GPCR/G-Protéine
Les inhibiteurs des GPCR/protéines G sont des composés qui ciblent les récepteurs couplés aux protéines G (GPCR) et les protéines G associées, qui jouent un rôle crucial dans la transmission des signaux de l'extérieur vers l'intérieur des cellules. Ces inhibiteurs sont essentiels pour étudier les voies de signalisation médiées par les GPCR, impliquées dans de nombreux processus physiologiques, y compris la perception sensorielle, la réponse immunitaire et la neurotransmission. Les inhibiteurs des GPCR sont également importants dans le développement de médicaments, car de nombreux agents thérapeutiques ciblent ces récepteurs. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de GPCR/protéines G de haute qualité pour soutenir vos recherches en pharmacologie, biologie cellulaire et domaines connexes.
Sous-catégories appartenant à la catégorie "GPCR/G-Protéine"
- récepteur 5-HT(1.025 produits)
- Récepteur d'adénosine(248 produits)
- Récepteur adrénergique(2.994 produits)
- Récepteur de la bombésine(35 produits)
- Récepteur de la bradykinine(61 produits)
- CXCR(154 produits)
- CaSR(34 produits)
- Récepteur cannabinoïde(216 produits)
- Cholécystokinine(1 produits)
- Récepteur de la dopamine(445 produits)
- Récepteur de l'endothéline(86 produits)
- Récepteur GNRH(84 produits)
- GPCR19(33 produits)
- GRK(33 produits)
- GTPase(22 produits)
- Récepteur du glucagon(191 produits)
- Hérisson/Smoothened(49 produits)
- Récepteur de l'histamine(385 produits)
- Récepteur LPA(21 produits)
- Récepteur de la mélatonine(26 produits)
- Récepteur OX(41 produits)
- Récepteur opioïde(325 produits)
- PAFR(14 produits)
- PKA(59 produits)
- Récepteur S1P(17 produits)
- SGLT(31 produits)
- Récepteur Sigma(46 produits)
Affichez 19 plus de sous-catégories
5963 produits trouvés pour "GPCR/G-Protéine"
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Noradrenaline bitartrate
CAS :Norepinephrine bitartrate acts directly on the α- and β-adrenergic receptors.Formule :C12H19NO10Degré de pureté :99.53% - >99.99%Couleur et forme :SolidMasse moléculaire :337.28Clopidogrel
CAS :Clopidogrel (SR-25990C), a P2Y12 receptor antagonist, decreases platelet aggregation.Formule :C16H16ClNO2SDegré de pureté :98.23% - 98.83%Couleur et forme :White PowderMasse moléculaire :321.82AH 6809
CAS :AH 6809 blocks EP1, EP2, EP3, DP receptors (Ki: 1217-1597 nM human, 350 nM mouse EP2).Formule :C17H14O5Degré de pureté :97.59%Couleur et forme :SolidMasse moléculaire :298.29Ref: TM-T14148
1mg35,00€5mg66,00€10mg96,00€25mg168,00€50mg264,00€100mg424,00€200mg612,00€1mL*10mM (DMSO)71,00€Vilazodone
CAS :Vilazodone (SB659746A): an SSRI and 5-HT-1A agonist, boosts serotonin to treat depression and anxiety.Formule :C26H27N5O2Degré de pureté :99.61%Couleur et forme :Light Yellow SolidMasse moléculaire :441.52YNT-185
CAS :YNT-185 is a nonpeptide, selective agonist of the orexin type-2 receptor (OX2R), demonstrating EC50 values of 0.028 μM and 2.75 μM for OX2R and OX1R,Formule :C33H37N5O5SDegré de pureté :99.67%Couleur et forme :SolidMasse moléculaire :615.74Quetiapine
CAS :Quetiapine treats schizophrenia and bipolar I, targeting serotonin, dopamine, and adrenoreceptor subtypes, plus H1 histamine receptor.Formule :C21H25N3O2SDegré de pureté :99.14% - 99.63%Couleur et forme :White To Off-White Crystalline PowderMasse moléculaire :383.51Urocortin (rat) acetate
Urocortin (rat) acetate: CRF receptor agonist; Ki=13nM (hCRF1), 1.5nM (rCRF2α), 0.97nM (mCRF2β); neuropeptide.Degré de pureté :97.76%Couleur et forme :SoildTerlipressin Acetate
CAS :Terlipressin Acetate, a highly selective vasopressin V1 receptor agonist, on OGD/R-induced damage in intestinal epithelial cells (IEC-6).Formule :C56H82N16O19S2Degré de pureté :98.50% - 99.69%Couleur et forme :SolidMasse moléculaire :1347.5Ro 10-5824 dihydrochloride
CAS :Ro 10-5824 dihydrochloride is a selective agonist of dopamine D4 receptor partial, (Ki of 5.2 nM).Formule :C17H22Cl2N4Degré de pureté :99.79%Couleur et forme :SolidMasse moléculaire :353.29(3aR,9aR)-Fluparoxan
CAS :(3aR,9aR)-Fluparoxan is a highly selective and potent adrenergic receptor α2B antagonist for the prevention, amelioration or treatment of neurodevelopmentalFormule :C10H10FNO2Degré de pureté :97.82%Couleur et forme :SoildMasse moléculaire :195.19Levodropropizine
CAS :Levodropropizine ((S)-(-)-Dropropizine) is a histamine receptor inhibitor. It is used as an effective and very well tolerated peripheral antitussive drug.Formule :C13H20N2O2Degré de pureté :99.87% - 99.93%Couleur et forme :White Or Off White Crystalline PowderMasse moléculaire :236.31Tegaserod maleate
CAS :Tegaserod (SDZ-HTF-919), a 5-HT4 agonist for irritable bowel syndrome, was withdrawn by FDA on March 30, 2007, due to heart risk concerns.Formule :C20H27N5O5Degré de pureté :98% - 99.06%Couleur et forme :White PowderMasse moléculaire :417.46Ref: TM-T1551
10mg44,00€25mg74,00€50mg113,00€100mg188,00€200mg285,00€500mg482,00€1mL*10mM (DMSO)48,00€Erenumab
CAS :Erenumab: human antibody blocking CGRP receptors to prevent migraines.Degré de pureté :99.43% (SEC-HPLC) - > 95%Couleur et forme :LiquidMasse moléculaire :146.2 kDaDipivefrin hydrochloride
CAS :Dipivefrin hydrochloride (Dipivefrin HCl) that is available as an ophthalmic solution is a prodrug of adrenaline, which is used to treat glaucoma.Formule :C19H27NO5·HClDegré de pureté :99.22% - 99.92%Couleur et forme :Less Gas With A Sweet Odor Colorless Gas With A Sweet OdorMasse moléculaire :387.9Betaxolol hydrochloride
CAS :Betaxolol HCl (SL 75212) is a cardioselective beta-blocker for hypertension without reported liver injury.Formule :C18H30ClNO3Degré de pureté :99.48% - 99.56%Couleur et forme :SolidMasse moléculaire :343.89Protriptyline hydrochloride
CAS :Protriptyline HCl: a tricyclic antidepressant that increases norepinephrine and serotonin levels and has anticholinergic effects.Formule :C19H21N·HClDegré de pureté :98.54% - 99.98%Couleur et forme :SolidMasse moléculaire :299.84Thioridazine hydrochloride
CAS :Thioridazine hydrochloride (Mellaril) , an antipsychotic drug, is used in the therapy of psychosis and schizophrenia and shows serotonin antagonism or D4Formule :C21H27ClN2S2Degré de pureté :99.55% - 99.957%Couleur et forme :White To Off-White SolidMasse moléculaire :407.04Urapidil hydrochloride
CAS :Urapidil hydrochloride (Urapidil HCl) is 5-HT1A receptor agonist and an α1-adrenoceptor antagonist.Formule :C20H29N5O3·HClDegré de pureté :99.58%Couleur et forme :White Or Off-White Crystalline PowderMasse moléculaire :423.94INCB-9471
CAS :INCB-9471 is a CCR5 antagonist with anti-HIV activity and inhibits the interaction between HIV-1 gp120.Formule :C30H40F3N5O2Degré de pureté :98.80%Couleur et forme :SolidMasse moléculaire :559.666MK-0812 Succinate
CAS :MK-0812 Succinate is an effective and selective CCR2 antagonist.Formule :C28H40F3N3O7Degré de pureté :98.62% - 99.93%Couleur et forme :SolidMasse moléculaire :587.63Indacaterol maleate
CAS :Indacaterol maleate (QAB149) is an ultra-long-acting β-adrenoceptor agonist.Formule :C28H32N2O7Degré de pureté :99.03% - 99.67%Couleur et forme :SolidMasse moléculaire :508.56PF429242 dihydrochloride
CAS :PF429242 dihydrochloride can reversibly inhibit S1P (IC50 of 175 nM).
