GPCR/G-Protéine
Les inhibiteurs des GPCR/protéines G sont des composés qui ciblent les récepteurs couplés aux protéines G (GPCR) et les protéines G associées, qui jouent un rôle crucial dans la transmission des signaux de l'extérieur vers l'intérieur des cellules. Ces inhibiteurs sont essentiels pour étudier les voies de signalisation médiées par les GPCR, impliquées dans de nombreux processus physiologiques, y compris la perception sensorielle, la réponse immunitaire et la neurotransmission. Les inhibiteurs des GPCR sont également importants dans le développement de médicaments, car de nombreux agents thérapeutiques ciblent ces récepteurs. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de GPCR/protéines G de haute qualité pour soutenir vos recherches en pharmacologie, biologie cellulaire et domaines connexes.
Sous-catégories appartenant à la catégorie "GPCR/G-Protéine"
- récepteur 5-HT(1.025 produits)
- Récepteur d'adénosine(249 produits)
- Récepteur adrénergique(3.018 produits)
- Récepteur de la bombésine(35 produits)
- Récepteur de la bradykinine(61 produits)
- CXCR(158 produits)
- CaSR(34 produits)
- Récepteur cannabinoïde(217 produits)
- Cholécystokinine(1 produits)
- Récepteur de la dopamine(445 produits)
- Récepteur de l'endothéline(86 produits)
- Récepteur GNRH(84 produits)
- GPCR19(33 produits)
- GRK(33 produits)
- GTPase(23 produits)
- Récepteur du glucagon(194 produits)
- Hérisson/Smoothened(49 produits)
- Récepteur de l'histamine(385 produits)
- Récepteur LPA(21 produits)
- Récepteur de la mélatonine(26 produits)
- Récepteur OX(41 produits)
- Récepteur opioïde(327 produits)
- PAFR(14 produits)
- PKA(60 produits)
- Récepteur S1P(18 produits)
- SGLT(31 produits)
- Récepteur Sigma(46 produits)
Affichez 19 plus de sous-catégories
5983 produits trouvés pour "GPCR/G-Protéine"
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Fluphenazine free base
CAS :Flufenazine: antipsychotic for schizophrenia, blocks dopamine D2 receptors, reduces hallucinations and delusions.Formule :C22H26F3N3OSCouleur et forme :SolidMasse moléculaire :437.52Orexin A (human, rat, mouse) acetate
Orexin A (human, rat, mouse) acetate (Hypocretin-1 (human, rat, mouse) acetate) is an excitatory neuropeptide with analgesic properties.Formule :C154H247N47O46S4Couleur et forme :SolidMasse moléculaire :3621.15Spantide I TFA
Spantide I TFA is a selective NK1 antagonist (230 nM); much less for NK2 (8150 nM); it modulates cytokines to prevent corneal perforation.Formule :C77H109F3N20O15Couleur et forme :SolidMasse moléculaire :1611.81Mosliciguat
CAS :Mosliciguat is a guanylate cyclase activator.Formule :C41H36ClF3N2O5Couleur et forme :SolidMasse moléculaire :729.19L-770644 dihydrochloride
CAS :L-770644 dihydrochloride is a potent and selective agonist of the human beta3 adrenergic receptor.Formule :C30H38ClN7O4SCouleur et forme :SolidMasse moléculaire :628.19Apelin-12 acetate
Apelin-12 acetate possesses a high affinity to orphan receptor APJ receptor.Formule :C66H107N21O16SDegré de pureté :98.82%Couleur et forme :SolidMasse moléculaire :1482.75Ref: TM-T39823L
1mg128,00€5mg172,00€10mg269,00€25mg429,00€50mg610,00€100mg820,00€1mL*10mM (DMSO)430,00€Anthramycin
CAS :Anthramycin: a PBD family antibiotic with antitumor effects and CNS cholecystokinin antagonist properties in mice.Formule :C16H17N3O4Couleur et forme :SolidMasse moléculaire :315.32APJ receptor agonist 10
CAS :APJ receptor agonist 10 (Compound I choline salt) modulates the activity of the APJ receptor, making it useful for pulmonary hypertension research. Compared to its free form, this compound exhibits improved bioavailability.Formule :C26H36N7O6SCouleur et forme :SolidMasse moléculaire :574.67L-796,778
CAS :L-796,778 is an SST3 agonist and a selective ligand of SST3, which can increase the level of cAMP in the body.Formule :C29H40N6O7Degré de pureté :99.24%Couleur et forme :SolidMasse moléculaire :584.66Ref: TM-T32511
1mg175,00€5mg404,00€10mg592,00€25mg888,00€50mg1.243,00€100mg1.701,00€500mg3.402,00€1mL*10mM (DMSO)522,00€PF-9184
CAS :PF-9184 inhibits human mPGES-1 selectively, with an IC50 of 16.5 nM, and reduces IL-1β-stimulated PGE2 production in vitro.Formule :C21H14Cl2N2O4SDegré de pureté :97.43%Couleur et forme :SolidMasse moléculaire :461.32GLP-1(7-37)
CAS :GLP-1 (7-37) is a truncated, bioactive form of GLP-1 that is the product of proglucagon processing in intestinal endocrine L cells.Formule :C151H228N40O47Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :3355.672-Furoyl-LIGRLO-amide
CAS :2-Furoyl-LIGRLO-amide TFA is a peptide that acts as a proteinase-activated receptor-2 (PAR2) agonist, and contains a furoyl group addition at its N-terminal.Formule :C36H63N11O8Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :777.95Cagrilintide acetate
.Cagrilintide is a long-acting amylin analog,treat diabetes and obesity by reducing appetite through activation of the AMY3R and calcitonin receptor.Formule :C196H316N54O61S2Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :4469.06Neurokinin B (TFA)
CAS :Neurokinin B TFA, a tachykinin, targets NK1R, NK2R, nk3r GPCRs, modulating effects.Formule :C59H81F6N13O18S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1438.47Phenoxybenzamine
CAS :Phenoxybenzamine blocks α-1 receptors, potentially reducing neuroinflammation post brain trauma.Formule :C18H22ClNODegré de pureté :98%Couleur et forme :Crystals From Petroleum Ether SolidMasse moléculaire :303.83Apigenin 6,8-di-C-α-L-arabinopyranoside
