GPCR/G-Protéine
Les inhibiteurs des GPCR/protéines G sont des composés qui ciblent les récepteurs couplés aux protéines G (GPCR) et les protéines G associées, qui jouent un rôle crucial dans la transmission des signaux de l'extérieur vers l'intérieur des cellules. Ces inhibiteurs sont essentiels pour étudier les voies de signalisation médiées par les GPCR, impliquées dans de nombreux processus physiologiques, y compris la perception sensorielle, la réponse immunitaire et la neurotransmission. Les inhibiteurs des GPCR sont également importants dans le développement de médicaments, car de nombreux agents thérapeutiques ciblent ces récepteurs. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de GPCR/protéines G de haute qualité pour soutenir vos recherches en pharmacologie, biologie cellulaire et domaines connexes.
Sous-catégories appartenant à la catégorie "GPCR/G-Protéine"
- récepteur 5-HT(1.025 produits)
- Récepteur d'adénosine(249 produits)
- Récepteur adrénergique(3.018 produits)
- Récepteur de la bombésine(35 produits)
- Récepteur de la bradykinine(61 produits)
- CXCR(158 produits)
- CaSR(34 produits)
- Récepteur cannabinoïde(217 produits)
- Cholécystokinine(1 produits)
- Récepteur de la dopamine(445 produits)
- Récepteur de l'endothéline(86 produits)
- Récepteur GNRH(84 produits)
- GPCR19(33 produits)
- GRK(33 produits)
- GTPase(23 produits)
- Récepteur du glucagon(194 produits)
- Hérisson/Smoothened(49 produits)
- Récepteur de l'histamine(385 produits)
- Récepteur LPA(21 produits)
- Récepteur de la mélatonine(26 produits)
- Récepteur OX(41 produits)
- Récepteur opioïde(327 produits)
- PAFR(14 produits)
- PKA(60 produits)
- Récepteur S1P(18 produits)
- SGLT(31 produits)
- Récepteur Sigma(46 produits)
Affichez 19 plus de sous-catégories
5983 produits trouvés pour "GPCR/G-Protéine"
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Cholic Acid 7-sulfate
CAS :Cholic acid 7-sulfate: a cholic acid metabolite with added sulfate at position 7, increased in feces of male mice with specific diets.Formule :C24H40O8SCouleur et forme :SolidMasse moléculaire :488.64ACT-373898
CAS :ACT-373898 is a metabolite of the endothelin (ET) receptor type A (ETA) and ETBdual antagonist macitentan .1Formule :C15H17BrN4O5SCouleur et forme :SolidMasse moléculaire :445.29[Des-Arg10]-HOE I40 TFA
[Des-Arg10]-HOE I40 TFA is a potent antagonist of the bradykinin B1 receptor.
Formule :C53H77N15O12S·xC2HF3O2Couleur et forme :Solidα-CGRP(human)
CAS :Endogenous calcitonin gene-related peptide receptor (CGRP) agonist.Formule :C163H267N51O49S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :3789.33RF9
CAS :RF9 is an effective and selective antagonist of the Neuropeptide FF receptor (Kis: 58±5 and 75±9 nM for hNPFF1R and hNPFF2R, respectively).Formule :C26H38N6O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :482.62Azaline B
CAS :Azaline B is an antagonist of the gonadotropin-releasing hormone (GnRH), with an IC50 of 1.37 nM. It is utilized in research related to pathologies associated with sex hormones, ovulation induction, and male contraception.Formule :C80H102ClN23O12Couleur et forme :SolidMasse moléculaire :1613.27Xenopus orexin B
CAS :Xenopus orexin B, a neuropeptide identified as an endogenous ligand for an orphan G-protein-coupled receptor, acts as a potent agonist of OX2R [1].Formule :C130H219N45O40S2Couleur et forme :SolidMasse moléculaire :3116.54TRAP-6 amide TFA
CAS :TRAP-6 amide TFA is a PAR-1 thrombin receptor agonist peptide.Formule :C36H58F3N11O10Couleur et forme :SolidMasse moléculaire :861.922Zovaglutide
CAS :Zovaglutide is a GLP-1 receptor agonist that is utilized in diabetes research.Couleur et forme :SolidRC-3095
CAS :RC-3095, a selective GRPR antagonist, has been shown to have anti-inflammatory properties in different models of inflammation.Formule :C56H79N15O9Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1106.32Rhazimine
