GPCR/G-Protéine
Les inhibiteurs des GPCR/protéines G sont des composés qui ciblent les récepteurs couplés aux protéines G (GPCR) et les protéines G associées, qui jouent un rôle crucial dans la transmission des signaux de l'extérieur vers l'intérieur des cellules. Ces inhibiteurs sont essentiels pour étudier les voies de signalisation médiées par les GPCR, impliquées dans de nombreux processus physiologiques, y compris la perception sensorielle, la réponse immunitaire et la neurotransmission. Les inhibiteurs des GPCR sont également importants dans le développement de médicaments, car de nombreux agents thérapeutiques ciblent ces récepteurs. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de GPCR/protéines G de haute qualité pour soutenir vos recherches en pharmacologie, biologie cellulaire et domaines connexes.
Sous-catégories appartenant à la catégorie "GPCR/G-Protéine"
- récepteur 5-HT(1.025 produits)
- Récepteur d'adénosine(249 produits)
- Récepteur adrénergique(3.004 produits)
- Récepteur de la bombésine(35 produits)
- Récepteur de la bradykinine(61 produits)
- CXCR(155 produits)
- CaSR(34 produits)
- Récepteur cannabinoïde(217 produits)
- Cholécystokinine(1 produits)
- Récepteur de la dopamine(445 produits)
- Récepteur de l'endothéline(86 produits)
- Récepteur GNRH(84 produits)
- GPCR19(33 produits)
- GRK(33 produits)
- GTPase(23 produits)
- Récepteur du glucagon(192 produits)
- Hérisson/Smoothened(49 produits)
- Récepteur de l'histamine(385 produits)
- Récepteur LPA(21 produits)
- Récepteur de la mélatonine(26 produits)
- Récepteur OX(41 produits)
- Récepteur opioïde(326 produits)
- PAFR(14 produits)
- PKA(60 produits)
- Récepteur S1P(17 produits)
- SGLT(31 produits)
- Récepteur Sigma(46 produits)
Affichez 19 plus de sous-catégories
5971 produits trouvés pour "GPCR/G-Protéine"
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Ala-parafluoroPhe-Arg-Cha-Cit-Tyr-NH2
CAS :Ala-parafluoroPhe-Arg-Cha-Cit-Tyr-NH2 is a biologically active peptide functioning as a selective agonist for Protease Activated Receptor 1 (PAR-1), a subtypeFormule :C42H63FN12O8Couleur et forme :SolidMasse moléculaire :883.02HL2-m5
CAS :HL2-m5 is an inhibitor of the sonic hedgehog/patched (Shh/PTCH1) interaction, with a Kd for Shh of 170 nM. It effectively inhibits the activation of the Hedgehog signaling pathway and the transcription of Gli-controlled genes, with an IC50 of 230 nM.Formule :C70H101N15O24S3Couleur et forme :SolidMasse moléculaire :1632.83Lys-Bradykinin
CAS :Endogenous bradykinin receptor agonistFormule :C56H85N17O12Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1188.38Tirzepatide hydrochloride
Tirzepatide HCl is a dual GIP and GLP-1 receptor agonist.Formule :C225H349N48O68ClDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :4849.91Desamino(D-3-(3′-pyridyl)-Ala2,Arg8)-Vasopressin
CAS :Desamino(D-3-(3′-pyridyl)-Ala2,Arg8)-Vasopressin, a synthetic analog of vasopressin (AVP), acts as a weak agonist at the antidiuretic receptor but is a potentFormule :C45H63N15O11S2Couleur et forme :SolidMasse moléculaire :1054.21Plozalizumab
CAS :Plozalizumab (MLN-1202) is a humanized selective and potent anti-CCR2 antibody.Plozalizumab has antitumor activity.Plozalizumab is used in the study of
Degré de pureté :96.4%Couleur et forme :LiquidMasse moléculaire :146.02 kDaYM 218
CAS :YM 218 is a novel, potent, selective antagonist of nonpeptide vasopressin V1A receptor.Formule :C35H38F2N4O4Couleur et forme :SolidMasse moléculaire :616.7Oxopurpureine
CAS :Oxopurpureine, classified as an oxoaporphine compound, functions to inhibit plant pathogens.Formule :C21H19NO6Couleur et forme :SolidMasse moléculaire :381.38Olanzapine Lactam Impurity
CAS :Olanzapine lactam impurity, found in olanzapine, forms under heat or oxidative stress.Formule :C17H20N4O2Couleur et forme :SolidMasse moléculaire :312.373Melanostatin, frog TFA
Melanostatin, frog TFA is an α-MSH release inhibitor, a 36 amino acid peptide isolated from the frog brain.Degré de pureté :99.23%Couleur et forme :Odour Solid[Des-Arg10]-HOE I40 TFA
[Des-Arg10]-HOE I40 TFA is a potent antagonist of the bradykinin B1 receptor.
Formule :C53H77N15O12S·xC2HF3O2Couleur et forme :SolidSpantide I TFA
Spantide I TFA is a selective NK1 antagonist (230 nM); much less for NK2 (8150 nM); it modulates cytokines to prevent corneal perforation.Formule :C77H109F3N20O15Couleur et forme :SolidMasse moléculaire :1611.81(D-Phe6,Leu-NHEt13,des-Met14)-Bombesin (6-14)
CAS :(D-Phe6,Leu-NHEt13,des-Met14)-Bombesin (6-14), a bombesin (BBN) antagonist, holds potential for cancer research applications [1].Formule :C49H69N13O9Couleur et forme :SolidMasse moléculaire :984.15P2Y14R antagonist 3
P2Y14R antagonist 3 (compound A) is an orally active P2Y14R antagonist with an IC50 of 23.60 nM and a Kd of 7.26 μM. It mitigates lung injury in mice induced by Lipopolysaccharides (LPS) and can be utilized in the study of inflammatory diseases.Formule :C26H25N5O5Couleur et forme :SolidMasse moléculaire :487.51T-10430
T-10430 is a potent and orally active agonist of the leukotriene B4 receptor 2 (BLT2). It shows potential for use in psoriasis research.Formule :C17H22N6OCouleur et forme :SolidMasse moléculaire :326.396RVD-Hpα
CAS :N-terminally extended form of human hemopressin that acts as a selective CB1 receptor agonist.Formule :C65H105N19O17Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1424.66Peptide YY (PYY), human
CAS :PYY: a 36-amino-acid hormone, amidated, part of neuroendocrine control, acts via Neuropeptide Y receptors.Formule :C194H295N55O57Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :4309.75Bradykinin (1-3)
CAS :Bradykinin (1-3) is a fragment of Bradykinin. Bradykinin is an activates pain receptors.
