GPCR/G-Protéine
Les inhibiteurs des GPCR/protéines G sont des composés qui ciblent les récepteurs couplés aux protéines G (GPCR) et les protéines G associées, qui jouent un rôle crucial dans la transmission des signaux de l'extérieur vers l'intérieur des cellules. Ces inhibiteurs sont essentiels pour étudier les voies de signalisation médiées par les GPCR, impliquées dans de nombreux processus physiologiques, y compris la perception sensorielle, la réponse immunitaire et la neurotransmission. Les inhibiteurs des GPCR sont également importants dans le développement de médicaments, car de nombreux agents thérapeutiques ciblent ces récepteurs. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de GPCR/protéines G de haute qualité pour soutenir vos recherches en pharmacologie, biologie cellulaire et domaines connexes.
Sous-catégories appartenant à la catégorie "GPCR/G-Protéine"
- récepteur 5-HT(1.025 produits)
- Récepteur d'adénosine(249 produits)
- Récepteur adrénergique(3.023 produits)
- Récepteur de la bombésine(35 produits)
- Récepteur de la bradykinine(61 produits)
- CXCR(158 produits)
- CaSR(34 produits)
- Récepteur cannabinoïde(217 produits)
- Cholécystokinine(1 produits)
- Récepteur de la dopamine(445 produits)
- Récepteur de l'endothéline(86 produits)
- Récepteur GNRH(84 produits)
- GPCR19(33 produits)
- GRK(33 produits)
- GTPase(23 produits)
- Récepteur du glucagon(194 produits)
- Hérisson/Smoothened(49 produits)
- Récepteur de l'histamine(385 produits)
- Récepteur LPA(21 produits)
- Récepteur de la mélatonine(26 produits)
- Récepteur OX(41 produits)
- Récepteur opioïde(327 produits)
- PAFR(14 produits)
- PKA(60 produits)
- Récepteur S1P(18 produits)
- SGLT(31 produits)
- Récepteur Sigma(46 produits)
Affichez 19 plus de sous-catégories
5986 produits trouvés pour "GPCR/G-Protéine"
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Physalaemin acetate
Physalaemin acetate is a non-mammalian tachykinin with high affinity when binding selectively to neurokinin-1 (NK1) receptor.Formule :C60H88N14O18SDegré de pureté :99.13%Couleur et forme :SolidMasse moléculaire :1325.49Tofogliflozin (hydrate)
CAS :Tofogliflozin hydrate (CSG-452 hydrate) is a potent and highly specific inhibitor of SGLT2(Ki of 2.9 nM, 14.9 nM, and 6.4 nM for human, rat, and mouse SGLT2).Formule :C22H28O7Degré de pureté :97.03% - 98.78%Couleur et forme :SolidMasse moléculaire :404.45Ref: TM-T5016
1mg35,00€2mg49,00€5mg74,00€1mL*10mM (DMSO)82,00€10mg109,00€25mg202,00€50mg324,00€100mg505,00€200mg717,00€Triptorelin acetate(57773-63-4 free base)
CAS :Triptorelin acetate is a GnRH agonist for hormone-responsive cancers, precocious puberty, and assisted reproduction.Formule :C66H86N18O15Degré de pureté :99.59% - 99.90%Couleur et forme :White PowderMasse moléculaire :1371.53Ref: TM-T21410
5mg52,00€10mg78,00€1mL*10mM (DMSO)116,00€25mg119,00€50mg172,00€100mg259,00€200mg388,00€Myristicin
CAS :Myristicin is a natural spice extract with antibacterial, anti-inflammatory, and hepatoprotective properties, and can induce apoptosis.
Formule :C11H12O3Degré de pureté :99.828%Couleur et forme :LiquidMasse moléculaire :192.21GR 94800 acetate
GR 94800 acetate is a potent and selective neurokinin 2(NK-2) antagonist.
Formule :C51H65N9O10Degré de pureté :97.86%Couleur et forme :SolidMasse moléculaire :964.12Hypidone hydrochloride
CAS :Hypidone hydrochloride (YL0919) is a novel antidepressant candidate with dual activity as a 5-HT1A receptor agonist and a selective serotonin reuptake inhibitorFormule :C18H23ClN2O2Degré de pureté :99.82% - 99.93%Couleur et forme :SolidMasse moléculaire :334.84Acrivastine
CAS :Acrivastine (Acrivastin) is a short-acting histamine 1 receptor antagonist.Formule :C22H24N2O2Degré de pureté :99.73% - >99.99%Couleur et forme :SolidMasse moléculaire :348.44Protease-Activated Receptor-4 diTFA
Protease-Activated Receptor-4 diTFA,2454 is the proteinase-activated receptor-4 (PAR4)agonistFormule :C37H48F6N8O11Degré de pureté :98.54%Couleur et forme :SolidMasse moléculaire :894.81Ref: TM-T7740
1mg46,00€2mg57,00€5mg81,00€10mg131,00€1mL*10mM (DMSO)161,00€25mg259,00€50mg389,00€100mg575,00€BML-190
CAS :BML-190 (Indomethacin morpholinylamide) 是一种 CB2 受体的配体，其对 CB2 受体 (Ki:435 nM) 和 CB1受体 (Ki> 2 μM)。Formule :C23H23ClN2O4Degré de pureté :97.70%Couleur et forme :SolidMasse moléculaire :426.89(±)-Ibipinabant
CAS :(±)-Ibipinabant ((±)-SLV319) has been used in trials studying the treatment of Obesity and Obesity and Type 2 Diabetes.Formule :C23H20Cl2N4O2SDegré de pureté :99.28% - 99.83%Couleur et forme :SolidMasse moléculaire :487.4Glucagon-like peptide 1 (1-37), human acetate
Glucagon-like peptide 1 (1-37), human acetate is a highly potent the GLP-1 receptor agonist.Degré de pureté :98%Couleur et forme :LiquidMasse moléculaire :N/AOxyntomodulin acetate
Oxyntomodulin acetate, a 37-amino acid peptide hormone, is a glucagon-like peptide 1 (GLP-1) receptor agonist[1].Degré de pureté :99.24%Couleur et forme :LiquidMasse moléculaire :N/ABRL 54443
CAS :BRL 54443 is a potent 5-HT1E/1F receptor agonist (pKi values are 8.7 and 8.9 respectively).Formule :C14H18N2ODegré de pureté :98.07%Couleur et forme :SolidMasse moléculaire :230.31BIBO3304
CAS :BIBO3304: Selective NPY Y1 blocker, IC50 of 0.38nM (human), 0.72nM (rat); curbs hunger from NPY/fasting when injected centrally.Formule :C29H35N7O3Couleur et forme :SolidMasse moléculaire :529.63Ufenamate
CAS :Ufenamate (Flufenamic acid butyl ester) is an anthranilic acid-based anti-inflammatory drug developed for skin diseasesFormule :C18H18F3NO2Degré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :337.34Pergolide mesylate
CAS :Pergolide mesylate (LY127809), a dopamine agonist for Parkinson's and hyperprolactinemia, was withdrawn for heart valve risk.Formule :C20H30N2O3S2Degré de pureté :99.70%Couleur et forme :White To Off-White SolidMasse moléculaire :410.59Cutamesine dihydrochloride
CAS :Cutamesine dihydrochloride is a σ1 receptor agonist, selective over σ2, combating cardiomyocyte hypertrophy and improving stroke recovery.Formule :C23H32N2O2·2HClDegré de pureté :99.96%Couleur et forme :SolidMasse moléculaire :441.43Ref: TM-T3597
2mg34,00€5mg50,00€1mL*10mM (DMSO)55,00€10mg86,00€25mg167,00€50mg260,00€100mg401,00€200mg580,00€Maropitant
CAS :Maropitant is a selective neurokinin (NK1) receptor antagonist.Formule :C32H40N2ODegré de pureté :97.35% - 99.75%Couleur et forme :SolidMasse moléculaire :468.67α-MSH
CAS :α-MSH (MSH, amide) is amide stimulates melanocortin 1 receptor that results in the activation of adenylyl cyclase.Formule :C77H109N21O19SDegré de pureté :99.10% - 99.67%Couleur et forme :White PowderMasse moléculaire :1664.89CID 16020046
