GPCR/G-Protéine
Les inhibiteurs des GPCR/protéines G sont des composés qui ciblent les récepteurs couplés aux protéines G (GPCR) et les protéines G associées, qui jouent un rôle crucial dans la transmission des signaux de l'extérieur vers l'intérieur des cellules. Ces inhibiteurs sont essentiels pour étudier les voies de signalisation médiées par les GPCR, impliquées dans de nombreux processus physiologiques, y compris la perception sensorielle, la réponse immunitaire et la neurotransmission. Les inhibiteurs des GPCR sont également importants dans le développement de médicaments, car de nombreux agents thérapeutiques ciblent ces récepteurs. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de GPCR/protéines G de haute qualité pour soutenir vos recherches en pharmacologie, biologie cellulaire et domaines connexes.
Sous-catégories appartenant à la catégorie "GPCR/G-Protéine"
- récepteur 5-HT(1.025 produits)
- Récepteur d'adénosine(249 produits)
- Récepteur adrénergique(3.024 produits)
- Récepteur de la bombésine(35 produits)
- Récepteur de la bradykinine(61 produits)
- CXCR(158 produits)
- CaSR(34 produits)
- Récepteur cannabinoïde(217 produits)
- Cholécystokinine(1 produits)
- Récepteur de la dopamine(445 produits)
- Récepteur de l'endothéline(86 produits)
- Récepteur GNRH(84 produits)
- GPCR19(33 produits)
- GRK(33 produits)
- GTPase(23 produits)
- Récepteur du glucagon(194 produits)
- Hérisson/Smoothened(49 produits)
- Récepteur de l'histamine(385 produits)
- Récepteur LPA(21 produits)
- Récepteur de la mélatonine(26 produits)
- Récepteur OX(41 produits)
- Récepteur opioïde(327 produits)
- PAFR(14 produits)
- PKA(60 produits)
- Récepteur S1P(18 produits)
- SGLT(31 produits)
- Récepteur Sigma(46 produits)
Affichez 19 plus de sous-catégories
5990 produits trouvés pour "GPCR/G-Protéine"
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Sumatriptan hydrochloride
CAS :Sumatriptan hydrochloride (GR 43175), an oral 5-HT1 receptor agonist, treats migraines; Ki: 5-HT1D - 17 nM, 5-HT1B - 27 nM, 5-HT1A - 100 nM.Formule :C14H22ClN3O2SCouleur et forme :SolidMasse moléculaire :331.86Dobutamine
CAS :Dobutamine, a synthetic catecholamine, boosts cardiac output and improves blood flow, mainly targeting β1-AR.Formule :C18H23NO3Couleur et forme :SolidMasse moléculaire :301.38Montelukast dicyclohexylamine
CAS :Montelukast (MK0476), a selective CysLT1 antagonist, treats asthma, liver injury, and is researched for COVID-19.Formule :C47H59ClN2O3SCouleur et forme :SolidMasse moléculaire :767.5Sarpogrelate
CAS :Sarpogrelate (MCI-9042), an oral 5-HT2 antagonist, boosts platelet aggregation and aids in studying Buerger's disease.Formule :C24H31NO6Couleur et forme :SolidMasse moléculaire :429.51Droxidopa hydrochloride
CAS :Droxidopa (L-DOPS) HCI is an oral norepinephrine precursor for nOH and ADHD research, raising standing BP and easing orthostatic hypotension.Formule :C9H12ClNO5Couleur et forme :SolidMasse moléculaire :249.65Cannabigerol
CAS :Cannabigerol is a high affinity α±2-adrenergic receptor agonist, moderate affinity 5-HT1A receptor antagonist, and low affinity CB1 receptor antagonist ; alsoFormule :C21H32O2Degré de pureté :99.59% - 99.92%Couleur et forme :SolidMasse moléculaire :316.48Ref: TM-TN1465
1mg138,00€2mg203,00€5mg298,00€1mL*10mM (DMSO)306,00€10mg449,00€25mg765,00€50mg1.054,00€100mg1.423,00€Romifidine hydrochloride
CAS :Romifidine hydrochloride, an α2 adrenergic receptor agonist, induces sedation effects in vivo.Formule :C9H10BrClFN3Couleur et forme :SolidMasse moléculaire :294.55Domperidone monomaleate
CAS :Domperidone monomaleate, a selective oral dopamine-2 antagonist, aids gastric motility and has antiemetic properties.Formule :C26H28ClN5O6Couleur et forme :SolidMasse moléculaire :541.98Mesdopetam
CAS :Mesdopetam (IRL790), a D3 antagonist, has Ki=90 nM, IC50=9.8 μM, stabilizes psychomotors, used in Parkinson's research.Formule :C12H18FNO3SCouleur et forme :SolidMasse moléculaire :275.34Bunazosin
CAS :Bunazosin is a potent and selective α1-adrenoceptor antagonist that can be used for antihypertensive and ocular hypotensive research [1].Formule :C19H27N5O3Couleur et forme :SolidMasse moléculaire :373.45Syk Inhibitor II dihydrochloride dihydrate
CAS :Potent, selective ATP-competitive Syk Inhibitor II (IC50: 41 nM), with anti-allergic properties, in dihydrochloride dihydrate form.Formule :C14H21Cl2F3N6O3Couleur et forme :SolidMasse moléculaire :449.26Cinaciguat hydrochloride
CAS :Cinaciguat( BAY582667, BAY58-2667) is a soluble guanosine cyclase activator that can prevent cardiac dysfunction in rat models of type 1 diabetes.Formule :C36H40ClNO5Couleur et forme :SolidMasse moléculaire :602.17Apraclonidine
CAS :Apraclonidine (ALO 2145), an α2/weak α1 agonist, lowers IOP; used as eye drops.Formule :C9H10Cl2N4Couleur et forme :SolidMasse moléculaire :245.11Napitane Mesylate
CAS :Napitane Mesylate inhibits norepinephrine transporter and blocks CNS CA uptake as an alpha 2-adrenoceptor antagonist.Formule :C23H29NO5SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :431.55PD 168568
CAS :PD 168568: Oral DRD4 antagonist, selective over D2/D3, K_i - 8.8 nM. Used in GBM research.Formule :C22H27N3OCouleur et forme :SolidMasse moléculaire :349.47Regadenoson hydrate
CAS :Regadenoson is an A2A adenosine receptor agonist, a coronary vasodilator commonly used in pharmacologic stress testing.Formule :C15H20N8O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :408.37Rolapitant hydrochloride hydrate
CAS :Rolapitant (SCH-619734) is a selective NK1-receptor antagonist that may prevent nausea and vomiting induced by chemotherapy.Formule :C25H29ClF6N2O3Couleur et forme :SolidMasse moléculaire :554.95Siponimod hemifumarate
CAS :Siponimod (BAF-312) is a potent S1P receptor modulator for multiple sclerosis research.Formule :C62H74F6N4O10Couleur et forme :SolidMasse moléculaire :1149.282Irdabisant hydrochloride
CAS :Irdabisant (CEP-26401) is a selective H3R inverse agonist, BBB-penetrable, with cognition-enhancing effects.Formule :C18H24ClN3O2Couleur et forme :SolidMasse moléculaire :349.86Tiapride
CAS :Tiapride, an atypical neuroleptic, is a selective dopamine D2-receptor antagonist with varying IC50 values for D1-D4.Formule :C15H24N2O4SCouleur et forme :SolidMasse moléculaire :328.43BRL-15572 hydrochloride
CAS :BRL-15572 hydrochloride: selective h5-HT1D antagonist with high affinity; useful for studying h5-HT1D responses.Formule :C25H28Cl2N2OCouleur et forme :SolidMasse moléculaire :443.41KB-5492 anhydrous
CAS :KB 5492 is an agent of anti-ulcer. It preventing cysteamine-induced duodenal ulcers by stimulating duodenal HCO3- secretion.Formule :C27H34N2O10Couleur et forme :SolidMasse moléculaire :546.57Melitracen hydrochloride
CAS :Melitracen hydrochloride (Thymeol hydrochloride) , an antidepressant, is used as potential dopamine D1/2 receptor antagonist to treat depression.Formule :C21H26ClNDegré de pureté :99.99%Couleur et forme :Crystalline SolidMasse moléculaire :327.90Ref: TM-T4274
10mg44,00€1mL*10mM (DMSO)48,00€25mg64,00€50mg93,00€100mg110,00€200mg161,00€500mg264,00€Triprolidine hydrochloride
CAS :Triprolidine hydrochloride anhydrous, a Histamine H1 antagonist, is used in asthma, allergic rhinitis, and urticaria.Formule :C19H23ClN2Couleur et forme :SolidMasse moléculaire :314.852RS 100329
CAS :RS 100329 HCl is a selective α1A-adrenoceptor antagonist (pKi = 9.6 for human cloned α1A receptors).Formule :C20H25F3N4O3Couleur et forme :SolidMasse moléculaire :426.43PF3274167
