GPCR/G-Protéine
Les inhibiteurs des GPCR/protéines G sont des composés qui ciblent les récepteurs couplés aux protéines G (GPCR) et les protéines G associées, qui jouent un rôle crucial dans la transmission des signaux de l'extérieur vers l'intérieur des cellules. Ces inhibiteurs sont essentiels pour étudier les voies de signalisation médiées par les GPCR, impliquées dans de nombreux processus physiologiques, y compris la perception sensorielle, la réponse immunitaire et la neurotransmission. Les inhibiteurs des GPCR sont également importants dans le développement de médicaments, car de nombreux agents thérapeutiques ciblent ces récepteurs. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de GPCR/protéines G de haute qualité pour soutenir vos recherches en pharmacologie, biologie cellulaire et domaines connexes.
Sous-catégories appartenant à la catégorie "GPCR/G-Protéine"
- récepteur 5-HT(1.025 produits)
- Récepteur d'adénosine(251 produits)
- Récepteur adrénergique(3.027 produits)
- Récepteur de la bombésine(35 produits)
- Récepteur de la bradykinine(61 produits)
- CXCR(158 produits)
- CaSR(34 produits)
- Récepteur cannabinoïde(218 produits)
- Cholécystokinine(1 produits)
- Récepteur de la dopamine(445 produits)
- Récepteur de l'endothéline(86 produits)
- Récepteur GNRH(84 produits)
- GPCR19(36 produits)
- GRK(33 produits)
- GTPase(23 produits)
- Récepteur du glucagon(195 produits)
- Hérisson/Smoothened(49 produits)
- Récepteur de l'histamine(385 produits)
- Récepteur LPA(21 produits)
- Récepteur de la mélatonine(26 produits)
- Récepteur OX(41 produits)
- Récepteur opioïde(327 produits)
- PAFR(14 produits)
- PKA(60 produits)
- Récepteur S1P(18 produits)
- SGLT(31 produits)
- Récepteur Sigma(46 produits)
Affichez 19 plus de sous-catégories
6011 produits trouvés pour "GPCR/G-Protéine"
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Bevantolol hydrochloride
CAS :Bevantolol hydrochloride (NC-1400 hydrochloride) is a β1-adrenoceptor antagonist that treatment angina pectoris and hypertension.Formule :C20H28ClNO4Degré de pureté :99.49%Couleur et forme :SolidMasse moléculaire :381.9Pimozide
CAS :Pimozide: antipsychotic that blocks type 2 dopamine, alpha-adrenergic, and 5-HT2 receptors, reducing tics and delusions.Formule :C28H29F2N3ODegré de pureté :99.63% - >99.99%Couleur et forme :SolidMasse moléculaire :461.55Chlorphenesin
CAS :Chlorphenesin (Chlorophenesin) is an antigen-associated immunosuppressant that inhibits IgE-mediated histamine release. It is also used as an antimycotic agent.Formule :C9H11ClO3Degré de pureté :99.59%Couleur et forme :SolidMasse moléculaire :202.63SBI-115
CAS :SBI-115 is an antagonist of TGR5. SBI-115 decreases hepatic cystogenesis with polycystic liver diseases via inhibiting TGR5Formule :C14H13ClN2O4SDegré de pureté :99.53% - 99.78%Couleur et forme :SolidMasse moléculaire :340.78ZK 756326
CAS :ZK 756326: Selective CCR8 agonist, IC50 1.8 μM (human), 2.6 μM (mouse), no CCR4/5, CXCR3/4 action, 28-fold selectivity vs 26 GPCRs, anti-HIV fusion.Formule :C21H28N2O3Degré de pureté :99.43%Couleur et forme :SolidMasse moléculaire :356.46Clemizole
CAS :Clemizole is an H1 histamine receptor antagonist, can inhibit NS4B's RNA binding and hepatitis C virus (HCV) replication.Formule :C19H20ClN3Degré de pureté :98% - 99.65%Couleur et forme :SolidMasse moléculaire :325.84Ref: TM-T1822
1mg42,00€5mg82,00€1mL*10mM (DMSO)93,00€10mg101,00€25mg152,00€50mg256,00€100mg460,00€500mg973,00€Taladegib
CAS :Taladegib (LY2940680), an oral Smo receptor antagonist, targets Hedgehog signaling for cancer treatment.Formule :C26H24F4N6ODegré de pureté :98.75% - >99.99%Couleur et forme :SolidMasse moléculaire :512.5Nitrobenzylthioinosine
CAS :Nitrobenzylthioinosine (NBMPR) is an inhibitor of ENT1 transporter that binds to ENT1 transporter with high affinity.Formule :C17H17N5O6SDegré de pureté :99.69% - 99.74%Couleur et forme :Off-White SolidMasse moléculaire :419.41(E)-3,4,5-Trimethoxycinnamic acid
CAS :(E)-3,4,5-Trimethoxycinnamic acid (O-Methylsinapic acid) is a natural product from the roots and rhizomes of Notopterygium incisum.Formule :C12H14O5Degré de pureté :99.83%Couleur et forme :SolidMasse moléculaire :238.24[Sar9] Substance P acetate(77128-75-7 free base)
[Sar9]-Substance P acetate, an NK-1 receptor agonist, mimics SP's effect on progesterone metabolism.Formule :C66H104N18O15SDegré de pureté :96.67%Couleur et forme :SolidMasse moléculaire :1421.71Amitriptyline
CAS :Amitriptyline: a tricyclic antidepressant used for depression and neuropathic pain.Formule :C20H23NDegré de pureté :98.24% - 99.64%Couleur et forme :Crystals SolidMasse moléculaire :277.4Neuropeptide S (Mouse) acetate
Neuropeptide S (Mouse) acetate is a bioactive peptide.Formule :C95H160N34O29Degré de pureté :98.25%Couleur et forme :SolidMasse moléculaire :2242.5MIPS521
CAS :MIPS521 ({2-Amino-4-[3,5-bis(trifluoromethyl)phenyl]thiophen-3-yl}(4-chlorophenyl)methanone) is a positive allosteric modulator of the A1R.Formule :C19H10ClF6NOSDegré de pureté :99.76%Couleur et forme :SolidMasse moléculaire :449.8Ref: TM-T9330
1mg35,00€2mg50,00€5mg74,00€1mL*10mM (DMSO)82,00€10mg105,00€25mg178,00€50mg313,00€100mg485,00€LP-211
CAS :LP-211 is a brain penetrant selective agonist for a 5-HT7 receptor (Ki: 0.58 nM), and >300-fold selectivity over the 5-HT1A receptor.Formule :C30H34N4ODegré de pureté :98.65%Couleur et forme :SolidMasse moléculaire :466.62Ref: TM-T5387
2mg44,00€5mg66,00€1mL*10mM (DMSO)73,00€10mg90,00€25mg170,00€50mg289,00€100mg462,00€200mg658,00€Pramipexole dihydrochloride hydrate
CAS :Pramipexole dihydrochloride hydrate (Mirapex) is a selective, blood-brain barrier-crossing D2 dopamine receptor agonist, and is used in the study of PD.Formule :C10H17N3S·2HCl·H2ODegré de pureté :99.68%Couleur et forme :White To Off-White Crystalline PowderMasse moléculaire :302.26Ref: TM-T6951
10mg44,00€1mL*10mM (DMSO)44,00€25mg71,00€50mg113,00€100mg166,00€200mg241,00€500mg408,00€Fexofenadine
CAS :Fexofenadine, a non-sedating antihistamine, treats allergies like hay fever and urticaria.Formule :C32H39NO4Degré de pureté :99.35%Couleur et forme :White To Off-White SolidMasse moléculaire :501.66PEN (human) aceate
PEN (human) aceate, one of the most abundant hypothalamic neuropeptide and derived from the proprotein ProSAAS, is an endogenous ligand of GPR83.Formule :C99H163N27O34Degré de pureté :99.25%Couleur et forme :SolidMasse moléculaire :2275.51Bradykinin (2-9)
CAS :Bradykinin (2-9) (Des-Arg1-bradykinin) is an amino-truncated peptide compound that is a metabolite of Bradykinin.Formule :C44H61N11O10Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :904.02Ref: TM-TP1181
1mg39,00€5mg88,00€10mg130,00€1mL*10mM (DMSO)144,00€25mg210,00€50mg313,00€100mg464,00€200mg660,00€Terazosin hydrochloride dihydrate
