GPCR/G-Protéine
Les inhibiteurs des GPCR/protéines G sont des composés qui ciblent les récepteurs couplés aux protéines G (GPCR) et les protéines G associées, qui jouent un rôle crucial dans la transmission des signaux de l'extérieur vers l'intérieur des cellules. Ces inhibiteurs sont essentiels pour étudier les voies de signalisation médiées par les GPCR, impliquées dans de nombreux processus physiologiques, y compris la perception sensorielle, la réponse immunitaire et la neurotransmission. Les inhibiteurs des GPCR sont également importants dans le développement de médicaments, car de nombreux agents thérapeutiques ciblent ces récepteurs. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de GPCR/protéines G de haute qualité pour soutenir vos recherches en pharmacologie, biologie cellulaire et domaines connexes.
Sous-catégories appartenant à la catégorie "GPCR/G-Protéine"
- récepteur 5-HT(1.025 produits)
- Récepteur d'adénosine(251 produits)
- Récepteur adrénergique(3.027 produits)
- Récepteur de la bombésine(35 produits)
- Récepteur de la bradykinine(61 produits)
- CXCR(158 produits)
- CaSR(34 produits)
- Récepteur cannabinoïde(218 produits)
- Cholécystokinine(1 produits)
- Récepteur de la dopamine(445 produits)
- Récepteur de l'endothéline(86 produits)
- Récepteur GNRH(84 produits)
- GPCR19(36 produits)
- GRK(33 produits)
- GTPase(23 produits)
- Récepteur du glucagon(195 produits)
- Hérisson/Smoothened(49 produits)
- Récepteur de l'histamine(385 produits)
- Récepteur LPA(21 produits)
- Récepteur de la mélatonine(26 produits)
- Récepteur OX(41 produits)
- Récepteur opioïde(327 produits)
- PAFR(14 produits)
- PKA(60 produits)
- Récepteur S1P(18 produits)
- SGLT(31 produits)
- Récepteur Sigma(46 produits)
Affichez 19 plus de sous-catégories
6011 produits trouvés pour "GPCR/G-Protéine"
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GRA Ex-25
CAS :GRA Ex-25 (GRA-Ex-25) is an inhibitor of glucagon receptor.Formule :C29H36F3N3O5Degré de pureté :98.2% - 98.88%Couleur et forme :SolidMasse moléculaire :563.61Ref: TM-T3422
1mg50,00€5mg105,00€1mL*10mM (DMSO)130,00€10mg161,00€25mg314,00€50mg470,00€100mg708,00€200mg964,00€BAY-545
CAS :BAY-545 is an antagonist of A2B adenosine receptor(IC50 : 59 nM).Formule :C18H22F3N3O4SDegré de pureté :98.05%Couleur et forme :SolidMasse moléculaire :433.45Ref: TM-T8512
1mg84,00€5mg161,00€1mL*10mM (DMSO)172,00€10mg235,00€25mg420,00€50mg605,00€100mg842,00€200mg1.134,00€Mequitazine
CAS :Mequitazine (Virginan) is an effective, nonsedative and long-acting histamine H1 antagonist.Formule :C20H22N2SDegré de pureté :99.98%Couleur et forme :SolidMasse moléculaire :322.47Lixisenatide acetate (320367-13-3 free base)
CAS :Lixisenatide acetate is a receptor agonist similar to glucagon-like peptide-1 (glp-1) for the treatment of type 2 diabetes mellitus (T2DM).Formule :C215H347N61O65S·6C2H4O2Degré de pureté :98% - 99.9%Couleur et forme :SolidMasse moléculaire :5218.88MF-766
CAS :MF-766: potent, selective oral EP4 antagonist, Ki=0.23 nM, IC50=1.4 nM; shifts to 1.8 nM with 10% HS. Useful in cancer, inflammation studies.Formule :C27H21F3N2O3Degré de pureté :99.54% - 99.59%Couleur et forme :SolidMasse moléculaire :478.46[D-Phe12,Leu14]-Bombesin acetate
[D-Phe12,Leu14]-Bombesin acetate inhibits bombesin-stimulated secretion.Formule :C77H118N22O20Degré de pureté :98.41% - 99.14%Couleur et forme :SolidMasse moléculaire :1671.9Chlorcyclizine
CAS :CHLORCYCLIZINE is a histamine H1 antagonist and a potent hepatitis C virus (HCV) entry inhibitor.Formule :C18H21ClN2Degré de pureté :98.75%Couleur et forme :SolidMasse moléculaire :300.83Ranitidine
CAS :Ranitidine (HSDB 3925) is a non-imidazole blocker of those histamine receptors that mediate gastric secretion (H2 receptors).Formule :C13H22N4O3SDegré de pureté :99.52%Couleur et forme :Solid SolidMasse moléculaire :314.40Orexin B, rat, mouse Acetate
Orexin B, rat, mouse Acetate (Rat orexin B) is an endogenous agonist at Orexin receptor with Kis of 420 and 36 nM for OX1 and OX2, respectively.Formule :C128H219N45O36SDegré de pureté :94.61%Couleur et forme :SolidMasse moléculaire :2996.45Metergoline
CAS :Metergoline (Methergoline) is a dopamine agonist and serotonin antagonist.Formule :C25H29N3O2Degré de pureté :99.83% - 99.97%Couleur et forme :SolidMasse moléculaire :403.52Ciproxifan maleate
CAS :Ciproxifan maleate (FUB 359)(FUB-359 maleate) is a highly potent and selective histamin H3-receptor antagonist with IC50 of 9.2 nM, with low apparent affinityFormule :C20H22N2O6Degré de pureté :99.39%Couleur et forme :SolidMasse moléculaire :386.4Ref: TM-T2004
1mg40,00€2mg52,00€5mg75,00€1mL*10mM (DMSO)82,00€10mg101,00€25mg205,00€50mg380,00€100mg565,00€Capadenoson
CAS :Capadenoson (BAY 68-4986) is a selective adenosine-A1 receptor agonist.Formule :C25H18ClN5O2S2Degré de pureté :98.85% - 99.57%Couleur et forme :SolidMasse moléculaire :520.03BWX 46 Acetate
BWX 46 Acetate is a potent, highly selective neuropeptide Y (NPY) receptor agonist with IC50 of 0.5 nM.Formule :C118H190N36O30S2Degré de pureté :96.86%Couleur et forme :SolidMasse moléculaire :2657.12ATC 0175 free base
CAS :ATC0175 is a potent, orally active MCH1R antagonist with high selectivity over MCH2R, demonstrating antidepressant and anxiolytic effects in animal models.Formule :C23H25F2N5ODegré de pureté :99.73%Couleur et forme :SolidMasse moléculaire :425.47Neurotensin(8-13) 3TFA(60482-95-3(free base))
CAS :Neurotensin(8-13) 3TFA is Neurotensin (NT) fragment. Neurotensin(8-13) 3TFA results in a decrease in cell-surface NT1 receptors (NTR1) density.Formule :C40H65F3N12O10Degré de pureté :98.31%Couleur et forme :SolidMasse moléculaire :931.03Ref: TM-T7617L
1mg35,00€5mg73,00€10mg107,00€1mL*10mM (DMSO)132,00€25mg207,00€50mg313,00€100mg447,00€200mg620,00€Piboserod
CAS :Piboserod (SB-207266) (SB 207266) is a selective 5-HT(4) receptor antagonist.Formule :C22H31N3O2Degré de pureté :97.21% - 99.49%Couleur et forme :SolidMasse moléculaire :369.5Ref: TM-T2278
1mg38,00€2mg50,00€5mg84,00€10mg118,00€1mL*10mM (DMSO)120,00€25mg220,00€50mg403,00€100mg582,00€500mg1.198,00€L-745870 trihydrochloride
CAS :L-745870 trihydrochloride is a highly potent and selective D4 dopamine receptor antagonist.Formule :C18H22Cl4N4Degré de pureté :97.52%Couleur et forme :SolidMasse moléculaire :436.21JNJ-7777120
CAS :JNJ-7777120 is the first potent and selective non-imidazole histamine H4 receptor antagonist, exhibits >1000-fold selectivity over the other histamin receptors.Formule :C14H16ClN3ODegré de pureté :99.83% - 99.96%Couleur et forme :SolidMasse moléculaire :277.754i
CAS :4i (CHEMBL1269981) is a 5-HT3 receptor antagonist,It modulates the serotonergic system.Formule :C16H12ClN3ODegré de pureté :99.49%Couleur et forme :SolidMasse moléculaire :297.74CGP71683 hydrochloride
CAS :CGP71683 hydrochloride: NPY5 receptor antagonist, Ki=1.3 nM; inactive at Y1 (Ki >4000 nM) and Y2 (Ki=200 nM).Formule :C26H30ClN5O2SDegré de pureté :99.92%Couleur et forme :SolidMasse moléculaire :512.07Bevantolol hydrochloride
CAS :Bevantolol hydrochloride (NC-1400 hydrochloride) is a β1-adrenoceptor antagonist that treatment angina pectoris and hypertension.Formule :C20H28ClNO4Degré de pureté :99.49%Couleur et forme :SolidMasse moléculaire :381.9Pimozide