Formule :C16H28N6O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :368.43Hemokinin 1, human
CAS :Endogenous P-like compound, NK1 receptor agonist; IC50: NK1-1.8 nM, NK3-370 nM, NK2-480 nM; boosts B-cell growth, antiapoptotic, lowers blood pressure in vivo.Formule :C54H84N14O14SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :1185.4M617
CAS :Galanin GAL1 agonist, Ki: GAL1 0.23 nM, GAL2 5.71 nM; boosts rat appetite, lessens inflammation pain.Formule :C112H161N29O28Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :2361.68α-MSH TFA
CAS :α-Melanocyte-stimulating hormone (α-MSH) is a 13-amino acid peptide hormone produced by post-translational processing of proopiomelanocortin (POMC) in theFormule :C79H110F3N21O21SCouleur et forme :SolidMasse moléculaire :1778.93GnRH Associated Peptide (1-24), human
CAS :GnRH Associated Peptide (GAP) (1-24), human, is the 1-24 fragment of hGAP linked to LH-RH via a 3 amino acid site.Formule :C117H190N32O43Couleur et forme :SolidMasse moléculaire :2732.95CKLF1-C27 TFA
CKLF1-C27 peptide activates ERK1/2 via CCR4, competes with CKLF1, promotes HUVEC growth, and has psoriasis research potential.Formule :C153H244F3N39O39Couleur et forme :SolidMasse moléculaire :3310.8sGnRH-A
CAS :sGnRH-A, a salmon GnRH analog, boosts growth hormone and induces ovulation for artificial insemination.Formule :C64H83N17O12Couleur et forme :SolidMasse moléculaire :1282.45Cinnamtannin A2
CAS :Cinnamtannin A2, a tetrameric procyanidin, boosts GLP-1, insulin, CRH expression, and has antioxidant, anti-diabetic, nephroprotective properties.
Formule :C60H50O24Couleur et forme :SolidMasse moléculaire :1155.02Imipramine N-oxide
CAS :Imipramine N-oxide is a tricyclic antidepressant (TCA) and imipramine analogue used to treat depression.Formule :C19H24N2ODegré de pureté :99.80%Couleur et forme :SolidMasse moléculaire :296.41Ref: TM-T74205
1mg72,00€5mg157,00€10mg241,00€25mg409,00€50mg565,00€100mg794,00€1mL*10mM (DMSO)167,00€Tezusomant
CAS :Tezusomant is an antagonist of the growth hormone receptor (growth hormone receptor). It is being investigated for potential use in conditions like acromegaly, which are caused by excessive secretion of growth hormone.Formule :C120H171N23O32SCouleur et forme :SolidMasse moléculaire :2479.84Osanetant
CAS :Osanetant produces anxiolytic- and antidepressant-like effects. Osanetant is a selective NK3 receptor antagonist. It is researched for schizophrenia.Formule :C35H41Cl2N3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :606.62RXFP3/4 agonist 1
CAS :RXFP3/4 agonist 1 is a relaxin family peptide 3/4 receptor (RXFP3/4) agonist(EC50s of 82/2 nM, respectivley).Formule :C20H22ClN5ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :383.88SphK1&2-IN-1
CAS :SphK1&2-IN-1 is a sphingosine kinase inhibitor with anti-inflammatory, antitumor and hemostatic effects.
Formule :C14H14N2O3SDegré de pureté :99.59%Couleur et forme :SolidMasse moléculaire :290.34Sar-[D-Phe8]-des-Arg9-Bradykinin
CAS :Potent bradykinin B1 agonist, EC50 = 9.02 nM, enzyme resistant, induces hypotension and angiogenesis.Formule :C47H66N12O11Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :975.11Methionyl-Lysyl-Bradykinin
CAS :Methionyl-Lysyl-Bradykinin (Met-Lys-Bradykinin), a Bradykinin analogue, is a kinin [1] [2] .Formule :C61H94N18O13SCouleur et forme :SolidMasse moléculaire :1319.581-39-Corticotropin (human)(TFA)
ACTH (1-39) human (TFA) is a melanocortin agonist that boosts adrenal CS production and affects the CNS and immune system.Formule :C207H308N56O58S·C2HF3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :4655.16MM 54
CAS :Potent apelin receptor antagonist (Ki=82 nM, IC50=93 nM), counters [Pyr1]-Apelin-13, inhibits glioblastoma growth in mice.Formule :C70H121N29O15S4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1737.15Mabuterol free base
CAS :Mabuterol: selective β2 agonist, inhibits isoprenaline, affects rat uterus and rabbit jejunum, alters intestinal propulsion.Formule :C13H18ClF3N2ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :310.74LTB4-IN-2
LTB4-IN-2 (Compound 6x) is a selective inhibitor of Leukotriene B4 (LTB4), acting by specifically targeting the 5-Lipoxygenase-activating protein (FLAP) with anFormule :C24H17N5S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :439.56Orexin A (human, rat, mouse)
CAS :Orexin A, a 33 AA neuropeptide in humans, rats, mice, influences various processes, studied in pancreatic function and as an OX1R antagonist.Formule :C152H243N47O44S4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :3561.1Somatostatin 1-28 acetate
Somatostatin 1-28 acetate circulates in human plasma.Degré de pureté :99.22%Couleur et forme :SoildSB 216641
CAS :SB 216641 is a 5-HT (1B/1D) antagonist with anxiolytic activity for the study of anxiety disorders and depression.Formule :C28H30N4O4Degré de pureté :98.09%Couleur et forme :SolidMasse moléculaire :486.56Palmitoyl tetrapeptide-20 TFA
Palmitoyl tetrapeptide-20 (PTP20) TFA is a biomimetic peptide and acts as an agonist of α-MSH. It protects follicular melanocytes by boosting catalase expression and activating melanogenesis.Formule :C38H70N6O8·xC2HF3O2GLP-1R agonist 20
GLP-1R agonist 20 (Compound I-132) is an agonist of the glucagon-like peptide-1 receptor (GLP-1 receptor), with an EC50 value of 0.0162 nM.Formule :C31H30Cl2F2N4O5Masse moléculaire :646.15613Relaxin H3 (human) TFA
Relaxin H3 (human) (TFA) is a relaxin peptide that exerts antifibrotic effects through the RXFP1 receptor.Formule :C237H374N70O69S6·xC2HF3O2palm11-PrRP31
Palm11-PrRP31 is a lipid-modified analog of the endogenous appetite-suppressing neuropeptide (PrRP). It functions as a potent dual agonist for GPR10 (EC50 = 39 pM) and NPFF-R2. By mimicking the natural activity of PrRP, palm11-PrRP31 binds to these receptors to reduce food intake. It has potential applications as an anti-obesity agent and is useful in studying neuropeptide and receptor interactions.Formule :C181H289N55O46SMasse moléculaire :4001.16865MR33317
MR33317 is an inhibitor of acetylcholinesterase with an IC50 value of 41 nM. Additionally, it acts as an agonist for brain 5-HT4 receptors.Formule :C22H28ClN3O2Masse moléculaire :401.187[D-Phe12]-Bombesin
CAS :Bombesin receptor antagonist