CAS :Terazosin hydrochloride dihydrate (Heitrin dihydrate) is a selective α1-adrenoceptor antagonist, used for treatment of symptoms of an enlarged prostate (BPH).Formule :C19H25N5O4·HCl·2H2ODegré de pureté :99.81%Couleur et forme :White Or Off-White Crystalline PowderMasse moléculaire :459.92CB1 antagonist 4
CAS :TM38837 is an antagonist of cannabinoid receptor type 1 (CB1), with potential for the treatment of obesity and type 2 diabetes.Formule :C30H25Cl2F3N4OSDegré de pureté :98.97%Couleur et forme :SolidMasse moléculaire :617.51Ref: TM-T8511
2mg46,00€5mg92,00€10mg152,00€1mL*10mM (DMSO)155,00€25mg259,00€50mg405,00€100mg597,00€200mg848,00€MK-3697
CAS :MK-3697, an isonicotinamide small molecule, acts as a potent and selective Orexin 2 receptor antagonist (Ki: 0.95 nM).Formule :C23H21N5O3SDegré de pureté :97.69% - 98.15%Couleur et forme :SolidMasse moléculaire :447.51Ref: TM-T1913
1mg49,00€2mg65,00€5mg90,00€1mL*10mM (DMSO)100,00€10mg113,00€25mg200,00€50mg333,00€100mg477,00€Talnetant hydrochloride
CAS :Talnetant (SB 223412) hydrochloride, an NK3 antagonist, selectively binds hNK-3 at 1.4 nM, much less to hNK-2, none to hNK-1 at 100 μM.Formule :C25H23ClN2O2Couleur et forme :SolidMasse moléculaire :418.92Quipazine
CAS :Quipazine: 5-HT agonist, Ki 1.4 nM at 5-HT3R, anti-SARS-CoV-2 (EC50 31.64 μM), for neurological research.Formule :C13H15N3Couleur et forme :SolidMasse moléculaire :213.28Raclopride tartrate
CAS :Raclopride is a selective antagonist on D2 dopamine receptor ( D2 Ki: 1.8 nm, D3 Ki: 3.5 nm, D4 Ki: 2400, D1 Ki: 18000 nM).Formule :C19H26Cl2N2O9Couleur et forme :SolidMasse moléculaire :497.32Urotensin I acetate (83930-33-0 Free base)
Urotensin I acetate, CRF1/CRF2 agonist: pEC50s - hCRF1 11.46, hCRF2 9.36, rCRF2α 9.85; KIs - hCRF1 0.4 nM, rCRF2α 1.8 nM, mCRF2β 5.7 nM.Degré de pureté :95.44% - 99.73%Couleur et forme :SolidMasse moléculaire :N/ABay 55-9837 acetate
Bay 55-9837 acetate is a potent and highly selective VPAC2 agonist(Kd = 0.65 nM) and can be used in type 2 diabetes studies.Degré de pureté :98.27%Couleur et forme :LiquidMasse moléculaire :N/AGSK 789472 hydrochloride
CAS :GSK 789472 hydrochloride is both a dopamine D3 receptor antagonist and a D2 partial agonist.Formule :C15H22ClN3ODegré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :295.81N-ACETYLTRYPTAMINE
CAS :N-ACETYLTRYPTAMINE is a partial agonist for melatonin receptors in the retina. Also used for determination of serotonin N-acetyl transferase.Formule :C12H14N2ODegré de pureté :98.79%Couleur et forme :PowderMasse moléculaire :202.25CYM-5520
CAS :CYM-5520 is a noncompetitive allosteric agonist of S1P2Formule :C21H19N3O2Degré de pureté :99.47%Couleur et forme :SolidMasse moléculaire :345.39Ref: TM-T22703
1mg46,00€2mg60,00€5mg88,00€1mL*10mM (DMSO)98,00€10mg135,00€25mg236,00€50mg354,00€100mg528,00€Bevantolol
CAS :Bevantolol, a selective β-1 adrenoceptor antagonist, is utilized for the investigation of angina pectoris and hypertension [1].Formule :C20H27NO4Couleur et forme :SolidMasse moléculaire :345.43Sigma-LIGAND-1 hydrochloride
CAS :Sigma-LIGAND-1 HCl: selective sigma receptor ligand; DTG IC50: 16 nM, PPP IC50: 19 nM; weak D2 receptor affinity, Ki: 4000 nM.Formule :C27H34ClNO4Couleur et forme :SolidMasse moléculaire :472.02Niaprazine
CAS :Niaprazine is a histamine H1-receptor antagonist with marked sedative properties.Formule :C20H25FN4ODegré de pureté :99.56%Couleur et forme :SolidMasse moléculaire :356.44ML-193
CAS :ML-193: GPR55 antagonist, IC50 221nM, 27x selective over GPR35/CB1/CB2, may aid Parkinson's symptoms.Formule :C28H25N5O4SDegré de pureté :97.74%Couleur et forme :SolidMasse moléculaire :527.59Prucalopride Succinate
CAS :Prucalopride Succinate is a 5-HT4 receptor agonist with Ki 2.5 nM (5-HT4a) and 8 nM (5-HT4b).Formule :C18H26ClN3O3·C4H6O4Degré de pureté :99.24%Couleur et forme :SolidMasse moléculaire :485.96Mecamylamine
CAS :Mecamylamine: oral, noncompetitive nAChR blocker, crosses blood-brain barrier, for neuropsychiatric and hypertension research.Formule :C11H21NCouleur et forme :SolidMasse moléculaire :167.29Trimethobenzamide hydrochloride
CAS :Trimethobenzamide hydrochloride (Ro 2-9578) is a blocker of the D2 receptor. Trimethobenzamide is an antiemetic used to prevent nausea and vomiting.Formule :C21H29ClN2O5Degré de pureté :99.52%Couleur et forme :SolidMasse moléculaire :424.92TNCA
CAS :TNCA (Lycoperodine-1) is a high-affinity CaSR ligand (CaSRL) with co-agonist activity.Formule :C12H12N2O2Degré de pureté :97.33% - 97.73%Couleur et forme :SolidMasse moléculaire :216.24Clobenpropit 2HBr
CAS :Clobenpropit 2HBr is a histamine H3 receptor antagonist. It has neuroprotective effects via stimulation of GABA release in the brain.Formule :C14H17ClN4SCouleur et forme :SolidMasse moléculaire :308.83Syk Inhibitor II dihydrochloride
CAS :Syk inhibitor II selectively blocks Syk (IC50 = 41 nM), impacting platelet function and inflammation, with lower potency against other kinases.Formule :C14H17Cl2F3N6ODegré de pureté :98.53%Couleur et forme :SolidMasse moléculaire :413.22Ref: TM-T4391
1mg130,00€2mg212,00€5mg455,00€1mL*10mM (DMSO)455,00€10mg647,00€25mg947,00€50mg1.264,00€100mg1.700,00€Ambrisentan
CAS :Ambrisentan, an endothelin antagonist for PAH, has a low risk of liver enzyme elevation, not linked to acute liver injury.Formule :C22H22N2O4Degré de pureté :99.65% - 99.86%Couleur et forme :SolidMasse moléculaire :378.421-Oleoyl lysophosphatidic acid sodium
CAS :1-Oleoyl lysophosphatidic acid sodium (1-Oleoyl lysophosphatidic acid sodium salt) salt is an Endogenous agonist of LPA1 and LPA2Formule :C21H40O7P·NaDegré de pureté :98.75% - 99.24%Couleur et forme :SolidMasse moléculaire :458.51Piboserod
CAS :Piboserod (SB-207266) (SB 207266) is a selective 5-HT(4) receptor antagonist.Formule :C22H31N3O2Degré de pureté :97.21% - 99.49%Couleur et forme :SolidMasse moléculaire :369.5Ref: TM-T2278
1mg38,00€2mg50,00€5mg84,00€10mg118,00€1mL*10mM (DMSO)120,00€25mg220,00€50mg403,00€100mg582,00€500mg1.198,00€Sumatriptan hydrochloride
CAS :Sumatriptan hydrochloride (GR 43175), an oral 5-HT1 receptor agonist, treats migraines; Ki: 5-HT1D - 17 nM, 5-HT1B - 27 nM, 5-HT1A - 100 nM.Formule :C14H22ClN3O2SCouleur et forme :SolidMasse moléculaire :331.86Dobutamine
CAS :Dobutamine, a synthetic catecholamine, boosts cardiac output and improves blood flow, mainly targeting β1-AR.Formule :C18H23NO3Couleur et forme :SolidMasse moléculaire :301.38Montelukast dicyclohexylamine
CAS :Montelukast (MK0476), a selective CysLT1 antagonist, treats asthma, liver injury, and is researched for COVID-19.Formule :C47H59ClN2O3SCouleur et forme :SolidMasse moléculaire :767.5Lidamidine Hydrochloride
CAS :Lidamidine HCl: α2-adrenergic agonist; lowers gut secretion, slows transit, stops muscle contractions.Formule :C11H17ClN4OCouleur et forme :SolidMasse moléculaire :256.73Vortioxetine hydrobromide