CAS :Rhazimine is an indole alkaloid. It is a dual inhibitor of arachidonic acid metabolism and platelet activating factor-induced platelet aggregation.Formule :C21H22N2O3Couleur et forme :SolidMasse moléculaire :350.418ACTH (1-17)
CAS :ACTH (1-17), a potent MC1 receptor agonist with a Ki of 0.21 nM, is a variant of corticotropin from the pituitary gland.Formule :C95H145N29O23SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :2093.41Mapenterol hydrochloride
CAS :Mapenterol hydrochloride is an agonist of β2-adrenergic receptor.Formule :C14H21Cl2F3N2ODegré de pureté :98.11% - 99.98%Couleur et forme :SolidMasse moléculaire :361.23Ref: TM-T40622
1mg49,00€5mg102,00€10mg149,00€25mg249,00€50mg358,00€100mg520,00€500mg1.035,00€1mL*10mM (DMSO)107,00€APC 366 TFA
CAS :APC 366 (TFA) is a potent irreversible inhibitor of mast cell tryptase. It is particularly useful in studies related to allergic diseases.Formule :C24H29F3N6O6Couleur et forme :SolidMasse moléculaire :554.527Neurokinin B (TFA)
CAS :Neurokinin B TFA, a tachykinin, targets NK1R, NK2R, nk3r GPCRs, modulating effects.Formule :C59H81F6N13O18S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1438.47Yohimbic acid, ethyl ester
CAS :Yohimbic acid, ethyl ester is a biochemical with possible effects on reserpine action.Formule :C22H28N2O3Couleur et forme :SolidMasse moléculaire :368.47WB4-24
CAS :WB4-24 is a GLP-1 receptor agonist that enhances the release of β-endorphin in microglia. It exhibits antiallodynic, anti-inflammatory, and analgesic effects in mouse models of inflammation induced by formalin, carrageenan, and CFA.Formule :C52H48N4O14S2Couleur et forme :SolidMasse moléculaire :1017.09Dexbrompheniramine
CAS :Dexbrompheniramine: oral H1 antagonist, antihistamine for hay fever and urticaria research.Formule :C16H19BrN2Couleur et forme :SolidMasse moléculaire :319.24Thioperamide maleate
CAS :Thioperamide maleate (MR-12842 maleate) is an effective and selective antagonist of H3 receptor (Ki = 4.3 nM) for inhibition of [3H]histamine synthesis (Ki = 31Formule :C19H28N4O4SDegré de pureté :98.48%Couleur et forme :SolidMasse moléculaire :408.52Alosetron
CAS :Alosetron, a 5-HT3 antagonist, is used for the management of severe diarrhea-predominant irritable bowel syndrome (IBS) in women only.Formule :C17H18N4ODegré de pureté :98%Couleur et forme :Crystalline PowderMasse moléculaire :294.36Rp-dUTPαS tetrasodium
Rp-dUTPαS (tetrasodium) is an isomer of the sulfur-containing nucleotide dUTP-α-S and acts as an agonist of the purinergic P2Y2 receptor. It selectively induces the accumulation of inositol phosphates in P2Y2-expressing 1321N1 cells with an EC50 of 12.5 μM.Couleur et forme :Odour Solid1,8-Cineole
CAS :Eucalyptol, a natural monoterpenoid and cyclic ether found in eucalyptus species, effectively controls excessive airway mucus secretion and asthma by inhibiting pro-inflammatory cytokines. It serves as an efficacious treatment for non-purulent sinusitis, reducing inflammation and pain when applied topically, and demonstrating leukemic cell-killing capabilities in vitro.Formule :C10H18ODegré de pureté :97.44% - 97.44%Couleur et forme :SolidMasse moléculaire :154.25L 152804
CAS :L 152804: Y5 receptor antagonist, reduces food intake/boosts energy, leads to weight loss in obese mice.Formule :C23H26O4Degré de pureté :99.82%Couleur et forme :SolidMasse moléculaire :366.45Ref: TM-T15679
5mg48,00€10mg75,00€25mg111,00€50mg170,00€100mg245,00€200mg349,00€1mL*10mM (DMSO)49,00€A 31472
CAS :A 31472 is a tetracyclic spiro amine that has affinity for dopamine D-2 receptors.Formule :C22H22ClNCouleur et forme :SolidMasse moléculaire :335.87Cortistatin-8 acetate
Cortistatin-8 acetate: synthetic corticosteroid analog, GHS-R antagonist; doesn't affect acyl GH release or hesperidin response.