CAS :PF3274167 (Cligosiban) is a potent and selective, high-affinity nonpeptide oxytocin receptor antagonist.Formule :C19H19ClFN5O3Degré de pureté :99.67% - 99.88%Couleur et forme :SolidMasse moléculaire :419.84Guanabenz hydrochloride
CAS :Guanabenz hydrochloride (NE56490) is an orally active α2-adrenoceptor agonist with hypotensive effects.Formule :C8H9Cl3N4Degré de pureté :99.45%Couleur et forme :SolidMasse moléculaire :267.54Deslorelin acetate(57773-65-6 free base)
Deslorelin acetate(57773-65-6 free base) is a gonadotropin releasing hormone super-agonist (GnRH agonist)Formule :C66H87N17O14Degré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :1342.5CYM-5541
CAS :CYM-5541 (ML249) is a selective and allosteric S1P3 receptor agonist.Formule :C19H28N2O2Degré de pureté :99.74% - 99.76%Couleur et forme :SolidMasse moléculaire :316.44Ref: TM-T3961
2mg38,00€5mg57,00€1mL*10mM (DMSO)64,00€10mg92,00€25mg160,00€50mg254,00€100mg373,00€500mg873,00€Ganirelix Acetate
CAS :Ganirelix Acetate is a gonadotropin-releasing hormone (GnRH) receptor antagonistFormule :C82H117ClN18O15Degré de pureté :96.05%Couleur et forme :SolidMasse moléculaire :1630.4Tesmilifene fumarate
CAS :Tesmilifene fumarate (DPPE fumarate) (DPPE fumarate) is an H1C receptor antagonist。Formule :C23H29NO5Degré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :399.48Ref: TM-T22746
5mg44,00€1mL*10mM (DMSO)49,00€10mg60,00€25mg110,00€50mg164,00€100mg235,00€200mg349,00€Dolasetron
CAS :Dolasetron (MDL-73147)(MDL-73147) is a serotonin 5-HT3 receptor antagonist. Dolasetron is used to treat nausea and vomiting following chemotherapy.Formule :C19H20N2O3Degré de pureté :99.84% - 99.86%Couleur et forme :White PowderMasse moléculaire :324.37ESI-09
CAS :ESI-09 is a new-typel noncyclic nucleotide EPAC antagonist.The IC50 values of ESI-09 for EPAC1 and EPAC2 is 3.2 and 1.4 μM, respectively.Formule :C16H15ClN4O2Degré de pureté :97.24% - 99.57%Couleur et forme :SolidMasse moléculaire :330.77CCG-50014
CAS :CCG-50014 is a potent and selective inhibitor of RGS4 with IC50 of 30 nM.Formule :C16H13FN2O2SDegré de pureté :98.53%Couleur et forme :SolidMasse moléculaire :316.35Dazoxiben
CAS :Dazoxiben (UK-37248) is a potent inhibitor of thromboxane (TX) synthase
Formule :C12H13ClN2O3Degré de pureté :99.99%Couleur et forme :SolidMasse moléculaire :268.7RG7713
CAS :RG7713 (RO 5028442) has been used in trials studying Autistic Disorder.Formule :C25H28ClN3O2Degré de pureté :99.74%Couleur et forme :SolidMasse moléculaire :437.96AnaMorelin hydrochloride
CAS :AnaMorelin hydrochloride (RC-1291 hydrochloride) is a novel ghrelin receptor agonist(EC50 : 0.74 nM, in the FLIPR assay).Formule :C31H43ClN6O3Degré de pureté :99.18% - ≥98%Couleur et forme :SolidMasse moléculaire :583.16Ref: TM-T7225
1mg34,00€2mg48,00€5mg70,00€10mg90,00€1mL*10mM (DMSO)90,00€25mg138,00€50mg168,00€100mg222,00€CS 2100
CAS :CS 2100 (1-[[4-Ethyl-5-[5-(4-phenoxyphenyl)-1,2,4-oxadiazol-3-yl]-2-thienyl]methyl]-3-azetidinecarboxylic acid) is an S1P1 agonist.
Formule :C25H23N3O4SDegré de pureté :99.19%Couleur et forme :SolidMasse moléculaire :461.53Gadolinium chloride
CAS :Gadolinium chloride is a calcium-sensing receptor (CaSR) agonistFormule :Cl3GdDegré de pureté :98%Couleur et forme :White Crystalline SolidMasse moléculaire :263.61Propionylpromazine hydrochloride
CAS :Propionylpromazine hydrochloride (Propiopromazine hydrochloride) is a dopamine receptor D2 (DRD2) antagonist.Formule :C20H25ClN2OSDegré de pureté :99.17%Couleur et forme :SolidMasse moléculaire :376.94Ebastine
CAS :Ebastine (Kestine) (trade names Evastin, Kestine, Ebastel, Aleva) is a non-sedating H1 antihistamine.Formule :C32H39NO2Degré de pureté :99.65% - 99.99%Couleur et forme :White To Off-White PowderMasse moléculaire :469.66Paltusotine
CAS :Paltusotine: nonpeptide SST2 agonist, orally bioavailable, regulates GH/IGF-1 in acromegaly.Formule :C27H22F2N4ODegré de pureté :99.91%Couleur et forme :SolidMasse moléculaire :456.49Ozanimod
CAS :Ozanimod (RPC-1063) (RPC1063) is a specific oral S1P Receptor 1 modulator.Formule :C23H24N4O3Degré de pureté :98.68% - 99.58%Couleur et forme :SolidMasse moléculaire :404.46Ref: TM-T6923
1mg46,00€5mg90,00€1mL*10mM (DMSO)90,00€10mg137,00€25mg268,00€50mg430,00€100mg622,00€200mg879,00€500mg1.305,00€Almotriptan Malate
CAS :Almotriptan Malate (PNU180638), a selective 5-HT1B/1D receptor agonist, is used in the therapy of Migraine attacks in adults.Formule :C17H25N3O2S·C4H6O5Degré de pureté :99.95%Couleur et forme :Pale Yellow SolidMasse moléculaire :469.55ELA-14(human) acetate
ELA-14(human) acetate, a fragment of ELA, targets APJ, activates Gαi1 and β-arrestin-2, and prompts receptor internalization like its parent peptide.Formule :C77H123N25O19S2Degré de pureté :97.2%Couleur et forme :SolidMasse moléculaire :1767.09Cetrorelix diacetate
CAS :Cetrorelix diacetate (NS-75A) is is a gonadotropin-releasing hormone antagonist.Formule :C74H100ClN17O18Degré de pureté :98.38%Couleur et forme :SolidMasse moléculaire :1551.17Ref: TM-T5520L
1mg50,00€5mg95,00€10mg142,00€1mL*10mM (DMSO)239,00€25mg276,00€50mg414,00€100mg608,00€500mg1.288,00€Azaphen
CAS :Azaphen (Pipofezin hydrochloride) is the reuptake of serotonin inhibitor.with antidepressant action and has sedative effects, suggesting antihistamine activity.Formule :C16H21Cl2N5ODegré de pureté :97.62%Couleur et forme :SolidMasse moléculaire :370.28Dasotraline hydrochloride
CAS :Dasotraline hydrochloride, a dopamine, norepinephrine, and serotonin reuptake inhibitor with IC50s: 4, 6, 11 nM.Formule :C16H16Cl3NDegré de pureté :98.92% - 99.6%Couleur et forme :SolidMasse moléculaire :328.66Alizapride hydrochloride
CAS :Alizapride hydrochloride (Alizapride HCl) is a dopamine receptor antagonist used for the treatment of nausea and vomiting.Formule :C16H21N5O2·HClDegré de pureté :99.35% - 99.48%Couleur et forme :CoaMasse moléculaire :351.83CYM2503
CAS :CYM2503 is a GAL2 receptor PAM enhancing galanin-induced IP1 without binding the galanin site.Formule :C45H55N5O7Degré de pureté :97.04%Couleur et forme :SolidMasse moléculaire :777.95ABT-724
CAS :ABT-724 is an agonist of dopamine D4 receptor(EC50: 12.4 nM)Formule :C17H19N5Degré de pureté :99.73%Couleur et forme :SolidMasse moléculaire :293.37HTMT dimaleate
CAS :HTMT dimaleate (Histamine Trifluoromethyl Toluidide Dimaleate) is an H1 and H2 receptor agonist.Formule :C27H33F3N4O9Degré de pureté :99.51%Couleur et forme :SolidMasse moléculaire :614.57Mozavaptan
CAS :Mozavaptan (OPC-31260) is a competitive vasopressin receptor antagonist for both V1 and V2 receptors with IC50 of 1.2 μM and 14 nM, respectively.Formule :C27H29N3O2Degré de pureté :98.98% - 99.12%Couleur et forme :SolidMasse moléculaire :427.54Etrasimod
CAS :Etrasimod (APD334) is a specific and orally available antagonist of the sphingosine-1-phosphate-1 (S1P1) receptor (IC50: 1.88 nM in CHO cells).Formule :C26H26F3NO3Degré de pureté :98.52% - 99.73%Couleur et forme :SolidMasse moléculaire :457.48Ref: TM-TQ0227
1mg50,00€5mg105,00€1mL*10mM (DMSO)107,00€10mg170,00€25mg230,00€50mg289,00€100mg401,00€Cinacalcet hydrochloride
CAS :Cinacalcet hydrochloride (AMG-073 hydrochloride) is a naphthalene derivative and CALCIMIMETIC AGENT that increases the sensitivity of PARATHYROID GLAND calcium-Formule :C22H23ClF3NDegré de pureté :99.96% - >99.99%Couleur et forme :Off-White To Tan SolidMasse moléculaire :393.87Ref: TM-T2406
10mg50,00€1mL*10mM (DMSO)52,00€25mg70,00€50mg88,00€100mg144,00€200mg185,00€500mg309,00€BAY 41-8543
CAS :BAY 41-8543 is a nitric oxide (NO)-independent stimulator of soluble guanylyl cyclase (sGC).