CAS :Vortioxetine hydrobromide (Lu AA21004 hydrobromide) is a serotonin (5-HT) modulator and stimulator (SMS), inhibits 5-HT1A/1B/3A/7 receptor and SERT (IC50: 15/33Formule :C18H22N2S·HBrDegré de pureté :98.85% - 99.98%Couleur et forme :SolidMasse moléculaire :379.36Vercirnon sodium
CAS :Vercirnon (GSK1605786A) sodium: oral CCR9 antagonist, inhibits Ca2+ mobilization/chemotaxis, IC50 = 2.6-5.4 nM, selective for CCR9 vs. CCR1-12/CX3CR1-7.Formule :C22H21ClN2NaO4SCouleur et forme :SolidMasse moléculaire :467.92MK-1064
CAS :MK-1064 (Urokinase inhibitor 1) is a selective orexin 2 receptor antagonist (2-SORA).Formule :C24H20ClN5O3Degré de pureté :99.19% - 99.82%Couleur et forme :SolidMasse moléculaire :461.9Bunazosin
CAS :Bunazosin is a potent and selective α1-adrenoceptor antagonist that can be used for antihypertensive and ocular hypotensive research [1].Formule :C19H27N5O3Couleur et forme :SolidMasse moléculaire :373.45Syk Inhibitor II dihydrochloride dihydrate
CAS :Potent, selective ATP-competitive Syk Inhibitor II (IC50: 41 nM), with anti-allergic properties, in dihydrochloride dihydrate form.Formule :C14H21Cl2F3N6O3Couleur et forme :SolidMasse moléculaire :449.26Cinaciguat hydrochloride
CAS :Cinaciguat( BAY582667, BAY58-2667) is a soluble guanosine cyclase activator that can prevent cardiac dysfunction in rat models of type 1 diabetes.Formule :C36H40ClNO5Couleur et forme :SolidMasse moléculaire :602.17Amperozide
CAS :Amperozide (FG 5606), an atypical antipsychotic, antagonizes 5-HT2A and modulates dopamine activity for schizophrenia treatment.Formule :C23H29F2N3ODegré de pureté :99.68%Couleur et forme :SolidMasse moléculaire :401.49Ref: TM-T23733
1mg87,00€5mg178,00€10mg295,00€1mL*10mM (DMSO)321,00€25mg497,00€50mg708,00€100mg964,00€500mg1.918,00€BD-1047 dihydrobromide
CAS :BD-1047 dihydrobromide (BD1047.2HBr) , a selective functional antagonist of sigma receptors, has antipsychotic activity in animal models predictive of efficacyFormule :C13H22Br2Cl2N2Degré de pureté :98.13% - 99.39%Couleur et forme :SolidMasse moléculaire :437.04Ref: TM-T1740
1mg37,00€2mg48,00€5mg73,00€1mL*10mM (DMSO)74,00€10mg95,00€25mg168,00€50mg290,00€100mg490,00€Laropiprant sodium
Laropiprant sodium is a potent and selective DP receptor antagonist with Ki values of 0.57 nM for TP receptors and 2.95 nM for DP receptors.Couleur et forme :SolidGSK2018682
CAS :GSK2018682 is an agonist of sphingosine-1-phosphate receptor (s1p1) and (s1p5) agonist(pEC50s of 7.7 and 7.2,respectively).Formule :C22H21ClN4O4Degré de pureté :99.04%Couleur et forme :SolidMasse moléculaire :440.88Guanfacine hydrochloride
CAS :Guanfacine hydrochloride (Intuniv) is a centrally acting antihypertensive agent with specificity towards ADRENERGIC ALPHA-2 RECEPTORS.Formule :C9H10Cl3N3ODegré de pureté :99.89% - 99.91%Couleur et forme :SolidMasse moléculaire :282.55Eltoprazine hydrochloride
CAS :Eltoprazine hydrochloride (DU 28853 hydrochloride) is a partial agonist at serotonin 5-HT1A, 5-HT1B, and 5-HT2B receptors (Ki value of 40, 52, and 81 nM,Formule :C12H17ClN2O2Degré de pureté :99.35%Couleur et forme :SolidMasse moléculaire :256.73Lerisetron
CAS :Lerisetron is an antagonist of serotonin type 3 (5-HT3) receptor, with antiemetic activity.Formule :C18H20N4Degré de pureté :99.15% - 99.82%Couleur et forme :SolidMasse moléculaire :292.38Elinzanetant
CAS :Elinzanetant is a dual antagonist of neurokinin (NK) receptors 1 and 3 and modulates reproductive hormone secretion.Formule :C33H35F7N4O3Degré de pureté :98% - 99.13%Couleur et forme :SolidMasse moléculaire :668.64Ref: TM-T38144
1mg92,00€2mg118,00€5mg192,00€1mL*10mM (DMSO)284,00€10mg313,00€25mg528,00€50mg740,00€100g4.977,00€Cerlapirdine
CAS :Cerlapirdine (PF-05212365), a 5-HT6 receptor antagonist, is in trials for Alzheimer's and schizophrenia cognition issues.Formule :C22H23N3O3SDegré de pureté :98.77%Couleur et forme :SolidMasse moléculaire :409.5Ref: TM-T30798
1mg81,00€5mg170,00€1mL*10mM (DMSO)198,00€10mg274,00€25mg543,00€50mg780,00€100mg1.074,00€Diquafosol tetrasodium
CAS :Diquafosol Tetrasodium is a P2Y2 receptor agonist that stimulates the secretion of mucins from ocular tissues Diquafosol tetrasodium (INS365) improves tear filmFormule :C18H22N4Na4O23P4Degré de pureté :98.25% - 99.97%Couleur et forme :SolidMasse moléculaire :878.23KB-5492 anhydrous
CAS :KB 5492 is an agent of anti-ulcer. It preventing cysteamine-induced duodenal ulcers by stimulating duodenal HCO3- secretion.Formule :C27H34N2O10Couleur et forme :SolidMasse moléculaire :546.57Melitracen hydrochloride
CAS :Melitracen hydrochloride (Thymeol hydrochloride) , an antidepressant, is used as potential dopamine D1/2 receptor antagonist to treat depression.Formule :C21H26ClNDegré de pureté :99.99%Couleur et forme :Crystalline SolidMasse moléculaire :327.90Ref: TM-T4274
10mg44,00€1mL*10mM (DMSO)48,00€25mg64,00€50mg93,00€100mg110,00€200mg161,00€500mg264,00€ABT-702 dihydrochloride
CAS :ABT-702 dihydrochloride is a potent adenosine kinase (AK) inhibitor.Formule :C22H21BrCl2N6ODegré de pureté :98.42% - 98.98%Couleur et forme :SolidMasse moléculaire :536.25Ref: TM-T4668
1mg58,00€2mg82,00€5mg113,00€1mL*10mM (DMSO)133,00€10mg177,00€25mg333,00€50mg502,00€100mg710,00€500mg1.494,00€Anisotropine Methylbromide
CAS :Anisotropine Methylbromide is an anticholinergic agent and has been used for relief of gastrointestinal spasm and for the suppression of gastric acid secretion.Formule :C17H32BrNO2Degré de pureté :99.73%Couleur et forme :Crystals From Acetone SolidMasse moléculaire :362.35Doxazosin
CAS :Doxazosin (UK 33274) is a long-lasting inhibitor of α1-adrenoceptors that is widely used to treat benign prostatic hyperplasia and lower urinary tract symptoms.Formule :C23H25N5O5Degré de pureté :99.47% - 99.87%Couleur et forme :SolidMasse moléculaire :451.48Peptide YY (PYY) (3-36), human
CAS :Peptide YY (PYY) (3-36), human (Peptide YY (3-36)) is a gut hormone peptide. Peptide YY (PYY) (3-36), human acts as a Y2 receptor agonist to reduce appetite.Formule :C176H272N52O54Degré de pureté :97.76%Couleur et forme :SolidMasse moléculaire :3980.42DORA-22
CAS :DORA-22 is a dual orexin receptor antagonist, improves mild stress-induced insomnia with minimal effect on memoryFormule :C23H22F2N4O2Degré de pureté :97.67%Couleur et forme :SolidMasse moléculaire :424.44Ref: TM-T5500
1mg131,00€2mg188,00€5mg284,00€1mL*10mM (DMSO)331,00€10mg430,00€25mg710,00€50mg998,00€100mg1.349,00€Deslorelin acetate(57773-65-6 free base)
Deslorelin acetate(57773-65-6 free base) is a gonadotropin releasing hormone super-agonist (GnRH agonist)Formule :C66H87N17O14Degré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :1342.5Midodrine
CAS :Midodrine ((±)-Midodrin), an adrenergic alpha-1 agonist, belongs to the class of medications known as vasopressors.Formule :C12H18N2O4Degré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :254.28Cariprazine hydrochloride