Formule :C49H72N12O11S2Degré de pureté :99.01%Couleur et forme :SoildMasse moléculaire :1069.3Ref: TM-TP2236L
1mg229,00€5mg560,00€10mg800,00€25mg1.216,00€50mg1.644,00€100mg2.213,00€500mg4.436,00€Peptide YY (PYY), human
CAS :PYY: a 36-amino-acid hormone, amidated, part of neuroendocrine control, acts via Neuropeptide Y receptors.Formule :C194H295N55O57Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :4309.75GRK2i
CAS :GRK2 inhibitory polypeptide that specifically inhibits Gβγ activation of GRK2. Corresponds to the Gβγ-binding domain and acts as a cellular Gβγ antagonist.Formule :C153H256N50O41SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :3484.08GV-150013X
CAS :GV-150013X ((S)-1-(1-(adamantan-1-ylmethyl)-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydro-1H-benzo[b][1,4]diazepin-3-yl)-3-phenylurea) is a potent CCKB antiagonist, pKiFormule :C33H34N4O3Degré de pureté :99.94%Couleur et forme :SoildMasse moléculaire :534.65Ref: TM-T27503L
1mg90,00€5mg190,00€10mg259,00€25mg394,00€50mg532,00€100mg698,00€200mg924,00€1mL*10mM (DMSO)270,00€HTR2A antagonist 1
HTR2A antagonist 1 (Compound 15f) is an HTR2A antagonist with an IC50 of 42.79 nM. It induces sub-G1 cell cycle arrest and apoptosis in colorectal cancer cells by activating the p53/p21/caspase 3 signaling pathway. HTR2A antagonist 1 exhibits good liver microsomal stability and is useful for colorectal cancer research.Formule :C35H43Cl2F2N5O4Couleur et forme :SolidMasse moléculaire :706.65ZM 253270
CAS :ZM 253270 is an nonpeptide neurokinin A antagonist.Formule :C22H26ClN7O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :471.95Tiflucarbine
CAS :Tiflucarbine is a potential non-selective 5-HT agonist with antidepressant activity.Tiflucarbine dose-dependently increased the specific activity of solubleFormule :C16H17FN2SDegré de pureté :97.71%Couleur et forme :SolidMasse moléculaire :288.38Israpafant
CAS :Israpafant: PAF receptor blocker, IC50 0.84nM, hinders platelet aggregation, eosinophil activation, boosts calcium transit, anti-nephrotoxic.Formule :C28H29ClN4SCouleur et forme :SolidMasse moléculaire :489.07Tebufelone
CAS :Tebufelone is a potent NSAID, inhibits CO, has anti-inflammatory and analgesic properties, and blocks lipoxygenase products (IC50 ~20-22 microM).Formule :C20H28O2Degré de pureté :99.61%Couleur et forme :SolidMasse moléculaire :300.44Ref: TM-T68155
1mg54,00€5mg114,00€10mg169,00€25mg268,00€50mg410,00€100mg592,00€500mg1.224,00€1mL*10mM (DMSO)177,00€15(S)-15-methyl Prostaglandin D2
CAS :15(S)-15-methyl PGD2 is a stable PGD2 analog that induces vasoconstriction, raises blood pressure, and shows strong antifertility effects.Formule :C21H34O5Couleur et forme :SolidMasse moléculaire :366.49AM-0466
CAS :AM-0466 has a wide range of applications in life science related research.Formule :C27H19F3N4O4SCouleur et forme :SolidMasse moléculaire :552.52Somatostatin 1-28 acetate
Somatostatin 1-28 acetate circulates in human plasma.Degré de pureté :99.22%Couleur et forme :SoildProstaglandin F2α Alcohol
CAS :Prostaglandin F2α Alcohol is a PGF2α (T15133) analogue. Prostaglandin F2α Alcohol is an orally active prostaglandin F receptor (FP receptor) agonist.Formule :C20H36O4Couleur et forme :SolidMasse moléculaire :340.5Sar-[D-Phe8]-des-Arg9-Bradykinin
CAS :Potent bradykinin B1 agonist, EC50 = 9.02 nM, enzyme resistant, induces hypotension and angiogenesis.Formule :C47H66N12O11Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :975.11Hydroxybupropion
CAS :Hydroxybupropion is the major active metabolite of Bupropion and an antagonist of nACh receptor. Hydroxybupropion inhibits norepinephrine uptake (IC50 = 1.7 μM).Formule :C13H18ClNO2Degré de pureté :99.73%Couleur et forme :Off-White SolidMasse moléculaire :255.74Ref: TM-T11588
1mg89,00€5mg204,00€10mg331,00€25mg545,00€50mg777,00€100mg1.063,00€1mL*10mM (DMSO)232,00€Methdilazine
CAS :Methdilazine: oral antibiotic, histamine antagonist, fights mycobacterium (MIC 5-15 μg/mL) for infectious disease research.Formule :C18H20N2SCouleur et forme :SolidMasse moléculaire :296.43[D-p-Cl-Phe6,Leu17]-VIP
CAS :Selective vasoactive intestinal peptide (VIP) receptor antagonist (IC50 = 125.8 nM). Displays no activity on glucagon, secretin or GRF receptors.Formule :C148H239ClN44O42Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :3342.24Bradykinin (1-7)