CAS :CID 16020046 (C390-0219) is a selective GPR55 antagonist, inhibiting GPR55 constitutive activity with IC50 of 0.15 μM in yeast.Formule :C25H19N3O4Degré de pureté :99.03%Couleur et forme :SolidMasse moléculaire :425.44NIBR189
CAS :NIBR189 is a potent and selective antagonist of EBI2 (GPR183) receptor (IC50 of 11 and 15 nM for human and mouse EBI2 receptors, respectively)Formule :C21H21BrN2O3Degré de pureté :97%Couleur et forme :ColourlessMasse moléculaire :429.31PNU 22394 hydrochloride
CAS :PNU 22394 hydrochloride is a 5-HT2C agonist and partial 5-HT2A/5-HT2B agonistFormule :C13H17ClN2Degré de pureté :97.83%Couleur et forme :SolidMasse moléculaire :236.74Alcaftadine
CAS :Alcaftadine (Lastacaft) is an H1 histamine receptor antagonist indicated for the prevention of itching associated with allergic conjunctivitis.Formule :C19H21N3ODegré de pureté :98% - 98.65%Couleur et forme :SolidMasse moléculaire :307.39[D-Trp8]-γ-MSH acetate(321351-81-9 free base)
[D-Trp8]-γ-MSH acetate(321351-81-9 free base) is a selective melanocortin 3 (MC3) receptor agonist (IC50 values are 6.7, 340 and 600 nM for human MC3, MC5 andFormule :C76H103N21O18SDegré de pureté :99.75%Couleur et forme :SolidMasse moléculaire :1630.82PAR-2-IN-1
CAS :PAR-2-IN-1 (IUN76750) is a PAR- 2 signaling pathway inhibitor with anti-inflammatory and anticancer effects.Formule :C12H14ClN3O2Degré de pureté :99.75%Couleur et forme :SolidMasse moléculaire :267.71Ref: TM-T8917
2mg34,00€5mg50,00€1mL*10mM (DMSO)52,00€10mg86,00€25mg161,00€50mg243,00€100mg355,00€200mg502,00€Bosentan (hydrate)
CAS :Bosentan hydrate (Ro 47-0203) is a competitive and dual antagonist of endothelin-1 at the endothelin-A (ET-A) and endothelin-B (ET-B) receptors.Formule :C27H29N5O6S·H2ODegré de pureté :99.31% - 99.86%Couleur et forme :White PowderMasse moléculaire :569.63Bexagliflozin
CAS :Bexagliflozin (EGT1442) is a potent, selective sodium glucose co-transporter 2 (SGLT2) inhibitor with IC50 values of 2 nM for human SGLT2.Formule :C24H29ClO7Degré de pureté :98.99% - 99.89%Couleur et forme :SolidMasse moléculaire :464.94Ref: TM-T7217
1mg67,00€2mg95,00€5mg129,00€1mL*10mM (DMSO)137,00€10mg187,00€25mg371,00€50mg552,00€100mg785,00€GW 405833
CAS :GW 405833 (L-768242) is an agonist of cannabinoid-2 (CB(2)) receptor-selectiveFormule :C23H24Cl2N2O3Degré de pureté :99.82% - 99.93%Couleur et forme :SolidMasse moléculaire :447.35Epinastine
CAS :Epinastine (WAL801) is an antihistamine, mast cell stabilizer, and H1 antagonist with anti-allergic properties.Formule :C16H15N3Degré de pureté :99.94%Couleur et forme :SolidMasse moléculaire :249.316-fluoro-DL-Tryptophan
CAS :6-fluoro-DL-Tryptophan is an inhibitor of serotonin (5-HT) synthesis.Formule :C11H11FN2O2Degré de pureté :99.25%Couleur et forme :Off-White PowderMasse moléculaire :222.22HS 014 acetate(207678-81-7 free base)
HS 014 acetate is a potent MC4R antagonist with Ki: 3.16 nM (MC4), and boosts food intake and nociception in animals.Formule :C73H98N20O19S2Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :1623.83Sertindole
CAS :Sertindole, atypical antipsychotic, targets D2, 5-HT1D, 5-HT2A, 5-HT2C receptors (Kds: 2.7, 20, 0.14, 6 nM).Formule :C24H26ClFN4ODegré de pureté :99.87% - 99.92%Couleur et forme :Off-White To Pale Yellow SolidMasse moléculaire :440.94GLPG2938
CAS :GLPG2938 (1-(2-Ethoxy-6-(trifluoromethyl)pyridin-4-yl)-3-((5-methyl-6-(1-methyl-3-(trifluoromethyl)-1H-pyrazol-4-yl)pyridazin-3-yl)methyl)urea) is a potent andFormule :C20H19F6N7O2Degré de pureté :98.25%Couleur et forme :SolidMasse moléculaire :503.4Ref: TM-T9199
1mg79,00€2mg92,00€5mg137,00€1mL*10mM (DMSO)152,00€10mg236,00€25mg520,00€50mg750,00€100mg1.035,00€Dioxopromethazine hydrochloride
CAS :Dioxopromethazine is a target-based classification of drug and available in a number of countries worldwide.Formule :C17H20N2O2S·HClDegré de pureté :99.58%Couleur et forme :SolidMasse moléculaire :352.88Nomifensine
CAS :Nomifensine ((±)-Nomifensin) is a norepinephrine-dopamine reuptake inhibitor that prevents dopamine reuptake into synaptosomes.Formule :C16H18N2Degré de pureté :99.83% - ≥95%Couleur et forme :SolidMasse moléculaire :238.33A-582941 dihydrochloride
CAS :A-582941 dihydrochloride (A 582941) is a Selective agonist of α7 nAChR partialFormule :C17H22Cl2N4Degré de pureté :99.55%Couleur et forme :SolidMasse moléculaire :353.29Ref: TM-T22016
1mg42,00€1mL*10mM (DMSO)87,00€5mg88,00€10mg120,00€25mg235,00€50mg354,00€100mg533,00€200mg743,00€Elagolix sodium
CAS :Elagolix sodium (NBI-56418 sodium) is a GnRH receptor (GnRHR) antagonist ( IC50 and Ki of 0.25 and 3.7 nM, respectively).Formule :C32H29F5N3NaO5Degré de pureté :99.71%Couleur et forme :SolidMasse moléculaire :653.57Ref: TM-T5031
2mg35,00€5mg52,00€1mL*10mM (DMSO)74,00€10mg80,00€25mg144,00€50mg227,00€100mg359,00€200mg532,00€Bimatoprost
CAS :Bimatoprost (AGN 192024) is a cloprostenol-derived amide that is used as an antihypertensive agent in the treatment of open-angle glaucoma and ocularFormule :C25H37NO4Degré de pureté :98% - >99.99%Couleur et forme :Crystalline SolidMasse moléculaire :415.57Ref: TM-T2538
2mg34,00€5mg48,00€1mL*10mM (DMSO)50,00€10mg75,00€25mg127,00€50mg219,00€100mg371,00€200mg547,00€Neuromedin N acetate(92169-45-4 free base)
Neuromedin N acetate(92169-45-4 free base) is a neuropeptide derived from the same precursor polypeptide as neurotensin, and with similar but subtly distinctFormule :C40H67N7O10Degré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :805.9Chlorphenoxamine
CAS :Chlorphenoxamine (Contristamine) is an antihistamine and anticholinergic used as an antipruritic and antiparkinsonian agent.Formule :C18H22ClNODegré de pureté :99.44% - 99.85%Couleur et forme :SolidMasse moléculaire :303.83Ref: TM-T7564
2mg35,00€5mg51,00€1mL*10mM (DMSO)63,00€10mg81,00€25mg106,00€50mg147,00€100mg207,00€200mg306,00€UFP 803 acetate
UFP 803 acetate is a potent ligand of urotensin-II (UT) receptor. UFP-803 displays the activity of a lower residual agonist.Formule :C52H68N10O14S2Degré de pureté :99.78%Couleur et forme :SolidMasse moléculaire :1121.29Vorapaxar
CAS :Vorapaxar (MK-5348) (SCH 530348) is an effective and orally active thrombin receptor (PAR-1) antagonist (Ki: 8.1 nM).Formule :C29H33FN2O4Degré de pureté :98.77% - 99.93%Couleur et forme :SolidMasse moléculaire :492.58Ref: TM-T7013
1mg71,00€5mg138,00€1mL*10mM (DMSO)152,00€10mg192,00€25mg326,00€50mg447,00€100mg642,00€200mg888,00€Octreotide Acetate
CAS :Octreotide Acetate (Sandostatin) is a potent, long-acting synthetic somatostatin octapeptide analog that inhibits secretion of growth hormone.Formule :C51H70N10O12S2Degré de pureté :99.03% - 99.87%Couleur et forme :Less To Off-White Lyophilised Solid Colourless To Off-White Lyophilised SolidMasse moléculaire :1079.30Betahistine