CAS :Apigenin 6,8-di-C-alpha-L-arabinopyranoside is a useful organic compound for research related to life sciences.Formule :C25H26O13Couleur et forme :SolidMasse moléculaire :534.47Alcaftadine carboxylic acid
CAS :Alcaftadine is a novel antihistamine for preventing allergic conjunctivitis.Formule :C19H21N3O2Couleur et forme :SolidMasse moléculaire :323.39Detomidine carboxylic acid
CAS :Detomidine carboxylic acid, a urine metabolite of detomidine, is a synthetic α2-agonist, animal analgesic, with cardiac, respiratory, and diuretic effects.Formule :C12H12N2O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :216.24Cortistatin 14, human, rat acetate
Cortistatin 14, human, rat acetate is a neuropeptide having structural similarity to somatostatin-14 and shows anticonvulsive, neuroprotective effects andFormule :C80H112N18O19S2Degré de pureté :97.86%Couleur et forme :SolidMasse moléculaire :1693.98MrgprX2 antagonist-2
CAS :MrgprX2 antagonist-2, from patent WO2021092262A1 E163, is potent for skin inflammation studies.Formule :C17H16F5N3O3Couleur et forme :SolidMasse moléculaire :405.325IRL-1620
CAS :IRL-1620 is an effective and selective agonist of endothelin receptor type B (ETB) (Ki: 16 pM).Formule :C86H117N17O27Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1820.974Apelin-17(human, bovine)
CAS :Endogenous apelin receptor agonist. Potently inhibits forskolin-stimulated cAMP accumulation (pIC50 = 9.94).Formule :C96H156N34O20SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :2138.56CB1R agonist 1
CB1R agonist 1 (Compound '1350) is a potent full agonist of the cannabinoid-1 receptor (CB1R) with a Ki value of 0.95 nM. It demonstrates significant pain-relieving effects in various pain models, including acute thermal pain, inflammatory pain, and neuropathic pain.Formule :C20H18F3N3O3SCouleur et forme :SolidMasse moléculaire :437.435SC 31391
CAS :SC 31391 is a PGE1 analog.Formule :C24H32O6Couleur et forme :SolidMasse moléculaire :416.515-trans Latanoprost (free acid)
CAS :Latanoprost, a prodrug eye drop, turns into active acid inside the body and treats high eye pressure. Its trans isomer also likely reduces eye pressure.Formule :C23H34O5Couleur et forme :SolidMasse moléculaire :390.52TT-OAD2 free base
CAS :TT-OAD2 free base, a non-peptide GLP-1 receptor agonist, can treat diabetes; has an EC50 of 5 nM.Formule :C50H47Cl2N3O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :856.83MRS 2365
CAS :Highly potent, selective P2Y1 receptor agonistFormule :C13H19N5O9P2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :483.33[D-Phe12]-Bombesin
CAS :Bombesin receptor antagonist
Formule :C74H112N22O18SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :1629.88APJ receptor agonist 1
CAS :Potent APJ-R agonist 1, biphenyl acid, EC50: 0.093 nM (human), 0.12 nM (rat), targets apelin-13, promising for heart failure study.Formule :C31H26ClN3O3Couleur et forme :SolidMasse moléculaire :524.02(R,R)-Palonosetron Hydrochloride
CAS :(R,R)-Palonosetron Hydrochloride is the active enantiomer of PalonosetronFormule :C19H25ClN2ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :332.875-HT2A receptor agonist-5
CAS :5-HT2A receptor agonist-5 (compound I-3) is a potent 5-HT2A agonist with a Ki value of 0.017 µM and exhibits antidepressant activity.Formule :C23H29N3OCouleur et forme :SolidMasse moléculaire :363.5PAR-4 Agonist Peptide, amide
CAS :PAR-4 Agonist Peptide, amide (AY-NH2) is an agonist of proteinase-activated receptor-4 (PAR-4).Formule :C34H48N8O7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :680.79(Ala13)-Apelin-13 TFA
'(Ala13)-Apelin-13 TFA acts as a potent antagonist of the apelin receptors (APJ) and impedes gastric motility via the vagal cholinergic pathway [1].'Formule :C63H107N23O16S·xC2HF3O2Couleur et forme :SolidMasse moléculaire :1474.73 (free acid)(d(CH2)51,Tyr(Me)2,Arg8)-Vasopressin
CAS :V1A receptor antagonist; blocks vasopressin & oxytocin, lowers Ca²⁺ levels (IC50: 5/30 nM); long-acting antivasopressor; anxiolytic in dorsal hippocampus.Formule :C52H74N14O12S2Degré de pureté :98%Couleur et forme :White Lyophilized PowderMasse moléculaire :1151.38HS014
CAS :Potent MC4 antagonist; Ki: 3.16 nM (MC4), 108 (MC1), 54.4 (MC3), 694 (MC5). Boosts rat appetite, mouse pain, blocks IL-1β Fos in hypothalamus.Formule :C71H94N20O17S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1563.77Pasireotide L-aspartate salt
CAS :Pasireotide L-aspartate, a stable cyclohexapeptide, mimics somatostatin with high affinity for sst1/2/3/4/5 receptors (pKi=8.2/9.0/9.1/<7.0/9.9).Formule :C62H73N11O13Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1180.336α-Prostaglandin I1
CAS :6α-Prostaglandin I1 (6α-PGI1) is a stable Prostaglandin I2 (PGI2) analog resistant to hydrolysis in aqueous solutions.Formule :C20H34O5Couleur et forme :SolidMasse moléculaire :354.487Xylamidine
CAS :Xylamidine is a biochemical.Formule :C19H24N2O2Couleur et forme :SolidMasse moléculaire :312.41PF-4348235 HCl
PF-4348235 HCl (β2AR/M-receptor agonist-2 HCl) is a muscarinic M3 receptor antagonist (Ki: 0.73 nM) and β2 adrenergic receptor agonist (MABA, EC50: 3.7 nM). PF-4348235 HCl is also a bronchial BM213 acetate is a bronchodilator used to study cardiovascular and respiratory diseases such as chronic obstructive pulmonary disease (COPD).