CAS :Bradykinin (1-7), an amino-truncated peptide derived from Bradykinin, is a metabolite formed through enzymatic cleavage by endopeptidase.Formule :C35H52N10O9Degré de pureté :98%Couleur et forme :White Lyophilized PowderMasse moléculaire :756.85γ-2-MSH (41-58), amide
CAS :Melanocortin (MC) 3-MSH (Melanocyte-Stimulating Hormone) is believed to signal through the MC 3 receptor.Formule :C74H100N22O15SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :1569.79Tirzepatide hydrochloride
Tirzepatide HCl is a dual GIP and GLP-1 receptor agonist.Formule :C225H349N48O68ClDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :4849.91meta-Fluoxetine (hydrochloride)
CAS :meta-Fluoxetine (hydrochloride) can be used in related research in the field of life sciences. Its product number is T37474 and CAS number is 79088-29-2.Formule :C17H19ClF3NOCouleur et forme :SolidMasse moléculaire :345.79Orexin B, human
CAS :Orexin B, human agonizes Orexin receptors (OX1 Ki=420 nM, OX2 Ki=36 nM), promotes feeding in rats, and is a neuropeptide.Formule :C123H212N44O35SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :2899.34Navafenterol
CAS :AZD-8871, a potential COPD and asthma treatment, may work well with ICS.Formule :C38H42N6O6S2Couleur et forme :SolidMasse moléculaire :742.91(Hyp³)-Bradykinin acetate
(Hyp³)-Bradykinin acetate is an agonist of bradykinin B2 receptor and stimulates inositol phosphate production in cultured human fibroblasts.Formule :C52H77N15O14Degré de pureté :99.46%Couleur et forme :SolidMasse moléculaire :1136.26Galanin (1-15) (porcine, rat)
CAS :N-terminal galanin fragment used to mediate central cardiovascular effectsFormule :C72H105N19O20Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1556.72PD 144418 oxalate
CAS :PD 144418 oxalate: σ1 receptor ligand, Ki=0.08 nM; 1377 nM for σ2, minimal affinity elsewhere; potential antipsychotic.Formule :C20H24N2O5Degré de pureté :98.76%Couleur et forme :SolidMasse moléculaire :372.42Urocortin II, human
Human urocortin (hUcn) II is a new member of the corticotropin-releasing-factor (CRF) family. It selectively binds to the CRF2 receptor.Formule :C194H339N63O54SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :4450.28Methicillin sodium hydrate
CAS :Methicillin sodium hydrate, a narrow-spectrum antibiotic, combats methicillin-resistant Staphylococcus strains and treats various infections.Formule :C17H21N2NaO7SCouleur et forme :SolidMasse moléculaire :420.41NR2E3 agonist 1
CAS :NR2E3 agonist 1 is an NR2E3 agonist with antitumor activity and can be used to study diseases caused by NR2E3 abnormalities.Formule :C24H19ClN4O2Degré de pureté :98.88%Couleur et forme :SoildMasse moléculaire :430.89AMI-193
CAS :AMI-193 (Spiramide) is a selective 5-HT2 & D2 receptor antagonist with antipsychotic properties.Formule :C22H26FN3O2Degré de pureté :99.65%Couleur et forme :SolidMasse moléculaire :383.46Orexin A (human, rat, mouse)
CAS :Orexin A, a 33 AA neuropeptide in humans, rats, mice, influences various processes, studied in pancreatic function and as an OX1R antagonist.Formule :C152H243N47O44S4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :3561.1MM 54
CAS :Potent apelin receptor antagonist (Ki=82 nM, IC50=93 nM), counters [Pyr1]-Apelin-13, inhibits glioblastoma growth in mice.Formule :C70H121N29O15S4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1737.15Pal-Glu(OSu)-OH
CAS :Pal-Glu(OSu)-OH is a Liraglutide side chain, a GLP-1 agonist for type 2 diabetes study.Formule :C25H42N2O7Couleur et forme :SolidMasse moléculaire :482.618ONO-0300302
CAS :ONO-0300302: LPA1 antagonist, treats Benign Prostatic Hyperplasia, IC50 = 0.16 nM, reduces IUP in rats and dogs for 12h.Formule :C29H35NO5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :477.59Terazosin dimer impurity dihydrochloride
CAS :Terazosin dimer impurity dihydrochloride is a chemical byproduct of the α1-antagonist Terazosin, derived from quinazoline.Formule :C24H30Cl2N8O4Couleur et forme :SolidMasse moléculaire :565.46GI-560192
CAS :GI-560192 (RL-0070933), a potent smo modulator, EC50: 0.02µM; affects smoothened in cilia via hedgehog signaling.Formule :C20H16N2O2Degré de pureté :99.53%Couleur et forme :SoildMasse moléculaire :316.35Ref: TM-T64351
1mg85,00€5mg170,00€10mg250,00€25mg371,00€50mg522,00€100mg712,00€200mg954,00€1mL*10mM (DMSO)170,00€PEN (rat)
CAS :PEN (rat) is an Endogenous peptide GPR83 agonist. ProSAAS-derived neuropeptide.Formule :C102H169N27O33Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :2301.62mPGES-1/sEH-IN-1