Formule :C74H112N22O18SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :1629.88Ivabradine-d3 hydrochloride
CAS :Ivabradine HCl: novel If blocker, IC50 2.9 μM, slows heart rate; D3 version is deuterium labeled.Formule :C27H37ClN2O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :508.07Guanylin TFA (mouse,rat)
Guanylin (mouse, rat) TFA is a peptide composed of 15 amino acids and acts as an activator of intestinal guanylate cyclase. This compound is utilized in research related to diarrhea.Formule :C60H90N16O22S4·xC2HF3O2Couleur et forme :SolidMasse moléculaire :1515.71 (free base)RAG8 peptide
RAG8 peptide is an antagonist of protease-activated receptor 4 (PAR 4), which inhibits late-stage platelet activation and reduces thrombosis without altering hemostasis or increasing bleeding risk. It is applicable in atherosclerosis research.Formule :C56H98N16O11Masse moléculaire :1170.760111-deoxy Prostaglandin E2
CAS :11-deoxy PGE2 is a synthetic PGE2 analog, a potent bronchoconstrictor, 5-30x stronger than PGF2α on human respiratory muscles.Formule :C20H32O4Couleur et forme :SolidMasse moléculaire :336.47Amisulpride hydrochloride
CAS :Amisulpride is an antagonist of 5-HT7 receptor and dopamine D2 and D3 receptors. It modulates beta 2- arresting signaling and increases neurite outgrowth.Formule :C17H28ClN3O4SCouleur et forme :SolidMasse moléculaire :405.94Cortagine
Potent CRF1 agonist, EC50 = 0.18 nM in rats. Exhibits in vivo anxiolytic and antidepressant effects; reduces mouse defensive behavior.Formule :C192H323N55O63SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :4442.06Labradimil
CAS :Labradimil, a bradykinin B2 agonist, boosts brain drug delivery and tumor survival rates.Formule :C49H75N15O12SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :1098.29β-CGRP (mouse)
β-CGRP (mouse), a calcitonin gene-related peptide, induces vasodilation and is applicable in research areas including cardiovascular, pro-inflammatory, migraine, and metabolic studies.Formule :C165H265N49O55S2Couleur et forme :SolidMasse moléculaire :3879.29L-803087 TFA
CAS :L-803087 TFA: potent sst4 agonist, Ki=0.7 nM, >280x selective vs other somatostatin receptors; boosts AMPA, heightens seizures.Formule :C27H30F5N5O5Couleur et forme :SolidMasse moléculaire :599.55Nebokitug
Nebokitug is a humanized IgG1κ antibody targeting CCL24, with HumanIgG1kappa, Isotype Control serving as its corresponding isotype control.Couleur et forme :Odour LiquidY1 receptor antagonist 1 formic
H 409-22 isomer formic, a formate salt of Y1 receptor antagonist 1, is an antagonist of the neuropeptide Y1 receptor (neuropeptide Y1 receptor). This compound effectively blocks the actions of the receptor, playing a crucial role in modulating physiological responses.Formule :C29H35N5O5Couleur et forme :SolidMasse moléculaire :533.62AR-C126313
CAS :AR-C126313 is a thiouracil derivative.
Formule :C28H23N7O3SCouleur et forme :SolidMasse moléculaire :537.5920-Carboxy-Leukotriene B4
CAS :20-COOH LTB4, a metabolite of LTB4, binds BLT1 receptor and inhibits LTB4-induced neutrophil responses.Formule :C20H30O6Couleur et forme :SolidMasse moléculaire :366.45NTRC-824
CAS :NTRC-824: NTS2 antagonist, 150x more selective than NTS1; IC50: 38 nM, Ki: 202 nM; nonpeptide, neurotensin-like.Formule :C25H26F3N3O6SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :553.55Abediterol napadisylate
CAS :Abediterol napadisylate is a novel long-acting β2-agonist in persistent asthma that is efficacy, safe, and tolerable.Formule :C60H68F4N4O14S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1209.32IRL-1038
CAS :ETB endothelin receptor antagonistFormule :C68H92N14O15S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1409.67A-286501
CAS :A-286501: Oral adenosine kinase inhibitor, IC50=0.47 nM, reduces pain via non-opioid, non-NSAID ADO receptors.Formule :C11H14BrN5O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :328.17Guanylate cyclase-IN-1
CAS :Guanylate cyclase-IN-1 (Example 46) is a specific inhibitor of guanylate cyclase, employed in research related to cardiovascular diseases.Formule :C20H17FN8OCouleur et forme :SolidMasse moléculaire :404.409AC-178335
CAS :AC-178335: SRIF antagonist, Ki=172 nM, inhibits SRIF's adenylate cyclase effects (IC50=5.1 µM), triggers GH release in rats.Formule :C49H63N13O7Couleur et forme :SolidMasse moléculaire :946.11L-779976
CAS :L-779,976 is an agonist of somatostatin receptor.Formule :C33H43N7O3Couleur et forme :SolidMasse moléculaire :585.74Avorelin
CAS :Avorelin, a luteinizing hormone releasing hormone (LH-RH) agonist, is used potentially for the treatment of prostate.Formule :C65H85N17O12Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1296.48Rubraxanthone
CAS :Rubraxanthone is a PAF inhibitor isolated from Garcinia parvifolia Miq.Formule :C24H26O6Couleur et forme :SolidMasse moléculaire :410.466Scyliorhinin II
CAS :Scyliorhinin II, a cyclic Tachykinin peptide, is a potent NK3 receptor agonist.Formule :C77H119N21O26S3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1851.09Thioperamide maleate
CAS :Thioperamide maleate (MR-12842 maleate) is an effective and selective antagonist of H3 receptor (Ki = 4.3 nM) for inhibition of [3H]histamine synthesis (Ki = 31Formule :C19H28N4O4SDegré de pureté :98.48%Couleur et forme :SolidMasse moléculaire :408.52Khusimol
CAS :Khusimol is a vasopressin V1a receptors non-peptide ligand that acts by inhibiting the binding of vasopressin.Formule :C15H24ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :220.35NF546
CAS :NF546 is a selective agonist of non-nucleotide P2Y11(pEC50 of 6.27).Formule :C47H44N6Na4O17P4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1180.74GRL093-22
GRL093-22 is an effective and selective inhibitor of G protein-coupled receptor kinases (GRK), with IC50 values of 60 nM for GRK5 and 40 nM for GRK6. It shows potential for research in heart failure and multiple myeloma.Formule :C33H29FN6O3Couleur et forme :SolidMasse moléculaire :576.62[cPP1-7,NPY19-23,Ala31,Aib32,Gln34]-hPancreatic Polypeptide
CAS :Potent, selective NPY Y5 receptor agonist; IC50: 0.24 nM (Y5), >500 nM (Y2), 530 nM (Y1), 51 nM (Y4); Ki: 0.1-0.15 nM (Y5); increases food intake in vivo.Formule :C183H281N57O54S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :4207.67O-2172