CAS :Betahistine treats vertigo and balance issues in Ménière's disease; it's a histamine analog and H1 receptor agonist.Formule :C8H12N2Degré de pureté :99.87% - 99.87%Couleur et forme :Yellowish Liquid Liquid LiquidMasse moléculaire :136.19Sotagliflozin
CAS :Sotagliflozin (LP-802034) is an orally bioavailable inhibitor of the sodium-glucose co-transporter subtype 1 (SGLT1) and 2 (SGLT2), with potentialFormule :C21H25ClO5SDegré de pureté :99% - 99.86%Couleur et forme :SolidMasse moléculaire :424.94Ref: TM-T3547
1mg46,00€2mg57,00€5mg87,00€1mL*10mM (DMSO)88,00€10mg131,00€25mg248,00€50mg378,00€100mg560,00€500mg1.198,00€M617 acetate
M617 acetate is a selective agonist of galanin receptor 1 (GAL1).Formule :C112H161N29O28Degré de pureté :96.02%Couleur et forme :SolidMasse moléculaire :2361.65HS024
CAS :HS024 is a highly potent melanocortin MC4 receptor antagonist, increases food intake, and blocks α-MSH- and MTII-induced hypotension and bradycardia in rats.Formule :C58H79N19O10S2Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :1266.5SB-222200
CAS :SB-222200 is a selective, reversible, and competitive antagonist of the human NK-3 receptor(Ki=4.4 nM).Formule :C26H24N2ODegré de pureté :97.13%Couleur et forme :SolidMasse moléculaire :380.48Guanabenz Acetate
CAS :Guanabenz Acetate (Wytensin) is a specific agonist of adrenergic receptor.Formule :C8H8Cl2N4·C2H4O2Degré de pureté :99% - 99.66%Couleur et forme :White Solid From Acetonitrile White SolidMasse moléculaire :291.13SKF38393 hydrobromide
CAS :SKF38393 hydrobromide is the salt form of SKF38393.a dopamine D1 receptor agonist that increases the expression of Shati/Nat8L mRNA in the NAc of mice;Formule :C16H18BrNO2Degré de pureté :98.99%Couleur et forme :SolidMasse moléculaire :336.22m-Chlorophenylbiguanide hydrochloride
CAS :m-Chlorophenylbiguanide hydrochloride is a 5-HT3 receptor agonist.Formule :C8H11Cl2N5Degré de pureté :99.43% - 99.87%Couleur et forme :SolidMasse moléculaire :248.11BQU57
CAS :BQU57 shows selective inhibition for Ral relative to Ras or Rho and inhibit xenograft tumor growth.Formule :C16H13F3N4ODegré de pureté :97.45% - 98.72%Couleur et forme :SolidMasse moléculaire :334.3[D-Phe12]-Bombesin acetate
[D-Phe12]-Bombesin acetate inhibits bombesin-stimulated secretion.Formule :C76H116N22O20SDegré de pureté :99.81%Couleur et forme :SolidMasse moléculaire :1689.94Tecadenoson
CAS :Tecadenoson (CVT-510) is a selective agonist of A1 adenosine receptor.
Formule :C14H19N5O5Degré de pureté :98.83%Couleur et forme :SolidMasse moléculaire :337.33AZD1283
CAS :AZD1283 is an effective P2Y12 receptor antagonist (EC50: 3.0 ug/kg/min, binding IC50: 11 nM).Formule :C23H26N4O5SDegré de pureté :98.37% - 99.63%Couleur et forme :SolidMasse moléculaire :470.542-Methoxyidazoxan monohydrochloride
CAS :L-Albizziin (2-Methoxyidazoxan monohydrochloride) is a highly potent selective antagonist of the alpha 2r adrenergic receptor.Formule :C12H14N2O3·HClDegré de pureté :98.99%Couleur et forme :SolidMasse moléculaire :270.72Urantide acetate(669089-53-6 free base)
Urantide acetate: selective UT receptor blocker, doesn't affect other contractions or relaxations, partial agonist in Ca²⁺ assay.Formule :C53H70N10O14S2Degré de pureté :99.22%Couleur et forme :SolidMasse moléculaire :1135.31(S)-Amisulpride
CAS :(S)-Amisulpride ((S) Amisulpride) (Esamisulpride) is a potent dopamine D2/D3 receptor antagonist.Formule :C17H27N3O4SDegré de pureté :98.38%Couleur et forme :SolidMasse moléculaire :369.48Ref: TM-T26375
1mg34,00€5mg84,00€1mL*10mM (DMSO)94,00€10mg123,00€25mg225,00€50mg358,00€100mg485,00€200mg622,00€Cinacalcet
CAS :Cinacalcet (AMG 073) is an orally active, allosteric Ca receptor (CaR) agonist, treatment of cardiovascular disease .Formule :C22H22F3NDegré de pureté :99.48%Couleur et forme :Yellow OilMasse moléculaire :357.41Nefazodone hydrochloride
CAS :Nefazodone hydrochloride (Serzone) is a serotoninergic modulating antidepressant that is used in therapy of depression, aggressive behavior and panic disorder.Formule :C25H33Cl2N5O2Degré de pureté :99% - 99.86%Couleur et forme :White SolidMasse moléculaire :506.47Ref: TM-T3275
5mg47,00€10mg70,00€1mL*10mM (DMSO)77,00€25mg120,00€50mg216,00€100mg325,00€200mg472,00€500mg775,00€RO 46-8443
CAS :RO 46-8443: First non-peptide ETB receptor antagonist, >2000-fold ETB selectivity in binding and function.Formule :C31H35N3O8SDegré de pureté :98.77% - 99.77%Couleur et forme :SolidMasse moléculaire :609.69Mizagliflozin
CAS :Mizagliflozin is an orally active, selective SGLT1 inhibitor with a Ki value of 27 nM for human SGLT1.Cost-effective and quality-assured.Formule :C28H44N4O8Degré de pureté :98.66% - 99.67%Couleur et forme :SolidMasse moléculaire :564.67Ref: TM-T16083
1mg66,00€2mg96,00€5mg144,00€1mL*10mM (DMSO)173,00€10mg227,00€25mg455,00€50mg645,00€100mg938,00€200mg1.264,00€Buclizine dihydrochloride
CAS :Buclizine dihydrochloride (Buclina) is the hydrochloride salt form of buclizine, a piperazine histamine H1 receptor antagonist with primarily antiemetic andFormule :C28H33ClN2·2HClDegré de pureté :98.05%Couleur et forme :Off-White PowderMasse moléculaire :505.95Naratriptan hydrochloride
CAS :Naratriptan Hydrochloride, a selective 5-HT1 receptor agonist with anti-migraine effect, induces vasoconstriction and reduces inflammation in migraines.Formule :C17H25N3O2S·HClDegré de pureté :99.17% - 99.93%Couleur et forme :Beige SolidMasse moléculaire :371.93Lofexidine
CAS :Lofexidine is a selective α2-receptor agonist, Lofexidine reduces narcotic withdrawal symptoms.
Formule :C11H12Cl2N2ODegré de pureté :98.78%Couleur et forme :SolidMasse moléculaire :259.13S 38093
CAS :S 38093 is a brain-penetrant antagonist of the H3 receptor (Ki: 8.8/1.44/1.2 μM, for rat/mouse/human).Formule :C17H24N2O2Degré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :288.38Ref: TM-T4099
2mg35,00€5mg50,00€1mL*10mM (DMSO)50,00€10mg75,00€25mg124,00€50mg198,00€100mg316,00€200mg442,00€Bepotastine Besilate
CAS :Bepotastine Besilate (TAU 284) is a non-sedating and selective H1 receptor antagonist (pIC50: 5.7).Formule :C21H25ClN2O3·C6H6O3SDegré de pureté :99.83% - 99.9%Couleur et forme :Brown Viscous LiquidMasse moléculaire :547.06CYM5442
CAS :CYM5442 is an S1P agonist, targeting to Sphingosine.Formule :C23H27N3O4Degré de pureté :98.02% - 99.48%Couleur et forme :SolidMasse moléculaire :409.48SBI-553
CAS :SBI-553 is an effective and brain penetrant NTR1 allosteric modulator (EC50: 0.34 μM).Formule :C26H31FN4O2Degré de pureté :99.33%Couleur et forme :SolidMasse moléculaire :450.55Bremelanotide Acetate
CAS :Bremelanotide Acetate (PT-141 Acetate) is an agonist of melanocortin receptor (MCR) .