CAS :Pimozide: antipsychotic that blocks type 2 dopamine, alpha-adrenergic, and 5-HT2 receptors, reducing tics and delusions.Formule :C28H29F2N3ODegré de pureté :99.63% - >99.99%Couleur et forme :SolidMasse moléculaire :461.55NPY 5RA972
CAS :NPY 5RA972 is a neuropeptide Y Y5 receptor antagonistFormule :C21H25N3O2Degré de pureté :99.02% - 99.56%Couleur et forme :SolidMasse moléculaire :351.44Ivabradine hydrochloride
CAS :Ivabradine HCl (S 16257-2) is an If inhibitor (IC50: 2.9 μM) and SA node HCN channel blocker that slows heart rate.Formule :C27H37ClN2O5Degré de pureté :99% - 99.73%Couleur et forme :SolidMasse moléculaire :505.05dasiglucagon acetate
Dasiglucagon acetate: new, stable glucagon for hypoglycemia with better absorption and longer half-life.Formule :C154H226N38O52Degré de pureté :99.63%Couleur et forme :SolidMasse moléculaire :3441.67Dimaprit dihydrochloride
CAS :Dimaprit dihydrochloride: selective H2 agonist, inhibits nNOS (IC50: 49 μM), boosts gastric acid.Formule :C6H15N3S·2HClDegré de pureté :99.79%Couleur et forme :SolidMasse moléculaire :234.19HPI 1
CAS :HPI 1 suppresses Hh pathway: IC50 = 1.5 μM (Shh, SAG), 4 μM (Gli2), 6 μM (Gli1) in Shh-LIGHT2 cells.Formule :C27H29NO6Degré de pureté :97.6%Couleur et forme :SolidMasse moléculaire :463.52Ref: TM-T22089
1mg44,00€2mg57,00€5mg96,00€1mL*10mM (DMSO)102,00€10mg128,00€25mg207,00€50mg308,00€100mg447,00€500mg973,00€N-Desmethylclozapine
CAS :N-Desmethylclozapine: 5-HT2C antagonist (IC50: 7.1 nM), dopamine D4 antagonist, δ-opioid agonist.Formule :C17H17ClN4Degré de pureté :97.25% - 99.83%Couleur et forme :Yellow Crystalline SolidMasse moléculaire :312.8Ref: TM-T5158
2mg34,00€5mg48,00€1mL*10mM (DMSO)58,00€10mg79,00€25mg152,00€50mg235,00€100mg344,00€200mg490,00€SBI-115
CAS :SBI-115 is an antagonist of TGR5. SBI-115 decreases hepatic cystogenesis with polycystic liver diseases via inhibiting TGR5Formule :C14H13ClN2O4SDegré de pureté :99.53% - 99.78%Couleur et forme :SolidMasse moléculaire :340.78ZK 756326
CAS :ZK 756326: Selective CCR8 agonist, IC50 1.8 μM (human), 2.6 μM (mouse), no CCR4/5, CXCR3/4 action, 28-fold selectivity vs 26 GPCRs, anti-HIV fusion.Formule :C21H28N2O3Degré de pureté :99.43%Couleur et forme :SolidMasse moléculaire :356.46OXOMEMAZINE
CAS :Oxomemazine: a phenothiazine antihistamine H1-blocker with strong antimuscarinic and selective M1 antagonist properties, used in cough research.Formule :C18H22N2O2SDegré de pureté :99.58%Couleur et forme :SolidMasse moléculaire :330.44Clemizole
CAS :Clemizole is an H1 histamine receptor antagonist, can inhibit NS4B's RNA binding and hepatitis C virus (HCV) replication.Formule :C19H20ClN3Degré de pureté :98% - 99.65%Couleur et forme :SolidMasse moléculaire :325.84Ref: TM-T1822
1mg42,00€5mg82,00€1mL*10mM (DMSO)93,00€10mg101,00€25mg152,00€50mg256,00€100mg460,00€500mg973,00€AC-55541
CAS :AC-55541 (AOB2796), a PAR2 agonist, activates PAR2 in cellular proliferation assays, phosphatidylinositol hydrolysis assays, and Ca(2+) mobilization assays.
Formule :C25H20BrN5O3Degré de pureté :98% - 99.33%Couleur et forme :SolidMasse moléculaire :518.36Litorin acetate(55749-97-8 Free base)
Litorin acetate, an amphibian bombesin peptide derivative, is an bombesin receptor agonist.Formule :C53H72N14O13SDegré de pureté :98.61%Couleur et forme :SolidMasse moléculaire :1145.29Tulobuterol hydrochloride
CAS :Tulobuterol hydrochloride (Hokunalin) is a long-acting beta2-adrenergic receptor agonist.Formule :C12H19Cl2NODegré de pureté :99.24% - >99.99%Couleur et forme :Appearance White Crystalline PowderMasse moléculaire :264.19LY334370
CAS :LY334370 is a selective 5-HT1F receptor agonist with a Ki of 1.6 nMFormule :C21H22FN3ODegré de pureté :99.32%Couleur et forme :SolidMasse moléculaire :351.42Ozagrel hydrochloride
CAS :Ozagrel hydrochloride (OKY-046 HCl) is a selective thromboxane A(2) synthetase inhibitor used for the improvement of postoperative cerebrovascular contractionFormule :C13H12N2O2·HClDegré de pureté :99.80%Couleur et forme :White Or Off White Crystalline PowderMasse moléculaire :264.71Aprepitant
CAS :Aprepitant (Aprepitant`) is a Substance P/Neurokinin-1 Receptor Antagonist.Formule :C23H21F7N4O3Degré de pureté :98% - 99.68%Couleur et forme :Off-White To Light Yellow Cyrstalline SolidMasse moléculaire :534.43Sevoflurane
CAS :Sevoflurane (Fluoromethyl), a noncompetitive inhibitor of 5-HT3 receptor, acts as a low-soluble inhalation anesthetics.Formule :C4H3F7ODegré de pureté :98%Couleur et forme :Less Oil Colorless OilMasse moléculaire :200.05Ref: TM-T22425
2mg39,00€5mg54,00€1mL*10mM (DMSO)56,00€10mg75,00€25mg110,00€50mg158,00€100mg226,00€200mg339,00€ML-SI3
CAS :CCG-143140 is a GLP-1 receptor inverse agonists.Formule :C23H31N3O3SDegré de pureté :99.75%Couleur et forme :SolidMasse moléculaire :429.58CCG215022
CAS :CCG215022 is a G protein-coupled receptor kinases (GRKs) inhibitor with IC50s of 0.15±0.07 μM, 0.38±0.06 μM and 3.9±1 μM for GRK2, 5 and 1, respectively.Formule :C26H22FN7O3Degré de pureté :97.63% - 99.69%Couleur et forme :SolidMasse moléculaire :499.5Ref: TM-T3498
1mg56,00€5mg114,00€1mL*10mM (DMSO)127,00€10mg178,00€25mg394,00€50mg655,00€100mg1.035,00€Clemizole hydrochloride
CAS :Clemizole hydrochloride blocks H1 histamine receptors and inhibits HCV replication and NS4B RNA binding.Formule :C19H21Cl2N3Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :362.3PF-4136309
CAS :PF-4136309 (INCB8761) is a specific, effective, and orally bioavailable CCR2 antagonist.Formule :C29H31F3N6O3Degré de pureté :98.85% - 99.47%Couleur et forme :SolidMasse moléculaire :568.59PGS-IN-1
CAS :PGS-IN-1 (KME-4) is a potent inhibitor of prostaglandin synthetase (PGS, IC50: 0.28 μM) and 5-lipoxygenase (IC50: 1.05 μM).Formule :C19H26O3Degré de pureté :99.39%Couleur et forme :SolidMasse moléculaire :302.41BMS-813160
CAS :BMS-813160 is the first dual CCR2/CCR5 antagonist to enter Clinical development for cardiovascular.Formule :C25H40N8O2Degré de pureté :99.66% - 99.79%Couleur et forme :SolidMasse moléculaire :484.64Ref: TM-T4584
1mg63,00€5mg137,00€1mL*10mM (DMSO)145,00€10mg187,00€25mg341,00€50mg567,00€100mg810,00€500mg1.644,00€HhAntag
CAS :HhAntag is a small molecule inhibitor of GLI1-mediated transcription, an essential down-stream element of the Hedgehog (Hh) pathway with the anti-tumor activityFormule :C24H23ClN4O3Degré de pureté :95.73%Couleur et forme :SolidMasse moléculaire :450.92BX471
CAS :BX471 (BX 471) is a potent, selective non-peptide CCR1 antagonist.Formule :C21H24ClFN4O3Degré de pureté :98% - 99.98%Couleur et forme :SolidMasse moléculaire :434.89Ref: TM-T2375
1mg35,00€5mg86,00€1mL*10mM (DMSO)95,00€10mg117,00€25mg200,00€50mg313,00€100mg489,00€200mg740,00€Glasdegib
CAS :Glasdegib (PF-04449913) (PF-04449913) is a potent, and orally bioavailable Smoothened (Smo) inhibitor with IC50 of 5 nM. Phase 2.Formule :C21H22N6ODegré de pureté :98.72%Couleur et forme :SolidMasse moléculaire :374.44RS102895
CAS :RS102895 is a potent CCR2 antagonist (IC50: 360 nM) and shows no effect on CCR1.Formule :C21H21F3N2O2Degré de pureté :97.64% - 99.80%Couleur et forme :SolidMasse moléculaire :390.4SAG
CAS :SAG (Smoothened Agonist) is a Smo receptor agonist (EC50=3 nM) that is cell-permeable and selective.