Formule :C36H50Cl2N4O7SDegré de pureté :98.81%Couleur et forme :SolidMasse moléculaire :753.785-HT1AR agonist 2
5-HT1AR Agonist 2 (Compound 4f) is a potent agonist of the 5-HT1A receptor with a Ki value of 10.0 nM. It also binds to SERT, D2, and 5-HT6 receptors with Ki values of 2.8 nM, 23 nM, and 192 nM, respectively. Furthermore, this compound demonstrates stability in microsomes and induces hypothermia in mice.Formule :C31H31N5O3Couleur et forme :SolidMasse moléculaire :521.61Calcitonin Gene Related Peptide (CGRP) II, rat TFA
Rat CGRP II TFA: potent vasodilator and CGRP receptor activator for cardiovascular research.Formule :C165H268F3N51O52S2Couleur et forme :SolidMasse moléculaire :3919.33Endothelin-3, human, mouse, rabbit, rat
CAS :Endothelin-3, human, mouse, rabbit, rat , is a cyclic 21 amino acid peptide. It is an endogenous neuropeptide and potent vasoconstrictor.Formule :C121H168N26O33S4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :2643.04Luteinizing Hormone Releasing Hormone (LH-RH), salmon
CAS :LH-RH: a hypothalamus-made pituitary hormone, key in reproductive control.Formule :C60H73N15O13Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1212.31Mitemcinal fumarate
CAS :Mitemcinal fumarate is a erythromycin derivative that is used to treat gastroesophageal reflux disease.Formule :C84H142N2O28Couleur et forme :SolidMasse moléculaire :1628.02Zoliprofen
CAS :Zoliprofen: potent, oral NSAID with anti-inflammatory, antipyretic, analgesic effects. Exceeds ibuprofen's efficacy in rats and rabbits.Formule :C12H11NO3SDegré de pureté :99.62%Couleur et forme :SolidMasse moléculaire :249.29Ref: TM-T68025
1mg85,00€5mg170,00€10mg256,00€25mg480,00€50mg655,00€100mg933,00€500mg1.872,00€1mL*10mM (DMSO)168,00€γ-Glu-Abu TFA
Gamma-Glu-AbuTFA is the TFA salt form of Gamma-Glu-Abu. This compound acts as an agonist for the calcium sensing receptor (CaSR), activating CaSR in HEK-293 cells with an EC50 of 0.21 μM.Formule :C11H17F3N2O7Couleur et forme :SolidMasse moléculaire :346.26Alosetron
CAS :Alosetron, a 5-HT3 antagonist, is used for the management of severe diarrhea-predominant irritable bowel syndrome (IBS) in women only.Formule :C17H18N4ODegré de pureté :98%Couleur et forme :Crystalline PowderMasse moléculaire :294.36tetranor-PGDM
CAS :PGD2, made by H-PGDS in mast cells and lipocalin-PGD-synthase in the brain, aids sleep, cools the body, and inhibits platelet aggregation.Formule :C16H24O7Couleur et forme :SolidMasse moléculaire :328.361PD 142893
CAS :PD 142893 is a functional endothelin-stimulated vasoconstriction antagonist.Formule :C50H65N7O10Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :924.09(Hyp³)-Bradykinin acetate
(Hyp³)-Bradykinin acetate is an agonist of bradykinin B2 receptor and stimulates inositol phosphate production in cultured human fibroblasts.Formule :C52H77N15O14Degré de pureté :99.46%Couleur et forme :SolidMasse moléculaire :1136.26G-Protein antagonist peptide
CAS :Peptide inhibits G protein-receptor binding; competitively blocks M2 and β-adrenoceptor-induced Gs/Gi/Go activation.Formule :C57H64N12O9SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :1093.271-Octadecyl Lysophosphatidic Acid
CAS :1-Octadecyl LPA, an LPA analog with stearic acid at sn-1, has strong platelet aggregation (EC50=9 nM) via G protein receptors.Formule :C21H45O6PCouleur et forme :SolidMasse moléculaire :424.559Ceruletide Ammonium Salt
Ceruletide Ammonium Salt is a decapeptide, originating from the skin of tropical frogs, which is a potent cholecystokinin receptor agonist and a safe andFormule :C58H77N14O21S2Degré de pureté :98.47% - 98.54%Couleur et forme :SoildMasse moléculaire :1370.44Ref: TM-T14932L1
1mg93,00€5mg313,00€10mg465,00€25mg742,00€50mg982,00€100mg1.333,00€500mg2.637,00€1mL*10mM (DMSO)34,00€MI 1544
CAS :MI 1544 is a LHRH antagonist.Formule :C71H94ClN17O13Couleur et forme :SolidMasse moléculaire :1429.09N6-Benzyl-5'-ethylcarboxamido adenosine
CAS :N6-Benzyl-5'-ethylcarboxamido adenosine is a selective A3 adenosine receptor agonist.Formule :C19H22N6O4Couleur et forme :SolidMasse moléculaire :398.42NPC 567
CAS :NPC 567 is an antagonist of the bradykinin receptor.Formule :C60H87N19O13Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1282.48Spantide I
CAS :Spantide antagonizes both bombesin & substance P. It is also tachykinin receptor antagonist.Formule :C75H108N20O13Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1497.79AC-263093
CAS :AC-263093 is an NPFFR2 agonist with anxiolytic activity that increases c-Fos protein expression in the paraventricular nucleus of the hypothalamus.Formule :C8H8Br2N4Degré de pureté :99.78%Couleur et forme :SoildMasse moléculaire :319.98(R)-(+)-Atenolol
CAS :(R)-(+)-Atenolol ((R)-Atenolol) is a cardioselective beta-1 adrenergic blocker, which properties are similar to propranolol, but without a negative inotropic effect.Formule :C14H22N2O3Degré de pureté :98.72%Couleur et forme :SolidMasse moléculaire :266.34Lintitript
CAS :Lintitript (SR 27897) is a selective antagonist of CCK1 with EC50s of 6 nM and 200 nM for CCK1 and CCK2. The Ki value is 0.2 nM for CCK1.Formule :C20H14ClN3O3SDegré de pureté :99.28%Couleur et forme :SolidMasse moléculaire :411.86Ref: TM-T15759
1mg50,00€2mg71,00€5mg105,00€10mg160,00€25mg344,00€50mg645,00€100mg864,00€1mL*10mM (DMSO)117,00€INCB 3284 dimesylate
CAS :INCB 3284 dimesylate: oral CCR2 antagonist, blocks MCP-1/hCCR2 binding (IC50: 3.7 nM), potential in acute liver failure research.Formule :C28H39F3N4O10S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :712.76(D-Ala2)-GRF (1-29) amide (human)
CAS :(D-Ala2)-GRF (1-29) amide (human) is a potent superagonist of Growth Hormone-Releasing Factor (GRF), demonstrating an exceptionally high Growth Hormone (GH)-Formule :C149H246N44O42SCouleur et forme :SolidMasse moléculaire :3357.88Hemopressin (human, mouse)
CAS :Endogenous peptide, inhibits ep24.15/24.16/ACE with Ki of 27.76/3.43/1.87 μM. Lowers blood pressure, CB1 inverse agonist, reduces pain in vivo.Formule :C50H79N13O12Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1054.26MGV354
MGV354 is a soluble activator of guanylate cyclase(sGC) with EC 50 s of <0.5 nM, and 5 nM in CHO and GTM-3 E cells, respectively [1] [2].Formule :C35H37N5O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :575.7[Arg-15,20,21,Leu17]-PACAP-Gly-Lys-Arg-NH2
CAS :[Arg-15,-20,-21, Leu17]-PACAP-Gly-Lys-Arg-NH2 (BM-PACAP) is a synthetic analogue of PACAP 1-27 that exhibits a relaxant effect [1].Formule :C157H253N53O42Couleur et forme :SolidMasse moléculaire :3555.02Biotin-NeurokininA
Biotin-NeurokininA: biotinylated peptide, NK-2 receptor agonist, key in human airway and gut function.Formule :C60H94N16O16S2Couleur et forme :SolidMasse moléculaire :1359.61Histamine H4 receptor antagonist-1