Formule :C21H21FN8ODegré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :420.44RO1138452
CAS :RO1138452 (CAY10441) blocks prostacyclin receptor; orally active, high affinity (Ki: 1.5 nM), analgesic in rats (2-20 mg/kg).Formule :C19H23N3ODegré de pureté :97.01% - 99.34%Couleur et forme :SolidMasse moléculaire :309.41Ref: TM-T4436
1mg49,00€2mg65,00€5mg90,00€1mL*10mM (DMSO)90,00€10mg144,00€25mg313,00€50mg537,00€100mg767,00€Bepotastine
CAS :Bepotastine (Bepotastine free base) free base is a histamine 1 (H1) receptor antagonis.Formule :C21H25ClN2O3Degré de pureté :99.75%Couleur et forme :SolidMasse moléculaire :388.89Ref: TM-T7893
2mg34,00€5mg50,00€1mL*10mM (DMSO)56,00€10mg78,00€25mg141,00€50mg205,00€100mg313,00€200mg464,00€Carcinine ditrifluoroacetate Acetate
Carcinine ditrifluoroacetate Acetate (β-Alanylhistamine dihydrochloride) is an H3 receptor antagonist.Formule :C14H20F6N4O7Degré de pureté :98.18%Couleur et forme :SolidMasse moléculaire :470.32β-MSH (1-22) (human) acetate
Beta-MSH (1-22) (human) acetate (Beta-MSH (1-22) (human) acetate (17908-57-5 Free base)) , is an endogenous melanocortin-4 receptor (MC4-R) agonist.Formule :C120H178N34O37SDegré de pureté :99.64%Couleur et forme :SolidMasse moléculaire :2720.97Rimegepant
CAS :View and buy Rimegepant from TargetMol.BMS-927711 is a highly potent, oral calcitonin gene-related peptide (CGRP) receptor antagonist with a Ki value of 0.027 nM.Cited in 1 publications.Formule :C28H28F2N6O3Degré de pureté :99.1% - 99.99%Couleur et forme :SolidMasse moléculaire :534.56ML-031
CAS :ML-031 activated S1P2 with an EC50 value of 1 μM in an S1P reporter assay.Formule :C19H20N2O3Degré de pureté :99.21%Couleur et forme :SolidMasse moléculaire :324.37JNJ-31020028
CAS :JNJ-31020028 is a selective brain penetrant antagonist of neuropeptide Y2 receptor with high affinity (pIC50=8.07, human; pIC50=8.22, rat).Formule :C34H36FN5O2Degré de pureté :95.92% - 99.65%Couleur et forme :SolidMasse moléculaire :565.68Tetrahydrozoline hydrochloride
CAS :Tetrahydrozoline hydrochloride (Murine Plus) is an imidazoline derivative with alpha receptor agonist activity.Formule :C13H16N2·HClDegré de pureté :99.90%Couleur et forme :Off-White SolidMasse moléculaire :236.74Cinitapride
CAS :Cinitapride (Blaston) treats acid reflux and gastric issues, targeting 5-HT2, 5-HT1, and 5-HT4 receptors.Formule :C21H30N4O4Degré de pureté :99.52%Couleur et forme :SolidMasse moléculaire :402.49Ref: TM-T21385
1mg73,00€5mg155,00€1mL*10mM (DMSO)177,00€10mg240,00€25mg479,00€50mg692,00€100mg973,00€JNJ-5207852 dihydrochloride
CAS :JNJ-5207852 dihydrochloride is a novel, non-imidazole histamine H3 receptor antagonist, with high affinity at the rat (pKi=8.9) and human (pKi=9.24) H3 receptorFormule :C20H34Cl2N2ODegré de pureté :99.51%Couleur et forme :SolidMasse moléculaire :389.4DPCPX
CAS :DPCPX (PD 116948) is an A1 adenosine receptor antagonistFormule :C16H24N4O2Degré de pureté :99.23% - 99.93%Couleur et forme :White SolidMasse moléculaire :304.39A-836339
CAS :A-836339: Potent cannabinoid, CB2-focused (Ki=0.64nM), lesser CB1 affinity (Ki=270nM); analgesic, anti-inflammatory in mice.Formule :C16H26N2O2SDegré de pureté :99.94%Couleur et forme :SolidMasse moléculaire :310.45Ref: TM-T7375
2mg34,00€1mL*10mM (DMSO)63,00€5mg67,00€10mg109,00€25mg177,00€50mg260,00€100mg369,00€200mg500,00€RBC8
CAS :RBC8 is a specific GTPases RalA/RalB inhibitor by inhibiting the binding of Ral to its effector RALBP1, no inhibition on the GTPases RhoA and Ras.Formule :C25H20N4O3Degré de pureté :98.44% - 99.81%Couleur et forme :SolidMasse moléculaire :424.45Ref: TM-T6634
1mg46,00€1mL*10mM (DMSO)92,00€5mg96,00€10mg147,00€25mg281,00€50mg447,00€100mg650,00€200mg888,00€Blarcamesine hydrochloride
CAS :Blarcamesine hydrochloride (AVex-73 hydrochloride) is a Sigma-1 Receptor agonist (IC50: 860 nM).Formule :C19H24ClNODegré de pureté :99.57% - 99.9%Couleur et forme :SolidMasse moléculaire :317.85Ref: TM-T4111
1mg34,00€2mg46,00€5mg66,00€1mL*10mM (DMSO)73,00€10mg99,00€25mg197,00€50mg340,00€100mg557,00€200mg790,00€MK 212 hydrochloride
CAS :MK 212 hydrochloride is a 5-HT2C receptor agonistFormule :C8H11ClN4·HClDegré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :235.12Melitracen
CAS :Melitracen is a tricyclic antidepressant.Formule :C21H25NCouleur et forme :SolidMasse moléculaire :291.43Donitriptan Mesylate
CAS :Donitriptan Mesylate, a 5-HT1B/1D agonist, is used potentially for the treatment of migraines.Formule :C24H29N5O5SCouleur et forme :SolidMasse moléculaire :499.58Bucindolol hydrochloride
CAS :Bucindolol, a 4th-gen β-blocker, prevents onset AF; effectiveness varies with β₁/α(2c) genes; best in β₁389 Arg homozygotes.Formule :C22H26ClN3O2Couleur et forme :SolidMasse moléculaire :399.91Fipamezole HCl
CAS :Fipamezole HCl, a α2-adrenoceptor antagonist, is used potentially for the treatment of dyskinesia associated with Parkinson's disease.Formule :C14H16ClFN2Couleur et forme :SolidMasse moléculaire :266.74Jatrorrhizine
CAS :Jatrorrhizine (neprotin) is a protoberberine alkaloid isolated from Enantia chlorantha (Annonaceae) and other species.Formule :C20H20NO4Degré de pureté :97.18% - 99.06%Couleur et forme :SolidMasse moléculaire :338.38Taprenepag
CAS :Taprenepag (CP-544326) (CP-544326) is a potent and selective prostaglandin E2 receptor agonist (EC50 = 2.8 nM).Formule :C24H22N4O5SDegré de pureté :98.89% - 99.15%Couleur et forme :SolidMasse moléculaire :478.52Ref: TM-T3174
1mg34,00€5mg62,00€1mL*10mM (DMSO)66,00€10mg92,00€25mg178,00€50mg295,00€100mg425,00€200mg595,00€LY 78335
CAS :LY 78335 (1-(2,3-Dichlorophenyl)ethanamine hydrochloride) is a phenylethanolamine-N-methyltransferase (PNMT) inhibitor.Formule :C8H10Cl3NDegré de pureté :99.30% - 99.81%Couleur et forme :SolidMasse moléculaire :226.539-Ethyladenine
CAS :9-Ethyladenine (6-Amino-9-ethylpurine) is a partially potent APRT (adenine phosphoribosyltransferase) inhibitor [1].Formule :C7H9N5Degré de pureté :99.35% - 99.37%Couleur et forme :SolidMasse moléculaire :163.18Fabomotizole
CAS :Fabomotizole (Obenoxazine) is an anxiolytic drug; produces anxiolytic and neuroprotective effects without any sedative or muscle relaxant actions.Formule :C15H21N3O2SDegré de pureté :99.4%Couleur et forme :SolidMasse moléculaire :307.412-ATHBI
CAS :2-ATHBI is a S1P lyase inhibitor.Formule :C9H14N2O5Degré de pureté :99.10%Couleur et forme :SolidMasse moléculaire :230.22TCS 1102