CAS :Cariprazine hydrochloride (RGH188 hydrochloride) is an antipsychotic drug, is a D3 and D2 receptor partial agonist((Ki of 0.085 nM and 0.49 nM, respectively)Formule :C21H33Cl3N4ODegré de pureté :99.78% - >99.99%Couleur et forme :SolidMasse moléculaire :463.87Talnetant
CAS :Talnetant (SB 223412) is a selective NK3 receptor antagonist that can penetrate the brain and modulate dopamine.Formule :C25H22N2O2Degré de pureté :97.88%Couleur et forme :SolidMasse moléculaire :382.45Ref: TM-T7549
1mg40,00€2mg52,00€5mg87,00€10mg123,00€1mL*10mM (DMSO)135,00€25mg251,00€50mg464,00€100mg705,00€Bradykinin (acetate)
CAS :Bradykinin (acetate) is an active peptide that is generated by the kallikrein-kinin system.Formule :C52H77N15O13Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :1120.26Talinolol
CAS :(±)-Talinolol is a selective β1 adrenoceptor antagonist well known for its cardioprotective and antihypertensive activity.Formule :C20H33N3O3Degré de pureté :98.8%Couleur et forme :SolidMasse moléculaire :363.49Ref: TM-T21640
2mg34,00€5mg52,00€1mL*10mM (DMSO)52,00€10mg92,00€25mg178,00€50mg313,00€100mg535,00€200mg775,00€LML134
CAS :LML134 (LML-134) is an inverse agonist of Histamine 3 receptor (H3R)(hH3R cAMP and hH3R bdg with Kis of 0.3 nM and 12 nM).Formule :C19H29N5O3Degré de pureté :99.36%Couleur et forme :SolidMasse moléculaire :375.47Ref: TM-T8514
1mg34,00€5mg78,00€1mL*10mM (DMSO)86,00€10mg112,00€25mg203,00€50mg299,00€100mg447,00€200mg600,00€Thonzylamine
CAS :Thonzylamine is an antihistamine/anticholinergic, combined with Clofedanol or Phenylephrine for cold, hay fever, or allergy relief.Formule :C16H22N4ODegré de pureté :99.45%Couleur et forme :SolidMasse moléculaire :286.375-Hydroxy-1-methylhydantoin
CAS :5-Hydroxy-1-methylhydantoin (HD-003) is an antioxidant potentially for the treatment of renal failure.Formule :C4H6N2O3Degré de pureté :99.99%Couleur et forme :SolidMasse moléculaire :130.1Dazoxiben
CAS :Dazoxiben (UK-37248) is a potent inhibitor of thromboxane (TX) synthaseFormule :C12H13ClN2O3Degré de pureté :99.99%Couleur et forme :SolidMasse moléculaire :268.7Ref: TM-T7968
1mg35,00€2mg50,00€1mL*10mM (DMSO)56,00€5mg75,00€10mg120,00€25mg236,00€50mg349,00€100mg485,00€500mg1.035,00€HJC0350
CAS :HJC0350 is an effective and specific EPAC2 inhibitor (IC50: 0.3 μM), and no inhibition of Epac1.Formule :C15H19NO2SDegré de pureté :99.27% - 99.65%Couleur et forme :SolidMasse moléculaire :277.38SB 242084
CAS :SB 242084 dihydrochloride hydrate is a psychoactive drug and research chemical which acts as a selective antagonist for the 5HT2C receptor.Formule :C21H19ClN4O2Degré de pureté :99.75% - ≥98%Couleur et forme :SolidMasse moléculaire :394.85PAR-2 Activating Peptide acetate
PAR-2 Activating Peptide acetate (SLIGRL-NH2 acetate) is an agonist of Protease-Activated Receptor-2 (PAR-2).Formule :C31H60N10O9Degré de pureté :98.5% - 99.92%Couleur et forme :SolidMasse moléculaire :716.88Pimavanserin tartrate
CAS :Pimavanserin tartrate is a potent 5-HT 2A receptor inverse agonist used to treat Parkinson's disease-related psychosis.Cost-effective and quality-assured.Formule :C50H68F2N6O4·C4H6O6Degré de pureté :99.24% - 99.98%Couleur et forme :SolidMasse moléculaire :1005.2Ocaperidone
CAS :Ocaperidona (Ocaperidone (Ocaperidona)), a very high affinity dopamine D2 antagonist.Formule :C24H25FN4O2Degré de pureté :99.33%Couleur et forme :SolidMasse moléculaire :420.48H2L 5765834
CAS :H2L 5765834 is a lysophosphatidic acid receptors antagonistFormule :C21H12N2O7Degré de pureté :98.25% - 99.47%Couleur et forme :SolidMasse moléculaire :404.33Ref: TM-T22834
1mg58,00€5mg113,00€1mL*10mM (DMSO)124,00€10mg177,00€25mg334,00€50mg497,00€100mg708,00€Thrombin Receptor Activator for Peptide
Thrombin Receptor Activator (TRAP) or Coagulation Factor II (1-5), used in CHD research.Formule :C32H51F3N8O9Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :748.79Paltusotine
CAS :Paltusotine: nonpeptide SST2 agonist, orally bioavailable, regulates GH/IGF-1 in acromegaly.Formule :C27H22F2N4ODegré de pureté :99.91%Couleur et forme :SolidMasse moléculaire :456.49Pitolisant hydrochloride
CAS :Pitolisant hydrochloride (Ciproxidine) is a potent and selective inverse agonist of the histamine H3 receptor(Ki : 0.16 nM).Formule :C17H27Cl2NODegré de pureté :99.72% - 99.91%Couleur et forme :SolidMasse moléculaire :332.31Ref: TM-T7176
5mg48,00€1mL*10mM (DMSO)50,00€10mg71,00€25mg117,00€50mg187,00€100mg295,00€200mg442,00€500mg708,00€5'-N-Ethylcarboxamidoadenosine
CAS :NECA, an adenosine receptor agonist, boosts brain extravasation of fluorescein and dextran without affecting the blood-brain barrier.Formule :C12H16N6O4Degré de pureté :98.95% - ≥95%Couleur et forme :PowderMasse moléculaire :308.29Namodenoson
CAS :Namodenoson (2-Cl-IB-MECA) is an adenosine A3 receptor agonist.Formule :C18H18ClIN6O4Degré de pureté :98.97%Couleur et forme :SolidMasse moléculaire :544.73Dapiprazole Hydrochloride
CAS :Dapiprazole Hydrochloride (Glamidolo Hydrochloride) is an alpha-1-adrenergic antagonist that acts by blocking alpha-adrenergic receptors.Formule :C19H28ClN5Degré de pureté :99.75% - 99.93%Couleur et forme :SolidMasse moléculaire :361.92ONO-AE3-208
CAS :ONO-AE3-208 (AE 3-208) is an EP4 antagonist. It suppresses cell migration, invasion, and metastasis of prostate cancer.Formule :C24H21FN2O3Degré de pureté :98.04% - 99.55%Couleur et forme :SolidMasse moléculaire :404.43Ref: TM-TQ0290
100mgÀ demander2mg39,00€5mg60,00€1mL*10mM (DMSO)66,00€10mg96,00€25mg148,00€50mg212,00€Harmine hydrochloride
CAS :Harmine hydrochloride (telepathine hydrochloride) is extracted from Peganum Harmala Genus.Formule :C13H13ClN2ODegré de pureté :99.61% - >99.99%Couleur et forme :Yellow To Slightly Green Crystalline PowderMasse moléculaire :248.71ABT-724
CAS :ABT-724 is an agonist of dopamine D4 receptor(EC50: 12.4 nM)Formule :C17H19N5Degré de pureté :99.73%Couleur et forme :SolidMasse moléculaire :293.37Riociguat
CAS :Riociguat (BAY 632521) is a stimulator of guanylate cyclase which causes relaxation of vascular smooth muscle and is used to treat severe pulmonary arterialFormule :C20H19FN8O2Degré de pureté :99.28% - 99.95%Couleur et forme :SolidMasse moléculaire :422.42Ondansetron hydrochloride
CAS :Ondansetron hydrochloride (Zofran) is a serotonin 5-HT3 receptor antagonist, used to prevent nausea and vomiting caused by cancer chemotherapy, and radiationFormule :C18H19N3O·HClDegré de pureté :99.78%Couleur et forme :White PowderMasse moléculaire :329.82ML401
CAS :ML401 is a selectively EBI2(GPR183) receptor antagonist(IC50 of 1.03 nM) .Formule :C20H20BrClN2ODegré de pureté :99.13%Couleur et forme :SolidMasse moléculaire :419.74Vericiguat
CAS :Vericiguat (BAY1021189) is a potent and orally available guanylate cyclase stimulator.Formule :C19H16F2N8O2Degré de pureté :98.86% - 99.93%Couleur et forme :SolidMasse moléculaire :426.38Rotigotine Hydrochloride
CAS :Rotigotine HCl, D3-preferential dopamine agonist, is 50x stronger than quinpirole in anti-Parkinson's efficacy.