CAS :Histamine H4 receptor antagonist-1 is a potent antagonist of the histamine H4 receptor.Formule :C30H38N8O2Couleur et forme :SolidMasse moléculaire :542.68Naratriptan D3 Hydrochloride
CAS :Naratriptan D3 Hydrochloride is the deuterium labeled Naratriptan, is a selective agonist of 5-HT1 receptor subtype.Formule :C17H26ClN3O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :374.94Exendin-4 (3-39)
CAS :Exendin-4 (3-39) is a truncated peptide missing first 2 amino acids of Exendin-4, a potent GLP-1r agonist used in diabetes and HPA axis research.Formule :C176H272N46O58SCouleur et forme :SolidMasse moléculaire :3992.4412(S)-HpEPE
CAS :12(S)-HpEPE, a fatty acid created by 12-lipoxygenase on EPA, has unclear biological activities but may resemble 12(S)-HpETE.Formule :C20H30O4Couleur et forme :SolidMasse moléculaire :334.456Orexin A (human, rat, mouse)
CAS :Orexin A, a 33 AA neuropeptide in humans, rats, mice, influences various processes, studied in pancreatic function and as an OX1R antagonist.Formule :C152H243N47O44S4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :3561.1CKLF1-C27 TFA
CKLF1-C27 peptide activates ERK1/2 via CCR4, competes with CKLF1, promotes HUVEC growth, and has psoriasis research potential.Formule :C153H244F3N39O39Couleur et forme :SolidMasse moléculaire :3310.8Glucagon (19-29), human
CAS :Glucagon, a 29-amino-acid hormone, is produced by alpha cells in the pancreas' islets of Langerhans.Formule :C61H89N15O18SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :1352.53α-MSH TFA
CAS :α-Melanocyte-stimulating hormone (α-MSH) is a 13-amino acid peptide hormone produced by post-translational processing of proopiomelanocortin (POMC) in theFormule :C79H110F3N21O21SCouleur et forme :SolidMasse moléculaire :1778.93LAS190792
CAS :LAS190792 (AZD8999) is a dual muscarinic antagonist/β2-agonist, pIC50s (M1-M5, β1-β3): 8.9-5.6; used as a bronchodilator.Formule :C39H43ClN4O9S2Couleur et forme :SolidMasse moléculaire :811.36Sarafotoxin S6a
CAS :Endothelin receptor agonist (EC50 values are 7.5 and > 150 nM for contraction of pig coronary artery and guinea pig aorta respectively). Nociceptive in vivo.Formule :C105H156N28O34S5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :2514.85Cannabidiolic acid methyl ester
CAS :Cannabidiolic acid methyl ester (HU-580) is an orally active analogue of cannabidiolic acid. It enhances the activation of 5-HT1A receptors and increases the expression of c-Fos and NeuN in specific hypothalamic nuclei in rats. Cannabidiolic acid methyl ester exhibits anti-nausea, anxiolytic, and anti-nociceptive effects.Formule :C23H32O4Couleur et forme :SolidMasse moléculaire :372.5a-Helical Corticotropin Releasing Factor (12-41)
CAS :α-Helical CRF (12-41), a 30-aa analog, curbs CRF's ACTH-stimulating effect.Formule :C152H251N43O47S2Couleur et forme :SolidMasse moléculaire :3497.01Uroguanylin (human) TFA
Uroguanylin (human) (TFA) is the natural ligand for the guanylate cyclase C (GCC) receptor expressed in metastatic colorectal cancer tumors. In animal models of human colon cancer, Uroguanylin (human) (TFA) demonstrates antitumor activity.Couleur et forme :Odour SolidPoly-D-lysine hydrobromide (MW 1000-5000)
Poly-D-lysine hydrobromide (PDLHB) (MW 1000-5000) is a synthetically produced polymeric substrate widely used in neural cell culture. Additionally, Poly-D-lysine hydrobromide acts as a CaSR agonist peptide.Couleur et forme :Odour Solid2-Methyl-N,N-dimethyltryptamine
CAS :2-Methyl-N,N-dimethyltryptamine (2,N,N-TMT, compound 15) exhibits binding affinity for the serotonin (5-HT) receptor, with a pA2 value of 6.04. It plays a significant role in neurological disease research.Formule :C13H18N2Couleur et forme :SolidMasse moléculaire :202.35-HT5AR/5-HT6R ligand-1
5-HT5AR/5-HT6R ligand-1 (Compound PP10) is a ligand for serotonin receptors, exhibiting high affinity for the 5-HT5A and 5-HT6 receptors with Ki values of 59 nM and 96 nM, respectively. It possesses some antiproliferative activity against tumor cells and can be utilized in cancer research.Formule :C25H30N4O2SCouleur et forme :SolidMasse moléculaire :450.6TGR5 agonist 2
TGR5 agonist 2 (compound 19) serves as a highly potent agonist of TGR5, demonstrating an EC50 value of 0.27 µM [1].Formule :C29H50NNaO6SCouleur et forme :SolidMasse moléculaire :563.77sGnRH-A
CAS :sGnRH-A, a salmon GnRH analog, boosts growth hormone and induces ovulation for artificial insemination.Formule :C64H83N17O12Couleur et forme :SolidMasse moléculaire :1282.45RXFP3/4 agonist 1
CAS :RXFP3/4 agonist 1 is a relaxin family peptide 3/4 receptor (RXFP3/4) agonist(EC50s of 82/2 nM, respectivley).Formule :C20H22ClN5ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :383.88(Trp7,β-Ala8)-Neurokinin A (4-10)
CAS :(Trp7,β-Ala8)-Neurokinin A (4-10) is a potent neurokinin-3 (NK3) antagonist [1] .Formule :C41H57N9O10SCouleur et forme :SolidMasse moléculaire :868.01Atrial natriuretic factor (1-28) (rat) TFA
ANP (1-28), rat (TFA) inhibits Ang II-induced endothelin-1 secretion; main circulating ANP form in rats.Formule :C130H206N45F3O41S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :3176.43Apraglutide
CAS :Apraglutide (FE 203799 is a synthetic 33-amino acid peptide and long-acting glp-2 analogue.Formule :C172H263N43O52Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :3765.2511-deoxy Prostaglandin F1α
CAS :11-deoxy PGF1α is a synthetic analog of PGF1α.Formule :C20H36O4Couleur et forme :SolidMasse moléculaire :340.504BQ-123 TFA
BQ-123 TFA: Potent ETA antagonist, IC50 = 7.3 nM, Ki = 25 nM, inhibits ET-1 cell proliferation, lowers rat BP.Formule :C33H43F3N6O9Couleur et forme :SolidMasse moléculaire :724.72RF9
CAS :RF9 is an effective and selective antagonist of the Neuropeptide FF receptor (Kis: 58±5 and 75±9 nM for hNPFF1R and hNPFF2R, respectively).Formule :C26H38N6O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :482.62MM 419447
CAS :MM 419447, a linaclotide metabolite, is a guanylate cyclase-C agonist showing potential in IBS-C research.Formule :C50H70N14O19S6Couleur et forme :SolidMasse moléculaire :1363.55(D-Phe12,Nle21,38,α-Me-Leu37)-CRF (12-41) (human, rat)
CAS :(D-Phe12,Nle21,38,α-Me-Leu37)-CRF (12-41) (human, rat) is a corticotropin-releasing factor (CRF) antagonist known to counteract the inhibitory effects of IL-1aFormule :C159H267N49O43Couleur et forme :SolidMasse moléculaire :3553.12Kisspeptin 13
CAS :Kisspeptin 13 activates GPR54 & GnRH receptors, boosts memory, and aids in Alzheimer's research.Formule :C78H107N21O18Couleur et forme :SolidMasse moléculaire :1626.81(D-Ser4,D-Ser(tBu)6,Azagly10)-LHRH
CAS :Analog of LHRH, stimulates LH and FSH release, controls reproduction.Formule :C59H84N18O14Couleur et forme :SolidMasse moléculaire :1269.418-iso Prostaglandin E1
CAS :8-iso Prostaglandin E1 causes spasm in the pulmonary veins of dogs and also acts as a vasodilator.