CAS :TCS 1102 is an effective, dual orexin receptor antagonist (Ki: 0.2/3 nM for OX2/1 receptors).Formule :C27H26N4O2SDegré de pureté :99.35% - 99.52%Couleur et forme :SolidMasse moléculaire :470.59Tribenoside
CAS :Tribenoside (BG-356) is a vasoprotectant with mild anti-inflammatory, analgesic, and wound healing properties.Formule :C29H34O6Degré de pureté :≥98%Couleur et forme :LiquidMasse moléculaire :478.58ARN272
CAS :ARN272 is a FAAH-like anandamide transporter (FLAT) inhibitor (IC50: 1.8 μM).Formule :C27H20N4O2Degré de pureté :98.23%Couleur et forme :SolidMasse moléculaire :432.47Endothelin-2 (49-69), human
CAS :Endothelin-2 (49-69), human (Human endothelin-2) is a 21-amino acid vasoactive peptide that binds to G-protein-linked transmembrane receptors, ET-RA and ET-RB.Formule :C115H160N26O32S4Degré de pureté :98.26%Couleur et forme :SolidMasse moléculaire :2546.92Reboxetine
CAS :Reboxetine (Norebox) is an antidepressant drug used in the treatment of clinical depression, panic disorder and ADD/ADHD.Formule :C19H23NO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :313.39Emorfazone
CAS :Emorfazone (PH011085) has an anti-nociceptive effect.Formule :C11H17N3O3Degré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :239.27Ref: TM-T9132
1mg84,00€1mL*10mM (DMSO)152,00€5mg168,00€10mg245,00€25mg404,00€50mg567,00€100mg767,00€200mg1.018,00€Opromazine hydrochloride
CAS :Opromazine hydrochloride, a phenothiazine antipsychotic, blocks brain dopamine receptors to treat schizophrenia and psychosis.Formule :C17H20Cl2N2OSDegré de pureté :98.03%Couleur et forme :SolidMasse moléculaire :371.32Ref: TM-T50054
1mg38,00€5mg82,00€1mL*10mM (DMSO)94,00€10mg111,00€25mg182,00€50mg269,00€100mg389,00€200mg555,00€EST64454 Maleic acid salt
CAS :EST64454 Maleic acid salt, a σ1 receptor antagonist, is a pain treatment candidate with high solubility.Formule :C22H26F2N4O6Degré de pureté :97.54%Couleur et forme :SolidMasse moléculaire :480.46Ref: TM-T9306
1mg84,00€5mg168,00€1mL*10mM (DMSO)197,00€10mg245,00€25mg404,00€50mg567,00€100mg767,00€200mg1.018,00€Darbufelone mesylate
CAS :Darbufelone mesylate blocks PGF2α, LTB4, PGHS-2 (IC50: 0.19 μM), and PGHS-1 (IC50: 20 μM).Formule :C19H28N2O5S2Degré de pureté :96.81% - 99.92%Couleur et forme :SolidMasse moléculaire :428.57Ref: TM-T10960L
1mg50,00€5mg99,00€1mL*10mM (DMSO)109,00€10mg167,00€25mg340,00€50mg557,00€100mg790,00€200mg1.063,00€Otenabant
CAS :Otenabant (CP-945598) has been investigated for the treatment of Obesity.Formule :C25H25Cl2N7ODegré de pureté :99.43%Couleur et forme :SolidMasse moléculaire :510.42GSK163090
CAS :GSK163090 is a specific and orally active 5-HT1A/B/D receptor antagonist (pKis: 9.4/8.5/9.7, and 6.3/6.7 for 5-HT1A/B/D, and dopamine D2/D3).Formule :C25H29N5ODegré de pureté :99.2%Couleur et forme :SolidMasse moléculaire :415.53Ref: TM-TQ0311
25mgÀ demander50mgÀ demander1mg34,00€2mg49,00€5mg75,00€1mL*10mM (DMSO)82,00€10mg118,00€Alprenolol benzoate
CAS :Alprenolol benzoate is the benzoate salt of Alprenolol -- a beta blocker.Formule :C22H29NO4Couleur et forme :SolidMasse moléculaire :371.48Tianeptine
CAS :Tianeptine (Tianeptine sodium) 是一种选择性5-HT 摄取促进剂，具有抗抑郁、抗焦虑和神经保护作用，可用于缓解疼痛的研究。Formule :C21H25ClN2O4SDegré de pureté :99.04%Couleur et forme :SolidMasse moléculaire :436.95Bromopride hydrochloride
CAS :Bromopride HCl: Salt of a D2 blocker used for upper GI disorders, like dyspepsia and emesis.Formule :C14H23BrClN3O2Couleur et forme :SolidMasse moléculaire :380.71PRX-08066
CAS :PRX-08066 is a selective 5-hydroxytryptamine receptor 2B (5-HT2BR, IC50= 3.4 nM) antagonist that induces selective vasodilation of pulmonary arteries.Formule :C19H17ClFN5SDegré de pureté :97.79% - 98.07%Couleur et forme :SolidMasse moléculaire :401.89Ref: TM-T16669
1mg57,00€1mL*10mM (DMSO)105,00€5mg113,00€10mg166,00€25mg333,00€50mg495,00€100mg710,00€200mg973,00€Zacopride hydrochloride
CAS :Zacopride is a highly potent 5-HT3 receptor antagonist (Kd = 0.38 nM) and 5-HT4 receptor agonist (Ki = 373 nM). It also is a selective IK1 channel agonist.Formule :C15H20ClN3O2·HClDegré de pureté :98.32%Couleur et forme :SolidMasse moléculaire :346.26Ref: TM-T5336
1mg34,00€5mg71,00€1mL*10mM (DMSO)79,00€10mg99,00€25mg212,00€50mg385,00€100mg618,00€200mg859,00€[Lys8, Lys9]-Neurotensin (8-13) acetate
[Lys8, Lys9]-Neurotensin (8-13) acetate, a Neurotensin analog, exerts its analgesic effects through activation of the G protein-coupled receptors NTS1 and NTS2Formule :C40H68N8O10Degré de pureté :99.31%Couleur et forme :SolidMasse moléculaire :821.02Ref: TM-T38807L
1mL*10mM (DMSO)À demander1mg87,00€2mg124,00€5mg187,00€10mg284,00€25mg452,00€50mg645,00€100mg867,00€200mg1.159,00€Facinicline (free base)
CAS :Facinicline (free base) is a partial agonist of the nicotinic alpha-7 (α7) receptor. It is used for the oral treatment of Alzheimer's.Formule :C15H18N4OCouleur et forme :SolidMasse moléculaire :270.33Carmoxirole (free base)
CAS :Carmoxirole: a dopamine D2 agonist, reduces pre-load/afterload, aids heart failure, lowers blood pressure by inhibiting noradrenaline release.Formule :C24H26N2O2Couleur et forme :SolidMasse moléculaire :374.48Milveterol
CAS :Milveterol is a long-acting β(2)-adrenoceptor agonist.Formule :C25H29N3O4Couleur et forme :SolidMasse moléculaire :435.52Vicriviroc
CAS :Vicriviroc, also known as MK4176 is a CCR5 antagonist.Formule :C28H38F3N5O2Couleur et forme :SolidMasse moléculaire :533.63Batefenterol Succinate
CAS :Batefenterol Succinate is a first-in-class inhaled bifunctional bronchodilator possessing muscarinic receptor antagonist and β2-adrenoceptor agonist properties.Formule :C44H48ClN5O11Couleur et forme :SolidMasse moléculaire :858.34Vortioxetine
CAS :Vortioxetine (Lu AA 21004) is a serotonergic antidepressant used for major depression disorders.Formule :C18H22N2SDegré de pureté :99.34% - 99.34%Couleur et forme :SolidMasse moléculaire :298.45Ref: TM-T2395
1mL*10mM (DMSO)46,00€10mg48,00€25mg65,00€50mg90,00€100mg117,00€200mg203,00€500mg333,00€1g477,00€PF-06882961 Tris
CAS :PF-06882961 Tris (UNII-2HJV78O0SS) is an orally bioavailable glucagon-like peptide-1 receptor (GLP-1R) agonist.Formule :C35H41FN6O7Degré de pureté :98.74% - 99.79%Couleur et forme :SolidMasse moléculaire :676.7Tecalcet Free Base
CAS :Tecalcet Free Base is an oral calcium receptor agonistFormule :C18H22ClNOCouleur et forme :SolidMasse moléculaire :303.83Clebopride
CAS :Clebopride is antidopaminergic. Clebopride also has an effect of antiemetic.Formule :C20H24ClN3O2Couleur et forme :SolidMasse moléculaire :373.88Evatanepag sodium