mPGES-1/sEH-IN-1 (compound 1f) is an sEH inhibitor with an IC50 value of 5 μM. It also exhibits antitumor activity by inhibiting mPGES-1, with an IC50 value of 25 µM.Formule :C20H16F3N3O2Couleur et forme :SolidMasse moléculaire :387.355β-Corticotropin (swine)
CAS :β-Corticotropin (swine), a synthetic analog of the peptide hormone corticotropin (ACTH), induces steroid release [1] [2].Couleur et forme :SolidEP3 antagonist 4
CAS :EP3 antagonist 4: hEP inhibitor, Ki = 2 nM, low clearance, high oral AUC, good bioavailability in rats, potential for diabetes research.Formule :C22H20Cl3FN4O3S2Degré de pureté :98%Couleur et forme :SoildMasse moléculaire :577.91Phoenixin-14 TFA
Phoenixin-14 TFA (PNX-14 TFA) is an endogenous neuropeptide that can modulate GnRH receptor expression and exerts anxiolytic effects.Formule :C75H110N18O20·xC2HF3O2Degré de pureté :99.11%Couleur et forme :SolidMasse moléculaire :1583.78 (free base)d[Cha4]-AVP
CAS :Potent human V1B vasopressin receptor agonist; Ki: V1B=1.2 nM; increases ACTH, corticosterone; low vasopressor effect.Formule :C50H71N13O11S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1094.31ADTN
CAS :ADTN is an agonist of the dopamine receptor.Formule :C10H13NO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :179.22BIIE-0246
CAS :BIIE-0246 is a selective NPY2R antagonist, IC50=15 nM at the rat [125I]PYY3-36 site, reduces NPY-stimulated expression of p-AKT S473 and P-p44/42 MAPK.Formule :C49H57N11O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :896.05ACTH (11-24)
CAS :ACTH (11-24) is an adrenocorticotrophin fragment, stimulates cortisol, and antagonizes ACTH (1-39)/(1-10) in adrenal cells.Formule :C77H134N24O16Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1652.04RWJ 676070
CAS :RWJ 676070 is an antagonist of vasopressin V1A/V2 receptor.Formule :C30H26ClFN2O5Couleur et forme :SolidMasse moléculaire :548.99Bromchlorbuterol hydrochloride
CAS :Bromchlorbuterol HCl, a potent β-agonist, is used to study lung diseases like asthma.Formule :C12H19BrCl2N2OCouleur et forme :SolidMasse moléculaire :358.1Uroguanylin (human)
CAS :Uroguanylin (human) serves as a natural ligand for the Guanylyl Cyclase C (GCC) receptor in metastatic colorectal cancer tumors and exhibits anti-tumor effectsFormule :C64H102N18O26S4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1667.86Phoenixin-14
CAS :Phoenixin-14 (PNX-14), an active endogenous isoform, induces an anxiolytic effect by activating the AHA GnRH system in mice and protects against ischemia/
Formule :C75H110N18O20Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1583.78CB2R agonist 2
CB2R agonist 2 (cis-17-para) is a CB2R agonist [1].Degré de pureté :98%Couleur et forme :Odour SolidSigma-1 receptor antagonist 5
Sigma-1 receptor antagonist 5 (compound 12), a 4-pyridylpiperidine derivative, exhibits analgesic properties through its antagonistic action on sigma receptorsFormule :C26H27N3ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :397.51human GALP (3-32)
Human GALP (3-32) (Galanin-like peptide (3-32)) serves as a high-affinity agonist for galanin receptors GalR1 (IC50 = 33 nM) and GalR2 (IC50 = 15 nM), asFormule :C137H213N43O38SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :3102.495-HT6 agonist 1
Compound 19, a 5-HT6 agonist with an affinity (K i : 5 nM), exhibits antidepressant-like effects and enhances cognitive function while also inhibiting plateletFormule :C17H22Cl2N6SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :413.37AB21 oxalate
AB21 oxalate, a potent and selective S1R antagonist, exhibits binding affinities (Kis) of 13 nM and 102 nM for S1R and S2R, respectively.Formule :C25H30N2O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :438.52Lys-[Des-Arg9]Bradykinin
CAS :Selective bradykinin B1 agonist with Ki 0.12 nM; inactive at B2 (>30,000 nM). Lowers blood pressure, more potent than Des-Arg9-Bradykinin.Formule :C50H73N13O11Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1032.21Muscarinic toxin 3
CAS :Muscarinic toxin 3 (MT3), a potent non-competitive antagonist of mAChR and adrenoceptors, exhibits pIC50 values of 6.71 for M1, 8.79 for M4, 8.86 for α1A, 7.57Formule :C319H489N89O97S8Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :7379.35PSB-1114 triethylamine
PSB-1114 triethylamine is a potent, enzymatically stable, P2Y2 receptor agonist with a 134 nM EC50, exhibiting greater than 50-fold selectivity over P2Y4 (EC50Formule :C10H15F2N3O13P3S·xC6H15NDegré de pureté :98%Couleur et forme :Solidα-CGRP (mouse, rat) TFA