Formule :C25H37Cl2N3O2Degré de pureté :99.68%Couleur et forme :SolidMasse moléculaire :482.49Ifenprodil
CAS :Ifenprodil (RC61-91) inhibits NMDA receptor subunits GluN1 & GluN2B, GIRK channels, and affects alpha1, serotonin, sigma receptors.Formule :C21H27NO2Degré de pureté :99.58%Couleur et forme :White Crystalline PowderMasse moléculaire :325.44Ref: TM-T1186L
1mg70,00€5mg150,00€10mg219,00€25mg358,00€50mg512,00€100mg707,00€200mg973,00€1mL*10mM (DMSO)157,00€Oxeladin citrate
CAS :Oxeladin citrate: potent, non-addictive cough suppressant safe for all ages and heart patients; no common antitussive side effects.Formule :C26H41NO10Degré de pureté :97.23%Couleur et forme :SolidMasse moléculaire :527.6Nylidrin hydrochloride
CAS :Nylidrin HCl inhibits IgG1-induced histamine release in guinea pigs and IgE-induced release in rat mast cells & human basophils.Formule :C19H26ClNO2Degré de pureté :99.35%Couleur et forme :SolidMasse moléculaire :335.87MP-A08
CAS :MP-A08 selectively inhibits SPHK1; targets SphK1 & SphK2 with Ki of 6.9 μM & 27 μM, respectively.Formule :C27H25N3O4S2Degré de pureté :97.44%Couleur et forme :SolidMasse moléculaire :519.64Dopexamine hydrochloride
CAS :Dopexamine hydrochloride (FPL60278AR) is a β2-adrenoceptor agonist that modulates inflammation and protects organs without affecting hemodynamics.Formule :C22H34Cl2N2O2Degré de pureté :98.55%Couleur et forme :SolidMasse moléculaire :429.42CGS 15943
CAS :CGS 15943 is an orally bioavailable non-xanthine antagonist of Adenosine Receptor.Formule :C13H8ClN5ODegré de pureté :97.4%Couleur et forme :SolidMasse moléculaire :285.69Ref: TM-T14944
2mg34,00€5mg50,00€10mg82,00€25mg147,00€50mg222,00€100mg334,00€200mg494,00€1mL*10mM (DMSO)55,00€PF-4348235 2HCl
PF-4348235 2HCl is an adrenergic agonist and muscarinic receptor antagonist, and is a bronchodilator.Formule :C36H51Cl3N4O7SDegré de pureté :99.85%Couleur et forme :SolidMasse moléculaire :790.24Alfuzosin hydrochloride
CAS :Alfuzosin hydrochloride (Alfuzosin HCl) is an α1 adrenergic receptor antagonist. It applies to treat benign prostatic hyperplasia (BPH).Formule :C19H27N5O4·HClDegré de pureté :99.78%Couleur et forme :White To Off-White SolidMasse moléculaire :425.912-Bromo-6-methoxynaphthalene
CAS :2-Bromo-6-methoxynaphthalene was used in the synthesis of nabumetone [4-(6-methoxy-2-naphthalenyl)-2-butanone] by Heck reaction.Formule :C11H9BrODegré de pureté :98.51%Couleur et forme :White To Off-White PowderMasse moléculaire :237.09Ketanserin
CAS :Ketanserin: quinazoline derivative, 5-HT2 receptor antagonist, may lower blood pressure and inhibit blood clots.Formule :C22H22FN3O3Degré de pureté :99.19% - 99.73%Couleur et forme :SolidMasse moléculaire :395.43Prucalopride
CAS :Prucalopride (R-93877), a selective 5-HT4A/4B agonist (Ki: 2.5/8 nM), is >290x more specific for these receptors.Formule :C18H26ClN3O3Degré de pureté :99.99% - >99.99%Couleur et forme :SolidMasse moléculaire :367.87Domperidone
CAS :Domperidone (R33812)(Motilium) is a dopamine blocker and an antidopaminergic reagent.
Formule :C22H24ClN5O2Degré de pureté :98% - 99.82%Couleur et forme :SolidMasse moléculaire :425.91Venlafaxine hydrochloride
CAS :Venlafaxine HCl, a cyclohexanol phenethylamine, acts as an SNRI antidepressant.Formule :C17H28ClNO2Degré de pureté :97.32% - 99.86%Couleur et forme :White Crystalline PowderMasse moléculaire :313.86Isothiuronium
CAS :Isothiouronium, a functional group, is the acid salt of isothiourea.Formule :C12H25IN2SDegré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :356.31Chlorprothixene hydrochloride
CAS :Chlorprothixene hydrochloride, a typical antipsychotic, blocks 5-HT2, D1-D3, H1, muscarinic, and alpha1 receptors.Formule :C18H18ClNS·HClDegré de pureté :99.76% - 99.97%Couleur et forme :White PowderMasse moléculaire :352.32Prochlorperazine Maleate
CAS :Prochlorperazine Maleate (Capazine) is a phenothiazine antipsychotic used principally in the treatment of NAUSEA; VOMITING; and VERTIGO.Formule :C28H32ClN3O8SDegré de pureté :99.78%Couleur et forme :Off-White PowderMasse moléculaire :606.09Talastine
CAS :Talastine is an antihistamine compound that can induce an allergic rash.Formule :C19H21N3ODegré de pureté :99.44% - 99.84%Couleur et forme :SolidMasse moléculaire :307.39CP-809101 hydrochloride
CAS :CP-809101 hydrochloride is a potent and selective 5-HT2C receptor agonist (pEC50: 9.96/7.19/6.81 for human 5-HT2C/5-HT2B/5-HT2A receptors).Formule :C15H18Cl2N4ODegré de pureté :99.5%Couleur et forme :SolidMasse moléculaire :341.24Methyldopa
CAS :Methyldopa (MK-351), an alpha-adrenergic agonist (selective for α2-adrenergic receptors) psychoactive medicine, is served as an antihypertensive orFormule :C10H13NO4Degré de pureté :98.95% - 99.86%Couleur et forme :Less Or Almost Colorless Crystals Or White To Yellowish-White FineMasse moléculaire :211.21Azasetron hydrochloride
CAS :Azasetron hydrochloride (Y-25130 HCl) is a 5-HT3 receptor antagonist which is used as an anti-emetic.Formule :C17H20ClN3O3·HClDegré de pureté :99.50%Couleur et forme :SolidMasse moléculaire :386.27(-)-GSK598809 hydrochloride
CAS :(-)-GSK598809 hydrochloride, a DRD3 selective antagonist, may correct reward deficits in substance dependence.