CAS :Evatanepag (CP-533536), an EP2-specific PGE2 agonist, promotes bone growth and heals fractures in rats with a single dose.Formule :C25H27N2NaO5SCouleur et forme :SolidMasse moléculaire :490.55Atrasentan sodium
CAS :Atrasentan (ABT-627) is an oral ETA receptor blocker with potential cancer-fighting properties, inhibiting angiogenesis and tumor growth.Formule :C29H37N2NaO6Couleur et forme :SolidMasse moléculaire :532.61Exo1
CAS :Exo1 is an inhibitor of the exocytic pathwayFormule :C15H12FNO3Degré de pureté :98.75%Couleur et forme :SolidMasse moléculaire :273.26Prazosin
CAS :Prazosin (Prazosine), an α1-blocker, acts as an inverse agonist at alpha-1 adrenergic receptors and is used to treat hypertension.
Formule :C19H21N5O4Degré de pureté :99.86%Couleur et forme :White To Tan Powder SolidMasse moléculaire :383.4Olanzapine HCl
CAS :Olanzapine HCl, an FDA-approved atypical antipsychotic for schizophrenia and bipolar disorder, resembles clozapine and quetiapine.Formule :C17H21ClN4SCouleur et forme :SolidMasse moléculaire :348.89MK-571 sodium
CAS :MK-571 sodium, a CysLT1 antagonist and MRP2 inhibitor, obstructs drug efflux and hampers enterocyte phase-2 conjugation of flavonoids.Formule :C26H27ClN2O3S2·NaDegré de pureté :97.86% - 99.58%Couleur et forme :SolidMasse moléculaire :537.07SKF 38393 hydrochloride
CAS :SKF 38393 hydrochloride (SKF38393 HCl) is a selective dopamine D1/D5 receptor agonist.Formule :C16H17NO2·HClDegré de pureté :99.1% - 99.51%Couleur et forme :SolidMasse moléculaire :291.77MEN 10207 acetate
MEN 10207 acetate is a selective antagonist for NK-2 tachykinin receptor.Formule :C59H72N14O12Degré de pureté :99.18%Couleur et forme :SolidMasse moléculaire :1169.29[Leu31,Pro34]-Neuropeptide Y (porcine)
CAS :[Leu31,Pro34]-Neuropeptide Y (porcine), is a selective and high affinity agonist of neuropeptide Y (NPY) Y1 receptor with anxiolytic effects.Formule :C190H286N54O56Degré de pureté :99.39%Couleur et forme :SolidMasse moléculaire :4223Isocorynoxeine
CAS :Isocorynoxeine reduces blood pressure, dilates vessels, and guards neurons against ischemia and glutamate toxicity.Formule :C22H26N2O4Degré de pureté :98% - 99.9%Couleur et forme :SolidMasse moléculaire :382.45Ref: TM-T6S0654
1mg62,00€2mg89,00€5mg132,00€1mL*10mM (DMSO)146,00€10mg226,00€25mg384,00€50mg557,00€100mg785,00€200mg1.054,00€Eprazinone dihydrochloride
CAS :Eprazinone dihydrochloride (NSC 317935) is a mucolytic with antitussive and mucolytic effect.Formule :C24H32N2O2·2HClDegré de pureté :99.25%Couleur et forme :A White Or Almost White CrysMasse moléculaire :453.44Azaperone
CAS :Azaperone, a sedative and antiemetic veterinary tranquilizer, belongs to pyridinylpiperazine and butyrophenone classes.Formule :C19H22FN3ODegré de pureté :98.73%Couleur et forme :White Or Off-White CrystallineMasse moléculaire :327.4Melanin Concentrating Hormone, salmon acetate
Melanin Concentrating Hormone, salmon acetate (MCH (salmon)) is a 19 amino acid cyclic peptide, is largely expressed in the hypothalamus.Formule :C91H143N27O26S4Degré de pureté :99.41%Couleur et forme :SolidMasse moléculaire :2157Rizatriptan sulfate
CAS :Rizatriptan sulfate is a selective serotonin 5-HTID receptor agonist derived from tryptamine.Formule :C15H21N5O4SCouleur et forme :SolidMasse moléculaire :367.42NLX-204 hydrochloride(2170405-10-2 free base)
NLX-204 hydrochloride is a potent and selective ERK1/2 phosphorylation-preferring serotonin 5 HT1A receptor agonist(pKi = 10.19).Formule :C20H23Cl2F2N3O2Degré de pureté :99.59%Couleur et forme :SolidMasse moléculaire :446.32CGP 71683 (free base)
CAS :CGP 71683 (free base) is a potent and highly selective non-peptide antagonist of the NPY Y(5) receptor in the study of obesity.Formule :C26H29N5O2SCouleur et forme :SolidMasse moléculaire :475.61Mini Gastrin I, human acetate
Mini Gastrin I, human acetate is a shorter version of human gastrin, consists of amino acids 5-17 of the parent peptide.Formule :C76H103N15O28SDegré de pureté :99.35% - 99.82%Couleur et forme :SolidMasse moléculaire :1706.78Taminadenant mesylate
CAS :Taminadenant (PBF-509/NIR-178) is an oral adenosine A2A receptor antagonist that activates T-cells to target tumor cells.Formule :C11H12BrN7O3SCouleur et forme :SolidMasse moléculaire :402.227Adoprazine hydrochloride
CAS :Adoprazine hydrochloride is a dopamine D2 receptor antagonist and 5-HT1A receptor agonist potential antipsychotic drug.Formule :C24H25ClFN3O2Couleur et forme :SolidMasse moléculaire :441.93Tetracosactide
CAS :Tetracosactide, a synthetic peptide, mirrors the 24-amino acid start of ACTH with sequence SYSMEHFRWGKPVGKKRRPVKVYP.Formule :C136H210N40O31SDegré de pureté :99.91%Couleur et forme :SolidMasse moléculaire :2933.44Pizuglanstat
CAS :Pizuglanstat is a hematopoietic prostaglandin synthase inhibitor.Formule :C27H36N6O4Degré de pureté :99.62%Couleur et forme :SolidMasse moléculaire :508.61SB-423562 HCl
CAS :SB-423562 is a calcium-sensing receptor antagonist.Formule :C26H33ClN2O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :473Betahistine EP Impurity C
CAS :Betahistine EP Impurity C (NSC19005) is structurally related to Betahistine. Betahistine EP Impurity C is a dimer of Betahistine.Formule :C15H19N3Degré de pureté :99.93% - ≥95%Couleur et forme :SolidMasse moléculaire :241.33Ataciguat
CAS :Ataciguat (HMR-1766) (HMR-1766) is a potent and specific soluble guanylate cyclase (sGC) activator.Formule :C21H19Cl2N3O6S3Degré de pureté :99.09%Couleur et forme :SolidMasse moléculaire :576.49Dimethocaine
CAS :Dimethocaine (Larocaine) is a local anesthetic which also effects on the central nervous system acting as dopamine-reuptake-inhibitor.Formule :C16H26N2O2Degré de pureté :99.52%Couleur et forme :SolidMasse moléculaire :278.39Rotundine
CAS :Rotundine (Gindarine) (L-tetrahydropalmatine, L-THP) is a selective dopamine D1 receptor antagonist with IC50 of 166 nM.Formule :C21H25NO4Degré de pureté :99.8% - 99.91%Couleur et forme :Off-White SolidMasse moléculaire :355.43Ursodeoxycholic acid sodium
CAS :Ursodeoxycholic acid sodium (Sodium Ursodeoxycholate) is a naturally occurring secondary bile acid with anti-inflammatory and cytoprotective activities.Formule :C24H40NaO4Degré de pureté :99.66% - 99.96%Couleur et forme :SolidMasse moléculaire :415.56BMY 7378 dihydrochloride
CAS :BMY 7378 dihydrochloride (BMY7378 HCl) , α1D-adrenergic receptor antagonist, is a weak partial agonist/antagonist of 5-HT1A receptor.Formule :C22H33Cl2N3O3Degré de pureté :97.32% - 99.08%Couleur et forme :SolidMasse moléculaire :458.42BMS 182874 hydrochloride