CAS :O-2172 is a carbocyclic analogue serving as an inhibitor of dopamine transporter (DAT), exhibiting IC50 values of 47 nM for DAT and 7000 nM for the serotonin transporter (SERT).Formule :C14H16Cl2O2Couleur et forme :SolidMasse moléculaire :287.18TGR5 agonist 7
TGR5 agonist 7 (Compound 22-Na) is an intestine-restricted, orally active agonist of the G protein-coupled bile acid receptor TGR5 (GPBAR1 or GPR131) with an EC50 of less than 1 μM. In mouse models, it demonstrates blood glucose-lowering effects, making it useful for diabetes research.Formule :C37H59N2NaO9SCouleur et forme :SolidMasse moléculaire :730.93Desmethyl Mirtazapine (hydrochloride)
CAS :Desmethyl mirtazapine is a metabolite of the antidepressant mirtazapine.1It is formed from mirtazapine by the cytochrome P450 (CYP) isoform CYP3A4.Formule :C16H18ClN3Couleur et forme :SolidMasse moléculaire :287.79PACAP (1-38), human, ovine, rat TFA
PACAP (1-38), neuropeptide from bovine brain, surpasses VIP in adenylate cyclase activation (EC50=7 nM), alters peptide release, affects gastrin and motility.Formule :C203H331N63O53S·C2HF3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :4648.28(d(CH2)51,Tyr(Me)2,Arg8)-Vasopressin
CAS :V1A receptor antagonist; blocks vasopressin & oxytocin, lowers Ca²⁺ levels (IC50: 5/30 nM); long-acting antivasopressor; anxiolytic in dorsal hippocampus.Formule :C52H74N14O12S2Degré de pureté :98%Couleur et forme :White Lyophilized PowderMasse moléculaire :1151.38S1PR1 modulator 1
CAS :S1PR1 modulator 1 is a selective inhibitor of S1PR1 with a pIC50 of 7.6.Formule :C23H24N2O3SDegré de pureté :99.69%Couleur et forme :SolidMasse moléculaire :408.51Apigenin 6,8-di-C-α-L-arabinopyranoside
CAS :Apigenin 6,8-di-C-alpha-L-arabinopyranoside is a useful organic compound for research related to life sciences.Formule :C25H26O13Couleur et forme :SolidMasse moléculaire :534.47Biotinyl-neuropeptide W-23 (human)
CAS :Biotinyl-neuropeptide W-23 (human) is a biotinylated form of neuropeptide W-23 (human), which functions as an agonist for the NPBW1 (GPR7) and NPBW2 (GPR8)Formule :C129H197N37O30S2Couleur et forme :SolidMasse moléculaire :2810.3Donetidine
CAS :Donetidine is a histamine H2 receptor antagonist used to treat digestive disorders.Formule :C20H25N5O3SDegré de pureté :99.32%Couleur et forme :SolidMasse moléculaire :415.51CAY10734
CAS :CAY10734 has a wide range of applications in life science related research.Formule :C23H25N3O3Couleur et forme :SolidMasse moléculaire :391.471Cholecystokinin (27-32)-amide
CAS :Cholecystokinin (27-32)-amide is a CCK receptor antagonist.Formule :C36H48N8O12S3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :881.01INCB3344 R-isomer
INCB3344 is a potent CCR2 antagonist. INCB3344 R-isomer is the R-isomer of INCB3344.Formule :C29H34F3N3O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :577.59Tafluprost ethyl amide
CAS :Tafluprost ethyl amide is a prostaglandin derivative.Formule :C24H33F2NO4Couleur et forme :SolidMasse moléculaire :437.52HCGRP-(8-37)
CAS :Rat CGRP-(8-37) (VTHRLAGLLSRSGGVVKDNFVPTNVGSEAF) is a highly selective CGRP receptor antagonistFormule :C139H230N44O38Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :3125.596α-Prostaglandin I1
CAS :6α-Prostaglandin I1 (6α-PGI1) is a stable Prostaglandin I2 (PGI2) analog resistant to hydrolysis in aqueous solutions.Formule :C20H34O5Couleur et forme :SolidMasse moléculaire :354.48717-phenyl trinor Prostaglandin F2α cyclopropyl amide
CAS :17-phenyl trinor Prostaglandin F2α cyclopropyl amide (17-phenyl trinor PGF2α cyclopropyl amide) is a novel analog of 17-phenyl trinor PGF2α ethyl amide.Formule :C26H37NO4Couleur et forme :SolidMasse moléculaire :427.585Nesiritide
CAS :Nesiritide, recombinant human B-type natriuretic peptide, binds NPR-A/C with Kd 7.3/13 pM.Formule :C143H244N50O42S4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :3464.04Ularitide
CAS :Ularitide is a 32-amino acid peptide from ANP prohormone, resistant to dog kidney cortex peptidase.Formule :C145H234N52O44S3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :3505.97Lipoxin B4 methyl ester
CAS :Lipoxin B4 methyl ester is a lipid-soluble prodrug of LXB4, inhibiting PMN migration/adhesion by LTB4 with IC50 of 0.3 nM.Formule :C21H34O5Couleur et forme :SolidMasse moléculaire :366.498Physalaemin
CAS :Physalaemin is a non-mammalian tachykinin.Formule :C58H84N14O16SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :1265.45GR 82334
CAS :Tachykinin NK1 receptor antagonist.Formule :C69H91N15O16Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1386.57Cagrilintide acetate
.Cagrilintide is a long-acting amylin analog,treat diabetes and obesity by reducing appetite through activation of the AMY3R and calcitonin receptor.Formule :C196H316N54O61S2Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :4469.06SRI-37330
CAS :SRI-37330 inhibits glucagon secretion and function, reduces hepatic glucose production, and reverses hepatic steatosis.
Formule :C16H19F3N4O2SDegré de pureté :99.65%Couleur et forme :SolidMasse moléculaire :388.41Amylin (IAPP), feline
Amylin (IAPP), feline is the peptide subunit of amyloid found in pancreatic islets of type 2 diabetic patients and in insulinomas.Formule :C165H270N52O54S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :3910.4517-phenyl trinor Prostaglandin F2α cyclopropyl methyl amide
CAS :Prostaglandin F2α (PGF2α) activates the FP receptor, promoting smooth muscle contraction and luteolysis.Formule :C27H39NO4Couleur et forme :SolidMasse moléculaire :441.612Flunarizine
CAS :Flunarizine is an orally administered peripheral vasodilator, a dual blocker of voltage-gated Na+/Ca2+ channels and a D2 dopamine receptor antagonist.Formule :C26H26F2N2Degré de pureté :99.9%Couleur et forme :SolidMasse moléculaire :404.505-HT7R antagonist 1 free base
CAS :5-HT7R antagonist 1 (free base) is a G protein-biased antagonist for the 5-HT 7 R receptor, with a dissociation constant (K i) of 6.5 nM.Formule :C14H17ClN4Couleur et forme :SolidMasse moléculaire :276.77Nebentan
CAS :Nebentan (YM598) is an oral, selective ETA antagonist; Ki: 0.697 nM (ETA), 569 nM (ETB); may slow cor pulmonale, myocardial infarction.