α-CGRP (mouse, rat) TFA, a neuropeptide belonging to the calcitonin gene-related peptide (CGRP) family, is predominantly located at neuromuscular junctions andFormule :C162H262N50O52S2·C2HF3O2Degré de pureté :98%Couleur et forme :SolidEmoghrelin
CAS :Emoghrelin, extracted from Heshouwu (Polygonum multiflorum), promotes the secretion of growth hormone by activating the ghrelin receptor [1].Formule :C24H22O13Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :518.42FFN246
CAS :FFN246, a fluorescent probe, concurrently targets the serotonin transporter (SERT) and vesicular monoamine transporter 2 (VMAT2), exhibiting excitation andFormule :C15H13FN2ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :256.27Arotinolol hydrochloride
CAS :Arotinolol HCl is a non-selective α/β-blocker, anti-hypertensive, anti-obesity, and improves aortic stiffness.Formule :C15H22ClN3O2S3Degré de pureté :99.82%Couleur et forme :SolidMasse moléculaire :408Bay 55-9837
CAS :Selective VPAC2 agonist; EC50: 0.4 nM (VPAC2), 100 nM (VPAC1), >1000 nM (PAC1). Enhances insulin secretion, reduces HIV-1 replication.Formule :C167H270N52O46Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :3742.29ONO-8711
CAS :ONO-8711 is a potent and selective competitive antagonist of EP1 receptor with Kis of 0.6 nM and 1.7 nM for human and mouse EP1, respectively.Formule :C22H30ClNO4SCouleur et forme :SolidMasse moléculaire :440Antipsychotic agent-2
Compound 11: potent antipsychotic, binds 5-HT1A/2A/2C, D2, H1 receptors; K is 56.6-1140 nM, BBB permeable.Formule :C22H26FN5OCouleur et forme :SolidMasse moléculaire :395.47Pafenolol
CAS :Pafenolol is a P-glycoprotein modulator with a Ki value of 5.5 µM. pafenolol is an orally available and selective beta-adrenergic receptor antagonist.Formule :C18H31N3O3Degré de pureté :98.33%Couleur et forme :SolidMasse moléculaire :337.46S1R agonist 2
CAS :S1R agonist 2 is a selective S1R agonist with a Ki of 88 nM for S2R and 1.1 nM for S1R and is protective against ROS and NMDA-induced neurotoxicity.Formule :C21H27NODegré de pureté :99.66%Couleur et forme :SolidMasse moléculaire :309.45CAY10509
CAS :CAY10509 is a PGF2α analogue and acts as an FP receptor inhibitor with an IC50 of 30 nM. It shows potential for use in studying the physiological regulatory mechanisms related to prostaglandins.Formule :C23H35FO5SCouleur et forme :SolidMasse moléculaire :442.58Glucagon-like peptide 1 (1-37), human TFA
Human Glucagon-like peptide 1 (1-37) TFA is a potent GLP-1 receptor agonist derived from proglucagon.Formule :C188H276N51F3O61Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :4283.5Neuromedin N
CAS :Neuromedin N is a neuropeptide derived from the same precursor polypeptide as neurotensin, and with similar but subtly distinct expression and effects.Formule :C38H63N7O8Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :745.95Lys-Bradykinin
CAS :Endogenous bradykinin receptor agonistFormule :C56H85N17O12Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1188.38GIP/GLP-1 dual receptor agonist-1 sodium
GIP/GLP-1 dual receptor agonist-1 (Compound 4) (sodium) functions as a GIP/GLP-1 receptor agonist. This compound is applicable for research into metabolic disorders and liver diseases, including non-alcoholic steatohepatitis (NASH) and non-alcoholic fatty liver disease (NAFLD).Couleur et forme :Odour SolidSulfatroxazole
CAS :Sulfatroxazole (Isosulfafurazole) (compound 12) is a selective antagonist of the ETA receptor with an IC50 of 0.26 μM.Formule :C11H13N3O3SCouleur et forme :SolidMasse moléculaire :267.3TT 232
CAS :sst1/sst4 somatostatin receptors agonistFormule :C45H58N10O9S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :947.13CACPD2011a-0001278239
CAS :CACPD2011a-0001278239 is a β2AR hybrid agonist with high affinity binding to both the wild-type and T164I β2AR variants. It exhibits neither cytotoxicity nor mutagenicity, making it suitable for asthma research.Formule :C21H22N4O4Couleur et forme :SolidMasse moléculaire :394.42Cetirizine Impurity C dihydrochloride
CAS :Cetirizine Impurity C dihydrochloride is a Cetirizine metabolite and long-acting H1-antihistamine.Formule :C21H27Cl3N2O3Couleur et forme :SolidMasse moléculaire :461.81BM213 acetate
BM213 acetate is a selective C5aR1 agonist with antitumor activity that induces C5aR1-mediated calcium mobilization and pERK1/2 signaling.