Formule :C28H28ClN3OSDegré de pureté :97.37% - 98.88%Couleur et forme :SolidMasse moléculaire :490.06Ciliobrevin A
CAS :Ciliobrevin A (HPI-4) is an inhibitor of hedgehog signaling pathway with an IC50 <10 μM.Formule :C17H9Cl2N3O2Degré de pureté :98.54% - 99.57%Couleur et forme :SolidMasse moléculaire :358.18Ref: TM-T3156
2mg39,00€5mg56,00€1mL*10mM (DMSO)65,00€10mg80,00€25mg165,00€50mg224,00€100mg314,00€200mg467,00€SANT-1
CAS :SANT-1 directly binds to Smoothened (Smo) receptor (Kd: 1.2 nM) and inhibits Smo agonist effects (IC50: 20 nM).Formule :C23H27N5Degré de pureté :99.93% - >99.99%Couleur et forme :SolidMasse moléculaire :373.49Vercirnon
CAS :Vercirnon (Traficet-EN) is a selective and potent antagonist of CCR9 (IC50: 10 nM). It is also used in the research of inflammatory bowel diseases.Formule :C22H21ClN2O4SDegré de pureté :99.23%Couleur et forme :SolidMasse moléculaire :444.93Ref: TM-T17225
1mg100,00€5mg245,00€1mL*10mM (DMSO)344,00€10mg385,00€25mg645,00€50mg888,00€100mg1.234,00€500mg2.457,00€SAG hydrochloride (912545-86-9(free base))
CAS :SAG hydrochloride (912545-86-9(free base)) (Smoothened Agonist HCl) acts as an SMO agonist.Formule :C28H29Cl2N3OSDegré de pureté :99.19% - 99.97%Couleur et forme :SolidMasse moléculaire :526.52Ref: TM-T4211
1mg49,00€2mg65,00€5mg90,00€1mL*10mM (DMSO)105,00€10mg114,00€25mg222,00€50mg334,00€100mg502,00€200mg717,00€R243
CAS :R243 is CCR8 signaling and chemotaxis inhibitor.Formule :C21H27NO4Degré de pureté :99.03%Couleur et forme :SolidMasse moléculaire :357.44Ref: TM-T24700
1mg40,00€2mg52,00€5mg80,00€1mL*10mM (DMSO)90,00€10mg117,00€25mg207,00€50mg333,00€100mg495,00€Sonidegib
CAS :Sonidegib (Erismodegib), a Smoothened (Smo) antagonist, inhibits Hedgehog (Hh) signaling with IC50 of 1.3 nM (mouse) and 2.5 nM (human), respectively.Formule :C26H26F3N3O3Degré de pureté :98% - 99.97%Couleur et forme :SolidMasse moléculaire :485.5Salmeterol Xinafoate
CAS :Salmeterol Xinafoate (GR 33343X xinafoate) is a long-acting β2-adrenergic receptor agonist with anti-inflammatory effects, used in the treatment of asthma.Formule :C36H45NO7Degré de pureté :98% - 98.24%Couleur et forme :White SolidMasse moléculaire :603.75MRT-81
CAS :MRT-81 blocks Smo receptors in Shh-light2 cells at 41 nM IC50, showing strong hedgehog pathway inhibition, useful in cancer research.Formule :C31H29N3O5SDegré de pureté :99.72%Couleur et forme :SolidMasse moléculaire :555.64Ref: TM-T9532
1mg46,00€5mg92,00€1mL*10mM (DMSO)110,00€10mg138,00€25mg241,00€50mg349,00€100mg479,00€200mg657,00€SB297006
CAS :SB297006 is an antagonist of C-C chemokine receptor 3, which normally is activated by eotaxin, eotaxin-3, MCP-3, MCP-4, RANTES, and MIP-1δ.Formule :C18H18N2O5Degré de pureté :99.59%Couleur et forme :SolidMasse moléculaire :342.35Felypressin
CAS :Felypressin, a Lypressin analog with a phenylalanine substitution, acts as a vasoconstrictor with less antidiuretic effect.Formule :C46H65N13O11S2Degré de pureté :99.65%Couleur et forme :SolidMasse moléculaire :1040.22Geissoschizine methyl ether
CAS :Geissoschizine methyl ether: an alkaloid from Uncaria hook, key in Yokukansan, impacts mood and social behavior enhancing serotonin activity.Formule :C22H26N2O3Degré de pureté :99.24% - 99.68%Couleur et forme :SolidMasse moléculaire :366.45Ref: TM-TN1032
1mg130,00€2mg187,00€5mg319,00€1mL*10mM (DMSO)326,00€10mg485,00€25mg770,00€50mg1.035,00€100mg1.395,00€VUF10460
CAS :VUF10460 is a non-imidazole histamine H4 receptor agonist.Formule :C15H19N5Degré de pureté :99.44% - 99.57%Couleur et forme :SolidMasse moléculaire :269.34Ansofaxine hydrochloride
CAS :Ansofaxine hydrochloride (LY03005) is a serotonin-norepinephrine-dopamine reuptake inhibitor (IC50s: 723, 763 and 491 nM, respectively).Formule :C24H32ClNO3Degré de pureté :99.57% - 99.77%Couleur et forme :SolidMasse moléculaire :417.97Treprostinil
CAS :Treprostinil (Orenitram) is a potent DP1, IP and EP2 agonist (EC50: 0.6/1.9/6.2 nM).Formule :C23H34O5Degré de pureté :99.29%Couleur et forme :SolidMasse moléculaire :390.51Ref: TM-T5150
1mg34,00€1mL*10mM (DMSO)60,00€5mg71,00€10mg108,00€25mg221,00€50mg355,00€100mg533,00€200mg755,00€BA 1 acetate(183241-31-8 free base)
BA 1 acetate: bombesin agonist, IC50s: 0.26/1.55/2.52 nM (BB1/BB2/BB3), boosts glucose transport, promotes lung cancer cell growth in vitro.Formule :C59H80N14O13Degré de pureté :95.3%Couleur et forme :SolidMasse moléculaire :1193.35Binodenoson
CAS :Binodenoson (WRC 0470), a selective A2A adenosine receptor agonist, aids in coronary imaging.Formule :C17H25N7O4Degré de pureté :99.74%Couleur et forme :SolidMasse moléculaire :391.42Ref: TM-T9516
1mg94,00€5mg222,00€1mL*10mM (DMSO)245,00€10mg334,00€25mg557,00€50mg745,00€100mg1.044,00€Asapiprant
CAS :Asapiprant (S-555739) is a potent and selective DP1 receptor antagonist (Ki: 0.44 nM). It exhibited high affinity and selectivity for the DP1 receptor.Formule :C24H27N3O7SDegré de pureté :99.64%Couleur et forme :SolidMasse moléculaire :501.55Ref: TM-T5386
1mg38,00€5mg92,00€1mL*10mM (DMSO)100,00€10mg147,00€25mg269,00€50mg424,00€100mg692,00€200mg888,00€Lecirelin acetate(61012-19-9 free base)
Lecirelin acetate is a synthetic GnRH (gonadotropin releasing hormone) analogue which shows a great efficacy in the treatment of bovine ovarian follicular cystsFormule :C61H88N16O14Degré de pureté :98.1%Couleur et forme :SolidMasse moléculaire :1269.45Nelociguat
CAS :Nelociguat (BAY60-4552) is an sGC stimulator, crucial in NO signal pathways.