Formule :C22H24ClF4N5OSDegré de pureté :98.36%Couleur et forme :SoildMasse moléculaire :517.97Amiselimod hydrochloride
CAS :Amiselimod hydrochloride (MT-1303 hydrochloride) is a sphingosine 1-phosphate receptor-1 (S1P1) modulator.Formule :C19H31ClF3NO3Degré de pureté :99.55%Couleur et forme :SolidMasse moléculaire :413.9Ref: TM-T10305
1mg35,00€2mg50,00€5mg75,00€10mg114,00€25mg203,00€50mg334,00€100mg485,00€200mg700,00€1mL*10mM (DMSO)84,00€Alverine citrate
CAS :Alverine citrate (NSC 35459) is utilized in functional gastrointestinal disorders.Formule :C26H35NO7Degré de pureté :98.53% - 99.43%Couleur et forme :CoaMasse moléculaire :473.57SR59230A
CAS :SR59230A is a potent, selective antagonist of β3-adrenergic receptor(β3, β1, and β2 receptors with IC50s of 40, 408, and 648 nM , respectively).Formule :C23H29NO6Degré de pureté :98.84%Couleur et forme :SolidMasse moléculaire :415.48Ref: TM-T13016
1mg50,00€2mg73,00€5mg102,00€10mg169,00€25mg324,00€50mg484,00€100mg697,00€1mL*10mM (DMSO)118,00€Filorexant
CAS :Filorexant (MK-6096) is an orally bioavailable effective and selective reversible antagonist of OX1 and OX2 receptor with (Ki <3 nM).Formule :C24H25FN4O2Degré de pureté :98.88%Couleur et forme :SolidMasse moléculaire :420.48Pizotifen
CAS :Pizotifen is a serotonin antagonist with mild anticholinergic effects, used in migraine prevention. Not available in the USA.Formule :C19H21NSDegré de pureté :99.93%Couleur et forme :SolidMasse moléculaire :295.44Clonidine hydrochloride
CAS :Clonidine hydrochloride (Catapres) is a centrally active α-adrenergic agonist used predominantly as an antihypertensive agent.Formule :C9H10Cl3N3Degré de pureté :99.16% - 99.86%Couleur et forme :SolidMasse moléculaire :266.55Quetiapine hemifumarate
CAS :Quetiapine hemifumarate (ICI-204636), an atypical antipsychotic, is used in the treatment of bipolar I mania, schizophrenia, bipolar I/II depression,.Formule :C46H54N6O8S2Degré de pureté :99.32% - >99.99%Couleur et forme :White Crystalline SolidMasse moléculaire :883.09Linaclotide
CAS :Linaclotide treats IBS-C & chronic constipation; it's a selective guanylate cyclase C agonist.Formule :C59H79N15O21S6Degré de pureté :97.93% - 98.71%Couleur et forme :SolidMasse moléculaire :1526.74Ref: TM-T11852
1mg50,00€5mg99,00€10mg177,00€25mg313,00€50mg465,00€100mg662,00€200mg888,00€1mL*10mM (DMSO)255,00€Pemirolast potassium
CAS :Pemirolast potassium, a pyrimidinone antiallergic, blocks antigen-induced Ca²⁺ influx in mast cells.Formule :C10H7KN6ODegré de pureté :98.91% - 99.63%Couleur et forme :Crystals From Dimethylformamide Crystalline SolidMasse moléculaire :266.31Ondansetron hydrochloride dihydrate
CAS :Ondansetron hydrochloride dihydrate (GR 38032) is a competitive serotonin type 3 receptor antagonist,which has reported anxiolytic and neuroleptic properties.Formule :C18H19N3O·HCl·2H2ODegré de pureté :99.92%Couleur et forme :White Crystal PowderMasse moléculaire :365.86Rimonabant
CAS :Rimonabant (SR141716) is an inverse agonist for the cannabinoid receptor CB1.Formule :C22H21Cl3N4ODegré de pureté :98% - 99.91%Couleur et forme :White Or Almost White Crystalline PowderMasse moléculaire :463.79Fluoxetine hydrochloride
CAS :Fluoxetine HCl (Lilly110140), a selective serotonin reuptake inhibitor (SSRI), is an antidepressant with fewer side effects.Formule :C17H19ClF3NODegré de pureté :99.6% - 99.98%Couleur et forme :White To Off-White Crystalline Solid White To Off-White PowderMasse moléculaire :345.787Palonosetron hydrochloride
CAS :Palonosetron hydrochloride (RS 25259) is a 5-HT3 antagonist used in the prevention and treatment of chemotherapy-induced nausea and vomiting.Formule :C19H24N2O·HClDegré de pureté :99.84% - 99.92%Couleur et forme :White SolidMasse moléculaire :332.87Desipramine hydrochloride
CAS :Desipramine hydrochloride (Norimipramine) ,a secondary amine tricyclic antidepressant (TCA), is the hydrochloride salt form of desipramine.Formule :C18H23ClN2Degré de pureté :99.58% - 99.96%Couleur et forme :White To Off-White PowderMasse moléculaire :302.84Carbetapentane citrate
CAS :Carbetapentane citrate (Pentoxyverine citrate) , an antitussive (cough suppressant), is frequently used for a cough related to illnesses like the common cold.Formule :C20H31NO3·C6H8O7Degré de pureté :99.46%Couleur et forme :White To Off-White SolidMasse moléculaire :525.59Dimenhydrinate
CAS :Dimenhydrinate (Vomex A) is an ethanolamine and histamine antagonist with anti-allergic activity.Formule :C24H28ClN5O3Degré de pureté :99.57% - 99.77%Couleur et forme :Crystals Physical Description Crystalline White Powder (Ntp 1992)Masse moléculaire :469.96Anatibant 2HCl
CAS :Anatibant 2HCl is a small molecule bradykinin B2 receptor antagonist for the treatment of neurological disorders and may be used in the study of brain injury.
Formule :C34H36Cl2N6O5S·2ClHDegré de pureté :99.17% - 99.58%Couleur et forme :SoildMasse moléculaire :784.58Promethazine hydrochloride
CAS :Promethazine HCl: First-gen antihistamine, H1 and mACh blocker, affects 5-HT2A/C, D2, α1 receptors.Formule :C17H20N2S·HClDegré de pureté :99.85%Couleur et forme :Crystals In Water Has A Ph Of 3 5-5 0 (Ntp 1992)Masse moléculaire :320.88YT 146
CAS :YT 146 is a biochemical.Formule :C18H25N5O4Degré de pureté :98.81% - 99.25%Couleur et forme :SolidMasse moléculaire :375.42GR 103691
CAS :GR 103691 is a potent, selective dopamine D3 receptor antagonist (Ki: 0.4 nM).Formule :C30H35N3O3Degré de pureté :98.94% - 99.29%Couleur et forme :SolidMasse moléculaire :485.62Ref: TM-T11463
2mg39,00€5mg58,00€10mg92,00€25mg177,00€50mg289,00€100mg462,00€200mg655,00€1mL*10mM (DMSO)63,00€Evocalcet
CAS :Evocalcet (KHK7580) has an activating effect on the calcium-sensing receptor (CaSR).Formule :C24H26N2O2Degré de pureté :98.88% - 99.68%Couleur et forme :SolidMasse moléculaire :374.48Abarelix
CAS :Abarelix (PPI 149) is a potent gonadotrophin-releasing hormone (GnRH) antagonist, which is used for prostate cancer treatment.Formule :C72H95ClN14O14Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :1416.06Atomoxetine hydrochloride
CAS :Atomoxetine HCl (LY 139603) is a selective non-stimulant ADHD drug that blocks norepinephrine reuptake, enhancing focus and reducing impulsivity.Formule :C17H22ClNODegré de pureté :99.86%Couleur et forme :White SolidMasse moléculaire :291.82p-MPPI hydrochloride
CAS :p-MPPI hydrochloride is a selective antagonist of 5-HT1A receptor, and has antidepressant and anxiolytic-like effects.Formule :C25H28ClIN4O2Degré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :578.87Ref: TM-T16421
2mg38,00€5mg56,00€10mg88,00€25mg138,00€50mg222,00€100mg351,00€200mg522,00€1mL*10mM (DMSO)94,00€Moxonidine
CAS :Moxonidine (BDF5895) is a selective agonist at the imidazoline receptor subtype 1, acting as an antihypertensive drug.Formule :C9H12ClN5ODegré de pureté :99.81% - 99.94%Couleur et forme :CrystalMasse moléculaire :241.68UCM-1306
CAS :UCM-1306: an oral dopamine D1 receptor PAM; boosts DA efficacy, may enhance motor and cognitive function in PD.Formule :C14H14FNO2SDegré de pureté :99.98%Couleur et forme :SoildMasse moléculaire :279.33Imidazolidinyl urea
CAS :Imidazolidinyl urea (Imidurea) is an antimicrobial preservative used in cosmetics.Formule :C11H16N8O8Degré de pureté :98.6%Couleur et forme :White Fluid Powder With Slight Characteristic OdorMasse moléculaire :388.29Avexitide acetate
CAS :Avexitide acetate (exendin 9-39) is a potent glucagon-like peptide 1 receptor (GLP-1R) antagonist for the study of post-obesity hypoglycemia.Formule :C155H246N40O53SDegré de pureté :96.64% - 98.65%Couleur et forme :SolidMasse moléculaire :3549.91Aripiprazole Lauroxil