Formule :C45H74N12O12Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :975.14Galanin (1-29)(rat, mouse)
CAS :Non-selective galanin agonist; Ki: GAL1-0.98, GAL2-1.48, GAL3-1.47 nM. Anticonvulsant, stops full seizures in rats.Formule :C141H211N43O41Degré de pureté :98%Couleur et forme :White Lyophilized PowderMasse moléculaire :3164.499FR252384
CAS :FR252384 is an antagonist of the neuropeptide Y-Y5 receptor (IC50: 2.3 nM).Formule :C18H17N3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :275.35Cannabidivarinic acid
CAS :Cannabidivarinic acid (CBDVA), the carboxylic acid precursor to cannabidivarin (CBDV), is a non-psychoactive cannabinoid found in Cannabis and known for its anti-inflammatory properties.Formule :C20H26O4Couleur et forme :SolidMasse moléculaire :330.42Esmolol acid hydrochloride
CAS :Esmolol acid (ASL-8123) hydrochloride is a mild antagonist of β-adrenergic receptors. It inhibits the heart rate and diastolic pressure responses induced by Isoproterenol in a dose-dependent manner and is applicable for renal failure research.Formule :C15H24ClNO4Couleur et forme :SolidMasse moléculaire :317.81ATMW-2
ATMW-2 is an antagonist engineered using NeuralGenThesis (NGT) technology, specifically targeting the melanocortin 2 receptor (MC2R).Formule :C27H29ClN2O4Couleur et forme :SolidMasse moléculaire :480.98Moperone
CAS :Moperone (R 1658) is an antagonist of both the D2 dopamine receptor (D2 dopamine receptor) and the D3 dopamine receptor (D3 dopamine receptor), with IC50 values for each of 1.0 nM.Formule :C22H26FNO2Couleur et forme :SolidMasse moléculaire :355.45VU0453379 hydrochloride
VU0453379 hydrochloride: selective CNS-penetrant GLP-1R PAM, EC50 1.3 μM.Formule :C26H35ClN4O2Couleur et forme :SolidMasse moléculaire :471.037-Methyl DMT
CAS :7-Methyl DMT (7-TMT) acts as a 5-HT2 receptor agonist. Structurally, it is a tryptamine derivative and serves as an analytical reference for the psychoactive substance DOM. It is also applicable in research related to neurological disorders.Formule :C13H18N2Couleur et forme :SolidMasse moléculaire :202.3Melatonin-Tamoxifen Conjugate
Melatonin-Tamoxifen Conjugate (compound 16c) is an anticancer drug conjugate made of Melatonin and Tamoxifen, serving as an effective antagonist of ERα (IC50 = 863 nM). In cells expressing the hMT1 receptor, it binds to MLT receptors (Ki = 3.1 nM) and exhibits the ability to promote β-arrestin activation (EC50 = 914 nM) and ERK activation (EC50 = 98 nM). The IC50 values for Melatonin-Tamoxifen Conjugate in MCF-7, MDA-MB-231, and HT-1080 cell lines are 6.8 μM, 6.4 μM, and 1.7 μM, respectively.Formule :C47H58N4O4Couleur et forme :SolidMasse moléculaire :742.99V1a/V2 antagonist 1
V1a/V2 antagonist 1 (Compound 18j) is an orally active dual-target antagonist of V1a and V2 receptors, exhibiting high binding affinity toward these receptors [Ki values are hV1a: 0.13 nM, hV2: 0.53 nM, and mV1a: 0.5 nM; IC50 for hV1a is 2.2 nM]. This compound can inhibit oxytocin-induced scratching behavior in mice.Formule :C25H26ClN5O3Couleur et forme :SolidMasse moléculaire :479.9625E-NBOMe hydrochloride
CAS :25E-NBOMe hydrochloride is a derivative of 2C-E, featuring an N-(2-methoxybenzyl) addition to the amine group, and acts as a selective agonist of the 5-HT2A receptor.Formule :C20H28ClNO3Couleur et forme :SolidMasse moléculaire :365.894-Iodoamphetamine hydrochloride
CAS :4-Iodoamphetamine (p-Iodoamphetamine) hydrochloride is a halogenated phenethylamine characterized by the presence of an iodine atom at the para position of the phenyl group. It selectively induces serotonin release and inhibits reuptake in rat brain synaptosomes.Formule :C9H13ClINCouleur et forme :SolidMasse moléculaire :297.56Δ8-THC methyl ether
CAS :Δ8-THC methyl ether (compound 3) demonstrates a strong docking score of -10.167 kcal/mol for the CB2 receptor. Additionally, Δ8-THC methyl ether exhibits antinociceptive activity in mice.Formule :C22H32O2Couleur et forme :SolidMasse moléculaire :328.49Pasireotide (diaspartate)
CAS :Pasireotide diaspartate (SOM230) has high agonist activity at sst1/2/3/5, less at sst4; it's antiproliferative and proapoptotic.Formule :C66H80N12O17Couleur et forme :SolidMasse moléculaire :1313.414-hydroxy DiPT hydrochloride
CAS :4-hydroxy DiPT (hydrochloride) is a 5-HT2A agonist that can induce head twitch response (HTR) in mice, indicating its hallucinogenic potential. This compound holds promise for research into hallucinogens.Formule :C16H25ClN2OCouleur et forme :SolidMasse moléculaire :296.84[18F]-Labeled L-dopa precursor
CAS :[18F]-Labeled L-dopa precursor is a precursor for synthesis of 18F-labeled L-dopa[1].Formule :C35H36N2O7Couleur et forme :SolidMasse moléculaire :596.67SBI-810
CAS :SBI-810 is a functional selective β-arrestin-biased allosteric modulator of the neurotensin receptor 1 (NTSR1). In the presence of the endogenous ligand neurotensin (NT), SBI-810 regulates NTSR1 signaling through a G protein-specific mechanism. It fully antagonizes NT-induced Gq activation and partially antagonizes NT-induced Gi1 activation, allowing NTSR1 to activate GoA and G12.Formule :C27H34N4O2Couleur et forme :SolidMasse moléculaire :446.59CB2 receptor agonist 9