Formule :C20H34O5Couleur et forme :Light Yellow Crystalline SolidMasse moléculaire :354.48Galanin (1-30), human
CAS :Galanin (1-30), human is a neuropeptide agonist for GalR1/R2 receptors with 1 nM affinity, influencing endocrine, metabolism, and neurotransmission.Formule :C139H210N42O43Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :3157.46Imipramine N-oxide
CAS :Imipramine N-oxide is a tricyclic antidepressant (TCA) and imipramine analogue used to treat depression.Formule :C19H24N2ODegré de pureté :99.80%Couleur et forme :SolidMasse moléculaire :296.41Ref: TM-T74205
1mg72,00€5mg157,00€10mg241,00€25mg409,00€50mg565,00€100mg794,00€1mL*10mM (DMSO)167,00€8-iso-15-keto Prostaglandin F2α
CAS :8-iso-15-keto Prostaglandin F2α (8-iso-15-keto PGF2α) is a metabolite of the isoprostane 8-iso PGF2α in rabbits, monkeys, and humans.Formule :C20H32O5Couleur et forme :SolidMasse moléculaire :352.471(Phe2,Orn8)-Oxytocin acetate
(Phe2,Orn8)-Oxytocin acetate: V1 agonist with EC50 of 280 nM for rabbit epididymis contractility.Formule :C44H69N13O13S2Couleur et forme :SolidMasse moléculaire :1052.23M871
CAS :GAL2 receptor antagonist; Ki: 13.1 nM (GAL2), 420 nM (GAL1); inhibits GAL2-induced pain.Formule :C108H163N27O28Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :2287.64σ1R-IN-1
σ1R-IN-1 ((R,R)-1a) is an effective σ-1R inhibitor with an IC50 of 110 nM. It shows promising potential for use in research related to neuropsychiatric disorders.Formule :C15H22N2Couleur et forme :SolidMasse moléculaire :230.35ALD1613
ALD1613 is a potent neutralizing monoclonal antibody targeting adrenocorticotropic hormone (ACTH). It neutralizes ACTH-induced signaling and inhibits cyclic adenosine monophosphate accumulation in ACTH-stimulated Y1 (mouse adrenal cell line) via all five melanocortin receptors. ALD1613 significantly reduces plasma corticosterone levels in wild-type rats and is applicable in studies involving elevated ACTH-related conditions.Couleur et forme :Odour LiquidKassinin
CAS :Kassinin is a peptide derived from the Kassina frog. It belongs to tachykinin family of neuropeptides.Formule :C59H95N15O18SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :1334.54CCZ01048 TFA
CCZ01048 TFA, α-MSH analog, binds MC1R with 0.31 nM affinity, internalizes in melanoma cells, and is stable for melanoma PET imaging.Formule :C73H106F3N21O18Couleur et forme :SolidMasse moléculaire :1622.755-HT6R antagonist 6
5-HT6R antagonist 6 (Compound PP15) exhibits high affinity and selectivity for the 5-HT6R receptor, with a Ki of 42 nM. It demonstrates weak antiproliferative activity on tumor cells and low toxicity toward normal cells. 5-HT6R antagonist 6 is applicable in tumor research.Formule :C24H26N4O2SCouleur et forme :SolidMasse moléculaire :434.55D5R agonist 1
D5R Agonist 1 (Compound 5j) is a selective, orally active partial agonist of the D5 receptor that can penetrate the blood-brain barrier (EC50: 269.7 nM). It has been demonstrated to enhance cognitive abilities in a scopolamine-induced amnesia model.Couleur et forme :Odour Solid1,8-Cineole
CAS :Eucalyptol, a natural monoterpenoid and cyclic ether found in eucalyptus species, effectively controls excessive airway mucus secretion and asthma by inhibiting pro-inflammatory cytokines. It serves as an efficacious treatment for non-purulent sinusitis, reducing inflammation and pain when applied topically, and demonstrating leukemic cell-killing capabilities in vitro.Formule :C10H18ODegré de pureté :97.44% - 97.44%Couleur et forme :SolidMasse moléculaire :154.25CRSP-1
CAS :Central CT receptor agonist, 350x stronger than CT, no CGRP or adrenomedullin action, inhibits osteoclasts, affects rat feeding, body temp, and calcium.Formule :C175H294N54O49S5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :4098.88γ-2-MSH (41-58), amide
CAS :Melanocortin (MC) 3-MSH (Melanocyte-Stimulating Hormone) is believed to signal through the MC 3 receptor.Formule :C74H100N22O15SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :1569.79Cloprostenol isopropyl ester
CAS :(+)-Chloprostol is a PGF2α agonist, mimics prostaglandin F2α, induces luteal dissolution in mares without side effects or stress.Formule :C25H35ClO6Couleur et forme :SolidMasse moléculaire :466.99BM213 acetate
BM213 acetate is a selective C5aR1 agonist with antitumor activity that induces C5aR1-mediated calcium mobilization and pERK1/2 signaling.
Formule :C45H74N12O12Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :975.14GLP-1(28-36)amide TFA
GLP-1(28-36)amide TFA, a nonapeptide cleavage product of GLP-1, shows antioxidant properties with anti-diabetic and cardioprotective effects.Formule :C56H86F3N15O11Couleur et forme :SolidMasse moléculaire :1202.37Ecnoglutide
CAS :Ecnoglutide (XW003) is a glucagon-like peptide 1 (GLP-1) receptor agonist [1] .Formule :C194H304N48O61Couleur et forme :SolidMasse moléculaire :4284.76[Nle11]-Substance P
CAS :'[Nle11]-Substance P is a gut and brain peptide, resisting methionine oxidation and causing excitatory neural effects.'