CAS :Aripiprazole lauroxil, the N-acyloxymethyl prodrug form of aripiprazole, a long-acting injectable (LAI) antipsychotic.Formule :C36H51Cl2N3O4Degré de pureté :99.64%Couleur et forme :SolidMasse moléculaire :660.71Ref: TM-T14319
10mg48,00€25mg72,00€50mg96,00€100mg130,00€200mg188,00€500mg318,00€1mL*10mM (DMSO)49,00€Prostaglandin E1
CAS :Alprostadil (PGE1) is a natural vasodilator that also inhibits platelets and induces bronchodilation, used in erectile dysfunction treatment.Formule :C20H34O5Degré de pureté :99.78% - >99.99%Couleur et forme :SolidMasse moléculaire :354.48Ref: TM-T1626
1mg34,00€5mg63,00€10mg94,00€25mg167,00€50mg276,00€100mg415,00€200mg595,00€1mL*10mM (DMSO)50,00€Mirabegron
CAS :Mirabegron (YM178) is a beta-3 adrenergic agonist that is used for treatment of overactive bladder syndrome.Formule :C21H24N4O2SDegré de pureté :99.64%Couleur et forme :Light Yellow To Yellow SolidMasse moléculaire :396.51Ciproquazone
CAS :Ciproquazone has analgesic activity and is used to treat spondylitis.Formule :C19H18N2O2Degré de pureté :99.66%Couleur et forme :SolidMasse moléculaire :306.36Pizotifen Malate
CAS :Pizotifen Malate (BC-105 malate), a highly selective 5-HT receptor blocking agent, is a drug based on benzocycloheptane.Formule :C19H21NS·C4H6O5Degré de pureté :99.96% - >99.99%Couleur et forme :SolidMasse moléculaire :429.53Mebhydrolin napadisylate
CAS :Mebhydrolin napadisylate (Incidal) is an antihistamine used to relieve allergic symptoms caused by histamine release, including nasal allergies and allergicFormule :C19H20N2C10H8O6S2Degré de pureté :99.35% - 99.96%Couleur et forme :White Or Almost White CrystallineMasse moléculaire :420.52JP1302 dihydrochloride
CAS :JP1302 dihydrochloride: selective α2C-adrenoceptor antagonist; Ki=28 nM, Kb=16 nM.Formule :C24H26Cl2N4Degré de pureté :99.61%Couleur et forme :SolidMasse moléculaire :441.4Ref: TM-T11726
1mg46,00€2mg59,00€5mg96,00€10mg127,00€25mg235,00€50mg379,00€100mg562,00€500mg1.216,00€1mL*10mM (DMSO)96,00€Capeserod
CAS :Capeserod is a potential 5-HT4 receptor (5-hydroxytryptamine receptor 4) agonist for the study of digestive disorders and neurological disorders.Formule :C23H25ClN4O4Degré de pureté :98.10% - 99.94%Couleur et forme :SolidMasse moléculaire :456.92Dapoxetine hydrochloride
CAS :Dapoxetine hydrochloride (LY-210448 hydrochloride) is a selectivity short-acting serotonin reuptake inhibitor, used for the therapy of premature ejaculation.Formule :C21H23NO·HClDegré de pureté :99.70% - 99.91%Couleur et forme :White To Off-White Crystalline SolidMasse moléculaire :341.87Ref: TM-T6461
10mg34,00€25mg49,00€50mg66,00€100mg90,00€200mg144,00€500mg234,00€1500mg309,00€1mL*10mM (DMSO)62,00€Tropanserin
CAS :Tropanserin (MDL 72422) is a 5-hydroxytryptamine receptor antagonist with anxiolytic activity that is used to treat depression and cognitive impairment.Formule :C17H23NO2Degré de pureté :99.74%Couleur et forme :SolidMasse moléculaire :273.37Methoxamine hydrochloride
CAS :Methoxamine hydrochloride (Methoxamine HCl) is an alpha-1 adrenergic agonist that causes prolonged peripheral VASOCONSTRICTION.Formule :C11H18ClNO3Degré de pureté :99.84% - >99.99%Couleur et forme :Colorless Or White Plate-Like Crystals Or White Crystalline Powder SolidMasse moléculaire :247.719Brefonalol HCl
Brefonalol HCl, ADRA blocker for neurological/cardiovascular issues, treats angina, arrhythmias, hypertension.Formule :C22H29ClN2O2Degré de pureté :99.98%Couleur et forme :SolidMasse moléculaire :388.93Tenilapine
CAS :Tenilapine is a neuroleptic compound that can be used to study atypical antipsychotics.Formule :C17H16N4S2Degré de pureté :99.58% - >99.99%Couleur et forme :SoildMasse moléculaire :340.47Doxepin hydrochloride
CAS :Doxepin hydrochloride, a dibenzoxepin tricyclic, blocks monoamine reuptake and has anticholinergic and antihistaminic effects. Mechanism partly unknown.Formule :C19H22ClNODegré de pureté :99.65% - 99.91%Couleur et forme :White To Off-White PowderMasse moléculaire :315.84Azelastine hydrochloride
CAS :Azelastine hydrochloride (Astelin) is a phthalazinone derivative with antihistaminergic activity.Formule :C22H24ClN3O·HClDegré de pureté :98% - >99.99%Couleur et forme :White Crystalline PowderMasse moléculaire :418.36Loratadine
CAS :Loratadine (SCH 29851) is a second-generation histamine H1 receptor antagonist used in the treatment of allergic rhinitis and urticaria.
Formule :C22H23ClN2O2Degré de pureté :99.71% - 99.98%Couleur et forme :White PowderMasse moléculaire :382.88Flopropione
CAS :Flopropione (Phloropropiophenone), a spasmolytic or antispasmodic agent, is used as a 5-HT1A receptor antagonist.Formule :C9H10O4Degré de pureté :99.93%Couleur et forme :SolidMasse moléculaire :182.17DREADD agonist 21
CAS :DREADD agonist 21 is a potent agonist of human muscarinic acetylcholine M3 receptors (EC50=1.7 nM).Formule :C17H18N4Degré de pureté :99.94%Couleur et forme :SolidMasse moléculaire :278.35Ref: TM-T11095L
5mg44,00€10mg59,00€25mg99,00€50mg160,00€100mg230,00€200mg330,00€1mL*10mM (DMSO)37,00€Lintopride HCl
CAS :Lintopride HCl is a 5HT-4 antagonist.Formule :C14H20Cl2N4O2Degré de pureté :98.42% - 98.81%Couleur et forme :SoildMasse moléculaire :347.24Duloxetine hydrochloride
CAS :Duloxetine hydrochloride is an SNRI used for depression, anxiety, and pain in diabetes and fibromyalgia.Formule :C18H20ClNOSDegré de pureté :99.93% - >99.99%Couleur et forme :White Or White Crystalline PowderMasse moléculaire :333.88Timonacic
CAS :Timonacic (Thioproline) has been used in trials studying the treatment of HIV Infections.Formule :C4H7NO2SDegré de pureté :99.99%Couleur et forme :SolidMasse moléculaire :133.17PIT
CAS :PIT (2,2'-Pyridylisatogen tosylate) is a specific and non-competitive antagonist of the Purinergic receptor P2Y1 with an IC50 of 0.14 μM for human P2Y1.Formule :C20H16N2O5SDegré de pureté :98.63%Couleur et forme :SolidMasse moléculaire :396.42Retatrutide sodium salt
Retatrutide sodium salt is a glucagon receptor and glucagon-like peptide-1 receptor agonist for the study of type 2 diabetes mellitus.Degré de pureté :99.97%Couleur et forme :SoildBenztropine mesylate
CAS :Benztropine mesylate (Benztropine methanesulfonate) is a centrally active muscarinic antagonist that has been used in the symptomatic treatment of PARKINSON
Formule :C21H25NO·CH4SO3Degré de pureté :98.41% - 99.96%Couleur et forme :White Crystalline Powder; Odourless Or Almost OdourlessMasse moléculaire :403.53Naftidrofuryl oxalate
CAS :Naftidrofuryl oxalate treats peripheral/cerebral vascular issues, boosts cell oxidation, is spasmolytic, and may block 5HT-2 serotonin receptors.Formule :C26H35NO7Degré de pureté :97.12% - 98.38%Couleur et forme :SolidMasse moléculaire :473.56Ketotifen fumarate
CAS :Ketotifen fumarate (HC 20511 fumarate) is a cycloheptathiophene blocker of histamine H1 receptors and release of inflammatory mediators.Formule :C23H23NO5SDegré de pureté :99.25% - 99.73%Couleur et forme :SolidMasse moléculaire :425.50Heptaminol hydrochloride
CAS :Heptaminol hydrochloride (RP-2831 hydrochloride), a vasoconstrictor, is used in the therapy of hypotension, especially orthostatic hypotension.Formule :C8H20ClNODegré de pureté :98.61%Couleur et forme :White Crystalline PowderMasse moléculaire :181.712',5'-Dideoxyadenosine
CAS :2',5'-Dideoxyadenosine is a potent and non-competitive adenylyl cyclase inhibitor via binding the P-site (IC50: 3 μM).Formule :C10H13N5O2Degré de pureté :99.55%Couleur et forme :White SolidMasse moléculaire :235.24Ref: TM-T10066
1mg39,00€5mg84,00€10mg119,00€25mg210,00€50mg354,00€100mg562,00€500mg1.225,00€1mL*10mM (DMSO)92,00€DSP-4 hydrochloride
CAS :DSP-4 hydrochloride is a neurotoxin that degrades noradrenergic neurons in rats and crosses the blood-brain barrier.