Formule :C52H72N14O12Degré de pureté :96.72% - >99.99%Couleur et forme :SolidMasse moléculaire :1085.22α-MSH, amide Acetate
a-MSH, amide Acetate as an endogenous neuropeptide.Formule :C79H113N21O21SDegré de pureté :98.67%Couleur et forme :SolidMasse moléculaire :1724.94Chemerin-9 (149-157) acetate
Chemerin-9 (149-157) acetate, a nonapeptide C-terminal fragment of chemerin, retains full protein's activity as chemerinR agonist.Formule :C56H70N10O15Degré de pureté :99.93%Couleur et forme :SolidMasse moléculaire :1123.23RFRP-1 (human) acetate(311309-25-8 free base)
RFRP-1 (human) acetate: potent NPFF2/1 agonist, alters rat/rabbit cardiac functions, and regulates rat prolactin.Formule :C69H105N19O16SDegré de pureté :96.84%Couleur et forme :SolidMasse moléculaire :1488.77Norfluoxetine Hydrochloride
CAS :Norfluoxetine Hydrochloride (Norfluoxetine HCl) is an active metabolite of fluoxetine. Fluoxetine is an antidepressant drug.Formule :C16H17ClF3NODegré de pureté :99.71%Couleur et forme :SolidMasse moléculaire :331.76BMS-986020
CAS :BMS-986020 (AM152) is a selective antagonist of LPA1.Formule :C29H26N2O5Degré de pureté :98.82% - >99.99%Couleur et forme :SolidMasse moléculaire :482.53Tandospirone citrate
CAS :Tandospirone citrate (SM-3997 citrate) is a potent and selective 5-HT1A receptor partial agonist (Ki : 27 nM)Formule :C27H37N5O9Degré de pureté :97.84% - 99.90%Couleur et forme :SolidMasse moléculaire :575.61HJC0350
CAS :HJC0350 is an effective and specific EPAC2 inhibitor (IC50: 0.3 μM), and no inhibition of Epac1.Formule :C15H19NO2SDegré de pureté :99.27% - 99.65%Couleur et forme :SolidMasse moléculaire :277.38RU 24969 free base
CAS :RU 24969 (5-methoxy-3-(1,2,3,6-tetrahydropyridin-4-yl)-1H-indole) is a selective agonist of 5-HT1A and 5-HT1B receptors.Formule :C14H16N2ODegré de pureté :97.38%Couleur et forme :SolidMasse moléculaire :228.29Neuropeptide FF acetate(99566-27-5 free base)
Neuropeptide FF acetate(99566-27-5 free base) (NPFF acetate) is an octapeptide belonging to the RF amide family.Formule :C56H80N14O12Degré de pureté :98.03%Couleur et forme :SolidMasse moléculaire :1141.32Conivaptan hydrochloride
CAS :Conivaptan hydrochloride (Vaprisol) is an orally active vasopressin V2 and V1A receptor antagonist, used in the therapy of hypervolemic hyponatremia andFormule :C32H26N4O2·HClDegré de pureté :98.33% - 99.86%Couleur et forme :SolidMasse moléculaire :535.04Ro 46-2005
CAS :Ro 46-2005: Synthetic non-peptide, blocks 125I-ET-1 at ETA receptors on human vascular cells (IC50: 220 nM).Formule :C23H27N3O6SDegré de pureté :98.02% - 98.8%Couleur et forme :SolidMasse moléculaire :473.54SORT-PGRN interaction inhibitor 1
CAS :SORT-PGRN interaction inhibitor 1 is a potent sortilin-progranulin interaction inhibitor(IC50 of 2 μM).Formule :C15H18N2O2Degré de pureté :98.72%Couleur et forme :SolidMasse moléculaire :258.32MDL 100009
CAS :MDL 100009, the S-enantiomer of MDL 100151 and the opposite enantiomer of MDL 100907, is a selective antagonist of 5-HT2A.Formule :C22H28FNO3Degré de pureté :98.96%Couleur et forme :SolidMasse moléculaire :373.46Ref: TM-T22359
1mg99,00€5mg187,00€1mL*10mM (DMSO)222,00€10mg280,00€25mg434,00€50mg585,00€100mg775,00€200mg1.054,00€Cotadutide acetate
Cotadutide acetate is a potent GLP-1 and glucagon receptor dual agonist with EC50s of 6.9 pM and 10.2 pM.Formule :C169H256N42O57Degré de pureté :98.28%Couleur et forme :SolidMasse moléculaire :3788.14Bosentan
CAS :Bosentan is a competitive endothelin receptor antagonist, used for treating pulmonary arterial hypertension.Formule :C27H29N5O6SDegré de pureté :99.74% - 99.84%Couleur et forme :Pale Yellow To Off-White SolidMasse moléculaire :551.614Ref: TM-T6264
10mg35,00€25mg52,00€50mg77,00€1mL*10mM (DMSO)84,00€100mg120,00€200mg195,00€500mg294,00€Neuropeptide SF(mouse,rat) acetate
Neuropeptide SF (mouse,rat) acetate is a NPFF receptor agonist with Ki of 48.4 nM (NPFF1) & 12.1 nM (NPFF2), enhancing ASIC3 current.Formule :C42H69N13O12Degré de pureté :98.37%Couleur et forme :SolidMasse moléculaire :948.08CJC-1295 acetate(863288-34-0 free base)
CJC-1295 acetate is a synthetic GHRH analogue and GHS.Formule :C154H256N44O44Degré de pureté :97.29%Couleur et forme :SolidMasse moléculaire :3428.01CP 376395
CAS :CP 376395 (CP-316311) is an effective and specific Corticotropin-releasing factor 1 (CRF1) receptor antagonist.Formule :C21H30N2ODegré de pureté :99.86% - 99.94%Couleur et forme :SolidMasse moléculaire :326.48Substance P 1-9 aceate
Substance P 1-9 aceate is nonapeptide, which decreases the inactivation of substance P by the guinea-pig ileum and urinary bladder.Formule :C54H81N15O14Degré de pureté :99.01%Couleur et forme :SolidMasse moléculaire :1164.31Protease-Activated Receptor-1, PAR-1 Agonist acetate
PAR-1 Agonist acetate is a selective PAR-1 agonist that mimics thrombin action.Formule :C37H62N10O11Degré de pureté :98.1800%Couleur et forme :SolidMasse moléculaire :822.95Etilevodopa hydrochloride
CAS :Etilevodopa hydrochloride (L-DOPA ethyl ester) is a prodrug of levodopa. It also has greater gastric solubility and significant brain penetration.Formule :C11H16ClNO4Degré de pureté :95.00%Couleur et forme :SolidMasse moléculaire :261.7Exendin-4
CAS :Exenatide: GLP-1 receptor agonist, 39-amino acid, longer half-life (2.4 hrs), IC50 of 3.22 nM.Formule :C184H282N50O60SDegré de pureté :97.71% - 99.78%Couleur et forme :SolidMasse moléculaire :4186.57Bay 59-3074
CAS :Bay 59-3074 is a CB1/CB2 receptor partial agonist (Ki: 48.3/45.5 nM).Formule :C18H13F6NO4SDegré de pureté :97.68% - 99.69%Couleur et forme :SolidMasse moléculaire :453.36Galanin (1-16), mouse, porcine, rat
CAS :Galanin (1-16), mouse, porcine, rat is a hippocampal galanin receptor agonist(Kd = 3 nM) with high biological activity on locus coeruleus neurons.Formule :C78H116N20O21Degré de pureté :98.65%Couleur et forme :White PowderMasse moléculaire :1669.88(+)-PD 128907 hydrochloride
CAS :(+)-PD 128907 hydrochloride is an agonist of D3 dopamine receptor .
Formule :C14H20ClNO3Degré de pureté :97.76%Couleur et forme :SolidMasse moléculaire :285.77Montelukast sodium
CAS :Montelukast sodium (MK0476), an oral leukotriene antagonist for asthma, can cause rare liver injury.Formule :C35H35ClNNaO3SDegré de pureté :99.14% - 99.89%Couleur et forme :White To Off-White Crystalline PowderMasse moléculaire :608.17RFRP3(human) acetate(311309-27-0 free base)
RFRP-3(human) acetate inhibits gonadotropin, blocks Ca2+ mobilization, acts on NPFF1 receptors, and has an IC50 of 0.7 nM against cAMP production.Formule :C47H76N14O12Degré de pureté :97.09%Couleur et forme :SolidMasse moléculaire :1029.19Dexmedetomidine
CAS :Dexmedetomidine: a central alpha-2 adrenergic agonist for general anesthesia.Formule :C13H16N2Degré de pureté :99% - >99.99%Couleur et forme :SolidMasse moléculaire :200.28Prucalopride Succinate
CAS :Prucalopride Succinate is a 5-HT4 receptor agonist with Ki 2.5 nM (5-HT4a) and 8 nM (5-HT4b).Formule :C18H26ClN3O3·C4H6O4Degré de pureté :99.24%Couleur et forme :SolidMasse moléculaire :485.96AM211
CAS :AM211 (AM211 free acid) is a potent and orally bioavailable antagonist of prostaglandin D2 (PGD2) receptor type 2 (DP2)Formule :C27H27F3N2O4Degré de pureté :≥95%Couleur et forme :SolidMasse moléculaire :500.51nifenalol.HCl
CAS :Nifenalol.HCl(INPEA) is a antagonist of β-adrenergic receptor.Formule :C11H17ClN2O3Degré de pureté :99.96%Couleur et forme :SolidMasse moléculaire :260.72GW627368
CAS :GW627368 (GW 627368X)X is a novel, potent and selective antagonist of prostanoid EP4 receptor.Formule :C30H28N2O6SDegré de pureté :99.75% - 99.92%Couleur et forme :SolidMasse moléculaire :544.62Flibanserin
CAS :Flibanserin (Girosa) is a serotonergic antidepressant used to treat hypoactive sexual desire disorder.