Formule :C19H26ClNOSDegré de pureté :99.53% - 99.56%Couleur et forme :Almost White To White Crystalline PowderMasse moléculaire :351.93Rotigotine-
CAS :Rotigotine (N-0923) is a non-ergot dopamine receptor agonist used in the therapy of Parkinson disease and restless leg syndrome.Formule :C19H25NOSDegré de pureté :98.08% - 99.59%Couleur et forme :SolidMasse moléculaire :315.47Ref: TM-T6647
5mg50,00€1mL*10mM (DMSO)52,00€10mg73,00€25mg138,00€50mg241,00€100mg358,00€200mg523,00€500mg822,00€RBC8
CAS :RBC8 is a specific GTPases RalA/RalB inhibitor by inhibiting the binding of Ral to its effector RALBP1, no inhibition on the GTPases RhoA and Ras.Formule :C25H20N4O3Degré de pureté :98.44% - 99.81%Couleur et forme :SolidMasse moléculaire :424.45Ref: TM-T6634
1mg46,00€1mL*10mM (DMSO)92,00€5mg96,00€10mg147,00€25mg281,00€50mg447,00€100mg650,00€200mg888,00€LY2828360
CAS :LY2828360: CB2 agonist, Ki=40.3 nM; biases CB2 over CB1 with EC50s of 20.1 nM and >100 μM.Formule :C22H27ClN6ODegré de pureté :98.45% - 99.51%Couleur et forme :SolidMasse moléculaire :426.94Conopressin S acetate(111317-90-9 free base)
Conopressin S acetate(111317-90-9 free base) (Con-S acetate) is a natural product isolated from Conus striatus, shows high affinity with vasopressin V1bFormule :C43H77N17O12S2Degré de pureté :99.79%Couleur et forme :SolidMasse moléculaire :1088.32Tiprenolol
CAS :Tiprenolol is a beta adrenergic receptor antagonist.[1]Formule :C13H21NO2SDegré de pureté :99.43%Couleur et forme :SolidMasse moléculaire :255.38Ref: TM-T50081
1mg52,00€1mL*10mM (DMSO)89,00€5mg98,00€10mg146,00€25mg235,00€50mg319,00€100mg447,00€200mg587,00€Ipsapirone hydrochloride
CAS :Ipsapirone, a pyrimidinylpiperazine ligand, is potent and specific for 5-HT1A receptors and has potential therapeutic use in affective disorders.Formule :C19H24ClN5O3SCouleur et forme :SolidMasse moléculaire :437.94Donitriptan Mesylate
CAS :Donitriptan Mesylate, a 5-HT1B/1D agonist, is used potentially for the treatment of migraines.Formule :C24H29N5O5SCouleur et forme :SolidMasse moléculaire :499.58Bucindolol hydrochloride
CAS :Bucindolol, a 4th-gen β-blocker, prevents onset AF; effectiveness varies with β₁/α(2c) genes; best in β₁389 Arg homozygotes.Formule :C22H26ClN3O2Couleur et forme :SolidMasse moléculaire :399.91Spexin acetate(1370290-58-6 free base)
Spexin acetate: GAL2/GAL3 agonist. EC50: 45.7/112.2 nM. Inactive at GAL1. Reduces appetite, fat uptake, and food intake; lowers LH in fish; anxiolytic.Formule :C76H117N19O22SDegré de pureté :95.43%Couleur et forme :SolidMasse moléculaire :1680.94PD-168077 maleate
CAS :PD-168077 maleate is a selective agonist of dopamine D4 receptor(Ki : 9 nM)Formule :C24H26N4O5Degré de pureté :99.13%Couleur et forme :SolidMasse moléculaire :450.49Ref: TM-T5047
2mg34,00€5mg50,00€1mL*10mM (DMSO)55,00€10mg75,00€25mg142,00€50mg231,00€100mg344,00€200mg490,00€JNJ-5207852
CAS :JNJ-5207852 is a novel, non-imidazole histamine H3 receptor antagonist, with high affinity at the rat (pKi=8.9) and human (pKi=9.24) H3 receptor.Formule :C20H32N2ODegré de pureté :97.19%Couleur et forme :SolidMasse moléculaire :316.48Thozalinone
CAS :Thozalinone is a psychostimulant agent inducing the release of norepinephrine and dopamine.Formule :C11H12N2O2Degré de pureté :99.68%Couleur et forme :SolidMasse moléculaire :204.23TCS 1102
CAS :TCS 1102 is an effective, dual orexin receptor antagonist (Ki: 0.2/3 nM for OX2/1 receptors).Formule :C27H26N4O2SDegré de pureté :99.35% - 99.52%Couleur et forme :SolidMasse moléculaire :470.59Empagliflozin
CAS :Empagliflozin (BI 10773) is an SGLT-2 inhibitor (IC50=3.1 nM) that is potent and selective, with more than 300-fold selectivity for SGLT-1/4/5/6.Formule :C23H27ClO7Degré de pureté :98% - 99.98%Couleur et forme :SolidMasse moléculaire :450.91Ref: TM-T1766
5mg44,00€1mL*10mM (DMSO)48,00€10mg57,00€50mg74,00€100mg90,00€200mg137,00€500mg178,00€1g263,00€Tribenoside
CAS :Tribenoside (BG-356) is a vasoprotectant with mild anti-inflammatory, analgesic, and wound healing properties.Formule :C29H34O6Degré de pureté :≥98%Couleur et forme :LiquidMasse moléculaire :478.58Tiaramide hydrochloride
CAS :Tiaramide hydrochloride (FK-1160) is an anti-inflammatory that blocks mast cell mediators and relaxes smooth muscles.Formule :C15H19Cl2N3O3SDegré de pureté :98.48%Couleur et forme :SolidMasse moléculaire :392.3Ref: TM-T28972
1mg66,00€5mg130,00€1mL*10mM (DMSO)137,00€10mg177,00€25mg299,00€50mg447,00€100mg623,00€200mg882,00€Buclizine
CAS :Buclizine is an orally active antihistamine, antiallergic compound. buclizine is also a strong teratogen in rats and exhibits antitumour effects.Formule :C28H33ClN2Couleur et forme :SolidMasse moléculaire :433.03cicloprofen
CAS :cicloprofen is Cell division cycle 7-related protein kinase (human) inhibitor.Formule :C16H14O2Degré de pureté :98.15%Couleur et forme :SolidMasse moléculaire :238.2812Ref: TM-T8586
1mg58,00€1mL*10mM (DMSO)105,00€5mg116,00€10mg172,00€25mg281,00€50mg396,00€100mg537,00€200mg712,00€Melperone
CAS :Melperone, a butyrophenone tranquillizer, caused bradycardia in vivo and in vitro.Formule :C16H22FNODegré de pureté :98.84%Couleur et forme :SolidMasse moléculaire :263.35[D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate
Broad-spectrum neuropeptide inverse agonist/antagonist; potent at ghrelin receptor (EC50 = 5.2 nM); inhibits cancer growth, induces apoptosis.Formule :C81H113N19O14Degré de pureté :97.68%Couleur et forme :SolidMasse moléculaire :1576.91Histrelin acetate
CAS :Histrelin acetate is a nonapeptide analog of gonadotropin-releasing hormone (GnRH) with added potency.Formule :C68H90N18O14Degré de pureté :99.92%Couleur et forme :SolidMasse moléculaire :1383.55TG4-155
CAS :TG4-155: brain-penetrant EP2 inhibitor, KB 2.4 nM; >1000x weaker at EP4, KB 11.4 μM; selective over other receptors/channels.Formule :C23H26N2O4Degré de pureté :97.2%Couleur et forme :SolidMasse moléculaire :394.46Ref: TM-T5482
2mg35,00€5mg52,00€1mL*10mM (DMSO)57,00€10mg94,00€25mg178,00€50mg313,00€100mg464,00€200mg660,00€Urapidil
CAS :Urapidil (Ebrantil), a sympatholytic antihypertensive drug, acts as a 5-HT1A receptor agonist and as an α1-adrenoceptor antagonist.Formule :C20H29N5O3Degré de pureté :99.85% - >99.99%Couleur et forme :SolidMasse moléculaire :387.48Brexpiprazole
CAS :Brexpiprazole (OPC-34712) is a partial agonist of human 5-hydroxytryptamine (5-HT) 5-HT1A and dopamine D2 receptors.Formule :C25H27N3O2SDegré de pureté :99.06% - 99.96%Couleur et forme :SolidMasse moléculaire :433.57Ref: TM-T2306
1mL*10mM (DMSO)À demander5mg50,00€10mg63,00€25mg75,00€50mg88,00€100mg94,00€200mg140,00€500mg259,00€FSLLRY-NH2 TFA(245329-02-6 free base)