Formule :C19H17FN8O2Degré de pureté :99.19%Couleur et forme :SolidMasse moléculaire :408.39Neurokinin A
CAS :Neurokinin A (NKA), formerly known as Substance K, is a neurologically active peptide translated from the pre-protachykinin gene.Formule :C50H80N14O14SDegré de pureté :>99.99%Couleur et forme :White To Off-White Lyophilized SolidMasse moléculaire :1133.32Phenylbiguanide
CAS :Phenylbiguanide (N-Phenylbiguanide) is a 5-HT3 receptor selective agonist(EC50 : 3.0±0.1 μM)Formule :C8H11N5Degré de pureté :99.54%Couleur et forme :SolidMasse moléculaire :177.21Lys-[Des-Arg9]Bradykinin acetate
Lys-[Des-Arg9]Bradykinin acetate is an endogenous potent and highly selective bradykinin B1 receptor agonist (Ki values are 0.12 and > 30000 nM at human B1 andFormule :C52H77N13O13Degré de pureté :99.93%Couleur et forme :SolidMasse moléculaire :1092.27I-191
CAS :I-191 is a potent antagonist of protease-activated receptor 2 (PAR2), inhibits multiple signaling functions in human cancer cells.Formule :C23H26FN5O2Degré de pureté :99.8%Couleur et forme :SolidMasse moléculaire :423.48M40 acetate(143896-17-7 free base)
M40 acetate is a potent, non-selective galanin receptor antagonist (Ki values are 1.82 and 5.1 nM at GAL1 and GAL2 respectively) that inhibits galanin (1-29)Formule :C96H149N23O26Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :2041.38Ticagrelor metabolite M5
CAS :Ticagrelor metabolite M5 (T437700) is a metabolite of Ticagrelor, the first reversible oral antagonist of P2Y12 receptor.Formule :C14H22N6O4SDegré de pureté :99.35%Couleur et forme :SolidMasse moléculaire :370.43AR-M 1896 Acetate
AR-M 1896 Acetate is the selective agonist of GalR2.Formule :C56H85N13O16Degré de pureté :99.76%Couleur et forme :SolidMasse moléculaire :1196.35Ref: TM-T21646L
1mg305,00€5mg605,00€10mg827,00€25mg1.215,00€1mL*10mM (DMSO)1.251,00€50mg1.603,00€100mg2.142,00€Eledoisin Related Peptide 2TFA
Eledoisin Related Peptide 2TFA (Eledoisin Related Peptide 2TFA (2990-43-4(free base))) is a tachykinin receptor ligand.Formule :C38H60F6N8O10SDegré de pureté :99%Couleur et forme :SolidMasse moléculaire :934.99Sitaxsentan sodium
CAS :Sitaxsentan sodium (TBC11251 sodium salt) is a highly selective antagonist of endothelin A receptors.Formule :C18H14ClN2O6S2·NaDegré de pureté :98.39% - 99.01%Couleur et forme :SolidMasse moléculaire :476.89Motilin (26-47), human, porcine
CAS :Motilin (26-47) binds Motilin receptors in hamster cells; Ki=2.3 nM, EC50=0.3 nM; same for humans, pigs.Formule :C120H188N34O35SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :2699.07Ref: TM-TP1425
500µg86,00€1mg111,00€5mg334,00€10mg504,00€25mg745,00€50mg999,00€100mg1.341,00€200mg1.773,00€LIXIVAPTAN
CAS :Lixivaptan (VPA-985) is an orally active and selective vasopressin receptor V2 antagonist(Ki = 2.3 nM)Formule :C27H21ClFN3O2Degré de pureté :98.36%Couleur et forme :SolidMasse moléculaire :473.93Ref: TM-T7303
2mg34,00€5mg66,00€1mL*10mM (DMSO)70,00€10mg99,00€25mg205,00€50mg334,00€100mg522,00€200mg743,00€Loxapine
CAS :Loxapine, a dibenzoxazepine antipsychotic, treats schizophrenia by blocking D2/D4 and serotonin receptors. Related to clozapine.Formule :C18H18ClN3ODegré de pureté :99.88%Couleur et forme :Pale Yellowish Crystals From Petroleum Ether SolidMasse moléculaire :327.81ACTH (1-17) acetate
ACTH (1-17) acetate is a potent agonist at the human melanocortin 1 (MC1) receptor with high affinity(Ki = 0.21 nM).Formule :C97H149N29O25SDegré de pureté :98.53%Couleur et forme :SolidMasse moléculaire :2153.47Pergolide
CAS :Pergolide is a long-acting and orally active dopamine receptor D1/D2 agonist and ergoline derivative, used in the study of Parkinson's diseaseFormule :C19H26N2SDegré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :314.49Ref: TM-T21340
2mg37,00€5mg54,00€1mL*10mM (DMSO)60,00€10mg77,00€25mg110,00€50mg164,00€100mg237,00€200mg350,00€Decloxizine
CAS :Decloxizine is a H1 receptor antagonistFormule :C21H28N2O2Degré de pureté :99.53%Couleur et forme :White Or Similar To White PowderMasse moléculaire :340.46FSLLRY-NH2 TFA(245329-02-6 free base)
FSLLRY-NH2 TFA inhibits PAR2, reverses taxol-induced pain, and reduces itch in mice; blocks ERK and collagen in fibroblasts.Formule :C41H61F3N10O10Degré de pureté :99.32%Couleur et forme :SolidMasse moléculaire :910.99PF-04418948
CAS :PF-04418948 is a potent EP2 receptor antagonist. Displays over 2000-fold selectivity for EP2 receptors over EP1, EP3, EP4, DP1 amd CRTH2 receptors.Formule :C23H20FNO5Degré de pureté :98.67% - 99.45%Couleur et forme :SolidMasse moléculaire :409.41d[Cha4]-AVP acetate(500170-27-4 free base)
'd[Cha4]-AVP acetate: strong V1B agonist, weak on V1A/Oxytocin/V2. Boosts ACTH, corticosterone; low blood pressure effect.'Formule :C52H75N13O13S2Degré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :1154.37Brexpiprazole
CAS :Brexpiprazole (OPC-34712) is a partial agonist of human 5-hydroxytryptamine (5-HT) 5-HT1A and dopamine D2 receptors.Formule :C25H27N3O2SDegré de pureté :99.06% - 99.96%Couleur et forme :SolidMasse moléculaire :433.57Ref: TM-T2306
1mL*10mM (DMSO)À demander5mg50,00€10mg63,00€25mg75,00€50mg88,00€100mg94,00€200mg140,00€500mg259,00€Urapidil
CAS :Urapidil (Ebrantil), a sympatholytic antihypertensive drug, acts as a 5-HT1A receptor agonist and as an α1-adrenoceptor antagonist.Formule :C20H29N5O3Degré de pureté :99.85% - >99.99%Couleur et forme :SolidMasse moléculaire :387.48Norepinephrine bitartrate salt
CAS :Norepinephrine bitartrate salt is an adrenergic neurotransmitter.Formule :C12H17NO9Degré de pureté :97.32% - 99.97%Couleur et forme :SolidMasse moléculaire :319.27Scyliorhinin II acetate
Scyliorhinin II acetate is a selective agonist of the neurokinin-3 (NK3) receptor (Ki = 2.5 nM) in rat cerebral cortex.Formule :C79H123N21O28S3Degré de pureté :99.06%Couleur et forme :SolidMasse moléculaire :1911.14Tolazoline
CAS :Tolazoline (Benzalolin), a vasodilator, treats vessel spasms and reverses 5-HT2A drug overdose effects.