Formule :C24H21N5O5SCouleur et forme :SolidMasse moléculaire :491.52Levitide
CAS :Levitide is a neurohormone-like peptide which is from the skin of Xenopus laevis.Formule :C66H119N21O19SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :1542.85NF157
CAS :NF157, a selective P2Y11 antagonist with pKi 7.35, lowers MMP-3/MMP-13, aiding OA treatment; IC50s: P2Y11 463 nM, P2Y1 1811 μM, P2Y2 170 μM.Formule :C49H28F2N6Na6O23S6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1437.1ACTH (34-39)
CAS :ACTH (34-39) is an adrenocorticotropic hormone fragment.Formule :C37H50N6O9Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :722.83Plecanatide acetate
CAS :Plecanatide acetate: GC-C receptor agonist, EC50=190 nM (T84 cells), anti-inflammatory in murine colitis.Formule :C67H108N18O28S4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1741.94Petrelintide acetate
Petrelintide (ZP8396) acetate is an amylin analog with potential for weight reduction, suitable for diabetes research.Formule :C185H305N49O61·xC2H4O2Couleur et forme :SolidMasse moléculaire :4191.69 (free base)Nemifitide diTFA
CAS :Nemifitide diTFA is a synthetic pentapeptide with antidepressant properties, resembling MIF, that crosses the blood-brain barrier.Formule :C37H45F7N10O10Degré de pureté :99.78% - 99.84%Couleur et forme :SolidMasse moléculaire :922.8[Gln8]-C517 (LH-RH), chicken
CAS :[Gln8] LH-RH: Avian hypothalamic peptide; prompts anterior pituitary to release gonadotropins, controlling reproduction.Formule :C54H71N15O14Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1154.23Meluadrine tartrate
CAS :Meluadrine tartrate is an endogenous metabolite.Formule :C16H24ClNO8Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :393.8216-phenoxy tetranor Prostaglandin F2α methyl ester
CAS :Prostaglandin F2α (PGF2α) drives luteolysis and smooth muscle contraction by activating the FP receptor.Formule :C23H32O6Couleur et forme :SolidMasse moléculaire :404.503Enuvaptan
CAS :Enuvaptan is a vasopressin receptor antagonist and has the potential for research into renal and cardiovascular diseases.Formule :C21H15ClF6N8O3Couleur et forme :SolidMasse moléculaire :576.84HAEGT
CAS :HAEGT is the first N-terminal 1-5 residues of GLP-1 peptide.
Formule :C20H31N7O9Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :513.5Neurokinin A(4-10) TFA
Neurokinin A (4-10) TFA is a tachykinin NK 2 receptor agonist [1] .Formule :C36H55F3N8O12SCouleur et forme :SolidMasse moléculaire :880.93Zevaquenabant
CAS :Zevaquenabant (S-MRI-1867): oral CB1/iNOS antagonist combatting obesity-induced CKD.Formule :C25H21ClF3N5O2SCouleur et forme :SolidMasse moléculaire :547.98(Ala13)-Apelin-13 TFA
'(Ala13)-Apelin-13 TFA acts as a potent antagonist of the apelin receptors (APJ) and impedes gastric motility via the vagal cholinergic pathway [1].'Formule :C63H107N23O16S·xC2HF3O2Couleur et forme :SolidMasse moléculaire :1474.73 (free acid)TGR5 agonist 1
Compound 18 (TGR5 agonist 1) is a potent agonist of TGR5, exhibiting an EC50 value of 0.31 µM [1].Formule :C28H48NNaO6SCouleur et forme :SolidMasse moléculaire :549.74Prepro VIP (81-122), human
CAS :Prepro VIP (81-122), human is a prepro-vasoactive intestinal polypeptide (VIP) derived peptide, corresponding to residues 81-122.Formule :C202H325N53O64SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :4552.13PG 931 acetate
PG 931 acetate is a potent agonist of melanocortin 4 (MC4) receptors.
Formule :C61H89N15O13Degré de pureté :98.74%Couleur et forme :SolidMasse moléculaire :1240.45Eletriptan
CAS :Eletriptan, second-generation triptans used to treat migraines, is used as an abortion drug.Formule :C22H26N2O2SCouleur et forme :SolidMasse moléculaire :382.52Amylin (1-37), human acetate
Amylin (1-37), human acetate, a peptide hormone containing 37 amino acids secreted by the pancreas in conjunction with insulin, inhibits glucagon secretion.Degré de pureté :96.21%Couleur et forme :Odour SolidPF-4348235 HCl
PF-4348235 HCl (β2AR/M-receptor agonist-2 HCl) is a muscarinic M3 receptor antagonist (Ki: 0.73 nM) and β2 adrenergic receptor agonist (MABA, EC50: 3.7 nM). PF-4348235 HCl is also a bronchial BM213 acetate is a bronchodilator used to study cardiovascular and respiratory diseases such as chronic obstructive pulmonary disease (COPD).