Formule :C64H100N18O13Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1329.59Zenagamtide sodium
Zenagamtide is an agonist for both glucagon-like peptide-1 (GLP-1) and amylin receptors.Couleur et forme :Odour SolidKB-5492 FA
KB-5492 FA is a selective sigma receptor inhibitor with antiulcerogenic effects.CAS 번호128-52-56-8Formule :C24H32N2O8Degré de pureté :98.12%Couleur et forme :SolidMasse moléculaire :476.52Msh (11-13)
CAS :Msh (11-13) is a bioactive chemical.Formule :C16H30N4O4Couleur et forme :SolidMasse moléculaire :342.43Pobilukast
CAS :Pobilukast (SKF 104353) is a cysteinyl leukotriene receptor antagonist that can be used to study limiting myocardial injury in MI/R rats.Formule :C26H34O5SDegré de pureté :99.65% - 99.84%Couleur et forme :SolidMasse moléculaire :458.61SAR441255
SAR441255 is a potent unimolecular peptide that acts as a GLP-1/GIP/GCG receptor triagonist, demonstrating balanced activation across all three target receptorsCouleur et forme :Odour SolidJNJ-10181457 (hydrochloride)
CAS :JNJ-10181457 (hydrochloride) is a non-imidazole H3 receptor antagonist that is brain-penetrating and selective, increasing NE and acetylcholine concentrationsFormule :C20H30Cl2N2OCouleur et forme :SolidMasse moléculaire :385.3715(S)-15-methyl Prostaglandin F2α methyl ester
CAS :15(S)-15-methyl Prostaglandin F2α methyl ester can be used in related research in the field of life sciences.Formule :C22H38O5Couleur et forme :SolidMasse moléculaire :382.53Urocortin II, human acetate
Urocortin II, human acetate, is a selective endogenous peptide agonist of type 2 corticotropin-releasing factor (CRF2) receptors, used to study the role of CRF2 receptors in feeding behavior.Couleur et forme :Odour SolidCorticotropin-releasing factor (human) acetate
Corticotropin-releasing factor (human) acetate stimulates to synthesize and secret adrenocorticotropin in the anterior pituitary.Degré de pureté :98.30%Couleur et forme :LiquidNXT-10796
NXT-10796 is an orally active, intestinally restricted agonist of the EP4 receptor [1].Formule :C23H31N3O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :445.51PA-8
CAS :PA-8: Selective PAC1 antagonist, orally active, blocks CREB phosphorylation & cAMP increase (IC50=2nM), reduces pain & aversive response in vivo.Formule :C17H18N4O4Degré de pureté :97.54%Couleur et forme :SolidMasse moléculaire :342.35Atrial natriuretic peptide (3-28) (human)
CAS :Atrial natriuretic peptide (3-28) (human) (ANP (3-28) (human)), a peptide hormone produced by the atrial myocardium, plays a critical role in the regulation ofFormule :C118H187N43O36S3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :2880.21Substance P (alligator)
CAS :Substance P from alligator: a neuropeptide with structure Arg-Pro-Arg-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH2.Formule :C63H98N20O13SCouleur et forme :SolidMasse moléculaire :1375.64ACTH (7-38) (human)
CAS :ACTH (7-38) (human) is a fragment (7-38) of the full human adrenocorticotropic hormone (ACTH (1-39)), also referred to as corticotropin inhibitory peptide (CIPFormule :C167H257N47O46Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :3659.11Conopeptide rho-TIA
CAS :Conopeptide rho-TIA, a peptide from Conus tulipa venom, acts as a selective, noncompetitive inhibitor at the human α1B-Adrenergic Receptor and as a competitiveFormule :C105H160N36O21S4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :2390.88Fasitibant chloride
CAS :Fasitibant chloride, a potent B2R blocker, alleviates pain and swelling in arthritis.
Formule :C36H49Cl3N6O6SCouleur et forme :SolidMasse moléculaire :800.23Dp[Tyr(methyl)2,Arg8]-Vasopressin
CAS :Dp[Tyr(Me)2,Arg8]-Vasopressin is a non-selective antagonist of the peptide arginine vasopressin V1b receptor [1].Formule :C49H70N14O12S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1111.3Pasireotide pamoate
CAS :Pasireotide pamoate is a stable cyclohexapeptide somatostatin mimic. Pasireotide pamoate exhibits antisecretory, antiproliferative, and proapoptotic activity.Formule :C81H82N10O15Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1435.58[Leu13]-Motilin
CAS :[Leu13]-Motilin (KW-5139) is an analogue of the gastrointestinal hormone motilin that induces concentration-dependent contractions in rabbit gastrointestinalFormule :C121H190N34O35Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :2681.014-Chloromethamphetamine hydrochloride
CAS :4-Chloromethamphetamine hydrochloride is a novel psychoactive substance belonging to the amphetamine class.Formule :C10H15Cl2NCouleur et forme :SolidMasse moléculaire :220.14Galanin-Like Peptide (rat)
CAS :Galanin-Like Peptide (rat), a neuropeptide comprising 60 amino acids, plays a crucial role in regulating feeding, body weight, and energy metabolism [1].Formule :C288H461N87O83SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :6502.34PACAP (6-38), human, ovine, rat acetate
PACAP (6-38), human, ovine, rat acetate is a potent PACAP receptor antagonist with IC50s of 30, 600, and 40 nM for PACAP type I receptor, PACAP type II receptorFormule :C184H303N55O48SDegré de pureté :99.84%Couleur et forme :SoildMasse moléculaire :4085.84(Ala13)-Apelin-13 acetate
(Ala13)-Apelin-13 acetate, an APJ antagonist, modulates CRF-induced enhanced colonic motility, visceral sensation, and gut barrier.Formule :C65H111N23O18SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :1534.79Ref: TM-T35374L
2mg116,00€5mg166,00€10mg259,00€25mg492,00€50mg740,00€100mg1.110,00€200mg1.668,00€500mg3.167,00€FR167344 free base
CAS :FR167344 free base: oral, nonpeptide B2 bradykinin receptor antagonist, high-affinity (IC50: 65 nM), no B1 affinity.Formule :C30H28BrCl2N5O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :673.38Des-Arg9-[Leu8]-Bradykinin acetate
CAS :Des-Arg9-[Leu8]-Bradykinin acetate is a potent antagonist of the bradykinin receptor 1 (B1R), utilized in renal fibrosis research [1].Formule :C43H67N11O12Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :930.06hA3AR agonist 2
hA3AR agonist 2 is a potent activator of A3AR, with a Ki value of 3.5 nM.Formule :C11H14ClN5O2SCouleur et forme :SolidMasse moléculaire :315.78Galanin-Like Peptide (human)
CAS :Galanin-Like Peptide (human) is a neuropeptide consisting of 60 amino acids, instrumental in regulating feeding, body weight, and energy metabolism [1].Formule :C292H451N83O84SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :6500.285-MeO-MET
CAS :5-MeO-MET (5-Methoxy-N-methyl-N-ethyltryptamine) is a compound belonging to the 5-methoxytryptamine class. It acts as an agonist for 5-HT1A and 5-HT2A receptors. In mice, 5-MeO-MET inhibits locomotion and has sedative effects.Formule :C14H20N2OCouleur et forme :SolidMasse moléculaire :232.32Bz-Dab(nbd)-awfpp-nle-NH2