Formule :C10H12N2Degré de pureté :99.52%Couleur et forme :SolidMasse moléculaire :160.22Ki16425
CAS :Ki16425 (Debio 0719) is a competitive, potent and reversible antagonist to LPA1, LPA2 and LPA3 with Ki of 0.34 μM, 6.5 μM and 0.93 μM, respectively.Formule :C23H23ClN2O5SDegré de pureté :97.6% - 97.78%Couleur et forme :SolidMasse moléculaire :474.96Perospirone hydrochloride
CAS :Perospirone hydrochloride (Perospirone HCl) is an atypical antipsychotic agent for the treatment of schizophrenia.Formule :C23H31ClN4O2SDegré de pureté :99.37%Couleur et forme :White SolidMasse moléculaire :463Serotonin
CAS :Serotonin (5-hydroxytryptamine) is a monoamine neurotransmitter in the CNS and an endogenous 5-HT receptor agonist. High-Quality, Low-Cost!Formule :C10H12N2ODegré de pureté :97.47% - 99.92%Couleur et forme :SolidMasse moléculaire :176.22Melatonin
CAS :Melatonin (Melatonine) is a natural hormone that activates melatonin receptors. Melatonin regulates the biological clock. Cost-effective and quality-assured.Formule :C13H16N2O2Degré de pureté :98% - 99.89%Couleur et forme :Pale Yellow Leaflets From Benzene SolidMasse moléculaire :232.28Verucerfont
CAS :Verucerfont (NBI77860) is an antagonist of corticotropin-releasing factor receptor 1 (CRF1) .Formule :C22H26N6O2Degré de pureté :99.90%Couleur et forme :SolidMasse moléculaire :406.48Ref: TM-T7361
1mg60,00€2mg87,00€5mg130,00€1mL*10mM (DMSO)142,00€10mg205,00€25mg376,00€50mg573,00€100mg803,00€Levalbuterol tartrate
CAS :Levalbuterol tartrate is a short-acting β2-adrenergic receptor agonist and the R enantiomer of salbutamol.Cost-effective and quality-assured.Formule :C17H27NO9Degré de pureté :99.28% - 99.98%Couleur et forme :SolidMasse moléculaire :389.39Ref: TM-T7164
2mg34,00€5mg50,00€1mL*10mM (DMSO)60,00€10mg88,00€25mg100,00€50mg124,00€100mg177,00€200mg259,00€PD-168077 maleate
CAS :PD-168077 maleate is a selective agonist of dopamine D4 receptor(Ki : 9 nM)Formule :C24H26N4O5Degré de pureté :99.13%Couleur et forme :SolidMasse moléculaire :450.49Ref: TM-T5047
2mg34,00€5mg50,00€1mL*10mM (DMSO)55,00€10mg75,00€25mg142,00€50mg231,00€100mg344,00€200mg490,00€IPSU
CAS :IPSU is an antagonist of OX2 receptor. IPSU Exhibits approximately six-fold selectivity for OX2 versus OX1 receptors.Formule :C23H27N5O2Degré de pureté :97.05%Couleur et forme :SolidMasse moléculaire :405.49Ref: TM-T5503
2mg51,00€5mg86,00€1mL*10mM (DMSO)92,00€10mg97,00€25mg200,00€50mg299,00€100mg432,00€200mg662,00€8-Cyclopentyl-1,3-dimethylxanthine
CAS :8-Cyclopentyl-1,3-dimethylxanthine (CPT) is a potent antagonist of adenosine A1 receptor.Formule :C12H16N4O2Degré de pureté :98.58% - 99.9%Couleur et forme :SolidMasse moléculaire :248.283-AQC
CAS :3-AQC is a competitive antagonist of 5-HT3.Formule :C20H21N5O4Degré de pureté :99.45%Couleur et forme :SolidMasse moléculaire :395.41Avexitide
CAS :Avexitide (Exendin-3 (9-39) amide) (Exendin (9-39)) is a specific and competitive antagonist of glucagon-like peptide-1 (GLP-1) receptor.Formule :C149H234N40O47SDegré de pureté :98% - 99.65%Couleur et forme :SolidMasse moléculaire :3369.76Methyldopa hydrate
CAS :Methyldopa hydrate (MK-351 hydrate) is a DOPA decarboxylase inhibitor and indirect α2-adrenergic receptor agonist used to treat hypertension.Formule :C10H13NO4H2ODegré de pureté :99.67%Couleur et forme :White SolidMasse moléculaire :238.24Tiprenolol
CAS :Tiprenolol is a beta adrenergic receptor antagonist.[1]Formule :C13H21NO2SDegré de pureté :99.43%Couleur et forme :SolidMasse moléculaire :255.38Ref: TM-T50081
1mg52,00€1mL*10mM (DMSO)89,00€5mg98,00€10mg146,00€25mg235,00€50mg319,00€100mg447,00€200mg587,00€Conopressin S acetate(111317-90-9 free base)
Conopressin S acetate(111317-90-9 free base) (Con-S acetate) is a natural product isolated from Conus striatus, shows high affinity with vasopressin V1bFormule :C43H77N17O12S2Degré de pureté :99.79%Couleur et forme :SolidMasse moléculaire :1088.32AVN-101
CAS :AVN-101 is a very potent 5-HT7 receptor antagonist.Cost-effective and quality-assured.Formule :C21H25ClN2Degré de pureté :99.61%Couleur et forme :SolidMasse moléculaire :340.89Ref: TM-T26690
1mg34,00€5mg75,00€1mL*10mM (DMSO)92,00€10mg114,00€25mg205,00€50mg334,00€100mg557,00€200mg790,00€Betahistine dihydrochloride
CAS :Betahistine dihydrochloride (Betahistine 2HCl) is a histamine analog and H1 receptor agonist that serves as a vasodilator.Formule :C8H14Cl2N2Degré de pureté :99.22% - 99.88%Couleur et forme :White To Light Yellow Crystalline PowderMasse moléculaire :209.12Mosapride
CAS :Mosapride (AS-4370) is a selective 5HT4 agonistFormule :C21H25ClFN3O3Degré de pureté :99.56%Couleur et forme :White To Off-White Crystalline SolidMasse moléculaire :421.89KH7
CAS :KH7 is a soluble inhibitor of adenylyl cyclase (sAC)-specific.Formule :C17H15BrN4O2SDegré de pureté :98.43%Couleur et forme :SolidMasse moléculaire :419.3Thrombin Receptor Activator for Peptide
Thrombin Receptor Activator (TRAP) or Coagulation Factor II (1-5), used in CHD research.Formule :C32H51F3N8O9Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :748.79HAEGTFT acetate(926018-95-3 free base)
HAEGTFT acetate is the first N-terminal 1-7 residues of GLP-1 peptide.Formule :C35H51N9O14Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :821.84Linzagolix
CAS :Linzagolix is a small-molecule, non-peptide, orally active gonadotropin-releasing hormone antagonist (GnRH antagonist) which is under development by KisseiFormule :C22H15F3N2O7SDegré de pureté :99.33%Couleur et forme :SolidMasse moléculaire :508.42ACH-000143
CAS :ACH-000143 是一种可口服的褪黑素受体激动剂，对 MT1 和 MT2 的EC50值分别为0.06 和0.32 nM。Formule :C13H16ClN3O3Degré de pureté :98.15%Couleur et forme :SolidMasse moléculaire :297.74Ref: TM-T9193
1mg50,00€5mg110,00€1mL*10mM (DMSO)122,00€10mg172,00€25mg304,00€50mg424,00€100mg583,00€200mg785,00€Ablukast
CAS :Ablukast (Ro 23-3544) is a leuktriene receptor antagonist. Ablukast acts as an anti-asthmatic.Formule :C28H34O8Degré de pureté :98.58%Couleur et forme :SolidMasse moléculaire :498.56GW842166X
CAS :GW842166X: Potent CB2 agonist, EC50=63 nM, inactive at CB1, in Phase 2 trials.Formule :C18H17Cl2F3N4O2Degré de pureté :99.47%Couleur et forme :SolidMasse moléculaire :449.25Thonzylamine
CAS :Thonzylamine is an antihistamine/anticholinergic, combined with Clofedanol or Phenylephrine for cold, hay fever, or allergy relief.Formule :C16H22N4ODegré de pureté :99.45%Couleur et forme :SolidMasse moléculaire :286.37LML134
CAS :LML134 (LML-134) is an inverse agonist of Histamine 3 receptor (H3R)(hH3R cAMP and hH3R bdg with Kis of 0.3 nM and 12 nM).Formule :C19H29N5O3Degré de pureté :99.36%Couleur et forme :SolidMasse moléculaire :375.47Ref: TM-T8514
1mg34,00€5mg78,00€1mL*10mM (DMSO)86,00€10mg112,00€25mg203,00€50mg299,00€100mg447,00€200mg600,00€Talinolol
CAS :(±)-Talinolol is a selective β1 adrenoceptor antagonist well known for its cardioprotective and antihypertensive activity.Formule :C20H33N3O3Degré de pureté :98.8%Couleur et forme :SolidMasse moléculaire :363.49Ref: TM-T21640
2mg34,00€5mg52,00€1mL*10mM (DMSO)52,00€10mg92,00€25mg178,00€50mg313,00€100mg535,00€200mg775,00€Ibutamoren Mesylate
CAS :Ibutamoren Mesylate (MK-0677) is a potent, non-peptide Growth hormone secretagogue receptor (GHSR) agonist.Formule :C28H40N4O8S2Degré de pureté :97.98% - ≥98%Couleur et forme :SolidMasse moléculaire :624.77SCH-23390 hydrochloride