Formule :C36H50Cl2N4O7SDegré de pureté :98.81%Couleur et forme :SolidMasse moléculaire :753.786β-Prostaglandin I1
CAS :6β-PGI1 is a stable PGI2 analog resistant to hydrolysis in aqueous solutions.Formule :C20H34O5Couleur et forme :SolidMasse moléculaire :354.487SR-31747 free base
CAS :SR-31747: immunosuppressive anti-inflammatory agent, inhibits cell growth by blocking sterol isomerase.Formule :C23H34ClNCouleur et forme :SolidMasse moléculaire :359.98meta-Fluoxetine (hydrochloride)
CAS :meta-Fluoxetine (hydrochloride) can be used in related research in the field of life sciences. Its product number is T37474 and CAS number is 79088-29-2.Formule :C17H19ClF3NOCouleur et forme :SolidMasse moléculaire :345.79Sauvagine
CAS :CRF receptor agonist; Ki: 9.4 nM (hCRF-R1), 9.9 nM (rCRF-R2a), 3.8 nM (mCRF-R2b) for 125I-[D-Tyr1]astressin binding inhibition.Formule :C202H346N56O63SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :4599.35SLP7111228
CAS :SLP7111228 is an effective and selective SphK1 inhibitor (Ki = 48 nM).Formule :C22H33N5OCouleur et forme :SolidMasse moléculaire :383.53ALD1910
ALD1910 is a humanized monoclonal antibody targeting PACAP38 and PACAP27. It inhibits PACAP signaling through pituitary adenylate cyclase-activating peptide type I receptor (PAC1-R), vasoactive intestinal peptide receptor 1 (VPAC1-R), and VPAC2-R. ALD1910 recognizes a non-linear epitope within PACAP and prevents its binding to cell surfaces. It is useful for studying PACAP-mediated migraines.Couleur et forme :Odour LiquidNR2E3 agonist 1
CAS :NR2E3 agonist 1 is an NR2E3 agonist with antitumor activity and can be used to study diseases caused by NR2E3 abnormalities.Formule :C24H19ClN4O2Degré de pureté :98.88%Couleur et forme :SoildMasse moléculaire :430.89tcY-NH2
CAS :Selective PAR4 antagonist peptide. Inhibits endostatin release and platelet aggregation induced by thrombin.Formule :C40H49N7O7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :739.87tetranor-PGDM
CAS :PGD2, made by H-PGDS in mast cells and lipocalin-PGD-synthase in the brain, aids sleep, cools the body, and inhibits platelet aggregation.Formule :C16H24O7Couleur et forme :SolidMasse moléculaire :328.361AM-0466
CAS :AM-0466 has a wide range of applications in life science related research.Formule :C27H19F3N4O4SCouleur et forme :SolidMasse moléculaire :552.52Filimelnotide
CAS :Filimelnotide is an agonist of the melanocortin receptor.Formule :C47H69N15O9S2Couleur et forme :SolidMasse moléculaire :1052.28GLP-1 receptor agonist 4
CAS :GLP-1 receptor agonist 4 targets GLP-1R, EC50 64.5 nM, potential diabetes treatment research.Formule :C51H44Cl2N4O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :879.82Linzagolix choline
CAS :Linzagolix choline is a GnRH antagonist. It can be used to study pain associated with uterine fibroids and endometriosis.Formule :C27H28F3N3O8SDegré de pureté :99.64%Couleur et forme :SolidMasse moléculaire :611.59Tirzepatide TFA
Tirzepatide TFA, a GIP and GLP-1 agonist, targets type 2 diabetes treatment.Formule :C227H349F3N48O70Couleur et forme :SolidMasse moléculaire :4927.47AP 811
CAS :AP 811: Selective NPR3 antagonist, Ki of 0.48 nM, >20,000x selective over NPR1, blocks ANP-induced pump stimulation.Formule :C46H66N12O8Couleur et forme :SolidMasse moléculaire :915.11SRA880 free base
CAS :SRA880: sst1-receptor antagonist, low affinity for other somatostatin receptors, binds to dopamine D4, may enhance antidepressant effects.Formule :C26H32N4O4Couleur et forme :SolidMasse moléculaire :464.56ANXA3 degrader 1
ANXA3 degrader 1 (Compound 18a5) is a highly selective ANXA3 degrader with activity against cancer cells. It demonstrates significant inhibitory effects in a triple-negative breast cancer (TNBC) tumor xenograft model, with a tumor growth inhibition (TGI) rate of 96%.Formule :C30H32N6O2S2Couleur et forme :SolidMasse moléculaire :572.74Moxilubant HCl
CAS :Moxilubant HCl: small molecule LTB4R antagonist for immune, skin, musculoskeletal disorders, and research in psoriasis, arthritis.Formule :C26H38ClN3O4Degré de pureté :99.94%Couleur et forme :SoildMasse moléculaire :492.05OXA(17-33) TFA
OXA(17-33) TFA: Potent OX1 agonist, ~23x more selective for OX1 (EC50=8.29nM) than OX2 (187nM).Formule :C81H126F3N23O24Couleur et forme :SolidMasse moléculaire :1863des-Gln14-Ghrelin TFA
Des-Gln14-Ghrelin TFA, a ligand for GHSR, boosts [Ca2+]i with an EC50 of 2.4 nM in CHO-GHSR62 cells.Formule :C144H238F3N43O42Couleur et forme :SolidMasse moléculaire :3300.69BMS-753426
CAS :BMS-753426 is a potent and orally bioavailable antagonist of CCR2 .
Formule :C25H33F3N6O2Couleur et forme :SolidMasse moléculaire :506.574Peptide YY (pig)
CAS :Peptide YY (pig), a 36 amino acid gut peptide from porcine duodenum, reduces appetite via Y2 receptor, affecting digestion and the heart.Formule :C190H288N54O57Couleur et forme :SolidMasse moléculaire :4240.72Thrombin Receptor Activator for Peptide 5 (TRAP-5)
CAS :Thrombin Receptor Activator for Peptide 5 (TRAP-5) is also called Coagulation Factor II Receptor (1-5), used in the research of coronary heart disease (CHD).Formule :C30H50N8O7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :634.77DD202-114
CAS :DD202-114 is an effective and selective agonist of GLP1R. It promotes the accumulation of cAMP, reduces blood glucose levels, and decreases food intake. Additionally, DD202-114 holds potential for research in type 2 diabetes mellitus (T2DM) and obesity studies.Formule :C33H35FN4O5Couleur et forme :SolidMasse moléculaire :586.65Contulakin G
CAS :Contulakin G: O-glycosylated neurotensin, weak neurotensin receptor agonist, strong antinociceptive.Formule :C88H140N20O37Masse moléculaire :2070.17d[Cha4]-AVP TFA
d[Cha4]-AVP TFA: potent, selective V1b agonist, K i 1.2 nM, favors V1b over V1a, V2, oxytocin receptors.Formule :C52H72F3N13O13S2Couleur et forme :SolidMasse moléculaire :1208.33JKC363
CAS :MC4 receptor antagonist; IC50: 0.5 nM (MC4), 44.9 nM (MC3). Blocks α-MSH, reduces TRH, food intake, and pain.