CAS :BMS 182874 hydrochloride is a nonpeptide endothelin (El) receptor antagonist.Formule :C17H20ClN3O3SDegré de pureté :97.01%Couleur et forme :SolidMasse moléculaire :381.88Ref: TM-T21790
1mg77,00€2mg92,00€5mg140,00€1mL*10mM (DMSO)146,00€10mg205,00€25mg343,00€50mg477,00€100mg665,00€200mg897,00€5-Benzyloxygramine
CAS :5-Benzyloxygramine blocks the Dopamin receptors and antagonizes the effects of 5-HT on the rat uterus and the rabbit ear.Formule :C18H20N2ODegré de pureté :99.13%Couleur et forme :SolidMasse moléculaire :280.36Detomidine hydrochloride
CAS :Detomidine hydrochloride (MPV-253 AII) produce dose-dependent sedative and analgesic effects, mediatated by activation of α2 catecholamine receptors.Formule :C12H14N2·HClDegré de pureté :99.97%Couleur et forme :SolidMasse moléculaire :222.71[Pyr1]-Apelin-13
CAS :[Pyr1]-Apelin-13 ([pGlu1]-Apelin-13) is a potent and selective endogenous Apelin receptor (APJ) agonist.Formule :C69H108N22O16SDegré de pureté :99.71%Couleur et forme :SolidMasse moléculaire :1533.8VPC171
CAS :VPC171 is a novel adenosine A1 receptor positive allosteric modulator (PAM).Formule :C18H12F3NOSDegré de pureté :99.78%Couleur et forme :SolidMasse moléculaire :347.35Ref: TM-T29112
1mg49,00€1mL*10mM (DMSO)88,00€5mg96,00€10mg124,00€25mg222,00€50mg309,00€100mg439,00€200mg592,00€BAY-545
CAS :BAY-545 is an antagonist of A2B adenosine receptor(IC50 : 59 nM).Formule :C18H22F3N3O4SDegré de pureté :98.05%Couleur et forme :SolidMasse moléculaire :433.45Ref: TM-T8512
1mg84,00€5mg161,00€1mL*10mM (DMSO)172,00€10mg235,00€25mg420,00€50mg605,00€100mg842,00€200mg1.134,00€A2B receptor antagonist 2
CAS :A2B receptor antagonist 2 is an antagonist of adenosine receptor A2B (Ki = 2.30 μM for rA1, 6.8 μM for rA2A, 3.44 μM for hA2B).Formule :C12H15N5Degré de pureté :100%Couleur et forme :SolidMasse moléculaire :229.28[D-Phe12,Leu14]-Bombesin acetate
[D-Phe12,Leu14]-Bombesin acetate inhibits bombesin-stimulated secretion.Formule :C77H118N22O20Degré de pureté :98.41% - 99.14%Couleur et forme :SolidMasse moléculaire :1671.9Regadenoson
CAS :Regadenoson (CVT-3146) is a selective A2A receptor agonist that increases coronary blood flow with a longer half-life than adenosine.Formule :C15H18N8O5Degré de pureté :99.57% - 99.81%Couleur et forme :Off-White SolidMasse moléculaire :390.35Ref: TM-T2671
2mg44,00€5mg62,00€1mL*10mM (DMSO)69,00€10mg96,00€25mg170,00€50mg259,00€100mg394,00€500mg887,00€Ranitidine
CAS :Ranitidine (HSDB 3925) is a non-imidazole blocker of those histamine receptors that mediate gastric secretion (H2 receptors).Formule :C13H22N4O3SDegré de pureté :99.52%Couleur et forme :Solid SolidMasse moléculaire :314.40Ciproxifan maleate
CAS :Ciproxifan maleate (FUB 359)(FUB-359 maleate) is a highly potent and selective histamin H3-receptor antagonist with IC50 of 9.2 nM, with low apparent affinityFormule :C20H22N2O6Degré de pureté :99.39%Couleur et forme :SolidMasse moléculaire :386.4Ref: TM-T2004
1mg40,00€2mg52,00€5mg75,00€1mL*10mM (DMSO)82,00€10mg101,00€25mg205,00€50mg380,00€100mg565,00€Epinastine hydrochloride
CAS :Epinastine hydrochloride (WAL-801CL HCl) is an antihistamine and mast cell stabilizer that is used in eye drops to treat allergic conjunctivitis.Formule :C16H15N3·HClDegré de pureté :99.26% - 99.62%Couleur et forme :White SolidMasse moléculaire :285.77AM095
CAS :AM095 is a potent LPA1 receptor antagonist with IC50 values of 0.98 and 0.73 μM for recombinant human or mouse LPA1 respectively.Formule :C27H23N2NaO5Degré de pureté :98.87%Couleur et forme :SolidMasse moléculaire :478.47Ref: TM-T2000
1mg34,00€2mg44,00€5mg63,00€1mL*10mM (DMSO)66,00€10mg92,00€25mg170,00€50mg268,00€100mg416,00€ATC 0175 free base
CAS :ATC0175 is a potent, orally active MCH1R antagonist with high selectivity over MCH2R, demonstrating antidepressant and anxiolytic effects in animal models.Formule :C23H25F2N5ODegré de pureté :99.73%Couleur et forme :SolidMasse moléculaire :425.47Neurotensin(8-13) 3TFA(60482-95-3(free base))
CAS :Neurotensin(8-13) 3TFA is Neurotensin (NT) fragment. Neurotensin(8-13) 3TFA results in a decrease in cell-surface NT1 receptors (NTR1) density.Formule :C40H65F3N12O10Degré de pureté :98.31%Couleur et forme :SolidMasse moléculaire :931.03Ref: TM-T7617L
1mg35,00€5mg73,00€10mg107,00€1mL*10mM (DMSO)132,00€25mg207,00€50mg313,00€100mg447,00€200mg620,00€4i
CAS :4i (CHEMBL1269981) is a 5-HT3 receptor antagonist,It modulates the serotonergic system.Formule :C16H12ClN3ODegré de pureté :99.49%Couleur et forme :SolidMasse moléculaire :297.74Perospirone
CAS :Perospirone (Lullan) is an antagonist of serotonin 5HT2A receptors and dopamine D2 receptors.Formule :C23H30N4O2SDegré de pureté :99.23%Couleur et forme :White PowderMasse moléculaire :426.57DAPTA
CAS :DAPTA (Adaptavir) is an inhibitor of CCR5, shows potent anti-HIV activities.Formule :C35H56N10O15Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :856.88Neurokinin A(4-10) TFA(97559-35-8 free base)
Neurokinin A(4-10) TFA(97559-35-8 free base) is a tachykinin NK2 receptor agonist[1].Formule :C36H55F3N8O12SDegré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :880.93NPY 5RA972
CAS :NPY 5RA972 is a neuropeptide Y Y5 receptor antagonistFormule :C21H25N3O2Degré de pureté :99.02% - 99.56%Couleur et forme :SolidMasse moléculaire :351.44HPI 1
CAS :HPI 1 suppresses Hh pathway: IC50 = 1.5 μM (Shh, SAG), 4 μM (Gli2), 6 μM (Gli1) in Shh-LIGHT2 cells.Formule :C27H29NO6Degré de pureté :97.6%Couleur et forme :SolidMasse moléculaire :463.52Ref: TM-T22089
1mg44,00€2mg57,00€5mg96,00€1mL*10mM (DMSO)102,00€10mg128,00€25mg207,00€50mg308,00€100mg447,00€500mg973,00€N-Desmethylclozapine
CAS :N-Desmethylclozapine: 5-HT2C antagonist (IC50: 7.1 nM), dopamine D4 antagonist, δ-opioid agonist.Formule :C17H17ClN4Degré de pureté :97.25% - 99.83%Couleur et forme :Yellow Crystalline SolidMasse moléculaire :312.8Ref: TM-T5158
2mg34,00€5mg48,00€1mL*10mM (DMSO)58,00€10mg79,00€25mg152,00€50mg235,00€100mg344,00€200mg490,00€AZD2098
CAS :AZD2098 is a potent CC-chemokine receptor 4 (CCR4) inhibitor used for asthma research.Formule :C11H9Cl2N3O3SDegré de pureté :99.80% - >99.99%Couleur et forme :SolidMasse moléculaire :334.18Ref: TM-T4300
1mg34,00€5mg66,00€1mL*10mM (DMSO)73,00€10mg105,00€25mg217,00€50mg334,00€100mg502,00€500mg1.063,00€AC-55541
CAS :AC-55541 (AOB2796), a PAR2 agonist, activates PAR2 in cellular proliferation assays, phosphatidylinositol hydrolysis assays, and Ca(2+) mobilization assays.