CAS :Bz-Dab(nbd)-ala-trp-phe-pro-pro-nle-NH2 is a fluorescent NK2 antagonist.Formule :C56H65N13O11Couleur et forme :SolidMasse moléculaire :1096.26-Fluoro-N,N-diethyltryptamine
CAS :6-Fluoro-N,N-diethyltryptamine (6-F-DET) exhibits affinity for the 5-HT2A receptor.Formule :C14H19FN2Couleur et forme :SolidMasse moléculaire :234.3125N-NBOMe hydrochloride
CAS :25N-NBOMe hydrochloride is a derivative of 2C-N and acts as an agonist for the 5-HT2A and 5-HT2C receptors, with Ki values of 0.144 nM and 1.06 nM, respectively. It has minimal effect on the release of preloaded neurotransmitters from recombinant dopamine, serotonin, and norepinephrine transporters.Formule :C18H23ClN2O5Couleur et forme :SolidMasse moléculaire :382.84(Leu31,Pro34)-Peptide YY (human) (TFA)
"(Leu31,Pro34)-Peptide YY (human) (TFA) is the trifluoroacetic acid (TFA) form of (Leu31,Pro34)-Peptide YY (human), a derivative of Peptide YY that acts as aFormule :C195H296N54O56·xC2HF3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :4292.75 (free base)[D-Trp8]-γ-MSH
CAS :[D-Trp8]-γ-MSH is a selective melanocortin 3 (MC3) receptor agonist (IC50 values are 6.7, 340 and 600 nM for human MC3, MC5 and MC4 receptors respectively).Formule :C74H99N21O16SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :1570.7915-keto Latanoprost
CAS :Latanoprost, a PG analog for ocular pressure, metabolizes into 15-keto latanoprost, a less potent variant reducing intraocular pressure and pupil size.Formule :C26H38O5Couleur et forme :SolidMasse moléculaire :430.584-Iodoamphetamine hydrochloride
CAS :4-Iodoamphetamine (p-Iodoamphetamine) hydrochloride is a halogenated phenethylamine characterized by the presence of an iodine atom at the para position of the phenyl group. It selectively induces serotonin release and inhibits reuptake in rat brain synaptosomes.Formule :C9H13ClINCouleur et forme :SolidMasse moléculaire :297.564-hydroxy DiPT hydrochloride
CAS :4-hydroxy DiPT (hydrochloride) is a 5-HT2A agonist that can induce head twitch response (HTR) in mice, indicating its hallucinogenic potential. This compound holds promise for research into hallucinogens.Formule :C16H25ClN2OCouleur et forme :SolidMasse moléculaire :296.84Casopitant
CAS :Casopitant (GW679769) is an orally active neurokinin-1 (NK1) receptor antagonist, researched for its potential use in managing chemotherapy-induced nausea and vomiting (CINV) and postoperative nausea and vomiting (PONV).Formule :C30H35F7N4O2Couleur et forme :SolidMasse moléculaire :616.61(Iso)-RJW100
CAS :Potent LRH-1/NR5A2 and SF-1/NR5A1 agonist; pEC50: 6.4 (LRH-1), 7.2 (SF-1).Formule :C28H34ODegré de pureté :99.79%Couleur et forme :SoildMasse moléculaire :386.57Ref: TM-T64363
1mg109,00€5mg241,00€10mg354,00€25mg532,00€50mg745,00€100mg1.018,00€500mg2.035,00€1mL*10mM (DMSO)259,00€Eloralintide
CAS :Eloralintide (LY 3841136) is an AMYR agonist, anticipated for research in type 2 diabetes and obesity.Formule :C201H319N49O65S2Couleur et forme :SolidMasse moléculaire :4526.1PACAP (6-38), human, ovine, rat
CAS :PACAP (6-38) in humans, sheep, rats: a strong inhibitor of PACAP 38, outperforms PACAP (6-27) in blocking PACAP-27-induced adenylate cyclase.Formule :C182H300N56O45SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :4024.744-Bromo-2,5-DMMA
CAS :4-Bromo-2,5-DMMA (Compound 2) demonstrates affinity for the 5-HT2 binding site and has an ED50 of 0.82 mg/kg in rat discrimination experiments.Formule :C12H18BrNO2Couleur et forme :SolidMasse moléculaire :288.18Arotinolol hydrochloride
CAS :Arotinolol HCl is a non-selective α/β-blocker, anti-hypertensive, anti-obesity, and improves aortic stiffness.Formule :C15H22ClN3O2S3Degré de pureté :99.82%Couleur et forme :SolidMasse moléculaire :408Latanoprost tris(triethylsilyl) ether
CAS :Latanoprosttris(triethylsilyl) ether is a precursor in the synthesis of Latanoprost, which serves as an agonist for the prostaglandin F2α (PGF2α) receptor, also known as the FP receptor.Formule :C44H82O5Si3Couleur et forme :SolidMasse moléculaire :775.38FXR/TGR5 agonist 1
CAS :FXR/TGR5 agonist 1 acts as an agonist on both FXR and TGR5 receptors and is utilized for treating fatty liver disease.Formule :C31H32ClN3O3Couleur et forme :SolidMasse moléculaire :530.07Amylin, amide, rat
CAS :Amylin: peptide, 50% similar to CGRP, found with somatostatin in stomach cells, reduces acid secretion in mice.Formule :C167H272N52O53S2Degré de pureté :99.92%Couleur et forme :SolidMasse moléculaire :3920.448-iso Prostaglandin A2
CAS :8-iso Prostaglandin A2 is an isoprostane produced by the nonenzymatic oxidation of arachidonic acid.Formule :C20H30O4Couleur et forme :SolidMasse moléculaire :334.45Ornipressin
CAS :Ornipressin is a vasoconstrictor, haemostatic and renal agent.Formule :C45H63N13O12S2Degré de pureté :98%Couleur et forme :White PowderMasse moléculaire :1042.19BQ-3020 ammonium
BQ-3020 ammonium, a selective endothelin receptor (ET B receptor) agonist, demonstrates inhibition of [125 I] ET-1 binding to ET B receptors with an IC50 of 0.2Formule :C96H140N20O25S·xNH3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :2006.32 (free base)TCMCB07 TFA
TCMCB07 TFA is a cyclic nonapeptide and an orally active, brain-penetrating antagonist of the melanocortin receptor 4 (MC4R), playing a significant role inFormule :C63H87N15O11·xC2HF3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1230.46 (free base)Adenosine 3'-monophosphate (sodium salt hydrate)
Adenosine 3'-monophosphate (sodium salt hydrate) (3'-AMP) is a nucleotide and cAMP-generating agonist that elevates cAMP levels in NG108-15 cells.Formule :C10H15N5NaO8PCouleur et forme :SolidMasse moléculaire :387.225-HT6R antagonist 1
Compound 8 (5-HT6R antagonist 1), a 5-HT6R antagonist (K i : 5 nM), not only demonstrates inhibition of platelet aggregation and excellent metabolic stabilityFormule :C17H22F2N6ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :364.39Δ8-THC methyl ether
CAS :Δ8-THC methyl ether (compound 3) demonstrates a strong docking score of -10.167 kcal/mol for the CB2 receptor. Additionally, Δ8-THC methyl ether exhibits antinociceptive activity in mice.Formule :C22H32O2Couleur et forme :SolidMasse moléculaire :328.49PZ-1922
PZ-1922 (Compound 16), able to cross the blood-brain barrier, is a dual antagonist for 5-HT6R and 5-HT3R with K i values of 17 nM and 0.45 nM, respectively.Degré de pureté :98%Couleur et forme :Odour SolidOsanetant
CAS :Osanetant produces anxiolytic- and antidepressant-like effects. Osanetant is a selective NK3 receptor antagonist. It is researched for schizophrenia.Formule :C35H41Cl2N3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :606.62GLP-1R agonist 4