Formule :C69H91N19O16S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1506.72(Pro34)-Peptide YY (human)
CAS :(Pro34)-Peptide YY (human) is a highly Y 1 -selective full agonist of Peptide YY /neuropeptide Y receptors [1] .Formule :C194H294N54O56Couleur et forme :SolidMasse moléculaire :4278.73Kisspeptin-10, human TFA
"Kisspeptin-10, human TFA: vasoconstrictor, angiogenesis inhibitor, metastasis suppressor via GPR54, key in kidney development & osteoblast differentiation."Formule :C63H83N17O14·C2HF3O2Couleur et forme :SolidMasse moléculaire :1416.46Ethylpropyltryptamine
CAS :Ethylpropyltryptamine (EPT) is an orally active novel psychoactive substance. It is predicted to act as a partial agonist of the 5-HT2A receptor.Formule :C15H22N2Couleur et forme :SolidMasse moléculaire :230.35LGnRH-III, lamprey
CAS :GnRH III triggers luteinizing and follicle-stimulating hormone release, part of the conserved GnRH family.Formule :C59H74N18O14Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1259.33Endothelin 1 (swine, human), Alexa Fluor 488-labeled
Synthetic human/swine Endothelin 1 peptide, tagged with Alexa Fluor 488, acts as a strong vasoconstrictor via ET A/B receptors.Couleur et forme :SolidMasse moléculaire :2848.4Veldoreotide
CAS :Veldoreotide (Somatoprim): a somatostatin analogue targeting receptors 2, 4, 5, reduces GH in pituitary adenomas.Formule :C60H74N12O10Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1123.3OXA(17-33)
CAS :Potent and selective peptide orexin OX1 receptor agonist (EC50 values are 8.29 and 187 nM for OX1 and OX2 receptors respectively). Truncated form of orexin A.Formule :C79H125N23O22Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1749a-Helical Corticotropin Releasing Factor (12-41)
CAS :α-Helical CRF (12-41), a 30-aa analog, curbs CRF's ACTH-stimulating effect.Formule :C152H251N43O47S2Couleur et forme :SolidMasse moléculaire :3497.01Blue FPG-A trisodium
CAS :Blue FPG-A trisodium is a P2X1 & P2Y1 receptor antagonist, IC50: 35.5 μM & 2.6 μM, related to RB2.Formule :C29H17ClN7Na3O11S3Couleur et forme :SolidMasse moléculaire :840.1Bay 55-9837 TFA
Bay 55-9837 TFA is a VPAC2 agonist with a 0.65 nM Kd, potential for type 2 diabetes research.Formule :C150H240F3ClN44O44Couleur et forme :SolidMasse moléculaire :3456.22Lys-[Hyp3]-Bradykinin
CAS :Lys-[Hyp3]-Bradykinin, a human urine-derived kinin and bradykinin agonist, is used for inflammation research.Formule :C56H85N17O13Couleur et forme :SolidMasse moléculaire :1204.38Neuropeptide W-23 (human) (TFA)
Neuropeptide W-23 (human) (NPW-23) TFA, representing the active form of Neuropeptide W, functions as an endogenous agonist for both NPBW1 (GPR7) and NPBW2 (GPR8Couleur et forme :Odour SolidVIP(6-28)(human, rat, porcine, bovine)
CAS :VIP(6-28) blocks VIP-induced cAMP signaling in humans, rats, pigs, and cows.Formule :C126H207N37O34SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :2816.2815(S)-Latanoprost
CAS :15(S)-Latanoprost, a latanoprost analog with inverted hydroxyl at C-15, has an IC50 of 24 nM and reduces IOP by 1 mmHg at 3 μg.Formule :C26H40O5Couleur et forme :SolidMasse moléculaire :432.59Pramlintide TFA
Pramlintide TFA, a polypeptide analogue of human amylin and an antidiabetic agent, exhibits antineoplastic properties in colorectal cancer [1].Formule :C173H268N51F3O55S2Couleur et forme :SolidMasse moléculaire :4063.4MrgprX2 antagonist-3
CAS :MrgprX2 antagonist-3 (compound E117) is a MrgprX2 antagonist applicable for investigating cutaneous inflammation.Formule :C16H20FN3O2SDegré de pureté :98.06%Couleur et forme :SolidMasse moléculaire :337.41Ref: TM-T40271
1mg57,00€5mg120,00€10mg190,00€25mg383,00€50mg604,00€100mg965,00€1mL*10mM (DMSO)134,00€Cortistatin 29
Cortistatin 29: neuropeptide, relieves neuropathic pain, binds SS receptors (IC50: 2.8-13.7 nM), anti-fibrotic.Formule :C161H242N46O41S2Couleur et forme :SolidMasse moléculaire :3539.77D[LEU4,LYS8]-VP TFA
D[LEU4,LYS8]-VP TFA: V1b receptor agonist; K_i: 0.16 nM (rat), 0.52 nM (human), 1.38 nM (mouse); weak antidiuretic/vasopressor/oxytocic.Formule :C49H68F3N11O13S2Couleur et forme :SolidMasse moléculaire :1140.25GLP-1 receptor agonist 13
Compound (S)-9, a GLP-1 receptor agonist, exhibits an EC50 of 76 nM for the glucagon GLP-1 receptor [1].Formule :C25H23ClF2N6OCouleur et forme :SolidMasse moléculaire :496.94Alsactide
CAS :Alsactide, an adrenocorticotropic hormone (ACTH) agonist and a heptadecapeptide analogue, is utilized in the study of the central nervous system [1].Formule :C99H155N29O21SCouleur et forme :SolidMasse moléculaire :2119.53Tecastemizole
CAS :Tecastemizole (R 43512) is a selective antagonist of H1 receptor and a major metabolite of astemizole with anti-inflammatory effects.Formule :C19H21FN4Degré de pureté :99.70%Couleur et forme :SolidMasse moléculaire :324.4Ref: TM-T26253
1mg54,00€5mg118,00€10mg168,00€25mg288,00€50mg414,00€100mg583,00€500mg1.161,00€1mL*10mM (DMSO)131,00€1a,1b-dihomo Prostaglandin E1
CAS :1a,1b-dihomo Prostaglandin E1 is a class of prostaglandin compounds.Formule :C22H38O5Couleur et forme :SolidMasse moléculaire :382.541JNJ-10181457 (hydrochloride)
CAS :JNJ-10181457 (hydrochloride) is a non-imidazole H3 receptor antagonist that is brain-penetrating and selective, increasing NE and acetylcholine concentrationsFormule :C20H30Cl2N2OCouleur et forme :SolidMasse moléculaire :385.37PG-931 TFA
PG-931 TFA, a potent MC4 receptor agonist (IC50 0.58 nM), excels in selectivity and helps reverse hemorrhagic shock in vivo.Formule :C61H86F3N15O13Couleur et forme :SolidMasse moléculaire :1294.42LP 12 hydrochloride
CAS :LP 12 hydrochloride is a selective 5-HT7 receptor agonist (Ki=0.13 nM).Formule :C32H40ClN3OCouleur et forme :SolidMasse moléculaire :518.14TRV045
CAS :TRV045 is a selective agonist of the sphingosine-1-phosphate (S1P) subtype 1 receptor and does not impact lymphocyte trafficking. It possesses antiepileptic properties.
Formule :C18H18N4O3Couleur et forme :SolidMasse moléculaire :338.36[Nle11]-Substance P
CAS :'[Nle11]-Substance P is a gut and brain peptide, resisting methionine oxidation and causing excitatory neural effects.'