FSLLRY-NH2 TFA inhibits PAR2, reverses taxol-induced pain, and reduces itch in mice; blocks ERK and collagen in fibroblasts.Formule :C41H61F3N10O10Degré de pureté :99.32%Couleur et forme :SolidMasse moléculaire :910.99Batefenterol Succinate
CAS :Batefenterol Succinate is a first-in-class inhaled bifunctional bronchodilator possessing muscarinic receptor antagonist and β2-adrenoceptor agonist properties.Formule :C44H48ClN5O11Couleur et forme :SolidMasse moléculaire :858.34Rimcazole
CAS :Rimcazole is a sigma receptor antagonist. It also binds to the dopamine transporter and inhibiting dopamine uptake.Formule :C21H27N3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :321.46Vortioxetine
CAS :Vortioxetine (Lu AA 21004) is a serotonergic antidepressant used for major depression disorders.Formule :C18H22N2SDegré de pureté :99.34% - 99.34%Couleur et forme :SolidMasse moléculaire :298.45Ref: TM-T2395
1mL*10mM (DMSO)46,00€10mg48,00€25mg65,00€50mg90,00€100mg117,00€200mg203,00€500mg333,00€1g477,00€GLP-1(7-36), amide
CAS :GLP-1 secretion by human enteroendocrine NCI-H716 cells is augmented in a dose-dependent manner by the addition of CPE.Cost-effective and quality-assured.Formule :C149H226N40O45Degré de pureté :99.85%Couleur et forme :White PowderMasse moléculaire :3297.63GBR 12935 dihydrochloride
CAS :GBR 12935 dihydrochloride (GBR 12935) can induce the increase of the extracellular levels of dopamine to basal levels.Formule :C28H36Cl2N2ODegré de pureté :99.09% - ≥95%Couleur et forme :SolidMasse moléculaire :487.5Eledoisin Related Peptide 2TFA
Eledoisin Related Peptide 2TFA (Eledoisin Related Peptide 2TFA (2990-43-4(free base))) is a tachykinin receptor ligand.Formule :C38H60F6N8O10SDegré de pureté :99%Couleur et forme :SolidMasse moléculaire :934.99Bindarit
CAS :Bindarit is a selective inhibitor of monocyte chemoattractant proteins MCP-1/CCL2, MCP-3/CCL7 and MCP-2/CCL8.Cost-effective and quality-assured.Formule :C19H20N2O3Degré de pureté :98.35% - 98.55%Couleur et forme :SolidMasse moléculaire :324.37Ref: TM-T6413
1mg35,00€2mg50,00€5mg75,00€1mL*10mM (DMSO)84,00€10mg110,00€25mg178,00€50mg314,00€100mg492,00€200mg710,00€Temanogrel hydrochloride
CAS :Temanogrel hydrochloride is a serotonin antagonist and anti-platelet agent.Formule :C24H29ClN4O4Couleur et forme :SolidMasse moléculaire :472.97Haloperidol lactate
CAS :Haloperidol lactate: a potent antipsychotic for acute/chronic schizophrenia and polyarousal syndrome research.Formule :C24H29ClFNO5Couleur et forme :SolidMasse moléculaire :465.95I-191
CAS :I-191 is a potent antagonist of protease-activated receptor 2 (PAR2), inhibits multiple signaling functions in human cancer cells.Formule :C23H26FN5O2Degré de pureté :99.8%Couleur et forme :SolidMasse moléculaire :423.48Pemirolast
CAS :Pemirolast: oral antiallergic, reduces paclitaxel reactions, inhibits neuropeptides, for asthma and conjunctivitis study.Formule :C10H8N6OCouleur et forme :SolidMasse moléculaire :228.21Hydroxyzine
CAS :Hydroxyzine (Hydroxyzine free base) is an antagonist of histamine H1-receptor.Formule :C21H27ClN2O2Degré de pureté :99.54% - ≥95%Couleur et forme :Oil SolidMasse moléculaire :374.9GUANABENZ
CAS :GUANABENZ is a Central alpha-2 Adrenergic Agonist. The mechanism of action of guanabenz is as an Adrenergic alpha2-Agonist.Formule :C8H8Cl2N4Degré de pureté :98.31%Couleur et forme :White Solid From Acetonitrile SolidMasse moléculaire :231.08Alprenolol hydrochloride
CAS :Alprenolol hydrochloride is a non-selective blocker of beta, and also is a antagonist of5-HT1A receptor.Formule :C15H24ClNO2Degré de pureté :99.79%Couleur et forme :SolidMasse moléculaire :285.81idalopirdine
CAS :Idalopirdine (Lu AE58054), a selective 5-HT6 receptor antagonist( Ki : 0.83 nM),as a treatment for Alzheimer's disease.Formule :C20H19F5N2ODegré de pureté :99.73%Couleur et forme :SolidMasse moléculaire :398.37Ref: TM-T7103
1mg88,00€2mg118,00€1mL*10mM (DMSO)187,00€5mg188,00€10mg254,00€25mg429,00€50mg630,00€100mg898,00€[Leu31,Pro34]-Neuropeptide Y (porcine)
CAS :[Leu31,Pro34]-Neuropeptide Y (porcine), is a selective and high affinity agonist of neuropeptide Y (NPY) Y1 receptor with anxiolytic effects.Formule :C190H286N54O56Degré de pureté :99.39%Couleur et forme :SolidMasse moléculaire :4223Isocorynoxeine
CAS :Isocorynoxeine reduces blood pressure, dilates vessels, and guards neurons against ischemia and glutamate toxicity.Formule :C22H26N2O4Degré de pureté :98% - 99.9%Couleur et forme :SolidMasse moléculaire :382.45Ref: TM-T6S0654
1mg62,00€2mg89,00€5mg132,00€1mL*10mM (DMSO)146,00€10mg226,00€25mg384,00€50mg557,00€100mg785,00€200mg1.054,00€Amylin, amide, rat acetate(124447-81-0,free base)
Amylin, amide, rat acetate is a potent and high affinity ligand of AMY1 and AMY3 receptors and variably of AMY2 receptors.Formule :C169H276N52O55S2Degré de pureté :98.93%Couleur et forme :SolidMasse moléculaire :3980.45AM-2232
CAS :AM-2232 (UNII-40KCH8YIKP) is a potent and unselective agonist of the cannabinoid receptors.Formule :C24H20N2ODegré de pureté :99.37%Couleur et forme :SolidMasse moléculaire :352.43GLP-1(7-37) acetate(106612-94-6 free base)
CAS :Glp-1(7-37) acetate is an intestinal insulin hormone that enhances glucose-induced insulin secretion.Formule :C151H228N40O47Degré de pureté :98.89%Couleur et forme :SolidMasse moléculaire :3355.67Ralinepag
CAS :Ralinepag (APD811) is a potent, orally bioavailable agonist of non-prostanoid prostacyclin (IP) receptor, with EC50s of 8.5 nM, 530 nM and 850 nM for human andFormule :C23H26ClNO5Degré de pureté :99.79% - 99.85%Couleur et forme :SolidMasse moléculaire :431.91Ref: TM-T4635
1mg50,00€2mg71,00€5mg105,00€1mL*10mM (DMSO)117,00€10mg167,00€25mg285,00€50mg401,00€100mg573,00€200mg803,00€Nelotanserin
CAS :Nelotanserin (APD125): strong 5-HT2A inverse agonist (IC50: 1.7 nM), moderate 5-HT2C (79 nM), weak 5-HT2B (791 nM).Formule :C18H15BrF2N4O2Degré de pureté :98.42% - 99.88%Couleur et forme :SolidMasse moléculaire :437.24Ref: TM-T7350
1mg38,00€2mg50,00€1mL*10mM (DMSO)80,00€5mg84,00€10mg113,00€25mg178,00€50mg333,00€100mg495,00€500mg1.071,00€CGP 71683 (free base)
CAS :CGP 71683 (free base) is a potent and highly selective non-peptide antagonist of the NPY Y(5) receptor in the study of obesity.Formule :C26H29N5O2SCouleur et forme :SolidMasse moléculaire :475.61Felypressin
CAS :Felypressin, a Lypressin analog with a phenylalanine substitution, acts as a vasoconstrictor with less antidiuretic effect.Formule :C46H65N13O11S2Degré de pureté :99.65%Couleur et forme :SolidMasse moléculaire :1040.22Etelcalcetide hydrochloride
CAS :Etelcalcetide HCl, a synthetic peptide modulator of CaSR, lowers PTH in dialysis patients with secondary hyperparathyroidism.Formule :C38H73N21O10S2HClDegré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :1353.33SRI-37330 hydrochloride