Formule :C20H21F3N4ODegré de pureté :99.37% - 99.93%Couleur et forme :White PowderMasse moléculaire :390.41-Oleoyl lysophosphatidic acid sodium
CAS :1-Oleoyl lysophosphatidic acid sodium (1-Oleoyl lysophosphatidic acid sodium salt) salt is an Endogenous agonist of LPA1 and LPA2Formule :C21H40O7P·NaDegré de pureté :98.75% - 99.24%Couleur et forme :SolidMasse moléculaire :458.51BAY 41-2272
CAS :BAY 41-2272 is a direct and NO-independent soluble guanylate cyclase (sGC) stimulator.Formule :C20H17FN6Degré de pureté :99.54%Couleur et forme :SolidMasse moléculaire :360.39SB-200646
CAS :SB-200646 is a selective and potent antagonist of 5-HT2B/5-HT2C receptorFormule :C15H14N4ODegré de pureté :99.61%Couleur et forme :SolidMasse moléculaire :266.3Decloxizine dihydrochloride
CAS :Decloxizine dihydrochloride (UCB 1402 dihydrochloride) is a histamine 1 receptor antagonist.Formule :C21H28N2O2·2ClHDegré de pureté :99.73%Couleur et forme :SolidMasse moléculaire :413.39ML221
CAS :ML221 is a potent apelin /APJ functional antagonist, inhibiting apelin-13-mediated activation of APJ, with IC50s of 0.70 μM in the cAMP assay, and 1.75 μM inFormule :C17H11N3O6SDegré de pureté :97.74%Couleur et forme :SolidMasse moléculaire :385.35Ref: TM-T4390
2mg34,00€5mg50,00€1mL*10mM (DMSO)52,00€10mg80,00€25mg137,00€50mg215,00€100mg349,00€200mg512,00€Piperacetazine
CAS :Piperacetazine (Piperacetazinum), an antipsychotic prodrug, is used forschizophrenia.Formule :C24H30N2O2SDegré de pureté :99.9% - 99.92%Couleur et forme :SolidMasse moléculaire :410.57Relugolix
CAS :Relugolix (RVT-601) is an orally available, non-peptide gonadotropin-releasing hormone (GnRH or luteinizing hormone-releasing hormone (LHRH)) antagonist, withFormule :C29H27F2N7O5SDegré de pureté :98.64% - 99.97%Couleur et forme :SolidMasse moléculaire :623.63Ref: TM-T3630
2mg39,00€5mg58,00€1mL*10mM (DMSO)81,00€10mg93,00€25mg167,00€50mg250,00€100mg408,00€200mg585,00€Obestatin (rat) acetate
Obestatin (rat) acetate is an endogenous ligand of G-protein coupled receptor 39 (GPR39).Formule :C114H174N34O31Degré de pureté :99.05%Couleur et forme :SolidMasse moléculaire :2516.81Ref: TM-TP2279L
1mg77,00€2mg97,00€5mg156,00€10mg225,00€25mg375,00€50mg535,00€100mg730,00€200mg938,00€Spexin acetate(1370290-58-6 free base)
Spexin acetate: GAL2/GAL3 agonist. EC50: 45.7/112.2 nM. Inactive at GAL1. Reduces appetite, fat uptake, and food intake; lowers LH in fish; anxiolytic.Formule :C76H117N19O22SDegré de pureté :95.43%Couleur et forme :SolidMasse moléculaire :1680.94Opiranserin hydrochloride
CAS :Opiranserin (VVZ-149) hydrochloride is a dual antagonist of glycine transporter type 2 (GlyT2) and serotonin receptor 2A (5HT2A), with IC50s of 0.86 and 1.3 μMFormule :C21H35ClN2O5Degré de pureté :99.33%Couleur et forme :SolidMasse moléculaire :430.97Ref: TM-T9833
1mg90,00€5mg215,00€1mL*10mM (DMSO)236,00€10mg340,00€25mg618,00€50mg879,00€100mg1.224,00€500mg2.457,00€AC-90179 HCl
CAS :AC-90179 HCl: selective 5-HT2A inverse agonist, atypical antipsychotic, reduces hallucinogen-induced vasoconstriction.Formule :C23H31ClN2O2Degré de pureté :99.71%Couleur et forme :SolidMasse moléculaire :402.96Melanotan (MT)-II
CAS :Melanotan (MT)-II, a synthetic melanocortin receptor agonist, is a synthetic analogue of the peptide hormone α-melanocyte-stimulating hormone (α-MSH).Formule :C50H69N15O9Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :1024.18FAUC-365
CAS :FAUC-365 is a D3 dopamine receptor agonist.Formule :C23H25Cl2N3OSDegré de pureté :99.62%Couleur et forme :SolidMasse moléculaire :462.44Ref: TM-T21667
1mg50,00€5mg105,00€1mL*10mM (DMSO)116,00€10mg160,00€25mg305,00€50mg485,00€100mg700,00€500mg1.459,00€AVN-492
CAS :AVN-49 is a potent and selective 5-HT6R Antagonist (Ki: 91 pM).Formule :C17H21N5O2SDegré de pureté :99.81%Couleur et forme :SolidMasse moléculaire :359.45Ref: TM-T5179
1mg37,00€2mg50,00€5mg77,00€1mL*10mM (DMSO)85,00€10mg114,00€25mg225,00€50mg335,00€100mg484,00€Vorapaxar sulfate
CAS :Vorapaxar sulfate (Zontivity) is a potent and orally active thrombin receptor (PAR-1) antagonist.Formule :C29H35FN2O8SDegré de pureté :99.9% - >99.99%Couleur et forme :SolidMasse moléculaire :590.66Ref: TM-T3098
1mg38,00€2mg49,00€5mg79,00€1mL*10mM (DMSO)99,00€10mg119,00€25mg210,00€50mg354,00€100mg528,00€500mg1.159,00€Tozadenant
CAS :Tozadenant (SYN115) is an adenosine A2A receptor antagonist(Ki of 11.5 nM and 6 nM on human and rhesus,respectively)Formule :C19H26N4O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :406.5Vipadenant
CAS :Vipadenant (CEB-4520)(BIIB-014) is an adenosine A2a antagonist with Ki of 1.3 nM; less potent for A1(Ki=69 nM).Formule :C16H15N7ODegré de pureté :97.25% - 97.36%Couleur et forme :SolidMasse moléculaire :321.34Ref: TM-T2373
2mg35,00€5mg51,00€10mg80,00€25mg131,00€50mg210,00€1mL*10mM (DMSO)215,00€100mg313,00€200mg445,00€γ-Mangostin
CAS :Gamma-Mangostin (Normangostin) has free radical scavenging activity, and antiproliferative and apoptotic activity. Gamma-Mangostin is an antihypertensive agent.Formule :C23H24O6Degré de pureté :98.55% - 99.08%Couleur et forme :SolidMasse moléculaire :396.43VUF 10166
CAS :VUF10166 is a novel, potent and competitive antagonist for 5-HT3A receptor with Ki of 0.04 nM, its affinity at 5-HT3AB receptor is significantly lower.Formule :C13H15ClN4Degré de pureté :99.66%Couleur et forme :SolidMasse moléculaire :262.74Buclizine
CAS :Buclizine is an orally active antihistamine, antiallergic compound. buclizine is also a strong teratogen in rats and exhibits antitumour effects.Formule :C28H33ClN2Couleur et forme :SolidMasse moléculaire :433.03Lurasidone
CAS :Lurasidone (SM-13496) is an antagonist of both dopamine D2 and 5-HT7(IC50=1.68 and 0.495 nM, respectively).It also a partial agonist of 5-HT1A receptor(IC50 : 6Formule :C28H36N4O2SDegré de pureté :99.78% - 99.91%Couleur et forme :SolidMasse moléculaire :492.68Ramosetron
CAS :Ramosetron 是一种血清素 5-HT3 受体拮抗剂，用于治疗恶心和呕吐。它被认为比其他一代 5-HT3 拮抗剂如昂丹司琼具有更高的效力和更长的止吐作用。它还适用于治疗“男性以腹泻为主的肠易激综合征”。它仅获准在日本和选定的东南亚国家使用。Formule :C17H17N3ODegré de pureté :98.84%Couleur et forme :SolidMasse moléculaire :279.34Nonapeptide-1 acetate salt (158563-45-2 free base)
Nonapeptide-1 acetate salt (158563-45-2 free base) (Melanostatine-5 acetate salt) , a peptide hormone, is a potent α-Melanocyte-stimulating hormone (α-MSH)Formule :C63H91N15O11SDegré de pureté :98.26%Couleur et forme :SolidMasse moléculaire :1266.58SR 57227 hydrochloride
CAS :SR 57227A (SR 57227 hydrochloride) is a potent, orally active and selective 5-HT3 receptor agonist. It with ability to cross the blood brain barrier.Formule :C10H14ClN3·HClDegré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :248.15BP 897
CAS :BP 897: potent selective dopamine D3 agonist, weak D2 antagonist. Ki: 0.92 nM (D3), 61 nM (D2), low affinity at D1/D4.Formule :C26H31N3O2Degré de pureté :99.44%Couleur et forme :SolidMasse moléculaire :417.54Ref: TM-T9100
1mg75,00€5mg154,00€1mL*10mM (DMSO)168,00€10mg215,00€25mg359,00€50mg512,00€100mg692,00€200mg888,00€Alloxazine