CAS :SCH-23390 hydrochloride (R-(+)-SCH23390 hydrochloride) is an effective dopamine receptor antagonist, and for the D1(Ki=0.2 nM) and D5(Ki=0.3 nM).Formule :C17H19Cl2NODegré de pureté :98% - 99.83%Couleur et forme :SolidMasse moléculaire :324.24Ref: TM-T4369
1mg39,00€2mg50,00€5mg78,00€1mL*10mM (DMSO)78,00€10mg97,00€25mg195,00€50mg369,00€100mg550,00€Clozapine N-Oxide
CAS :View and buy CLOZAPINE N-OXIDE from TargetMol.Clozapine N-oxide is a major metabolite of clozapine also known as DREADDs, technology to modulate synthetic receptors in vivo.Cited in 2 publications.Formule :C18H19ClN4ODegré de pureté :98.65% - 99.94%Couleur et forme :SolidMasse moléculaire :342.82OXA (17-33) acetate
OXA (17-33) acetate is a more potent agonist of orexin-1 receptor (OX1, EC50 = 8.29 nM)) over OX2 (EC50 = 187 nM).Formule :C79H125N23O22Degré de pureté :98.52%Couleur et forme :SolidMasse moléculaire :1748.98MK-0557
CAS :MK-0557 is a selective and orally available antagonist of the neuropeptide Y5 receptor (Ki: 1.6 nM).Formule :C22H19FN4O3Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :406.41Ref: TM-TQ0286
1mg34,00€5mg67,00€1mL*10mM (DMSO)75,00€10mg92,00€25mg166,00€50mg264,00€100mg371,00€200mg517,00€Bradykinin (acetate)
CAS :Bradykinin (acetate) is an active peptide that is generated by the kallikrein-kinin system.Formule :C52H77N15O13Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :1120.26Cariprazine hydrochloride
CAS :Cariprazine hydrochloride (RGH188 hydrochloride) is an antipsychotic drug, is a D3 and D2 receptor partial agonist((Ki of 0.085 nM and 0.49 nM, respectively)Formule :C21H33Cl3N4ODegré de pureté :99.78% - >99.99%Couleur et forme :SolidMasse moléculaire :463.87Ditolylguanidine
CAS :Ditolylguanidine (Di-o-tolylguanidine) is an agonist of sigma receptor (σ1/σ2 receptor).Formule :C15H17N3Degré de pureté :98.42%Couleur et forme :White To Pinkish Solid PowderMasse moléculaire :239.32Tetradecyl Phosphonate
CAS :Tetradecyl Phosphonate 是溶血磷脂酸 1 (LPA1)、LPA2 和 LPA3 受体的泛拮抗剂。Formule :C14H31O3PDegré de pureté :99.95%Couleur et forme :White To Off-White PowderMasse moléculaire :278.37Midodrine
CAS :Midodrine ((±)-Midodrin), an adrenergic alpha-1 agonist, belongs to the class of medications known as vasopressors.Formule :C12H18N2O4Degré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :254.281-[(5-methylisoxazol-3-yl)methyl]piperazine
CAS :1-[(5-methylisoxazol-3-yl)methyl]piperazine (Piperazine, 1-[(5-methyl-3-isoxazolyl)methyl]- (9CI)) is a P2Y12 inhibitor.Formule :C9H15N3ODegré de pureté :95%Couleur et forme :SolidMasse moléculaire :181.23Ref: TM-T8582
1mL*10mM (DMSO)À demander1mg58,00€5mg116,00€10mg172,00€25mg281,00€50mg396,00€100mg537,00€200mg712,00€VKGILS-NH2 Acetate
VKGILS-NH2 Acetate is a reversed amino acid sequence control peptide for SLIGKV-NH2, a protease-activated receptor 2 (PAR2) agonist.Formule :C30H58N8O9Degré de pureté :98.83%Couleur et forme :SolidMasse moléculaire :674.83Ref: TM-T21699L
1mg33,00€2mg49,00€5mg62,00€10mg92,00€1mL*10mM (DMSO)92,00€25mg155,00€50mg224,00€100mg331,00€200mg470,00€Hydroxyzine dihydrochloride
CAS :Hydroxyzine dihydrochloride treats allergies, pruritus, anxiety; causes drowsiness; also an antiemetic and sedative.Formule :C21H27ClN2O2·2HClDegré de pureté :99.46% - 99.79%Couleur et forme :Oil PowderMasse moléculaire :447.83Dapagliflozin ((2S)-1,2-propanediol, hydrate)
CAS :Dapagliflozin ((2S)-1,2-propanediol, hydrate) (BMS-512148 (2S)-1,2-propanediol, hydrate) is a selective, orally active inhibitor of the renal sodium-glucose co-Formule :C24H35ClO9Degré de pureté :99.88% - 99.94%Couleur et forme :SolidMasse moléculaire :502.98DORA-22
CAS :DORA-22 is a dual orexin receptor antagonist, improves mild stress-induced insomnia with minimal effect on memoryFormule :C23H22F2N4O2Degré de pureté :97.67%Couleur et forme :SolidMasse moléculaire :424.44Ref: TM-T5500
1mg131,00€2mg188,00€5mg284,00€1mL*10mM (DMSO)331,00€10mg430,00€25mg710,00€50mg998,00€100mg1.349,00€lumateperone Tosylate
CAS :lumateperone Tosylate (ITI-007) is a 5-HT2A receptor antagonist, a partial agonist of presynaptic D2 receptors and an antagonist of postsynaptic D2 receptors.Formule :C31H36FN3O4SDegré de pureté :95.83% - 99.95%Couleur et forme :SolidMasse moléculaire :565.7Peptide YY (PYY) (3-36), human
CAS :Peptide YY (PYY) (3-36), human (Peptide YY (3-36)) is a gut hormone peptide. Peptide YY (PYY) (3-36), human acts as a Y2 receptor agonist to reduce appetite.Formule :C176H272N52O54Degré de pureté :97.76%Couleur et forme :SolidMasse moléculaire :3980.42Doxazosin
CAS :Doxazosin (UK 33274) is a long-lasting inhibitor of α1-adrenoceptors that is widely used to treat benign prostatic hyperplasia and lower urinary tract symptoms.Formule :C23H25N5O5Degré de pureté :99.47% - 99.87%Couleur et forme :SolidMasse moléculaire :451.48Ropinirole hydrochloride
CAS :Ropinirole HCl (SKF-101468A) is a selective D2 dopamine agonist (Ki: 29 nM) with antiparkinsonian effects.Formule :C16H24N2O·HClDegré de pureté :99.87% - 99.98%Couleur et forme :Off-White SolidMasse moléculaire :296.84D3-βArr
CAS :D3-βArr (NCGC00379308) is a positive allosteric modulator for thyrotropin receptor (TSHR), which initiates translocation of β-Arr 1 (EC50: 11.6 μM) by directFormule :C20H23N5Degré de pureté :98.82%Couleur et forme :SolidMasse moléculaire :333.43Vilazodone Hydrochloride
CAS :Vilazodone Hydrochloride (EMD 68843) , a partial agonist of 5-HT1A receptors and specific serotonin reuptake inhibitor (SSRI), is utilized in treating of theFormule :C26H27N5O2·HClDegré de pureté :99.56% - >99.99%Couleur et forme :SolidMasse moléculaire :477.99PF-06291874
CAS :PF-06291874 (Glucagon receptor antagonists-4) (Glucagon receptor antagonists-4) is a highly effective and orally active antagonist of the glucagon receptor.Formule :C26H28F3N3O4Degré de pureté :99.12% - 99.27%Couleur et forme :SolidMasse moléculaire :503.51S 38093 HCl
CAS :S 38093 is a novel brain-penetrant antagonist/inverse agonist of H3 receptors.Formule :C17H25ClN2O2Degré de pureté :97.91%Couleur et forme :SolidMasse moléculaire :324.85Ref: TM-T4087
1mg37,00€5mg71,00€1mL*10mM (DMSO)71,00€10mg92,00€25mg164,00€50mg225,00€100mg323,00€200mg437,00€Cetirizine Impurity B dihydrochloride
CAS :Cetirizine Impurity B dihydrochloride is a Cetirizine antihistamine byproduct with anti-allergic properties.Formule :C19H23Cl3N2O2Degré de pureté :97.33%Couleur et forme :SolidMasse moléculaire :417.76Anisotropine Methylbromide
CAS :Anisotropine Methylbromide is an anticholinergic agent and has been used for relief of gastrointestinal spasm and for the suppression of gastric acid secretion.Formule :C17H32BrNO2Degré de pureté :99.73%Couleur et forme :Crystals From Acetone SolidMasse moléculaire :362.35ABT-702 dihydrochloride
CAS :ABT-702 dihydrochloride is a potent adenosine kinase (AK) inhibitor.Formule :C22H21BrCl2N6ODegré de pureté :98.42% - 98.98%Couleur et forme :SolidMasse moléculaire :536.25Ref: TM-T4668
1mg58,00€2mg82,00€5mg113,00€1mL*10mM (DMSO)133,00€10mg177,00€25mg333,00€50mg502,00€100mg710,00€500mg1.494,00€Parmodulin 2
CAS :ML161 (Parmodulin 2) inhibits PAR1, blocking platelet activation and thrombin-induced activity (IC50: 0.26μM).Formule :C17H17BrN2O2Degré de pureté :97.35% - 99.95%Couleur et forme :SolidMasse moléculaire :361.23Derenofylline
CAS :Derenofylline is a selective and potent adenosine A(1) antagonist in vitro (Ki=1 nM)Formule :C18H20N4ODegré de pureté :98.09%Couleur et forme :SolidMasse moléculaire :308.38NNC-0640