CAS :SRI-37330 hydrochloride is an orally active thioredoxin-interacting protein (TXNIP) inhibitor. hydrochloride can be used to study type 2 diabetes.Formule :C16H20ClF3N4O2SCouleur et forme :SolidMasse moléculaire :424.87Diclofensine hydrochloride
CAS :Diclofensine hydrochloride (Ro 8-4650 hydrochloride) 是一种高效单胺再摄取抑制剂，在大鼠脑突触体中能够阻断多巴胺 (IC50=0.74 nM)、去甲肾上腺素 (IC50=2.3 nM) 和 5-羟色胺 (IC50=3.7 nM)。Formule :C17H18Cl3NODegré de pureté :98.86% - 99.93%Couleur et forme :SolidMasse moléculaire :358.69NAV-2729
CAS :NAV-2729 inhibits six ArfGEFs (human ARNO, EFA6, BIG1, and BRAG2 and Legionella and Rickettsia RalF), the strongest effects being against BRAG2, Arf1 and Arf6.Formule :C25H17ClN4O3Degré de pureté :98.83% - 98.91%Couleur et forme :SolidMasse moléculaire :456.88Ref: TM-T5142
2mg43,00€5mg63,00€1mL*10mM (DMSO)71,00€10mg90,00€25mg193,00€50mg286,00€100mg429,00€500mg888,00€Vercirnon
CAS :Vercirnon (Traficet-EN) is a selective and potent antagonist of CCR9 (IC50: 10 nM). It is also used in the research of inflammatory bowel diseases.Formule :C22H21ClN2O4SDegré de pureté :99.23%Couleur et forme :SolidMasse moléculaire :444.93Ref: TM-T17225
1mg100,00€5mg245,00€1mL*10mM (DMSO)344,00€10mg385,00€25mg645,00€50mg888,00€100mg1.234,00€500mg2.457,00€Ataciguat
CAS :Ataciguat (HMR-1766) (HMR-1766) is a potent and specific soluble guanylate cyclase (sGC) activator.Formule :C21H19Cl2N3O6S3Degré de pureté :99.09%Couleur et forme :SolidMasse moléculaire :576.49Dimethocaine
CAS :Dimethocaine (Larocaine) is a local anesthetic which also effects on the central nervous system acting as dopamine-reuptake-inhibitor.Formule :C16H26N2O2Degré de pureté :99.52%Couleur et forme :SolidMasse moléculaire :278.39Cenicriviroc
CAS :Cenicriviroc (TAK-652), oral CCR2/CCR5 blocker, inhibits HIV-1/HIV-2, with strong anti-infective/anti-inflammatory effects.Formule :C41H52N4O4SDegré de pureté :97.87%Couleur et forme :SolidMasse moléculaire :696.94Ref: TM-TQ0297
1mg63,00€2mg90,00€5mg133,00€1mL*10mM (DMSO)200,00€10mg212,00€25mg423,00€50mg550,00€100mg715,00€200mg964,00€Maraviroc
CAS :Maraviroc: a CCR5 antagonist blocking HIV-1 entry; IC50s—MIP-1α: 3.3nM, MIP-1β: 7.2nM, RANTES: 5.2nM.Formule :C29H41F2N5ODegré de pureté :97.13% - 99.59%Couleur et forme :Brown SolidMasse moléculaire :513.67Ref: TM-T6016
5mg49,00€1mL*10mM (DMSO)56,00€10mg90,00€25mg152,00€50mg259,00€100mg465,00€200mg600,00€500mg945,00€AZD-4818
CAS :AZD-4818 (CCR1 antagonist) is a chemokine CCR1 antagonist for the treatment of chronic obstructive pulmonary disease.Formule :C27H32Cl2N2O7Degré de pureté :99.01%Couleur et forme :SolidMasse moléculaire :567.46JK184
CAS :JK184 is a potent Hedgehog (Hh) pathway inhibitor.
Formule :C19H18N4OSDegré de pureté :98.93% - 99.89%Couleur et forme :SolidMasse moléculaire :350.44Vicriviroc maleate
CAS :Vicriviroc maleate (SCH-417690 (maleate))(Sch-417690) is a piperazine-based CCR5 receptor antagonist with activity against human immunodeficiency virus.Formule :C32H42F3N5O6Degré de pureté :98.16% - 98.37%Couleur et forme :SolidMasse moléculaire :649.7[Pyr1]-Apelin-13
CAS :[Pyr1]-Apelin-13 ([pGlu1]-Apelin-13) is a potent and selective endogenous Apelin receptor (APJ) agonist.Formule :C69H108N22O16SDegré de pureté :99.71%Couleur et forme :SolidMasse moléculaire :1533.8VPC171
CAS :VPC171 is a novel adenosine A1 receptor positive allosteric modulator (PAM).Formule :C18H12F3NOSDegré de pureté :99.78%Couleur et forme :SolidMasse moléculaire :347.35Ref: TM-T29112
1mg49,00€1mL*10mM (DMSO)88,00€5mg96,00€10mg124,00€25mg222,00€50mg309,00€100mg439,00€200mg592,00€SAX-187
CAS :SAX-187 (SAX-187) has high-affinity binding at the human 5-HT6 receptor.Formule :C15H13ClN4O2S2Degré de pureté :97.82% - 98%Couleur et forme :SolidMasse moléculaire :380.87Ref: TM-T3183
1mg79,00€5mg152,00€1mL*10mM (DMSO)166,00€10mg245,00€25mg398,00€50mg532,00€100mg735,00€200mg973,00€Clemizole hydrochloride
CAS :Clemizole hydrochloride blocks H1 histamine receptors and inhibits HCV replication and NS4B RNA binding.Formule :C19H21Cl2N3Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :362.3MF-766
CAS :MF-766: potent, selective oral EP4 antagonist, Ki=0.23 nM, IC50=1.4 nM; shifts to 1.8 nM with 10% HS. Useful in cancer, inflammation studies.Formule :C27H21F3N2O3Degré de pureté :99.54% - 99.59%Couleur et forme :SolidMasse moléculaire :478.46CCG215022
CAS :CCG215022 is a G protein-coupled receptor kinases (GRKs) inhibitor with IC50s of 0.15±0.07 μM, 0.38±0.06 μM and 3.9±1 μM for GRK2, 5 and 1, respectively.Formule :C26H22FN7O3Degré de pureté :97.63% - 99.69%Couleur et forme :SolidMasse moléculaire :499.5Ref: TM-T3498
1mg56,00€5mg114,00€1mL*10mM (DMSO)127,00€10mg178,00€25mg394,00€50mg655,00€100mg1.035,00€Ranitidine
CAS :Ranitidine (HSDB 3925) is a non-imidazole blocker of those histamine receptors that mediate gastric secretion (H2 receptors).Formule :C13H22N4O3SDegré de pureté :99.52%Couleur et forme :Solid SolidMasse moléculaire :314.40Capadenoson
CAS :Capadenoson (BAY 68-4986) is a selective adenosine-A1 receptor agonist.Formule :C25H18ClN5O2S2Degré de pureté :98.85% - 99.57%Couleur et forme :SolidMasse moléculaire :520.03ACEPROMAZINE MALEATE
CAS :ACEPROMAZINE MALEATE is a dopamine receptor antagonistFormule :C23H26N2O5SDegré de pureté :98.87% - 99.51%Couleur et forme :Off White Or Yellow Crystalline PowderMasse moléculaire :442.53Vilazodone Hydrochloride
CAS :Vilazodone Hydrochloride (EMD 68843) , a partial agonist of 5-HT1A receptors and specific serotonin reuptake inhibitor (SSRI), is utilized in treating of theFormule :C26H27N5O2·HClDegré de pureté :99.56% - >99.99%Couleur et forme :SolidMasse moléculaire :477.99Ivabradine hydrochloride
CAS :Ivabradine HCl (S 16257-2) is an If inhibitor (IC50: 2.9 μM) and SA node HCN channel blocker that slows heart rate.Formule :C27H37ClN2O5Degré de pureté :99% - 99.73%Couleur et forme :SolidMasse moléculaire :505.05Opromazine hydrochloride
CAS :Opromazine hydrochloride, a phenothiazine antipsychotic, blocks brain dopamine receptors to treat schizophrenia and psychosis.Formule :C17H20Cl2N2OSDegré de pureté :98.03%Couleur et forme :SolidMasse moléculaire :371.32Ref: TM-T50054
1mg38,00€5mg82,00€1mL*10mM (DMSO)94,00€10mg111,00€25mg182,00€50mg269,00€100mg389,00€200mg555,00€[Lys5,MeLeu9,Nle10]-NKA(4-10)
CAS :Highy selective and potent NK2 receptor agonist (IC50 = 6.1 nM). Induces contraction of the rat fundus and bladder (EC50 values are 117 and 10 nM respectively).Formule :C39H65N9O9Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :803.99Ritanserin