CAS :GLP-1R agonist 4, potentially for diabetes research, is a potent GLP-1R stimulator linked to hypoglycemia.Formule :C32H30ClF2N3O5Couleur et forme :SolidMasse moléculaire :610.054-Methylhistamine
CAS :4-Methylhistamine serves as a potent agonist for the histamine 4 receptor (H4R), holding promise for research into immune-related diseases, including cancer andFormule :C6H11N3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :125.17L-797,591
CAS :L-797,591 is a selective agonist of somatostatin receptor subtype 1.Formule :C38H49N5O2Couleur et forme :SolidMasse moléculaire :607.83Sigma-1 receptor antagonist 4
Sigma-1 receptor antagonist 4 (Compound 32) is a potent σ1R antagonist that significantly enhances morphine's analgesic effects and reverses morphine-inducedFormule :C22H26N2OCouleur et forme :SolidMasse moléculaire :334.45PACAP-related Peptide (human) (trifluoroacetate salt)
Endogenous 29-amino acid PRP belongs to secretin/glucagon family, found in pancreas, adrenal glands, and some VIP tumors; secreted by CHO-K1 cells.Couleur et forme :LiquidBrexpiprazole S-oxide
CAS :Brexpiprazole S-oxide is the main metabolite of Brexpiprazole, a human 5-HT1A and dopamine receptor partial agonist (Ki: 0.12, 0.3 nM).Formule :C25H27N3O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :449.575-HT2C agonist-4
CAS :Compound 3i, a 5-HT2C agonist-4, acts as an agonist for the 5-HT2C receptor with an EC50 of 5.7 nM. It is capable of reducing locomotor activity in zebrafish larvae.Formule :C24H25N5OCouleur et forme :SolidMasse moléculaire :399.49TE-8105
TE-8105 is a GLP-1 receptor agonist that demonstrates prolonged and enhanced efficacy in models of diabetes, obesity, and non-alcoholic steatohepatitis (NASH).Couleur et forme :Odour SolidPAF C-18
CAS :PAF C-18 is a natural phospholipid molecule belonging to the platelet-activating factor (PAF) family,, involved in hemostasis and thrombosis by binding to PAFR.Formule :C28H58NO7PDegré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :551.74BIM-23190 hydrochloride
BIM-23190 hydrochloride, somatostatin analog, SSRT2/5 agonist, Ki: 0.34 nM (SSTR2), 11.1 nM (SSTR5). Used in cancer, acromegaly research.Couleur et forme :Liquid(+)-Oxypeucedanin methanolate
CAS :(+)-Oxypeucedanin methanolate (compound 9) is a natural compound that inhibits prostaglandin E2 production [1].Formule :C17H18O6Couleur et forme :SolidMasse moléculaire :318.32KSK94 FA
KSK94 FA is a potent histamine H3 receptor antagonist that inhibits H3 receptors and is used in the study of neuropathic pain and obesity.Formule :C26H28N4O3Degré de pureté :97.51%Couleur et forme :SoildMasse moléculaire :444.53TRPV1/CB2 agonist 1
TRPV1/CB2 agonist 1 (compound 41) is a dual agonist targeting hTRPV1 and CB2 receptors, with an EC50 value of 26.8 μM for hTRPV1. It is applicable in research related to the nervous system.Couleur et forme :Odour SolidBim 21009
CAS :Bim 21009 is an inhibitor of gonadorelin.Formule :C74H92ClN17O13Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1463.08HS024 TFA
HS024, a selective MC4 receptor antagonist, exhibits affinity with Ki values of 0.29, 3.29, 5.45, and 18.6 nM for MC4, MC5, MC3, and MC1 receptors, respectivelyFormule :C60H80F3N19O12S2Couleur et forme :SolidMasse moléculaire :1380.52LH-RH (7-10)
CAS :LH-RH (7-10), a tetrapeptide, is a key LHRH degradation product found in macrophages and pneumocytes.Formule :C19H36N8O4Couleur et forme :SolidMasse moléculaire :440.54SLP7111228
CAS :SLP7111228 is an effective and selective SphK1 inhibitor (Ki = 48 nM).Formule :C22H33N5OCouleur et forme :SolidMasse moléculaire :383.53N-Nitroso Atenolol
CAS :N-Nitroso Atenolol is a derivative of Atenolol. At concentrations ranging from 0.1 to 1 mM, it induces DNA fragmentation in rat hepatocytes.Formule :C14H21N3O4Couleur et forme :SolidMasse moléculaire :295.33ANQ-11125 TFA
ANQ-11125 TFA is a motilin antagonist with a pKd of 8.24, inhibiting motilide contractions in rabbits.Formule :C88H126F3N19O23Couleur et forme :SolidMasse moléculaire :1875.05Neuropeptide Y (18-36) (porcine)
CAS :"Neuropeptide Y (18-36) (porcine) is a NPY heart receptor blocker, halts I-NPY binding, aids in heart failure research."Formule :C112H174N36O27Couleur et forme :SolidMasse moléculaire :2456.8RS 56812
CAS :RS 56812 is a 5-HT3 receptor antagonist and agonist used in the study of cognitive disorders.Formule :C18H21N3O2Degré de pureté :99.38%Couleur et forme :SoildMasse moléculaire :311.38(±)-9-Nor-9α-hydroxy Hexahydrocannabinol
CAS :(±)-9-Nor-9α-hydroxy Hexahydrocannabinol is a cannabinoid-structured compound that exhibits potent cannabinoid-like activity in both dogs and mice.Formule :C20H30O3Couleur et forme :SolidMasse moléculaire :318.45Bodilisant
CAS :Bodilisant: nanomolar-affinity hH3R ligand, derived from piperidine, with BODIPY fluorophore.Formule :C27H34BF2N3OCouleur et forme :SolidMasse moléculaire :465.4Pancreatic Polypeptide, bovine
CAS :Agonist at Y4 neuropeptide Y receptors.Formule :C186H287N53O56S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :4225.78MRS2500 tetraammonium
CAS :Highly potent and selective antagonist of the platelet P2Y1 receptorFormule :C13H21IN6O8P2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :578.19Serazapine
CAS :Serazapine is a highly specific serotonin (5-HT2) binding inhibitor with anxiolytic activity for the treatment of anxiety disorders.
Formule :C22H23N3O2Degré de pureté :98.71% - 99.57%Couleur et forme :SolidMasse moléculaire :361.44Alsactide
CAS :Alsactide, an adrenocorticotropic hormone (ACTH) agonist and a heptadecapeptide analogue, is utilized in the study of the central nervous system [1].Formule :C99H155N29O21SCouleur et forme :SolidMasse moléculaire :2119.53Neuropeptide SF(mouse,rat) TFA
Neuropeptide SF TFA is a potent agonist for NPFF1 (Ki=48.4 nM) and NPFF2 (Ki=12.1 nM) and enhances ASIC3 current.Formule :C42H66F3N13O12Couleur et forme :SolidMasse moléculaire :1002.05BAM(8-22)
CAS :Potent MRGPRX1 agonist peptide; first found in bovine adrenal glands. Non-opioid, lacking met-enkephalin motif. EC50: 8-150 nM.Formule :C91H127N25O23SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :1971.22Peptide YY (PYY) (3-36), porcine TFA
Peptide YY (PYY) (3-36), porcine TFA, functions as a gut hormone that serves as a Y2 receptor agonist, effectively reducing appetite [1].Formule :C176H272N52O54·C2HF3O2Couleur et forme :SolidMasse moléculaire :4094.44CCK (26-30) (sulfated)
CAS :CCK (26-30) is a digestive and satiety-related peptide fragment inhibiting [125I]CCK-33 binding by 10% at 0.1 mM.Formule :C33H41N7O12S2Couleur et forme :SolidMasse moléculaire :791.85
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