CAS :NNC-0640 is a negative allosteric modulator of Human Glucagon Receptor with an IC50 of 69.2 nM.Formule :C29H31N7O4SDegré de pureté :97.04%Couleur et forme :SolidMasse moléculaire :573.67Ref: TM-T7364
1mg46,00€2mg62,00€5mg90,00€1mL*10mM (DMSO)90,00€10mg160,00€25mg281,00€50mg430,00€100mg620,00€Org 27569
CAS :Org 27569, an allosteric modulator of cannabinoid CB1 receptor, can induce a CB1 receptor state that is characterized by decreased inverse agonist affinity andFormule :C24H28ClN3ODegré de pureté :>99.99% - ≥95%Couleur et forme :SolidMasse moléculaire :409.95Antalarmin
CAS :Antalarmin is a CRHR1 antagonist that blocks adrenocorticotropin-releasing hormone-induced hypertension, blocks CRF activation.Formule :C24H34N4Degré de pureté :99.99%Couleur et forme :SolidMasse moléculaire :378.55Ref: TM-T70433
1mg81,00€5mg170,00€1mL*10mM (DMSO)173,00€10mg241,00€25mg408,00€50mg552,00€100mg745,00€Xaliproden hydrochloride
CAS :Xaliproden is a compound that mimics the effects of nerve growth factor and is also a serotonin 5-HT1A receptor agonist.Formule :C24H23ClF3NDegré de pureté :99.99%Couleur et forme :SolidMasse moléculaire :417.89Ref: TM-T9272
1mg38,00€5mg80,00€1mL*10mM (DMSO)92,00€10mg114,00€25mg222,00€50mg356,00€100mg512,00€200mg735,00€CAY10526
CAS :CAY10526 (BTH) is a selective mPGES-1 inhibitor that acts as an inhibitor of the NF-κB signaling pathway.Formule :C12H7BrO3SDegré de pureté :98.75%Couleur et forme :SolidMasse moléculaire :311.15Cerlapirdine
CAS :Cerlapirdine (PF-05212365), a 5-HT6 receptor antagonist, is in trials for Alzheimer's and schizophrenia cognition issues.Formule :C22H23N3O3SDegré de pureté :98.77%Couleur et forme :SolidMasse moléculaire :409.5Ref: TM-T30798
1mg81,00€5mg170,00€1mL*10mM (DMSO)198,00€10mg274,00€25mg543,00€50mg780,00€100mg1.074,00€Elinzanetant
CAS :Elinzanetant is a dual antagonist of neurokinin (NK) receptors 1 and 3 and modulates reproductive hormone secretion.Formule :C33H35F7N4O3Degré de pureté :98% - 99.13%Couleur et forme :SolidMasse moléculaire :668.64Ref: TM-T38144
1mg92,00€2mg118,00€5mg192,00€1mL*10mM (DMSO)284,00€10mg313,00€25mg528,00€50mg740,00€100g4.977,00€Hemokinin 1 (human) acetate(491851-53-7 free base)
Hemokinin 1 acetate: Human SP homolog, NK1 agonist (IC50: NK1 1.8 nM), proliferates B-cells, antihypertensive.Formule :C56H88N14O16SDegré de pureté :97.82%Couleur et forme :SolidMasse moléculaire :1245.45Lerisetron
CAS :Lerisetron is an antagonist of serotonin type 3 (5-HT3) receptor, with antiemetic activity.Formule :C18H20N4Degré de pureté :99.15% - 99.82%Couleur et forme :SolidMasse moléculaire :292.38M871 acetate
M871 acetate is a selective galanin GAL2 receptor antagonist (Ki values are 13.1 and 420 nM at GAL2 and GAL1 receptors, respectively).It blocks pronociceptiveFormule :C110H167N27O30Degré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :2347.67Eltoprazine hydrochloride
CAS :Eltoprazine hydrochloride (DU 28853 hydrochloride) is a partial agonist at serotonin 5-HT1A, 5-HT1B, and 5-HT2B receptors (Ki value of 40, 52, and 81 nM,Formule :C12H17ClN2O2Degré de pureté :99.35%Couleur et forme :SolidMasse moléculaire :256.73Guanfacine hydrochloride
CAS :Guanfacine hydrochloride (Intuniv) is a centrally acting antihypertensive agent with specificity towards ADRENERGIC ALPHA-2 RECEPTORS.Formule :C9H10Cl3N3ODegré de pureté :99.89% - 99.91%Couleur et forme :SolidMasse moléculaire :282.55Plecanatide
CAS :Plecanatide acetate is an analogue of Uroguanylin. It is an orally active guanylate cyclase-C (GC-C) receptor agonist.Formule :C65H104N18O26S4Degré de pureté :97.51%Couleur et forme :SolidMasse moléculaire :1681.89Metoclopramide hydrochloride hydrate
CAS :Metoclopramide hydrochloride hydrate (Metoclopramide monohydrochloride monohydrate) is a dopamine D2 antagonist that is a drug used for digestive dysfunction.Formule :C14H25Cl2N3O3Degré de pureté :99.33%Couleur et forme :SolidMasse moléculaire :354.27TY-52156
CAS :TY-52156 is an effective and selective S1P3 receptor antagonist (Ki: 110 nM).Formule :C18H19Cl2N3ODegré de pureté :99.91% - 99.91%Couleur et forme :SolidMasse moléculaire :364.27Ref: TM-T17183
2mg38,00€5mg57,00€1mL*10mM (DMSO)63,00€10mg93,00€25mg158,00€50mg281,00€100mg484,00€200mg647,00€BD-1047 dihydrobromide
CAS :BD-1047 dihydrobromide (BD1047.2HBr) , a selective functional antagonist of sigma receptors, has antipsychotic activity in animal models predictive of efficacyFormule :C13H22Br2Cl2N2Degré de pureté :98.13% - 99.39%Couleur et forme :SolidMasse moléculaire :437.04Ref: TM-T1740
1mg37,00€2mg48,00€5mg73,00€1mL*10mM (DMSO)74,00€10mg95,00€25mg168,00€50mg290,00€100mg490,00€Amperozide
CAS :Amperozide (FG 5606), an atypical antipsychotic, antagonizes 5-HT2A and modulates dopamine activity for schizophrenia treatment.Formule :C23H29F2N3ODegré de pureté :99.68%Couleur et forme :SolidMasse moléculaire :401.49Ref: TM-T23733
1mg87,00€5mg178,00€10mg295,00€1mL*10mM (DMSO)321,00€25mg497,00€50mg708,00€100mg964,00€500mg1.918,00€HT-2157
CAS :HT-2157 (SNAP-37889) is a selective, high-affinity competitive antagonist of the galanin-3 receptor (Gal3), demonstrating effective inhibition of this target.Formule :C21H13F3N2ODegré de pureté :98.33%Couleur et forme :SolidMasse moléculaire :366.34L-732138
CAS :L-732138 is a potent and competitive antagonist of neurokinin-1 (NK-1) receptor(IC50 : 2.3 nM)Formule :C22H18F6N2O3Degré de pureté :99.77%Couleur et forme :SolidMasse moléculaire :472.38Ref: TM-T8235
1mL*10mM (DMSO)À demander5mg50,00€10mg80,00€25mg135,00€50mg192,00€100mg286,00€200mg416,00€Indophagolin
CAS :Indophagolin: autophagy inhibitor, IC50 140 nM; blocks P2X4, P2X1, P2X3 receptors, IC50s 2.71, 2.40, 3.49 μM.Formule :C19H15BrClF3N2O3SDegré de pureté :99.76%Couleur et forme :SolidMasse moléculaire :523.75Phenelzine
CAS :Phenelzine is a MAOI antidepressant, boosting brain catecholamines, effective for endogenous depression.Formule :C8H12N2Degré de pureté :98%Couleur et forme :LiquidMasse moléculaire :136.19Ref: TM-T9540
5mgÀ demander10mgÀ demander25mgÀ demander50mgÀ demander100mgÀ demander200mgÀ demander500mgÀ demanderMK-1064
CAS :MK-1064 (Urokinase inhibitor 1) is a selective orexin 2 receptor antagonist (2-SORA).Formule :C24H20ClN5O3Degré de pureté :99.19% - 99.82%Couleur et forme :SolidMasse moléculaire :461.9Vortioxetine hydrobromide
CAS :Vortioxetine hydrobromide (Lu AA21004 hydrobromide) is a serotonin (5-HT) modulator and stimulator (SMS), inhibits 5-HT1A/1B/3A/7 receptor and SERT (IC50: 15/33Formule :C18H22N2S·HBrDegré de pureté :98.85% - 99.98%Couleur et forme :SolidMasse moléculaire :379.36Desmopressin acetate (16679-58-6 free base)
CAS :Desmopressin (16679-58-6), a synthetic vasopressin analog, treats nocturia, enuresis, and diabetes insipidus by reducing urine production.Formule :C48H68N14O14S2Degré de pureté :98.84% - >99.99%Couleur et forme :SolidMasse moléculaire :1129.26Zatebradine
CAS :Zatebradine is a potent hyperpolarization-activated cyclic nucleotide-gated (HCN) channels inhibitor(IC50 of 1.96 μM).Formule :C26H36N2O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :456.57RS-67333
CAS :RS-67333 is a partial agonist of 5-HT4R with neuroprotective effects.Formule :C19H29ClN2O2Degré de pureté :99.24%Couleur et forme :SolidMasse moléculaire :352.9Bay 55-9837 acetate
Bay 55-9837 acetate is a potent and highly selective VPAC2 agonist(Kd = 0.65 nM) and can be used in type 2 diabetes studies.Degré de pureté :98.27%Couleur et forme :LiquidMasse moléculaire :N/ANeuropeptide Y (29-64), amide, human acetate