Formule :C64H100N18O13Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1329.59GLP-1(9-36)amide TFA
GLP-1(9-36)amide TFA, a DPP-4 metabolite of GLP-1(7-36) amide, antagonizes human pancreatic GLP-1 receptor.Formule :C142H215F3N36O45Couleur et forme :SolidMasse moléculaire :3203.43AMK (hydrochloride)
CAS :AMK, a melatonin metabolite, scavenges oxygen, inhibits prostaglandin production, reduces lipid peroxidation, and affects Parkinson's in mouse studies.Formule :C12H17ClN2O3Couleur et forme :SolidMasse moléculaire :272.73TAK-683 acetate
TAK-683 acetate: potent KISS1R agonist (IC50=170 pM), stable, nonapeptide. Affects GnRH, FSH, LH, testosterone; potential in prostate cancer research.Formule :C66H87N17O15Couleur et forme :SolidMasse moléculaire :1358.58-iso-15-keto Prostaglandin F2α
CAS :8-iso-15-keto Prostaglandin F2α (8-iso-15-keto PGF2α) is a metabolite of the isoprostane 8-iso PGF2α in rabbits, monkeys, and humans.Formule :C20H32O5Couleur et forme :SolidMasse moléculaire :352.471Acetyl-Amylin (8-37) (human)
CAS :Acetyl-Amylin (8-37) (human) is a specific amylin antagonist [1] .Formule :C140H218N42O46Couleur et forme :SolidMasse moléculaire :3225.48DOTA-JR11
CAS :DOTA-JR11 is a somatostatin receptor 2 (SSTR2) antagonist that can be radiolabeled with 68Ga.Formule :C74H98ClN19O21S2Couleur et forme :SolidMasse moléculaire :1689.27SAE-14
CAS :GPR183, a chemotactic receptor aiding B cell maturation, binds 7α,25-OHC; studied in IBD research.Formule :C19H19F3N2O2Degré de pureté :99.85%Couleur et forme :SolidMasse moléculaire :364.36Neuropeptide SF(mouse,rat) TFA
Neuropeptide SF TFA is a potent agonist for NPFF1 (Ki=48.4 nM) and NPFF2 (Ki=12.1 nM) and enhances ASIC3 current.Formule :C42H66F3N13O12Couleur et forme :SolidMasse moléculaire :1002.05Human glucagon-like peptide-1-(7-36)-Lys(Biotin) amide
Biotin-labeled GLP-1-(7-36) amide; a gut peptide that enhances insulin release.Formule :C165H252N44O48SCouleur et forme :SolidMasse moléculaire :3652.1CCZ01048 TFA
CCZ01048 TFA, α-MSH analog, binds MC1R with 0.31 nM affinity, internalizes in melanoma cells, and is stable for melanoma PET imaging.Formule :C73H106F3N21O18Couleur et forme :SolidMasse moléculaire :1622.75Amylin, amide, human TFA
Amylin, a 37-amino acid human hormone, moderates glucose regulation by reducing glucagon, delaying digestion, and increasing satiety.Formule :C167H262F3N51O57S2Couleur et forme :SolidMasse moléculaire :4017.3(Phe2,Orn8)-Oxytocin acetate
(Phe2,Orn8)-Oxytocin acetate: V1 agonist with EC50 of 280 nM for rabbit epididymis contractility.Formule :C44H69N13O13S2Couleur et forme :SolidMasse moléculaire :1052.23Paynantheine
CAS :Paynantheine is an alkaloid with antinociceptive properties, found in Mitragyna speciosa. It also acts as an agonist at 5-HT1AR and 5-HT2BR receptors, inducing lower lip contraction and providing antinociception in rats.Formule :C23H28N2O4Couleur et forme :SolidMasse moléculaire :396.48M871
CAS :GAL2 receptor antagonist; Ki: 13.1 nM (GAL2), 420 nM (GAL1); inhibits GAL2-induced pain.Formule :C108H163N27O28Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :2287.64RC-3095
CAS :RC-3095, a selective GRPR antagonist, has been shown to have anti-inflammatory properties in different models of inflammation.Formule :C56H79N15O9Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1106.32CART(55-102)(rat) TFA
Rat CART(55-102) TFA suppresses appetite, links to leptin/neuropeptide Y, and may induce anxiety/stress.Formule :C228H368F3N65O67S7Couleur et forme :SolidMasse moléculaire :5373.2PAMP-12 (unmodified) (TFA)
PAMP-12 (unmodified) TFA, an endogenous peptide and potent MRGPRX2 (MrgX2) agonist (EC50=20-50 nM), induces hypotension by inhibiting catecholamine secretionFormule :C79H119F3N24O17Couleur et forme :SolidMasse moléculaire :1733.94(D-His(Bzl)6)-LHRH (1-7) (free acid)
CAS :(D-His(Bzl)6)-LHRH (1-7) free acid is a synthetic peptide derived from luteinizing hormone-releasing hormone (LHRH). It achieves enhanced stability and biological activity through the introduction of non-natural amino acid residues at specific positions within the LHRH molecule. This modification extends the drug's half-life in the body, reduces its rate of rapid metabolism and clearance, and subsequently increases its efficacy in inhibiting cell proliferation.Formule :C53H62N12O11Masse moléculaire :1043.13Acetyl-(D-Phe2,Lys15,Arg16,Leu27)-VIP (1-7)-GRF (8-27)
CAS :Acetyl-(D-Phe2,Lys15,Arg16,Leu27)-VIP(1-7)-GRF(8-27) is a selective antagonist [1] for the vasoactive intestinal peptide 1 (VIP 1) receptor.Formule :C150H246N44O38Couleur et forme :SolidMasse moléculaire :3273.83Galanin (1-30), human
CAS :Galanin (1-30), human is a neuropeptide agonist for GalR1/R2 receptors with 1 nM affinity, influencing endocrine, metabolism, and neurotransmission.Formule :C139H210N42O43Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :3157.46SR142948A
CAS :SR142948A is a selective and reversible non-peptide neurotensin receptor antagonist blocking hypothermia and analgesic effects, NMDA-induced dopamine release.Formule :C39H52ClN5O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :722.31K-(D-1-Nal)-FwLL-NH2 TFA
K-(D-1-Nal)-FwLL-NH2 TFA: potent ghrelin inverse agonist; Ki=4.9 nM (COS7), 31 nM (HEK293T); blocks Gq/G13 signaling.Formule :C53H68F3N9O8Couleur et forme :SolidMasse moléculaire :1016.16PF-07062119
PF-07062119 is a bispecific antibody targeting CD3 and GUCY2C and can be used for cancer research.Couleur et forme :Odour LiquidCRF, bovine
CAS :CRF, bovine is a potent agonist of CRF receptor, and displaces [125I-Tyr]ovine CRF with a Ki of 3.52 nM.Formule :C206H340N60O63SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :4697.34SB-206606
CAS :SB-206606 is a novel, highly specific radioactive ligand for the β3-adrenergic receptor.
Formule :C19H22ClNO4Couleur et forme :SolidMasse moléculaire :363.83
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