Formule :C11H16BrCl2NDegré de pureté :99.9%Couleur et forme :SolidMasse moléculaire :313.06HJC0197
CAS :HJC0197 is a selective Epac antagonist; blocks cAMP-induced activation with IC50=5.9 μM for Epac2.Formule :C19H21N3OSDegré de pureté :98.05%Couleur et forme :SolidMasse moléculaire :339.45Ref: TM-T15485
2mg38,00€5mg54,00€10mg86,00€25mg135,00€50mg188,00€100mg283,00€200mg426,00€1mL*10mM (DMSO)64,00€Midodrine hydrochloride
CAS :Midodrine, metabolized to desglymidodrine, activates alpha-1 receptors, raising blood pressure without CNS effects. It's a prodrug in hydrochloride form.
Formule :C12H19ClN2O4Degré de pureté :99.79% - >99.99%Couleur et forme :Crystalline SolidMasse moléculaire :290.74Maprotiline hydrochloride
CAS :Maprotiline hydrochloride (Psymion) is a tetracyclic antidepressant akin to tricyclics with similar side effects.Formule :C20H24ClNDegré de pureté :99.68% - 99.84%Couleur et forme :White PowderMasse moléculaire :313.864Benserazide hydrochloride
CAS :Benserazide hydrochloride (Ro 4-4602) is a peripherally-acting L-amino acid decarboxylase (AAAD) or DOPA decarboxylase inhibitor.Formule :C10H15N3O5·HClDegré de pureté :98.63% - 99.74%Couleur et forme :White Crystalline SolidMasse moléculaire :293.7Traxanox
CAS :Traxanox: oral diuretic, boosts phagocytosis in mice/rats, reverses antibody production inhibition in BALB/c mice.Formule :C13H6ClN5O2Degré de pureté :98.37%Couleur et forme :SolidMasse moléculaire :299.67CE3F4
CAS :CE3F4 is a selective antagonist of exchange protein directly activated by cAMP (Epac1; IC50s of 10.7 μM and 66 μM for Epac1 and Epac2(B), respectively).Formule :C11H10Br2FNODegré de pureté :97.15% - 98.06%Couleur et forme :SolidMasse moléculaire :351.01PHM-27 (human) acetate
PHM-27 (human) acetate is the endogenous peptide product of prepro-VIP (human), an agonist of the calcitonin receptor (EC 50 = 11 nM). enhanced insulin secretion.
Formule :C137H215F3N34O42SDegré de pureté :99.20%Couleur et forme :SoildMasse moléculaire :3099.44Nepafenac
CAS :Nepafenac (AHR 9434) is an NSAID that acts as a cyclooxygenase inhibitor.Formule :C15H14N2O2Degré de pureté :98.94% - 99.43%Couleur et forme :SolidMasse moléculaire :254.28Desvenlafaxine
CAS :Desvenlafaxine, a venlafaxine metabolite, is an SNRI used as an antidepressant.Formule :C16H25NO2Degré de pureté :99.46% - 99.81%Couleur et forme :White Crystalline PowderMasse moléculaire :263.38Frovatriptan succinate hydrate
CAS :Frovatriptan treats all migraine types, nausea, vomiting, light/sound sensitivity, and prevents menstrual migraines; it targets 5-HT1B/D and 5-HT7 receptors.Formule :C18H25N3O6Degré de pureté :99.66%Couleur et forme :SolidMasse moléculaire :379.41Azacyclonol
CAS :Azacyclonol (MER 17) is a drug used to diminish hallucinations in psychotic individuals.Formule :C18H21NODegré de pureté :99.46%Couleur et forme :Solid PowderMasse moléculaire :267.37(S)-(-)-Atenolol
CAS :(S)-(-)-Atenolol has beta-adrenergic blocking effects.Formule :C14H22N2O3Degré de pureté :99.31% - 99.81%Couleur et forme :SolidMasse moléculaire :266.34Rebamipide
CAS :Rebamipide (OPC12759) is a drug enhancing gastric defense by stimulating COX2, prostaglandins, and mucus, while reducing TNF alpha and free radicals.Formule :C19H15ClN2O4Degré de pureté :99.48% - 99.61%Couleur et forme :White PowderMasse moléculaire :370.79PF-04995274
CAS :PF-04995274: potent, selective partial 5-HT4R agonist; EC50 0.26-0.47 nM; brain penetrant; may treat Alzheimer's cognitive issues.Formule :C23H32N2O6Degré de pureté :99.52%Couleur et forme :SolidMasse moléculaire :432.51Iobenguane sulfate
CAS :Iobenguane sulfate is used in radioiodinated form to diagnose and treat adrenergic tumors.Formule :C8H10IN3H2O4SDegré de pureté :99.04%Couleur et forme :SolidMasse moléculaire :324.12Ref: TM-T15588
5mg66,00€10mg96,00€25mg197,00€50mg354,00€100mg530,00€500mg1.153,00€1mL*10mM (DMSO)73,00€Naftifine hydrochloride
CAS :Naftifine HCl: synthetic antifungal; inhibits squalene epoxidase, disrupting fungal cell sterol synthesis.Formule :C21H22ClNDegré de pureté :98.75% - 99.84%Couleur et forme :SolidMasse moléculaire :323.86N6-Ethyladenosine
CAS :N6-Ethyladenosine is an adenosine derivative, acts as an agonist of Adenosine receptor(hA1AR and hA3AR with Kis of 4.9 and 4.7 nM , respectively).Formule :C12H17N5O4Degré de pureté :99.96%Couleur et forme :SolidMasse moléculaire :295.29Ornidazole
CAS :Ornidazole (Tiberal) is a nitroimidazole antiprotozoal agent used in ameba and trichomonas infections.Formule :C7H10ClN3O3Degré de pureté :99.47%Couleur et forme :Crystalline SolidMasse moléculaire :219.63Amisulpride
CAS :Amisulpride (Solian/Deniban), a dopamine antagonist antipsychotic, treats psychosis and schizophrenia in Europe/Australia, not in the US.Formule :C17H27N3O4SDegré de pureté :99.97% - 99.99%Couleur et forme :White Or Almost White Crystalline PowderMasse moléculaire :369.48Doxofylline
CAS :Doxofylline (Doxophylline) is a methylxanthine derivative with the presence of a dioxolane group in position 7.Formule :C11H14N4O4Degré de pureté :99.958% - >99.99%Couleur et forme :SolidMasse moléculaire :266.25Molindone hydrochloride
CAS :Molindone hydrochloride (EN-1733A) is an indole derivative effective in schizophrenia and other psychoses by blocking the effects of dopamine in the brain.