CAS :Ritanserin (R 55667) is a long-acting, highly potent, relatively selective, orally bioavailable 5-HT2 receptor antagonist.Cost-effective and quality-assured.Formule :C27H25F2N3OSDegré de pureté :99.77% - 99.89%Couleur et forme :SolidMasse moléculaire :477.57TRAP-6 amide acetate
TRAP-6 amide acetate is a PAR-1 thrombin receptor agonist peptide[1].Formule :C36H61N11O10Degré de pureté :98.55%Couleur et forme :SolidMasse moléculaire :807.94Mini Gastrin I, human acetate
Mini Gastrin I, human acetate is a shorter version of human gastrin, consists of amino acids 5-17 of the parent peptide.Formule :C76H103N15O28SDegré de pureté :99.35% - 99.82%Couleur et forme :SolidMasse moléculaire :1706.78Metiamide
CAS :Metiamide (SK&F 92058) is a histamine H2-receptor antagonist .Formule :C9H16N4S2Degré de pureté :97.41%Couleur et forme :SolidMasse moléculaire :244.38SORT-PGRN interaction inhibitor 1
CAS :SORT-PGRN interaction inhibitor 1 is a potent sortilin-progranulin interaction inhibitor(IC50 of 2 μM).Formule :C15H18N2O2Degré de pureté :98.72%Couleur et forme :SolidMasse moléculaire :258.32Darbufelone mesylate
CAS :Darbufelone mesylate blocks PGF2α, LTB4, PGHS-2 (IC50: 0.19 μM), and PGHS-1 (IC50: 20 μM).Formule :C19H28N2O5S2Degré de pureté :96.81% - 99.92%Couleur et forme :SolidMasse moléculaire :428.57Ref: TM-T10960L
1mg50,00€5mg99,00€1mL*10mM (DMSO)109,00€10mg167,00€25mg340,00€50mg557,00€100mg790,00€200mg1.063,00€PF-06291874
CAS :PF-06291874 (Glucagon receptor antagonists-4) (Glucagon receptor antagonists-4) is a highly effective and orally active antagonist of the glucagon receptor.Formule :C26H28F3N3O4Degré de pureté :99.12% - 99.27%Couleur et forme :SolidMasse moléculaire :503.51Sultopride hydrochloride
CAS :Sultopride hydrochloride (LIN-1418 hydrochloride) is a selective dopamine D2 and D3 receptor antagonist.Formule :C17H27ClN2O4SDegré de pureté :≥95%Couleur et forme :White Or Yellowish PowderMasse moléculaire :390.93A-381393
CAS :A-381393 is a selective and brain penetrate dopamine D4 receptor antagonist (Kis: 1.9/1.5/1.6 nM for human dopamine D4.2/D4.4/D4.7 receptor).Formule :C20H24N4Degré de pureté :99.00%Couleur et forme :SolidMasse moléculaire :320.43Ref: TM-T5397
1mg38,00€5mg75,00€1mL*10mM (DMSO)84,00€10mg111,00€25mg198,00€50mg288,00€100mg414,00€200mg583,00€Otenabant
CAS :Otenabant (CP-945598) has been investigated for the treatment of Obesity.Formule :C25H25Cl2N7ODegré de pureté :99.43%Couleur et forme :SolidMasse moléculaire :510.42Procaterol hydrochloride hydrate
CAS :Short-acting β2-adrenergic receptor agonist used to treat asthma.Formule :C32H48Cl2N4O7Degré de pureté :99.71% - 99.97%Couleur et forme :SolidMasse moléculaire :671.65Ref: TM-T4548
1mg54,00€5mg114,00€1mL*10mM (DMSO)156,00€10mg167,00€25mg289,00€50mg485,00€100mg690,00€200mg888,00€Neurokinin A(4-10) TFA(97559-35-8 free base)
Neurokinin A(4-10) TFA(97559-35-8 free base) is a tachykinin NK2 receptor agonist[1].Formule :C36H55F3N8O12SDegré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :880.93[Sar9,Met(O2)11]-Substance P acetate
[Sar9,Met(O2)11]-Substance P acetate is an NK1 agonist, raising MAP and HR equally to septide but with unique timing and behaviors.Formule :C66H106N18O18SDegré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :1471.75TGR5 Receptor Agonist
CAS :TGR5 is a potent TGR5(GPCR19) agonist.Formule :C18H14Cl2N2O2Degré de pureté :99.77% - ≥95%Couleur et forme :SolidMasse moléculaire :361.22BMY-25368
CAS :BMY-25368 is a long-acting antagonist of the H2-receptor.Formule :C19H25N3O3Couleur et forme :SolidMasse moléculaire :343.42Nonapeptide-1 acetate salt (158563-45-2 free base)
Nonapeptide-1 acetate salt (158563-45-2 free base) (Melanostatine-5 acetate salt) , a peptide hormone, is a potent α-Melanocyte-stimulating hormone (α-MSH)Formule :C63H91N15O11SDegré de pureté :98.26%Couleur et forme :SolidMasse moléculaire :1266.58Dolasetron Mesylate hydrate
CAS :Dolasetron Mesylate hydrate blocks 5HT3 to prevent chemo and radiotherapy nausea.Formule :C20H26N2O7SDegré de pureté :99.86% - 99.99%Couleur et forme :SolidMasse moléculaire :438.49Alprenolol benzoate
CAS :Alprenolol benzoate is the benzoate salt of Alprenolol -- a beta blocker.Formule :C22H29NO4Couleur et forme :SolidMasse moléculaire :371.48Neuropeptide S (Rat) acetate
Neuropeptide S (Rat) acetate is an endogenous ligand of a previously orphan G-protein-coupled receptor now named NPS receptor.Formule :C97H164N34O29Degré de pureté :95.36%Couleur et forme :SolidMasse moléculaire :2270.59Ref: TM-TP1982L
1mg93,00€2mg117,00€5mg182,00€10mg269,00€25mg429,00€50mg610,00€100mg820,00€200mg1.099,00€BRL-15572 dihydrochloride
CAS :BRL-15572 dihydrochloride: 5-HT1D antagonist, pKi 7.9, also binds 5-HT1A/2B, 60x selective over 5-HT1B.Formule :C25H27ClN2O·2HClDegré de pureté :99.74%Couleur et forme :SolidMasse moléculaire :479.87Brimonidine Tartrate
CAS :Brimonidine Tartrate (AGN190342 tartrate) is a quinoxaline derivative and adrenergic α-2 receptor agonist (EC50: 0.45 nM).Formule :C15H16BrN5O6Degré de pureté :99.95%Couleur et forme :Off-White Crystalline SolidMasse moléculaire :442.22Tolazoline
CAS :Tolazoline (Benzalolin), a vasodilator, treats vessel spasms and reverses 5-HT2A drug overdose effects.
Formule :C10H12N2Degré de pureté :99.52%Couleur et forme :SolidMasse moléculaire :160.22Lanreotide acetate
CAS :Lanreotide acetate (BIM 23014 acetate) is a somatostatin analogue with antineoplastic activity, used for carcinoid syndromeFormule :C56H73N11O12S2Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :1156.39RS-127445 hydrochloride
CAS :RS-127445 hydrochloride (MT 500) is a selective, high affinity, orally bioavailable 5-HT2B receptor antagonist(pKi : 9.5).Formule :C17H17ClFN3Degré de pureté :99.48%Couleur et forme :SolidMasse moléculaire :317.79Zatebradine
CAS :Zatebradine is a potent hyperpolarization-activated cyclic nucleotide-gated (HCN) channels inhibitor(IC50 of 1.96 μM).Formule :C26H36N2O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :456.57Zacopride hydrochloride
CAS :Zacopride is a highly potent 5-HT3 receptor antagonist (Kd = 0.38 nM) and 5-HT4 receptor agonist (Ki = 373 nM). It also is a selective IK1 channel agonist.Formule :C15H20ClN3O2·HClDegré de pureté :98.32%Couleur et forme :SolidMasse moléculaire :346.26Ref: TM-T5336
1mg34,00€5mg71,00€1mL*10mM (DMSO)79,00€10mg99,00€25mg212,00€50mg385,00€100mg618,00€200mg859,00€NNC-0640
CAS :NNC-0640 is a negative allosteric modulator of Human Glucagon Receptor with an IC50 of 69.2 nM.Formule :C29H31N7O4SDegré de pureté :97.04%Couleur et forme :SolidMasse moléculaire :573.67Ref: TM-T7364
1mg46,00€2mg62,00€5mg90,00€1mL*10mM (DMSO)90,00€10mg160,00€25mg281,00€50mg430,00€100mg620,00€
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