CAS :Alloxazine (Isoalloxazine) is an A2 receptor antagonist, which is approximately 10-fold more selective for the A2B receptor than for the A2A receptor.Formule :C10H6N4O2Degré de pureté :99.75%Couleur et forme :SolidMasse moléculaire :214.18Hemopressin (rat) acetate(568588-77-2 free base)
Hemopressin is a nonapeptide, CB2 agonist, derived from rat hemoglobin, with antinociceptive properties.Formule :C5H81N13O14Degré de pureté :99.37%Couleur et forme :SolidMasse moléculaire :1148.31Droxidopa
CAS :Droxidopa (L-DOPS), an oral prodrug, treats symptomatic orthostatic hypotension from neurogenic autonomic failure.Formule :C9H11NO5Degré de pureté :97.27% - 99.88%Couleur et forme :SolidMasse moléculaire :213.19TC-G-1008
CAS :TC-G-1008 (GPR39-C3) is a GPR39 (zinc receptor) agonist (EC50 values are 0.4 and 0.8 nM for rat and human receptors respectively).Formule :C18H19ClN6O2SDegré de pureté :97.37% - 99%Couleur et forme :SolidMasse moléculaire :418.9Ref: TM-T4648
1mg35,00€5mg75,00€1mL*10mM (DMSO)84,00€10mg114,00€25mg203,00€50mg334,00€100mg557,00€200mg790,00€NPS-2143 hydrochloride
CAS :NPS-2143 hydrochloride (NPS-2143 HCL) is a selective potent calcium ion-sensing receptor antagonist.Formule :C24H25ClN2O2·HClDegré de pureté :99.38% - 99.67%Couleur et forme :SolidMasse moléculaire :445.38Ref: TM-T4967
1mg43,00€2mg56,00€5mg87,00€1mL*10mM (DMSO)95,00€10mg119,00€25mg203,00€50mg320,00€100mg475,00€AF38469
CAS :AF38469 is a new, specific and orally bioavailable Sortilin inhibitor (IC50: 330 nM).Formule :C15H11F3N2O3Degré de pureté :99.18%Couleur et forme :SolidMasse moléculaire :324.25Ref: TM-TQ0086
1mg93,00€2mg114,00€5mg170,00€1mL*10mM (DMSO)178,00€10mg268,00€25mg522,00€50mg802,00€100mg1.099,00€200mg1.468,00€Adenosine amine congener
CAS :Adenosine amine congener (ADAC) (ADAC) is an agonist of selective A1 adenosine receptor,.Formule :C28H32N8O6Degré de pureté :97.86%Couleur et forme :SolidMasse moléculaire :576.6Exenatide
CAS :Exenatide (Extendin-4) is a glucagon-like protein-1 (GLP-1) receptor agonist.Formule :C186H286N50O62SDegré de pureté :99.42%Couleur et forme :SolidMasse moléculaire :4247Fluphenazine decanoate
CAS :Fluphenazine decanoate is dopamine D2 receptor blocke,and is a long-acting phenothiazine neuroleptic that used to treat schizophrenia.Formule :C32H44F3N3O2SDegré de pureté :98.14%Couleur et forme :SolidMasse moléculaire :591.77Amezinium methylsulfate
CAS :Amezinium methylsulfate (Lu-1631) has multiple mechanisms, including stimulation of α and β-1 receptors and inhibition of noradrenaline and tyramine uptake.Formule :C12H15N3O5SDegré de pureté :99.64% - 99.99%Couleur et forme :SolidMasse moléculaire :313.33Levobetaxolol hydrochloride
CAS :Levobetaxolol hydrochloride ((S)-Betaxolol hydrochloride) is a beta blocker, used to lower the pressure in the eye in treating conditions such as glaucoma.Formule :C18H29NO3·HClDegré de pureté :98.80% - 99.69%Couleur et forme :SolidMasse moléculaire :343.89FAUC 213
CAS :FAUC 213 is a selective full antagonist of the dopamine D4 receptor.Formule :C18H19ClN4Degré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :326.82Eptapirone
CAS :Eptapirone (F 11440) is a highly effective and selective 5-HT1A receptor agonist with marked antidepressant and anxiolytic potential.Formule :C16H23N7O2Degré de pureté :99.39% - 99.65%Couleur et forme :SolidMasse moléculaire :345.4(E)-3,4,5-Trimethoxycinnamic acid
CAS :(E)-3,4,5-Trimethoxycinnamic acid (O-Methylsinapic acid) is a natural product from the roots and rhizomes of Notopterygium incisum.Formule :C12H14O5Degré de pureté :99.83%Couleur et forme :SolidMasse moléculaire :238.24Loxiglumide
CAS :Loxiglumide (CR-1505) is an antagonist of cholecystokinin (CCK-1) receptor.
Formule :C21H30Cl2N2O5Degré de pureté :97.55% - 99.81%Couleur et forme :SolidMasse moléculaire :461.38Opaganib
CAS :Opaganib (ABC294640) is an orally active and specific sphingosine kinase-2 (SphK2) inhibitor (IC50: 60 μM).Formule :C23H25ClN2ODegré de pureté :98.86% - 99.85%Couleur et forme :SolidMasse moléculaire :380.91Ref: TM-T6750
1mg38,00€2mg50,00€5mg80,00€1mL*10mM (DMSO)82,00€10mg117,00€25mg227,00€50mg394,00€100mg583,00€BETP
CAS :BETP is an agonist of GLP-1 receptor (EC50s: 0.66 and 0.755 μM for human and rat GLP-1 receptor).Formule :C20H17F3N2O2SDegré de pureté :98.51%Couleur et forme :SolidMasse moléculaire :406.42Sar-[D-Phe8]-des-Arg9-Bradykinin acetate
Sar-[D-Phe8]-des-Arg9-Bradykinin acetate is a potent and selective bradykinin B1 receptor agonist (EC50 = 9.02 nM in rabbit aorta) that is resistant toFormule :C49H70N12O13Degré de pureté :99.93%Couleur et forme :SolidMasse moléculaire :1035.15Preladenant
CAS :Preladenant (SCH-420814) is an orally bioavailable antagonist of the adenosine A2A receptor (Ki: 1.1 nM) and has >1000-fold selectivity over all other adenosineFormule :C25H29N9O3Degré de pureté :98.02% - 99.68%Couleur et forme :SolidMasse moléculaire :503.56AM1241
CAS :AM-1241 is a selective cannabinoid CB2 receptor agonist with Ki of 3.4 nM, exhibits 82-fold selectivity over CB1 receptor.Formule :C22H22IN3O3Degré de pureté :98.937% - 99.1%Couleur et forme :SolidMasse moléculaire :503.33Ref: TM-T6755
2mg35,00€5mg49,00€10mg84,00€1mL*10mM (DMSO)87,00€25mg168,00€50mg275,00€100mg495,00€500mg1.071,00€[Sar9] Substance P acetate(77128-75-7 free base)
[Sar9]-Substance P acetate, an NK-1 receptor agonist, mimics SP's effect on progesterone metabolism.Formule :C66H104N18O15SDegré de pureté :96.67%Couleur et forme :SolidMasse moléculaire :1421.71Ponesimod
CAS :Ponesimod (ACT-128800) is an orally available sphingosine-1-phosphate receptor 1 (S1PR1, S1P1) agonist with potential immunomodulating activity.Formule :C23H25ClN2O4SDegré de pureté :99.42% - 99.96%Couleur et forme :SolidMasse moléculaire :460.97Ref: TM-T3258
1mg43,00€2mg56,00€5mg88,00€1mL*10mM (DMSO)92,00€10mg124,00€25mg221,00€50mg383,00€100mg565,00€500mg1.215,00€HCGRP-(8-37) acetate
HCGRP-(8-37) acetate is a human calcitonin gene-related peptide (hCGRP) fragment acetate and also an antagonist of CGRP receptor.Formule :C141H234N44O40Degré de pureté :99.29%Couleur et forme :SolidMasse moléculaire :3185.64Ibrolipim
CAS :Ibrolipim (NO-1886) attenuates high glucose-induced endothelial dysfunction in cultured human umbilical vein endothelial cells via PI3K/Akt pathway.Formule :C19H20BrN2O4PDegré de pureté :98.04%Couleur et forme :SolidMasse moléculaire :451.25Amitriptyline
CAS :Amitriptyline: a tricyclic antidepressant used for depression and neuropathic pain.Formule :C20H23NDegré de pureté :98.24% - 99.64%Couleur et forme :Crystals SolidMasse moléculaire :277.4Siramesine
CAS :Siramesine (Lu 28-179)(Lu 28-179) is a selective sigma-2 receptor agonist, which has been shown to trigger cell death of cancer cells and to exhibit a potentFormule :C30H31FN2ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :454.58[Sar9,Met(O2)11]-Substance P acetate
[Sar9,Met(O2)11]-Substance P acetate is an NK1 agonist, raising MAP and HR equally to septide but with unique timing and behaviors.Formule :C66H106N18O18SDegré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :1471.75BD 1008 dihydrobromide
CAS :BD 1008 dihydrobromide: selective σ1 receptor antagonist (Ki=2 nM), high σ1 and moderate σ2 affinity.