Formule :C16H24N2O2·HClDegré de pureté :99% - 99.99%Couleur et forme :SolidMasse moléculaire :312.84Ritodrine hydrochloride
CAS :Ritodrine hydrochloride (NSC 291565), a phenethylamine derivative, reduces uterine contractions by increasing cAMP and decreasing calcium in myometrial cells.Formule :C17H21NO3·HClDegré de pureté :99% - 99.52%Couleur et forme :SolidMasse moléculaire :323.82Phenoxybenzamine hydrochloride
CAS :Phenoxybenzamine hydrochloride: non-selective, irreversible alpha-blocker; antihypertensive, vasodilator, may cause tachycardia, potential carcinogen.Formule :C18H23Cl2NODegré de pureté :98.04% - >99.99%Couleur et forme :Antihypertensive DrugMasse moléculaire :340.3GTS-21 dihydrochloride
CAS :GTS-21 dihydrochloride (DMBX-anabaseine) is a nAChRs agonist. nAChRs are neuron receptor proteins that activated by the binding of the neurotransmitter ACh.Formule :C19H20N2O2·2HClDegré de pureté :98.54% - >99.99%Couleur et forme :SolidMasse moléculaire :381.3Ref: TM-T2663
5mg51,00€10mg85,00€25mg115,00€50mg144,00€100mg216,00€200mg325,00€500mg545,00€1mL*10mM (DMSO)57,00€Famotidine
CAS :Famotidine, a histamine H2-blocker, curbs gastric acid production, lowering volume and acidity.Formule :C8H15N7O2S3Degré de pureté :98.93% - 99.91%Couleur et forme :White To Off-White Crystalline PowderMasse moléculaire :337.45Mirtazapine
CAS :Mirtazapine is a unique tetracyclic antidepressant, may cause temporary liver enzyme elevation, and is linked to rare liver injury.Formule :C17H19N3Degré de pureté :99.98%Couleur et forme :SolidMasse moléculaire :265.35Paroxetine hydrochloride
CAS :Paroxetine hydrochloride (Paroxetine HCl) is a serotonin uptake inhibitor that is effective in the treatment of depression.Formule :C19H21ClFNO3Degré de pureté :98% - 99.99%Couleur et forme :White Crystalline PowderMasse moléculaire :365.826Evatanepag
CAS :Evatanepag (CP-533536) is a selective EP2 agonist for bone formation with 0.3 nM EC50, promoting fracture healing in rats.Formule :C25H28N2O5SDegré de pureté :97.09%Couleur et forme :SolidMasse moléculaire :468.57Ref: TM-T15259
1mg66,00€5mg152,00€10mg236,00€25mg409,00€50mg587,00€100mg802,00€1mL*10mM (DMSO)167,00€Pimethixene
CAS :Pimethixene (Calmixen) blocks 5-HT1A, 2A/B/C, H1, D2/D4.4 & muscarinic M1/M2 receptors; potent with pKis 7.54-10.44.Formule :C19H19NSDegré de pureté :97.50%Couleur et forme :SolidMasse moléculaire :293.43Ref: TM-T12489
2mg34,00€5mg50,00€10mg65,00€25mg106,00€50mg158,00€100mg226,00€200mg339,00€1mL*10mM (DMSO)52,00€Pipamperone
CAS :Pipamperone (McN-JR 3345) binds 5-HT2A closely as receptor.Formule :C21H30FN3O2Degré de pureté :99.85%Couleur et forme :White PowderMasse moléculaire :375.48Ref: TM-T12480
1mg62,00€2mg85,00€5mg119,00€10mg170,00€25mg283,00€50mg430,00€100mg622,00€1mL*10mM (DMSO)131,00€Ciliobrevin D
CAS :Ciliobrevin D is a AAA+ ATPase motor cytoplasmic dynein inhibitor.Formule :C17H8Cl3N3O2Degré de pureté :98.09%Couleur et forme :SolidMasse moléculaire :392.62Ref: TM-T14965
1mg60,00€2mg87,00€5mg133,00€10mg203,00€25mg401,00€50mg592,00€100mg827,00€1mL*10mM (DMSO)148,00€Ramelteon
CAS :Ramelteon (TAK-375) is a Melatonin Receptor Agonist. The mechanism of action of ramelteon is as a Melatonin Receptor Agonist.Formule :C16H21NO2Degré de pureté :97.21% - 99.92%Couleur et forme :Crystalline SolidMasse moléculaire :259.34Ref: TM-T1463
2mg42,00€5mg62,00€10mg84,00€25mg129,00€50mg192,00€100mg309,00€500mg485,00€1mL*10mM (DMSO)67,00€Ranitidine Hydrochloride
CAS :Ranitidine Hydrochloride (AH19065) is a competitive and reversible inhibitor of histamine H2-receptor antagonists with antacid activity.Formule :C13H23ClN4O3SDegré de pureté :99.30% - 99.49%Couleur et forme :SolidMasse moléculaire :350.86Isoxsuprine hydrochloride
CAS :Isoxsuprine hydrochloride (Isolait) is a beta-adrenergic agonist that causes direct relaxation of uterine and vascular smooth muscle.Formule :C18H24ClNO3Degré de pureté :99.38%Couleur et forme :Crystals From Water SolidMasse moléculaire :337.84Mianserin hydrochloride
CAS :Mianserin HCl (Org GB 94): a tetracyclic antidepressant; blocks alpha-adrenergic, H1, serotonin receptors; may induce drowsiness, hematological issues.Formule :C18H21ClN2Degré de pureté :99.63% - 99.82%Couleur et forme :White And Film Coated Tablet And Seem To Be White Or White-Like After Removing It'S Film CoatedMasse moléculaire :300.83Pramipexole
CAS :Pramipexole (SND 919), a dopamine agonist for Parkinson's, may cause mild, temporary enzyme spikes, not acute liver injury.Formule :C10H17N3SDegré de pureté :98% - 99.96%Couleur et forme :SolidMasse moléculaire :211.33Strontium ranelate
CAS :Strontium ranelate (S12911), a strontium (II) salt of the ranelic acid, is a medication for osteoporosis and can slow the course of osteoarthritis of the knee.Formule :C12H6N2O8S·2SrDegré de pureté :98.97%Couleur et forme :Crystalline SolidMasse moléculaire :513.49Ziprasidone hydrochloride monohydrate
CAS :Ziprasidone hydrochloride monohydrate (CP 88059) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of the antipsychoticFormule :C21H21ClN4OS·HCl·H2ODegré de pureté :98% - 99.83%Couleur et forme :Off-White PowderMasse moléculaire :467.12Lamotrigine
CAS :Lamotrigine (BW430C) is an Anti-epileptic Agent and Mood Stabilizer.Formule :C9H7Cl2N5Degré de pureté :99.76% - 99.95%Couleur et forme :White To Pale Cream-Colored Powder Crystals From Isopropanol SolidMasse moléculaire :256.09Itopride hydrochloride
CAS :Itopride hydrochloride (Ganaton) is an AChE and D2DR inhibitor.Formule :C20H27ClN2O4Degré de pureté :99.59%Couleur et forme :White Or Pale Brownish CrystalMasse moléculaire :394.9CYM50308
CAS :CYM50308 is a high affinity agonist of sphingosine-1-phosphate receptor 4 (S1P4-R) (EC50: 56 nM).Formule :C20H21F2N3O2SDegré de pureté :99.43% - 99.77%Couleur et forme :SolidMasse moléculaire :405.46Ref: TM-T15032
1mg62,00€5mg140,00€10mg202,00€25mg324,00€50mg455,00€100mg597,00€200mg842,00€500mg1.225,00€Tolazoline hydrochloride
CAS :Tolazoline hydrochloride (NSC35110 (hydrochloride)) is a non-selective competitive α-adrenergic receptor antagonist used in treatment of persistent pulmonaryFormule :C10H13ClN2Degré de pureté :99.67%Couleur et forme :Pale Yellow Crystalline SolidMasse moléculaire :196.68GANT 58
CAS :GANT 58 (NSC-75503) is a potent antagonist of Gli. Which inhibits GLI1-induced transcription (IC50: 5 μM).Formule :C24H16N4SDegré de pureté :99.53%Couleur et forme :SolidMasse moléculaire :392.48CB1 antagonist 2
CAS :CB1 antagonist 2 (AM4113) is caimabinoid 1 (CB1) antagonist which inhibits CB1 in vivo with an IC50 of 25.5 nM.Formule :C17H12Cl3N3ODegré de pureté :99.75%Couleur et forme :SolidMasse moléculaire :380.66[Leu15]-Gastrin I, human
CAS :[Leu15]-Gastrin I, human is a variant of Gastrin I, modulating the binding of cholecystokinin to mucosal membranes.Formule :C98H126N20O31Degré de pureté :98.02% - 98.84%Couleur et forme :SolidMasse moléculaire :2080.16Somatostatin acetate
Somatostatin acetate is an endogenously secreted inhibitor of cell proliferation with potential antitumor activity for the study of cancer and neurological disorders.