Neuropeptide Y (29-64), amide, human acetate is involved in Alzheimer's disease (AD) and protects rat cortical neurons against β-Amyloid toxicity.Degré de pureté :98.42%Couleur et forme :LiquidMasse moléculaire :N/APancreatic Polypeptide (human) acetate
Pancreatic Polypeptide (human) acetate is a C-terminally amidated 36 amino acid peptide, which acts as a neuropeptide Y (NPY) Y4/Y5 receptor agonist.Degré de pureté :97.26%Couleur et forme :LiquidMasse moléculaire :N/AHuman growth hormone-releasing factor acetate
Human growth hormone-releasing factor acetate is a hypothalamic polypeptide and stimulates GH production and release by binding to the GHRH Receptor (GHRHR) onDegré de pureté :99.26%Couleur et forme :LiquidMasse moléculaire :N/AK 41498 aceate
K41498 acetate, a potent CRF2 antagonist (Ki: 0.66/0.62 nM for CRF2α/β) with 425 nM for CRF1; blocks aSvg-30 effect on cAMP in cells.Degré de pureté :96.4%Couleur et forme :LiquidMasse moléculaire :N/APACAP 1-38 acetate
PACAP 1-38 acetate, a PACAP analog, targets PACAP type I (IC50=4nM) and VIP2 receptors (IC50=1nM), not VIP1.Degré de pureté :98.16%Couleur et forme :LiquidMasse moléculaire :N/AML382
CAS :ML382 is a potent and selective MrgX1 positive allosteric modulator(EC50 : 190 nM).Formule :C18H20N2O4SDegré de pureté :99.79%Couleur et forme :SolidMasse moléculaire :360.43Ketanserin tartrate
CAS :Ketanserin tartrate (KJK-945 tartrate) is a 5-HT2A receptor and α1-adrenergic receptor antagonist for the study of systemic sclerosis.Formule :C26H28FN3O9Degré de pureté :99.68%Couleur et forme :SolidMasse moléculaire :545.51Fenoprofen
CAS :Fenoprofen (LILLY-5385) is a non-steroidal anti-inflammatory compound and a modifier enhancer of the melanocortin receptor, increasing ERK1/2 activation.Formule :C15H14O3Degré de pureté :98.4%Couleur et forme :SolidMasse moléculaire :242.27Atogepant
CAS :Atogepant (MK-8031) is an orally available, selective and potent calcitonin gene-related peptide receptor (CGRP) antagonist for the study of migraine.Formule :C29H23F6N5O3Degré de pureté :99.66%Couleur et forme :SolidMasse moléculaire :603.52Ref: TM-T26682
1mg147,00€5mg250,00€10mg313,00€1mL*10mM (DMSO)334,00€25mg620,00€50mg1.108,00€100mg1.611,00€200mg2.178,00€KB-5492 free base
CAS :KB-5492 free base is an antiulcer agent that inhibits sigma receptors and can be used to study gastric lesions and gastric secretion.Formule :C23H30N2O6Degré de pureté :97.10% - 97.94%Couleur et forme :SolidMasse moléculaire :430.49Ref: TM-T62396
2mg39,00€5mg58,00€1mL*10mM (DMSO)64,00€10mg82,00€25mg119,00€50mg168,00€100mg249,00€500mg613,00€Benzylthiouracil
CAS :Benzylthiouracil (6-Benzyl-2-thiouracil) induces ANCA-associated glomerulonephritis in Graves' disease patients and is used to study hyperthyroidism.Formule :C11H10N2OSDegré de pureté :99.65%Couleur et forme :SolidMasse moléculaire :218.28Rolofylline
CAS :Rolofylline (KW-3902) is an adenosine A1 receptor antagonist used to study acute congestive heart failure and renal dysfunction.Formule :C20H28N4O2Degré de pureté :99.53%Couleur et forme :SolidMasse moléculaire :356.46Alfuzosin
CAS :Alfuzosin (SL 77499) is an alpha-1 adrenergic antagonist used to treat benign prostatic hypertrophy and urethral dysfunction.Formule :C19H27N5O4Degré de pureté :99.64%Couleur et forme :White Crystaline PowderMasse moléculaire :389.45Trabodenoson
CAS :Trabodenoson (INO-8875) is a selective and potent adenosine A1 receptor agonist, an adenosine analog, for the study of primary open-angle glaucoma.Formule :C15H20N6O6Degré de pureté :99.94%Couleur et forme :SolidMasse moléculaire :380.36Ref: TM-T34914
1mg40,00€1mL*10mM (DMSO)88,00€5mg89,00€10mg116,00€25mg187,00€50mg285,00€100mg411,00€200mg577,00€INCB 3284
CAS :INCB 3284, a potent human CCR2 antagonist with an IC50 of 3.7 nM, is researchable for acute liver failure and inhibits MCP-1/hCCR2 binding.Formule :C26H31F3N4O4Degré de pureté :97.81% - 99.42%Couleur et forme :SolidMasse moléculaire :520.54Protein deglycase DJ-1 against-1
CAS :Protein deglycase DJ-1 against-1 penetrate the BBB and bind to DJ-1 protein,restoring neuronal cellular death in a neurotoxin MPTP-induced model of PD.Formule :C24H23N3O4Degré de pureté :97.23%Couleur et forme :SolidMasse moléculaire :417.46GRK6-IN-2
CAS :GRK6-IN-2 is a potent G protein-coupled receptor kinase 6 (GRK6) inhibitor with potential antitumor activity.GRK6-IN-2 has been studied in multiple myeloma.Formule :C21H21FN6Degré de pureté :98.94%Couleur et forme :SolidMasse moléculaire :376.43Medetomidine
CAS :Medetomidine (MPV785 free base) is a selective α2-adrenoceptor agonist, with sedative and analgesic and vasoconstrictive hypoxic , in small animal anesthesia.Formule :C13H16N2Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :200.28Ref: TM-T21492
2mg38,00€5mg57,00€1mL*10mM (DMSO)62,00€10mg77,00€25mg128,00€50mg193,00€100mg290,00€200mg447,00€Poly-D-lysine hydrobromide (MW 30000-70000)
CAS :Poly-D-lysine hydrobromide (MW 30000-70000) (Poly-D-lysine HBr) is a peptide CaSR agonist that removes proteinase K-resistant PrP from SN56 neuroblastoma cells.Formule :(C6H14N2O2)x·xHBrCouleur et forme :SolidMasse moléculaire :227.102GAT211
CAS :GAT211 (AZ-4) is a cannabinoid 1 receptor (CB1R) positive allosteric modulator (PAM) for the study of epilepsy.Formule :C22H18N2O2Degré de pureté :99.7%Couleur et forme :SolidMasse moléculaire :342.39Ref: TM-T27405
1mg34,00€5mg66,00€1mL*10mM (DMSO)73,00€10mg90,00€25mg148,00€50mg210,00€100mg310,00€500mg750,00€ACT-462206
CAS :ACT-462206 is a Orexin 1/Orexin 2 receptor antagonist.ACT-462206 is highly potent and can be used to study sleep and anxiety.Formule :C20H24N2O4SDegré de pureté :99.45%Couleur et forme :SolidMasse moléculaire :388.48Ref: TM-T26559
1mg42,00€1mL*10mM (DMSO)87,00€5mg88,00€10mg130,00€25mg264,00€50mg423,00€100mg670,00€500mg1.341,00€Canagliflozin hemihydrate
CAS :Canagliflozin hemihydrate (TA 7284) treats type 2 diabetes by blocking SGLT2, leading to glucose excretion in urine.Formule :C48H52F2O11S2Degré de pureté :99.42% - 99.96%Couleur et forme :SolidMasse moléculaire :907.05Nebentan potassium
CAS :Nebentan potassium (YM598) is an ETA receptor antagonist that inhibits pulmonary arterial hypertension and is used in the study of neurologic diseases.Formule :C24H20KN5O5SDegré de pureté :99.05%Couleur et forme :SolidMasse moléculaire :529.61Ref: TM-T36008
1mg52,00€2mg77,00€5mg111,00€1mL*10mM (DMSO)133,00€10mg177,00€25mg313,00€50mg502,00€100mg680,00€200mg888,00€Maropitant citrate
CAS :Maropitant citrate is a synthetic neurokinin-1 receptor antagonist and substance P inhibitor, used for controlling vomiting in cats and dogs.Formule :C38H50N2O9Degré de pureté :98.91%Couleur et forme :SolidMasse moléculaire :678.81Pentoxyverine
CAS :Pentoxyverine (Carbetapentan) is an orally available cough suppressant, an antagonist of muscarinic receptor M1 and an agonist of the σ1 receptor.Formule :C20H31NO3Degré de pureté :97.11%Couleur et forme :SolidMasse moléculaire :333.47Clopidogrel thiolactone
CAS :Clopidogrel thiolactone (2-oxoclopidogrel), a P2Y12 receptor inhibitor, is an antiplatelet aggregation compound.Formule :C16H16ClNO3SDegré de pureté :98.79%Couleur et forme :SolidMasse moléculaire :337.82Ref: TM-T5501
1mg96,00€5mg205,00€1mL*10mM (DMSO)227,00€10mg326,00€25mg557,00€50mg803,00€100mg1.063,00€200mg1.459,00€
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