Formule :C25H20BrN5O3Degré de pureté :98% - 99.33%Couleur et forme :SolidMasse moléculaire :518.36Litorin acetate(55749-97-8 Free base)
Litorin acetate, an amphibian bombesin peptide derivative, is an bombesin receptor agonist.Formule :C53H72N14O13SDegré de pureté :98.61%Couleur et forme :SolidMasse moléculaire :1145.29Nitrobenzylthioinosine
CAS :Nitrobenzylthioinosine (NBMPR) is an inhibitor of ENT1 transporter that binds to ENT1 transporter with high affinity.Formule :C17H17N5O6SDegré de pureté :99.69% - 99.74%Couleur et forme :Off-White SolidMasse moléculaire :419.41Chlorprothixene
CAS :Chlorprothixene (Truxal) is a typical antipsychotic drug of the thioxanthene class, which was the first of the series to be synthesized.Formule :C18H18ClNSDegré de pureté :98.77% - 99.756%Couleur et forme :Pale Yellow Crystals SolidMasse moléculaire :315.86LY334370
CAS :LY334370 is a selective 5-HT1F receptor agonist with a Ki of 1.6 nMFormule :C21H22FN3ODegré de pureté :99.32%Couleur et forme :SolidMasse moléculaire :351.42CCG215022
CAS :CCG215022 is a G protein-coupled receptor kinases (GRKs) inhibitor with IC50s of 0.15±0.07 μM, 0.38±0.06 μM and 3.9±1 μM for GRK2, 5 and 1, respectively.Formule :C26H22FN7O3Degré de pureté :97.63% - 99.69%Couleur et forme :SolidMasse moléculaire :499.5Ref: TM-T3498
1mg56,00€5mg114,00€1mL*10mM (DMSO)127,00€10mg178,00€25mg394,00€50mg655,00€100mg1.035,00€Clemizole hydrochloride
CAS :Clemizole hydrochloride blocks H1 histamine receptors and inhibits HCV replication and NS4B RNA binding.Formule :C19H21Cl2N3Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :362.3Vicriviroc maleate
CAS :Vicriviroc maleate (SCH-417690 (maleate))(Sch-417690) is a piperazine-based CCR5 receptor antagonist with activity against human immunodeficiency virus.Formule :C32H42F3N5O6Degré de pureté :98.16% - 98.37%Couleur et forme :SolidMasse moléculaire :649.7JK184
CAS :JK184 is a potent Hedgehog (Hh) pathway inhibitor.
Formule :C19H18N4OSDegré de pureté :98.93% - 99.89%Couleur et forme :SolidMasse moléculaire :350.44AZD-4818
CAS :AZD-4818 (CCR1 antagonist) is a chemokine CCR1 antagonist for the treatment of chronic obstructive pulmonary disease.Formule :C27H32Cl2N2O7Degré de pureté :99.01%Couleur et forme :SolidMasse moléculaire :567.46BX471
CAS :BX471 (BX 471) is a potent, selective non-peptide CCR1 antagonist.Formule :C21H24ClFN4O3Degré de pureté :98% - 99.98%Couleur et forme :SolidMasse moléculaire :434.89Ref: TM-T2375
1mg35,00€5mg86,00€1mL*10mM (DMSO)95,00€10mg117,00€25mg200,00€50mg313,00€100mg489,00€200mg740,00€Glasdegib
CAS :Glasdegib (PF-04449913) (PF-04449913) is a potent, and orally bioavailable Smoothened (Smo) inhibitor with IC50 of 5 nM. Phase 2.Formule :C21H22N6ODegré de pureté :98.72%Couleur et forme :SolidMasse moléculaire :374.44SAG
CAS :SAG (Smoothened Agonist) is a Smo receptor agonist (EC50=3 nM) that is cell-permeable and selective.