Degré de pureté :99.11%Couleur et forme :Odour SolidAstemizole
CAS :Astemizole (Laridal) is a long-acting antihistamine for allergies like rhinitis and asthma, with fewer anticholinergic effects.Formule :C28H31FN4ODegré de pureté :98.24% - 99.67%Couleur et forme :White Crystals SolidMasse moléculaire :458.57Terbutaline
CAS :Terbutaline is a short-acting agonist of β2-adrenergic receptor (β2-AR) . It is an active metabolite of bambuterolFormule :C12H19NO3Degré de pureté :99.12%Couleur et forme :SolidMasse moléculaire :225.3AZ084
CAS :AZ084 is a potent, selective, allosteric, and oral active CCR8 antagonist (Ki: 0.9 nM). It has the potential to treat asthma.Formule :C26H34N4O2Degré de pureté :97.12%Couleur et forme :SolidMasse moléculaire :434.57Ref: TM-T10425
1mg84,00€5mg161,00€10mg245,00€25mg406,00€50mg572,00€100mg772,00€200mg1.035,00€1mL*10mM (DMSO)172,00€Ogerin
CAS :Ogerin: GPR68 modulator, blocks mice fear recall, A2A inverse agonist/antagonist (Ki 220 nM), weak 5-HT2B antagonist (Ki 736 nM).Formule :C17H17N5ODegré de pureté :99.5% - 99.75%Couleur et forme :SolidMasse moléculaire :307.35Tipepidine hydrochloride
CAS :Tipepidine hydrochloride: reversible DA D2 receptor inhibitor, IC50 7.0 μM, with antidepressant effects.Formule :C15H18ClNS2Degré de pureté :99.97%Couleur et forme :SolidMasse moléculaire :311.89Asenapine Maleate
CAS :Asenapine Maleate (Org 5222 maleate) is a second generation (atypical) antipsychotic agent that is taken sublingually.Formule :C21H20ClNO5Degré de pureté :99.28%Couleur et forme :SolidMasse moléculaire :401.84JNJ-39758979
CAS :JNJ-39758979: selective H4 receptor antagonist, Kis 12.5/5.3/25 nM (human/mouse/monkey), blocks histamine cAMP inhibition (pA2 7.9).Formule :C11H19N5Degré de pureté :98.33% - 99.62%Couleur et forme :SolidMasse moléculaire :221.3Ref: TM-T11723L
1mg46,00€5mg92,00€10mg147,00€25mg241,00€50mg350,00€100mg515,00€200mg700,00€1mL*10mM (DMSO)100,00€Clozapine
CAS :Clozapine (HF 1854) is a tricylic dibenzodiazepine, classified as an atypical antipsychotic agent.Formule :C18H19ClN4Degré de pureté :99.91% - 99.93%Couleur et forme :Yellow Crystals From Acetone-Petroleum Ether SolidMasse moléculaire :326.82Ref: TM-T0455
1g425,00€10mg34,00€25mg49,00€50mg66,00€100mg90,00€200mg161,00€500mg286,00€1mL*10mM (DMSO)44,00€Paliperidone
CAS :Paliperidone (9-hydroxyrisperidone)(Invega) is used as an atypical antipsychotic.
Formule :C23H27FN4O3Degré de pureté :95% - 99.08%Couleur et forme :Off White To Light Orange Coloured SolidMasse moléculaire :426.48Mepyramine maleate
CAS :Mepyramine maleate is a mild hypnotic, local anesthetic, and H1 histamine antagonist for allergies and colds.Formule :C21H27N3O5Degré de pureté :99.51% - 99.7%Couleur et forme :White Crystalline PowderMasse moléculaire :401.47Carvedilol EP IMpurity E
CAS :Carvedilol EP IMpurity E (Carvedilol USP E) is used as a pharmaceutical intermediate.Formule :C9H14ClNO2Degré de pureté :99.53%Couleur et forme :White To Almost White Solid CrystallineMasse moléculaire :203.666Tolnaftate
CAS :Tolnaftate (NP-27) is a synthetic antifungal agent.Formule :C19H17NOSDegré de pureté :98.85%Couleur et forme :White PowderMasse moléculaire :307.41Isoprenaline hydrochloride
CAS :Isoprenaline hydrochloride (NCI-c55630) is a potent beta-adrenergic agonist with the peripheral vasodilator, bronchodilator, and cardiac stimulating properties.Formule :C11H18ClNO3Degré de pureté :98% - 99.65%Couleur et forme :Turn Brownish-Pink Upon Prolonged Exposure To Air (Ntp 1992)Masse moléculaire :247.719Flunarizine dihydrochloride
CAS :Flunarizine dihydrochloride: a calcium blocker also targeting calmodulin and histamine H1, used for migraine, vertigo, vascular disease, and epilepsy aid.
Formule :C26H28Cl2F2N2Degré de pureté :99.53% - 99.89%Couleur et forme :White Crystalline Powder Odorless And TastelessMasse moléculaire :477.42Vabicaserin hydrochloride
CAS :Vabicaserin hydrochloride (SCA 136) is a selective agonist of 5-hydroxytryptamine 2C (5-HT2C) receptor (EC50: 8 nM).Formule :C15H21ClN2Degré de pureté :98.32%Couleur et forme :SolidMasse moléculaire :264.79Ref: TM-T13275
1mg79,00€5mg170,00€10mg250,00€25mg403,00€50mg532,00€100mg735,00€200mg973,00€1mL*10mM (DMSO)178,00€Eletriptan hydrobromide
CAS :Eletriptan hydrobromide (Eletriptan HBr) is an orally active agonist with specific affinity for the 5-hydroxytriptamine1B/1D receptor.Formule :C22H27BrN2O2SDegré de pureté :99.69% - 99.85%Couleur et forme :Tan SolidMasse moléculaire :463.43Ref: TM-T0216
2mg37,00€5mg54,00€10mg66,00€25mg127,00€50mg205,00€100mg341,00€200mg504,00€1mL*10mM (DMSO)59,00€Glycerol phenylbutyrate
CAS :Glycerol phenylbutyrate (HPN-100) (GPB) is a new generation ammonia scavenger drug and it also is a sigma-2 (σ2) receptor ligand (pKi: 8.02).Formule :C33H38O6Degré de pureté :98.54% - 99.74%Couleur et forme :SolidMasse moléculaire :530.65NS-2028
CAS :NS-2028 is a selective sGC inhibitor, affecting both basal and NO-activated activities; used in nitric oxide research.Formule :C9H5BrN2O3Degré de pureté :99.44%Couleur et forme :A Crystalline SolidMasse moléculaire :269.05Ref: TM-T16344
1mg39,00€5mg88,00€10mg143,00€25mg250,00€50mg378,00€100mg543,00€200mg738,00€1mL*10mM (DMSO)87,00€BIBO3304 TFA
CAS :BIBO3304 TFA: Oral, selective NPY Y1 receptor blocker; IC50: 0.38 nM (human), 0.72 nM (rat).Formule :C31H36F3N7O5Degré de pureté :99.5%Couleur et forme :SolidMasse moléculaire :643.66Ref: TM-T10539
1mg63,00€5mg137,00€10mg243,00€25mg550,00€50mg757,00€100mg1.018,00€1mL*10mM (DMSO)187,00€Tropisetron hydrochloride
CAS :Tropisetron hydrochloride (Tropisetron HCl) is a selective, competitive serotonin 5-HT3 receptor antagonist, with antinauseant and antiemetic activities.
