracosactide, a synthetic peptide, mirrors the 24-amino acid start of ACTH with sequence SYSMEHFRWGKPVGKKRRPVKVYP.Formule :C136H210N40O31SDegré de pureté :99.91%Couleur et forme :SolidMasse moléculaire :2933.44Ralmitaront
CAS :Ralmitaront (RO6889450) is a potent, orally active partial agonist of the trace amine-associated receptor 1 (TAAR1).Formule :C17H22N4O2Degré de pureté :99.71% - 99.79%Couleur et forme :SolidMasse moléculaire :314.38Ref: TM-T9183
1mg105,00€5mg260,00€1mL*10mM (DMSO)286,00€10mg401,00€25mg668,00€50mg897,00€100mg1.243,00€200mg1.693,00€RO 46-8443
CAS :RO 46-8443: First non-peptide ETB receptor antagonist, >2000-fold ETB selectivity in binding and function.Formule :C31H35N3O8SDegré de pureté :98.77% - 99.77%Couleur et forme :SolidMasse moléculaire :609.69GSK189254A
CAS :GSK189254A (GSK189254) is a potent and specific histamine H3 receptor antagonist (pKi values: 9.59-9.90 and 8.51-9.17 for human and rat H3).Formule :C21H25N3O2Degré de pureté :98.71% - 99.858%Couleur et forme :SolidMasse moléculaire :351.44Ref: TM-TQ0066
1mg50,00€1mL*10mM (DMSO)64,00€5mg84,00€10mg114,00€25mg205,00€50mg333,00€100mg477,00€200mg690,00€Adoprazine hydrochloride
CAS :Adoprazine hydrochloride is a dopamine D2 receptor antagonist and 5-HT1A receptor agonist potential antipsychotic drug.Formule :C24H25ClFN3O2Couleur et forme :SolidMasse moléculaire :441.93FAUC 346
CAS :FAUC 346 is a highly selective D3 partial agonist with EC50 of 1.5 nM.Formule :C24H29N3O2SDegré de pureté :99.46%Couleur et forme :SolidMasse moléculaire :423.57Ref: TM-T9081
2mg34,00€5mg50,00€1mL*10mM (DMSO)52,00€10mg77,00€25mg138,00€50mg224,00€100mg359,00€200mg490,00€AdipoRon
CAS :AdipoRon (SC-396658) is an orally bioavailable adiponectin receptor agonist. It can combine with AdipoR1/2 (KD: 1.8/3.1 μM).Formule :C27H28N2O3Degré de pureté :97.90% - 99.86%Couleur et forme :SolidMasse moléculaire :428.52Ref: TM-T2257
5mg34,00€10mg50,00€1mL*10mM (DMSO)55,00€25mg102,00€50mg161,00€100mg203,00€200mg264,00€500mg445,00€1g647,00€SRI-37330 hydrochloride
CAS :SRI-37330 hydrochloride is an orally active thioredoxin-interacting protein (TXNIP) inhibitor. hydrochloride can be used to study type 2 diabetes.Formule :C16H20ClF3N4O2SCouleur et forme :SolidMasse moléculaire :424.87Pizuglanstat
CAS :Pizuglanstat is a hematopoietic prostaglandin synthase inhibitor.Formule :C27H36N6O4Degré de pureté :99.62%Couleur et forme :SolidMasse moléculaire :508.61Nefazodone hydrochloride
CAS :Nefazodone hydrochloride (Serzone) is a serotoninergic modulating antidepressant that is used in therapy of depression, aggressive behavior and panic disorder.Formule :C25H33Cl2N5O2Degré de pureté :99% - 99.86%Couleur et forme :White SolidMasse moléculaire :506.47Ref: TM-T3275
5mg47,00€10mg70,00€1mL*10mM (DMSO)77,00€25mg120,00€50mg216,00€100mg325,00€200mg472,00€500mg775,00€Myristicin
CAS :Myristicin is a natural spice extract with antibacterial, anti-inflammatory, and hepatoprotective properties, and can induce apoptosis.
Formule :C11H12O3Degré de pureté :99.828%Couleur et forme :LiquidMasse moléculaire :192.21Mini Gastrin I, human acetate
Mini Gastrin I, human acetate is a shorter version of human gastrin, consists of amino acids 5-17 of the parent peptide.Formule :C76H103N15O28SDegré de pureté :99.35% - 99.82%Couleur et forme :SolidMasse moléculaire :1706.78Taminadenant mesylate
CAS :Taminadenant (PBF-509/NIR-178) is an oral adenosine A2A receptor antagonist that activates T-cells to target tumor cells.Formule :C11H12BrN7O3SCouleur et forme :SolidMasse moléculaire :402.227Ajmalicine hydrochloride
CAS :Ajmalicine hydrochloride is a potent α1-adrenoceptor blocker, non-competitive nicotine receptor inhibitor, anti-hypertensive, and sedative. IC50: 72.3 μM.Formule :C21H25ClN2O3Couleur et forme :SolidMasse moléculaire :388.89SCH-37370
CAS :SCH-37370 is an effective and orally active dual antagonist of platelet-activating factor and histamine.Formule :C21H21ClN2ODegré de pureté :99.07%Couleur et forme :SolidMasse moléculaire :352.86Ref: TM-T19686
1mg46,00€5mg85,00€1mL*10mM (DMSO)86,00€10mg109,00€25mg185,00€50mg275,00€100mg371,00€200mg494,00€JD-5037
CAS :JD-5037 is a novel, peripherally restricted CB1R antagonist with an IC50 of 1.5 nM.Formule :C27H27Cl2N5O3SDegré de pureté :99.54% - 99.84%Couleur et forme :SolidMasse moléculaire :572.51Ref: TM-T4453
1mg42,00€2mg55,00€5mg90,00€1mL*10mM (DMSO)101,00€10mg133,00€25mg234,00€50mg350,00€100mg522,00€[Lys5,MeLeu9,Nle10]-NKA(4-10)
CAS :Highy selective and potent NK2 receptor agonist (IC50 = 6.1 nM). Induces contraction of the rat fundus and bladder (EC50 values are 117 and 10 nM respectively).Formule :C39H65N9O9Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :803.99
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