Formule :C28H28ClN3OSDegré de pureté :97.37% - 98.88%Couleur et forme :SolidMasse moléculaire :490.06Ciliobrevin A
CAS :Ciliobrevin A (HPI-4) is an inhibitor of hedgehog signaling pathway with an IC50 <10 μM.Formule :C17H9Cl2N3O2Degré de pureté :98.54% - 99.57%Couleur et forme :SolidMasse moléculaire :358.18Ref: TM-T3156
2mg39,00€5mg56,00€1mL*10mM (DMSO)65,00€10mg80,00€25mg165,00€50mg224,00€100mg314,00€200mg467,00€SANT-1
CAS :SANT-1 directly binds to Smoothened (Smo) receptor (Kd: 1.2 nM) and inhibits Smo agonist effects (IC50: 20 nM).Formule :C23H27N5Degré de pureté :99.93% - >99.99%Couleur et forme :SolidMasse moléculaire :373.49SAG hydrochloride (912545-86-9(free base))
CAS :SAG hydrochloride (912545-86-9(free base)) (Smoothened Agonist HCl) acts as an SMO agonist.Formule :C28H29Cl2N3OSDegré de pureté :99.19% - 99.97%Couleur et forme :SolidMasse moléculaire :526.52Ref: TM-T4211
1mg49,00€2mg65,00€5mg90,00€1mL*10mM (DMSO)105,00€10mg114,00€25mg222,00€50mg334,00€100mg502,00€200mg717,00€R243
CAS :R243 is CCR8 signaling and chemotaxis inhibitor.Formule :C21H27NO4Degré de pureté :99.03%Couleur et forme :SolidMasse moléculaire :357.44Ref: TM-T24700
1mg40,00€2mg52,00€5mg80,00€1mL*10mM (DMSO)90,00€10mg117,00€25mg207,00€50mg333,00€100mg495,00€Sonidegib
CAS :Sonidegib (Erismodegib), a Smoothened (Smo) antagonist, inhibits Hedgehog (Hh) signaling with IC50 of 1.3 nM (mouse) and 2.5 nM (human), respectively.Formule :C26H26F3N3O3Degré de pureté :98% - 99.97%Couleur et forme :SolidMasse moléculaire :485.5Salmeterol Xinafoate
CAS :Salmeterol Xinafoate (GR 33343X xinafoate) is a long-acting β2-adrenergic receptor agonist with anti-inflammatory effects, used in the treatment of asthma.Formule :C36H45NO7Degré de pureté :98% - 98.24%Couleur et forme :White SolidMasse moléculaire :603.75MRT-81
CAS :MRT-81 blocks Smo receptors in Shh-light2 cells at 41 nM IC50, showing strong hedgehog pathway inhibition, useful in cancer research.Formule :C31H29N3O5SDegré de pureté :99.72%Couleur et forme :SolidMasse moléculaire :555.64Ref: TM-T9532
1mg46,00€5mg92,00€1mL*10mM (DMSO)110,00€10mg138,00€25mg241,00€50mg349,00€100mg479,00€200mg657,00€BA 1 acetate(183241-31-8 free base)
BA 1 acetate: bombesin agonist, IC50s: 0.26/1.55/2.52 nM (BB1/BB2/BB3), boosts glucose transport, promotes lung cancer cell growth in vitro.Formule :C59H80N14O13Degré de pureté :95.3%Couleur et forme :SolidMasse moléculaire :1193.35Binodenoson
CAS :Binodenoson (WRC 0470), a selective A2A adenosine receptor agonist, aids in coronary imaging.Formule :C17H25N7O4Degré de pureté :99.74%Couleur et forme :SolidMasse moléculaire :391.42Ref: TM-T9516
1mg94,00€5mg222,00€1mL*10mM (DMSO)245,00€10mg334,00€25mg557,00€50mg745,00€100mg1.044,00€Lecirelin acetate(61012-19-9 free base)
Lecirelin acetate is a synthetic GnRH (gonadotropin releasing hormone) analogue which shows a great efficacy in the treatment of bovine ovarian follicular cystsFormule :C61H88N16O14Degré de pureté :98.1%Couleur et forme :SolidMasse moléculaire :1269.45Phenylbiguanide
CAS :Phenylbiguanide (N-Phenylbiguanide) is a 5-HT3 receptor selective agonist(EC50 : 3.0±0.1 μM)Formule :C8H11N5Degré de pureté :99.54%Couleur et forme :SolidMasse moléculaire :177.21Lys-[Des-Arg9]Bradykinin acetate
Lys-[Des-Arg9]Bradykinin acetate is an endogenous potent and highly selective bradykinin B1 receptor agonist (Ki values are 0.12 and > 30000 nM at human B1 andFormule :C52H77N13O13Degré de pureté :99.93%Couleur et forme :SolidMasse moléculaire :1092.27I-191
CAS :I-191 is a potent antagonist of protease-activated receptor 2 (PAR2), inhibits multiple signaling functions in human cancer cells.Formule :C23H26FN5O2Degré de pureté :99.8%Couleur et forme :SolidMasse moléculaire :423.48AM966
CAS :AM966, a excellent affinity, specific, oral LPA1(IC50=17 nM) antagonist, suppresses LPA-stimulated intracellular calcium release.Formule :C27H23ClN2O5Degré de pureté :98.06% - 99.79%Couleur et forme :SolidMasse moléculaire :490.93Lurasidone hydrochloride
CAS :Lurasidone HCl: Atypical antipsychotic, treats schizophrenia & bipolar, affects dopamine, serotonin & adrenergic receptors.Formule :C28H36N4O2S·HClDegré de pureté :99.51%Couleur et forme :SolidMasse moléculaire :529.14Ref: TM-T1735
5mg39,00€1mL*10mM (DMSO)54,00€10mg59,00€25mg75,00€50mg90,00€100mg137,00€200mg213,00€500mg447,00€2-Pyridylethylamine dihydrochloride
CAS :2-Pyridylethylamine dihydrochloride is a Histamine H1 receptor agonist.Formule :C7H12Cl2N2Degré de pureté :99.42%Couleur et forme :SolidMasse moléculaire :195.09Motilin (26-47), human, porcine
CAS :Motilin (26-47) binds Motilin receptors in hamster cells; Ki=2.3 nM, EC50=0.3 nM; same for humans, pigs.Formule :C120H188N34O35SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :2699.07Ref: TM-TP1425
500µg86,00€1mg111,00€5mg334,00€10mg504,00€25mg745,00€50mg999,00€100mg1.341,00€200mg1.773,00€LIXIVAPTAN
CAS :Lixivaptan (VPA-985) is an orally active and selective vasopressin receptor V2 antagonist(Ki = 2.3 nM)Formule :C27H21ClFN3O2Degré de pureté :98.36%Couleur et forme :SolidMasse moléculaire :473.93Ref: TM-T7303
2mg34,00€5mg66,00€1mL*10mM (DMSO)70,00€10mg99,00€25mg205,00€50mg334,00€100mg522,00€200mg743,00€GLP-1(7-36), amide
CAS :GLP-1 secretion by human enteroendocrine NCI-H716 cells is augmented in a dose-dependent manner by the addition of CPE.Cost-effective and quality-assured.Formule :C149H226N40O45Degré de pureté :99.85%Couleur et forme :White PowderMasse moléculaire :3297.63FSLLRY-NH2 TFA(245329-02-6 free base)
FSLLRY-NH2 TFA inhibits PAR2, reverses taxol-induced pain, and reduces itch in mice; blocks ERK and collagen in fibroblasts.Formule :C41H61F3N10O10Degré de pureté :99.32%Couleur et forme :SolidMasse moléculaire :910.99PF-04418948
CAS :PF-04418948 is a potent EP2 receptor antagonist. Displays over 2000-fold selectivity for EP2 receptors over EP1, EP3, EP4, DP1 amd CRTH2 receptors.Formule :C23H20FNO5Degré de pureté :98.67% - 99.45%Couleur et forme :SolidMasse moléculaire :409.41d[Cha4]-AVP acetate(500170-27-4 free base)
'd[Cha4]-AVP acetate: strong V1B agonist, weak on V1A/Oxytocin/V2. Boosts ACTH, corticosterone; low blood pressure effect.'Formule :C52H75N13O13S2Degré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :1154.37Brexpiprazole
CAS :Brexpiprazole (OPC-34712) is a partial agonist of human 5-hydroxytryptamine (5-HT) 5-HT1A and dopamine D2 receptors.Formule :C25H27N3O2SDegré de pureté :99.06% - 99.96%Couleur et forme :SolidMasse moléculaire :433.57Ref: TM-T2306
1mL*10mM (DMSO)À demander5mg50,00€10mg63,00€25mg75,00€50mg88,00€100mg94,00€200mg140,00€500mg259,00€Urapidil
CAS :Urapidil (Ebrantil), a sympatholytic antihypertensive drug, acts as a 5-HT1A receptor agonist and as an α1-adrenoceptor antagonist.Formule :C20H29N5O3Degré de pureté :99.85% - >99.99%Couleur et forme :SolidMasse moléculaire :387.48Norepinephrine bitartrate salt
CAS :Norepinephrine bitartrate salt is an adrenergic neurotransmitter.Formule :C12H17NO9Degré de pureté :97.32% - 99.97%Couleur et forme :SolidMasse moléculaire :319.27Perospirone hydrochloride
CAS :Perospirone hydrochloride (Perospirone HCl) is an atypical antipsychotic agent for the treatment of schizophrenia.Formule :C23H31ClN4O2SDegré de pureté :99.37%Couleur et forme :White SolidMasse moléculaire :463Serotonin
CAS :Serotonin (5-hydroxytryptamine) is a monoamine neurotransmitter in the CNS and an endogenous 5-HT receptor agonist. High-Quality, Low-Cost!Formule :C10H12N2ODegré de pureté :97.47% - 99.92%Couleur et forme :SolidMasse moléculaire :176.22Melatonin
CAS :Melatonin (Melatonine) is a natural hormone that activates melatonin receptors. Melatonin regulates the biological clock. Cost-effective and quality-assured.Formule :C13H16N2O2Degré de pureté :98% - 99.89%Couleur et forme :Pale Yellow Leaflets From Benzene SolidMasse moléculaire :232.28Verucerfont
CAS :Verucerfont (NBI77860) is an antagonist of corticotropin-releasing factor receptor 1 (CRF1) .Formule :C22H26N6O2Degré de pureté :99.90%Couleur et forme :SolidMasse moléculaire :406.48Ref: TM-T7361
1mg60,00€2mg87,00€5mg130,00€1mL*10mM (DMSO)142,00€10mg205,00€25mg376,00€50mg573,00€100mg803,00€
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