Formule :C17H21ClN2O2Degré de pureté :99.72% - 99.83%Couleur et forme :SolidMasse moléculaire :320.82REV 5901A
CAS :REV 5901A (REV 5901 HCl) is a leukotriene receptor antagonist and 5-LOX inhibitor with antimicrobial activity that attenuates the growth of colon cancer in miceFormule :C22H26ClNO2Degré de pureté :98.04%Couleur et forme :SoildMasse moléculaire :371.90Sarizotan 2HCl
CAS :Sarizotan 2HCl is an hERG channel inhibitor and 5-hydroxytryptamine 5-HT1A receptor agonist with potential antidepressant effects for the study of Parkinsonian movement disorders.Formule :C22H23Cl2FN2ODegré de pureté :98.83%Couleur et forme :SoildMasse moléculaire :421.34Degarelix acetate(214766-78-6 free base)
CAS :Degarelix acetate is a competitive and reversible antagonist of gonadotropin-releasing hormone receptor (GnRHR) .Formule :C84H107ClN18O18Degré de pureté :98.66%Couleur et forme :SolidMasse moléculaire :1692.34BF-1
CAS :BF-1 blocks 5-HT2B, may prevent migraines by hindering BW723C86/mCPP in guinea pigs.Formule :C22H25NO2SDegré de pureté :>99.99% - >99.99%Couleur et forme :SolidMasse moléculaire :367.50Delequamine
CAS :Delequamine (RS 15385-197) is a TNIK inhibitor (IC50: 8 nM).TINK-IN-1 inhibits colorectal cancer cell viability and can be used to study mental retardation.Formule :C18H26N2O3SDegré de pureté :99.39%Couleur et forme :SolidMasse moléculaire :350.48EMPA
CAS :EMPA is a selective, high-affinity and reversible antagonist of orexin OX2 receptor(human and rat OX2-HEK293 membranes with KD values of 1.1 and 1.4 nMFormule :C23H26N4O4SDegré de pureté :99.11%Couleur et forme :SolidMasse moléculaire :454.54Ref: TM-T11186
1mg49,00€2mg69,00€5mg92,00€10mg142,00€25mg250,00€50mg375,00€100mg563,00€200mg795,00€1mL*10mM (DMSO)104,00€ML-109
CAS :ML-109 is a potent agonist of thyroid stimulating hormone receptor (TSHR) (EC50 of 40 nM)
Formule :C31H29N3O5Degré de pureté :98.63%Couleur et forme :SolidMasse moléculaire :523.58Ebalzotan
CAS :NAE-086 is a high-affinity and selective 5-HT(1A) receptor ligand with a K(i) value of 4.5 nM in membranes from rat hippocampus.Formule :C19H30N2O2Degré de pureté :98.09% - 99.41%Couleur et forme :SolidMasse moléculaire :318.45Nardeterol HCl
Nardeterol HCl is a β-adrenergic receptor partial agonist used in the study of the central nervous system.CAS 번호13460-73-83-4
Formule :C20H25ClFN3O2Degré de pureté :97.72% - 98.65%Couleur et forme :SoildMasse moléculaire :393.88Ifenprodil Tartrate
CAS :Ifenprodil is a selective NMDA receptor (glutamate) antagonist.Formule :C21H27NO2C4H6O6Degré de pureté :99.02% - 99.55%Couleur et forme :SolidMasse moléculaire :400.49SBI-477
CAS :SBI-477 deactivates MondoA, inhibits TAG synthesis, and boosts glucose uptake in human muscle cells.Formule :C24H25N3O6SDegré de pureté :99.3%Couleur et forme :SolidMasse moléculaire :483.54Ref: TM-T12853
1mg153,00€5mg378,00€10mg560,00€25mg898,00€50mg1.216,00€100mg1.644,00€500mg3.287,00€1mL*10mM (DMSO)400,00€Nortriptyline hydrochloride
CAS :Nortriptyline HCl, a metabolite of amitriptyline, treats major and atypical depression, dysthymia.Formule :C19H22ClNDegré de pureté :99.85% - ≥95%Couleur et forme :SolidMasse moléculaire :299.84Orphenadrine hydrochloride
CAS :Orphenadrine hydrochloride (Mephenamin) is a muscarinic antagonist used to treat drug-induced parkinsonism and to relieve pain from muscle spasm.Formule :C18H23NO·HClDegré de pureté :99.88%Couleur et forme :Liquid About 5 5 Bitter Numbing Taste (Ntp 1992)Masse moléculaire :305.85Labetalol hydrochloride
CAS :Labetalol hydrochloride (Sch-15719W), a salicylamide derivative, is a non-cardioselective blocker of β-adrenergic receptors and α1-adrenergic receptors.Formule :C19H25ClN2O3Degré de pureté :99.54% - 99.85%Couleur et forme :SolidMasse moléculaire :364.87Vibozilimod
CAS :Vibozilimod (SCD-044) is S1P receptor-1 (S1PR1) agonist .Formule :C29H36ClN3O5Degré de pureté :99.97%Couleur et forme :SolidMasse moléculaire :542.07Sulpiride
CAS :Sulpiride (Aiglonyl) is a dopamine D2-receptor antagonist, used therapeutically as an antidepressant, antipsychotic, and as a digestive aid.Formule :C15H23N3O4SDegré de pureté :99.94%Couleur et forme :White Crystalline PowderMasse moléculaire :341.43Ozagrel
CAS :Ozagrel (Domenan) is a selective thromboxane A(2) (TXA(2)) synthetase inhibitor with IC50 of 11 nM for rabbit platelet, used for the improvement of
Formule :C13H12N2O2Degré de pureté :97.90% - 99.38%Couleur et forme :White PowderMasse moléculaire :228.25Trimipramine maleate
CAS :Trimipramine maleate, a tricyclic antidepressant, blocks serotonin and norepinephrine reuptake, boosting their levels and duration.Formule :C24H30N2O4Degré de pureté :99.47%Couleur et forme :SolidMasse moléculaire :410.51AM095 free acid
CAS :AM095 (free acid) is a potent LPA1 receptor antagonist (IC50s: 0.98 and 0.73 μM for recombinant human or mouse LPA1).Formule :C27H24N2O5Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :456.49Ref: TM-T10293
1mg34,00€5mg63,00€10mg92,00€25mg170,00€50mg268,00€100mg416,00€200mg625,00€1mL*10mM (DMSO)70,00€DF-1012 FA
DF-1012 FA is a structural analog of DF-1012, a neuropeptide inhibitor used in the study of asthma and cough.Formule :C17H22N4O3Degré de pureté :99.15% - 99.97%Couleur et forme :SolidMasse moléculaire :330.382Roluperidone
CAS :Roluperidone (CYR-101) is a novel cyclic amide derivative.Formule :C22H23FN2O2Degré de pureté :96.08% - 97.77%Couleur et forme :SolidMasse moléculaire :366.43Pheniramine maleate
CAS :Pheniramine maleate (Trimetose), an alkylamine derivative with antihistaminic and vasodilatory properties, binds to histamine H1 receptors.Formule :C16H20N2·C4H4O4Degré de pureté :99.85%Couleur et forme :Physical Description White Powder With A Faint Amine-Like Odor Melting Point 107°CMasse moléculaire :356.42Pancreatic Polypeptide, bovine
CAS :Agonist at Y4 neuropeptide Y receptors.Formule :C186H287N53O56S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :4225.78Melanostatin, frog TFA
Melanostatin, frog TFA is an α-MSH release inhibitor, a 36 amino acid peptide isolated from the frog brain.Degré de pureté :99.23%Couleur et forme :Odour SolidYM 218
CAS :YM 218 is a novel, potent, selective antagonist of nonpeptide vasopressin V1A receptor.Formule :C35H38F2N4O4Couleur et forme :SolidMasse moléculaire :616.7NPC 567 acetate
NPC 567 acetate is a bradykinin B2 antagonist and can be used in studies about the treatment of allergic airway disease.Formule :C62H91N19O15Degré de pureté :97.72%Couleur et forme :SolidMasse moléculaire :1342.5Org 13011
CAS :Org 13011 has CNS activity and induces conditioned taste aversion by mediating 5-HT 1A receptors.Formule :C18H25F3N4ODegré de pureté :98.02%Couleur et forme :SoildMasse moléculaire :370.41Ref: TM-T28258L
1mg115,00€5mg275,00€10mg394,00€25mg615,00€50mg848,00€100mg1.121,00€200mg1.510,00€1mL*10mM (DMSO)281,00€GLP-1R Antagonist 1
CAS :GLP-1R Antagonist 1 is an orally active, CNS penetrant and non-competitive glucagon-like peptide 1 receptor (GLP-1R) antagonist (IC50: 650 nM).Formule :C16H11ClF6N4O2Degré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :440.739-deoxy-9-methylene-16,16-dimethyl Prostaglandin E2
CAS :Meteneprost is a strong, long-lasting Prostaglandin E2 analog effective in ending early monkey pregnancies without causing fever or GI issues.Formule :C23H38O4Couleur et forme :SolidMasse moléculaire :378.553Khusimol
CAS :Khusimol is a vasopressin V1a receptors non-peptide ligand that acts by inhibiting the binding of vasopressin.Formule :C15H24ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :220.35Dabelotine, (R)-
CAS :Dabelotine, (R)- is the R-isomer of Dabelotine. Dabelotine is an adrenergic agonist used in the study of dementia.Formule :C15H22N2O2Couleur et forme :SolidMasse moléculaire :262.35GLI1-IN-3
GLI1-IN-3 (Compound 11a) is a triterpenoid-like compound that inhibits Hedgehog signaling in cancer cells with GLI1 overexpression. It suppresses the proliferation of non-small cell lung cancer and prostate cancer cell lines with excessive Hh signaling activation. Additionally, GLI1-IN-3 reduces the expression of GLI1 protein and its target genes associated with tumor progression and proliferation in A549 and DU-145 cancer cells.Couleur et forme :Odour SolidApelin-12 acetate
Apelin-12 acetate possesses a high affinity to orphan receptor APJ receptor.Formule :C66H107N21O16SDegré de pureté :98.82%Couleur et forme :SolidMasse moléculaire :1482.75Ref: TM-T39823L
1mg216,00€5mg304,00€10mg472,00€25mg753,00€50mg1.074,00€100mg1.444,00€1mL*10mM (DMSO)757,00€Add 4743
CAS :Add 4743 is an analog of sitoglitazone, which is also a fat-forming agent.Formule :C18H23NO4SCouleur et forme :SolidMasse moléculaire :349.44
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