Formule :C15H24Br2Cl2N2Degré de pureté :97.81%Couleur et forme :SolidMasse moléculaire :463.08Almotriptan
CAS :Almotriptan (LAS 31416), a triptan and 5-HT1B/1D agonist, treats migraines by constricting cranial vessels and altering blood flow.Formule :C17H25N3O2SDegré de pureté :99.85%Couleur et forme :Light Yellow Or White PowerMasse moléculaire :335.46[Lys5,MeLeu9,Nle10]-NKA(4-10)
CAS :Highy selective and potent NK2 receptor agonist (IC50 = 6.1 nM). Induces contraction of the rat fundus and bladder (EC50 values are 117 and 10 nM respectively).Formule :C39H65N9O9Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :803.99FAUC 346
CAS :FAUC 346 is a highly selective D3 partial agonist with EC50 of 1.5 nM.Formule :C24H29N3O2SDegré de pureté :99.46%Couleur et forme :SolidMasse moléculaire :423.57Ref: TM-T9081
2mg34,00€5mg50,00€1mL*10mM (DMSO)52,00€10mg77,00€25mg138,00€50mg224,00€100mg359,00€200mg490,00€Neuropeptide S (Mouse) acetate
Neuropeptide S (Mouse) acetate is a bioactive peptide.Formule :C95H160N34O29Degré de pureté :98.25%Couleur et forme :SolidMasse moléculaire :2242.5S26131
CAS :S26131 (N-[2-[7-[3-[8-(2-acetamidoethyl)naphthalen-2-yl]oxypropoxy]naphthalen-1-yl]ethyl]acetamide) behaves as an antagonist on MT1 and MT2 receptors with Ki ofFormule :C31H34N2O4Degré de pureté :99.77%Couleur et forme :SolidMasse moléculaire :498.61PU02
CAS :PU02 (6-[(1-Naphthalenylmethyl)thio]-9H-purine) is a potent and selective antagonist of 5-HT3 receptor.Formule :C16H12N4SDegré de pureté :99.35%Couleur et forme :SolidMasse moléculaire :292.36MIPS521
CAS :MIPS521 ({2-Amino-4-[3,5-bis(trifluoromethyl)phenyl]thiophen-3-yl}(4-chlorophenyl)methanone) is a positive allosteric modulator of the A1R.Formule :C19H10ClF6NOSDegré de pureté :99.76%Couleur et forme :SolidMasse moléculaire :449.8Ref: TM-T9330
1mg35,00€2mg50,00€5mg74,00€1mL*10mM (DMSO)82,00€10mg105,00€25mg178,00€50mg313,00€100mg485,00€ML-178
CAS :ML-178: selective S1PR4 agonist, EC50 of 46 nM; inactive on other S1P receptors at 25 μM.Formule :C13H9Br2Cl2NO2Degré de pureté :95.92%Couleur et forme :SolidMasse moléculaire :441.93ML417
CAS :ML417 is a selective and brain penetrant agonist of D3 Dopamine (EC50 : 38 nM).Formule :C22H25N3O3Degré de pureté :98.4% - 99.42%Couleur et forme :SolidMasse moléculaire :379.45Rizatriptan benzoate
CAS :Rizatriptan benzoate (MK-462 Benzoate) selectively binds to and activates serotonin (5-HT) 1B receptors and 5-HT 1D receptors providing relief of migraineFormule :C22H25N5O2Degré de pureté :99% - 99.79%Couleur et forme :White To Off-White Crystalline PowderMasse moléculaire :391.47Ref: TM-T1512
10mg44,00€1mL*10mM (DMSO)48,00€25mg74,00€50mg119,00€100mg173,00€200mg259,00€500mg437,00€SB 204741
CAS :SB 204741 is a selective 5-HT2B antagonist with high affinity and pKi value of 7.1.Formule :C14H14N4OSDegré de pureté :99.83%Couleur et forme :SolidMasse moléculaire :286.35Ref: TM-T23312
1mg38,00€2mg50,00€5mg84,00€1mL*10mM (DMSO)84,00€10mg119,00€25mg234,00€50mg439,00€100mg600,00€200mg837,00€Istradefylline
CAS :Istradefylline (KW-6002)(Ki of 2.2 nM) is a selective adenosine A2A receptor (A2AR) antagonist, which is under development in Phase 3 trails.Formule :C20H24N4O4Degré de pureté :98.18% - 99.95%Couleur et forme :SolidMasse moléculaire :384.43H4 Receptor antagonist 1
CAS :H4 Receptor antagonist 1 is a potent and selective histamine H4 receptor inverse agonist, with an IC50 of 19 nM.Formule :C16H17ClN4ODegré de pureté :98.81%Couleur et forme :SolidMasse moléculaire :316.791-(2,3-DIHYDRO-BENZO[1,4]DIOXIN-6-YL)-5-OXO-PYRROLIDINE-3-CARBOXYLIC ACID
CAS :1-(2,3-DIHYDRO-BENZO[1,4]DIOXIN-6-YL)-5-OXO-PYRROLIDINE-3-CARBOXYLIC ACID targets GRK2.
Formule :C13H13NO5Degré de pureté :99.55%Couleur et forme :SolidMasse moléculaire :263.25AZD4635
CAS :AZD4635 (HTL1071) is a new-type adenosine 2A receptor (A2AR) inhibitor(Ki=1.7 nM).Formule :C15H11ClFN5Degré de pureté :99.15% - 99.90%Couleur et forme :SolidMasse moléculaire :315.73Ref: TM-T4265
1mg37,00€2mg52,00€5mg79,00€1mL*10mM (DMSO)87,00€10mg116,00€25mg188,00€50mg296,00€100mg457,00€500mg1.008,00€RVD-Hpα acetate(1193362-76-3 free base)
RVD-Hpα acetate is the N-terminally extended form of human hemopressin that acts as a selective CB1 receptor agonist.Formule :C67H109N19O19Degré de pureté :99.87%Couleur et forme :SolidMasse moléculaire :1484.71BIM-23190 aceate
BIM-23190 aceate, a somatostatin analog, a selective agonist of SSTR2 and SSTR5. BIM-23190 can be used in cancer and acromegaly studies.
Formule :C59H83N13O14S2Degré de pureté :99.7%Couleur et forme :SolidMasse moléculaire :1262.5Trazodone
CAS :Trazodone (AF-1161), a 5-HT 2A/2C receptor antagonist, is used as an antidepressant for treating major anxiety disorders and depressive disorder.Formule :C19H22ClN5ODegré de pureté :99.79% - 99.92%Couleur et forme :White To Off-White Crystalline PowderMasse moléculaire :371.86LP-211
CAS :LP-211 is a brain penetrant selective agonist for a 5-HT7 receptor (Ki: 0.58 nM), and >300-fold selectivity over the 5-HT1A receptor.Formule :C30H34N4ODegré de pureté :98.65%Couleur et forme :SolidMasse moléculaire :466.62Ref: TM-T5387
2mg44,00€5mg66,00€1mL*10mM (DMSO)73,00€10mg90,00€25mg170,00€50mg289,00€100mg462,00€200mg658,00€Montelukast
CAS :Montelukast (Singular), oral asthma med, linked to rare liver injury.Formule :C35H36ClNO3SDegré de pureté :98.56% - >99.99%Couleur et forme :SolidMasse moléculaire :586.18Ramosetron hydrochloride
CAS :Ramosetron hydrochloride (YM-060) is a serotonin 5-HT3 receptor antagonist. It is used to treat diarrhea-predominant irritable bowel syndrome and nausea.Formule :C17H18ClN3ODegré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :315.8Harmine
CAS :Harmine (Telepathine) is an alkaloid isolated from seeds of Peganum harmala.Formule :C13H12N2ODegré de pureté :98.29% - 99.92%Couleur et forme :Off-White SolidMasse moléculaire :212.25(R)-Propranolol hydrochloride
CAS :(R)-Propranolol hydrochloride (Dexpropranolol hydrochloride) is the less active enantiomer of the anti-adrenoceptor (β-adrenoceptor) antagonist propranolol.Formule :C16H22ClNO2Degré de pureté :98.63% - 99.01%Couleur et forme :SolidMasse moléculaire :295.8Capromorelin Tartrate
CAS :Capromorelin Tartrate (CP 424391-18) is a potent, orally active growth hormone secretagogue receptor (GHSR) agonist (Ki: 7 nM for hGHS-R1a).Formule :C32H41N5O10Degré de pureté :97.69%Couleur et forme :SolidMasse moléculaire :655.7Ref: TM-TQ0022
5mg39,00€1mL*10mM (DMSO)52,00€10mg64,00€25mg126,00€50mg215,00€100mg319,00€200mg455,00€Vanoxerine dihydrochloride
CAS :Vanoxerine dihydrochloride (GBR-12909 dihydrochloride) is a potent inhibitor that blocks dopamine uptake (IC50 : 1-51 nM)Formule :C28H34Cl2F2N2ODegré de pureté :98.16% - 98.35%Couleur et forme :White SolidMasse moléculaire :523.49Pramipexole dihydrochloride hydrate
CAS :Pramipexole dihydrochloride hydrate (Mirapex) is a selective, blood-brain barrier-crossing D2 dopamine receptor agonist, and is used in the study of PD.Formule :C10H17N3S·2HCl·H2ODegré de pureté :99.68%Couleur et forme :White To Off-White Crystalline PowderMasse moléculaire :302.26Ref: TM-T6951
10mg44,00€1mL*10mM (DMSO)44,00€25mg71,00€50mg113,00€100mg166,00€200mg241,00€500mg408,00€Sultopride hydrochloride
CAS :Sultopride hydrochloride (LIN-1418 hydrochloride) is a selective dopamine D2 and D3 receptor antagonist.Formule :C17H27ClN2O4SDegré de pureté :≥95%Couleur et forme :White Or Yellowish PowderMasse moléculaire :390.93SHU 9119 acetate
SHU 9119 acetate: hMC3R & hMC4R antagonist, hMC5R partial agonist. IC50: MC3R 0.23nM, MC4R 0.06nM, MC5R 0.09nM.Formule :C56H75N15O11Degré de pureté :99.8%Couleur et forme :SolidMasse moléculaire :1134.29TGR5 Receptor Agonist
CAS :TGR5 is a potent TGR5(GPCR19) agonist.Formule :C18H14Cl2N2O2Degré de pureté :99.77% - ≥95%Couleur et forme :SolidMasse moléculaire :361.22Metoclopramide
CAS :Metoclopramide: dopamine D2 antagonist, treats nausea, vomiting, gastroparesis, GERD; safe for pregnancy.Formule :C14H22ClN3O2Degré de pureté :99.75%Couleur et forme :SolidMasse moléculaire :299.80GR-73632
CAS :Potent and selective tachykinin NK1 receptor agonist (EC50 = 2 nM in guinea pig vas deferens).Formule :C40H59N7O6SDegré de pureté :99.68%Couleur et forme :SolidMasse moléculaire :766Naftopidil dihydrochloride
CAS :Naftopidil dihydrochloride (KT-611 2HCl) is a selective 5-HT1A and α1-adrenergic receptor antagonist with IC50 of 0.1 μM and 0.2 μM, respectively.Formule :C24H28N2O3·2HClDegré de pureté :99.76%Couleur et forme :White SolidMasse moléculaire :465.415-Iodotubercidin
CAS :5-Iodotubercidin (NSC-113939) is a potent adenosine kinase inhibitor with IC50 of 26 nM.Formule :C11H13IN4O4Degré de pureté :99.88% - 99.98%Couleur et forme :Tan SolidMasse moléculaire :392.15Ref: TM-T6745
1mg43,00€1mL*10mM (DMSO)92,00€5mg96,00€10mg137,00€25mg268,00€50mg429,00€100mg685,00€200mg888,00€Zotepine
CAS :Zotepine, an antipsychotic agent, is a potent antagonist of 5-HT2A, 5-HT2C, Histamine H1, α1-adrenergic, and Dopamine D2 receptors, with Kds of 2.6 nM, 3.2 nM,Formule :C18H18ClNOSDegré de pureté :99.78%Couleur et forme :SolidMasse moléculaire :331.86Exo-1
CAS :Exo-1 (Methyl 3-(4-fluorobenzoyl)-6-methyl-2-pyridinecarboxylate) is a synthetic compound that has been shown to affect the metabolism of various nutrients, asFormule :C15H12FNO3Degré de pureté :99.45%Couleur et forme :SolidMasse moléculaire :273.26Ref: TM-T9200
5mg52,00€1mL*10mM (DMSO)65,00€10mg78,00€25mg119,00€50mg172,00€100mg259,00€200mg388,00€500mg642,00€Mebhydrolin
CAS :Mebhydrolin (Mebhydroline) is a specific histamine H1 receptor antagonist.Formule :C19H20N2Degré de pureté :99.3% - ≥98%Couleur et forme :SolidMasse moléculaire :276.38Fexofenadine
CAS :Fexofenadine, a non-sedating antihistamine, treats allergies like hay fever and urticaria.Formule :C32H39NO4Degré de pureté :99.35%Couleur et forme :White To Off-White SolidMasse moléculaire :501.66Idalopirdine Hydrochloride
CAS :Idalopirdine Hydrochloride (Lu AE58054 Hydrochloride) is an in-vivo binding affinity and effect, in-vitro selectivity and potency of 5-HT(6)R antagonist (Ki: 0.Formule :C20H20ClF5N2ODegré de pureté :99.77%Couleur et forme :SolidMasse moléculaire :434.83Dimemorfan phosphate
CAS :Dimemorfan phosphate (3,17-dimethylmorphinan) is a sigma 1 receptor agonist. Dimemorfan phosphate is used as a potent antitussive.Formule :C18H25N·H3O4PDegré de pureté :99.65%Couleur et forme :SolidMasse moléculaire :353.4TG6-10-1
CAS :TG6-10-1 is an EP2 antagonist.Formule :C23H23F3N2O4Degré de pureté :99.66% - ≥95%Couleur et forme :SolidMasse moléculaire :448.43BAR501
CAS :BAR501是高效选择性的 GPBAR1激动剂(EC50:1 μM)。Formule :C26H46O3Degré de pureté :99.29% - 99.68%Couleur et forme :SolidMasse moléculaire :406.64ANP(1-28) Acetate (human, porcine)
CAS :Carperitide acetate: 28-amino acid hormone from human heart, counters cardiac injury/stretch, reduces endothelin-1.Formule :C129H207N45O41S3Degré de pureté :98.24%Couleur et forme :SolidMasse moléculaire :3140.5Ref: TM-TP1220L
1mg185,00€5mg459,00€10mg657,00€25mg1.026,00€50mg1.388,00€100mg1.872,00€200mg2.527,00€ACTH 11-24 acetate(4237-93-8 free base)
CAS :ACTH 11-24 acetate is a cortisol-stimulating adrenocorticotrophin fragment and a competitive antagonist of ACTH 1-39 and 1-10.Formule :C79H138N24O18Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :1712.12PEN (human) aceate
PEN (human) aceate, one of the most abundant hypothalamic neuropeptide and derived from the proprotein ProSAAS, is an endogenous ligand of GPR83.Formule :C99H163N27O34Degré de pureté :99.25%Couleur et forme :SolidMasse moléculaire :2275.51
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