CAS :CB2 receptor agonist 9 (Compound 33) is an orally active agonist of cannabinoid receptor 2 (CB2 receptor) with an EC50 of 16.2 nM. It inhibits the expression of TNF-α, IL-1β, and IL-6, demonstrating anti-inflammatory activity in a DSS-induced acute colitis model in mice.Formule :C16H23N3O2SCouleur et forme :SolidMasse moléculaire :321.44N6-Benzyl-5'-ethylcarboxamido adenosine
CAS :N6-Benzyl-5'-ethylcarboxamido adenosine is a selective A3 adenosine receptor agonist.Formule :C19H22N6O4Couleur et forme :SolidMasse moléculaire :398.42GIP/GLP-1 dual receptor agonist-1
CAS :Compound 4: GIP/GLP-1 agonist for metabolic/fatty liver disease research.Couleur et forme :Solid(±)-9-Nor-9α-hydroxy Hexahydrocannabinol
CAS :(±)-9-Nor-9α-hydroxy Hexahydrocannabinol is a cannabinoid-structured compound that exhibits potent cannabinoid-like activity in both dogs and mice.Formule :C20H30O3Couleur et forme :SolidMasse moléculaire :318.45Bamosiran
CAS :Bamosiran, a small interfering RNA (siRNA), specifically targets the β-adrenergic receptor 2 to reduce intraocular pressure.Couleur et forme :SolidPobilukast
CAS :Pobilukast (SKF 104353) is a cysteinyl leukotriene receptor antagonist that can be used to study limiting myocardial injury in MI/R rats.Formule :C26H34O5SDegré de pureté :99.65% - 99.84%Couleur et forme :SolidMasse moléculaire :458.61Human growth hormone-releasing factor
CAS :GHRH from the hypothalamus prompts the pituitary to produce/release GH by attaching to the GHRHR.Formule :C215H358N72O66SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :5039.65N-Nitroso Atenolol
CAS :N-Nitroso Atenolol is a derivative of Atenolol. At concentrations ranging from 0.1 to 1 mM, it induces DNA fragmentation in rat hepatocytes.Formule :C14H21N3O4Couleur et forme :SolidMasse moléculaire :295.33Alosetron-d3
CAS :Alosetron D3 (GR 68755 D3) is a deuterium-labeled Alosetron. Alosetron is an antagonist of 5HT3-receptor.Formule :C17H18N4ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :297.3715(S)-HpEPE
CAS :15(S)-HpEPE, a monohydroperoxy fatty acid, forms when 15-lipoxygenase acts on EPA, with expected biological activities akin to 15(S)-HpETE.Formule :C20H30O4Couleur et forme :SolidMasse moléculaire :334.456Albenatide
CAS :Albenatide is a modified analog of exendin 4 conjugated to recombinant human albumin.
Formule :C26H47N7O9SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :633.76CB2R/FAAH modulator-3
CAS :CB2R/FAAH modulator-3 (compound 27) is a modulator targeting at CB2R and FAAH.Formule :C22H31NO2Degré de pureté :99.81%Couleur et forme :SoildMasse moléculaire :341.49Satavaptan
CAS :Satavaptan is a vasopressin V2 receptor antagonist. Satavaptan improves the control of ascites in cirrhosis.Formule :C33H45N3O8SCouleur et forme :SolidMasse moléculaire :643.79Norisoboldine hydrochloride
CAS :Norisoboldine hydrochloride: an oral AhR agonist from Radix Linderae, for Rheumatoid arthritis and Ulcerative colitis research.Formule :C18H20ClNO4Couleur et forme :SolidMasse moléculaire :349.81GLP-1(7-37)
CAS :GLP-1 (7-37) is a truncated, bioactive form of GLP-1 that is the product of proglucagon processing in intestinal endocrine L cells.Formule :C151H228N40O47Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :3355.67(S)-Osanetant
CAS :(S)-Osanetant, an S-enantiomer, is a selective NK3 antagonist with potential for treating schizophrenia and has anxiolytic and antidepressant effects.Formule :C35H41Cl2N3O2Couleur et forme :SolidMasse moléculaire :606.62RC-3095 TFA
CAS :RC-3095 TFA (RC-3095 (TFA)) is a bombesin/gastrin-releasing peptide (BN/GRP) antagonist with potential anticancer activity.Formule :C58H80F3N15O11Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1220.34KSK67
CAS :KSK67 is a selective dual antagonist of sigma-2 and histamine H3 receptors with inhibitory effects on H3 receptors, sigma-1, and sigma-2 receptors, with KiFormule :C22H27N3O2Degré de pureté :99.94%Couleur et forme :SoildMasse moléculaire :365.47SB 258585
CAS :SB 258585: Selective 5-HT6 antagonist, binds human receptors, used in cognitive and antipsychotic assays.Formule :C18H22IN3O3SDegré de pureté :99.77%Couleur et forme :SoildMasse moléculaire :487.36H4R antagonist 3
CAS :H4R antagonist 3 is a novel histamine-4 receptor (H4R) antagonist with an EC50 <10 mM.H4R antagonist 3 has potential inflammatory activity for the study ofFormule :C19H21ClN4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :372.92CB2R/FAAH modulator-2
CAS :CB2R/FAAH modulator-2 (compound 26) is a dual modulator targeting at CB2R and FAAH.Formule :C24H33NO2Degré de pureté :99.15%Couleur et forme :SoildMasse moléculaire :367.52WAY-620645
CAS :WAY-620645 is a CCK antagonist with antitumor and analgesic activities.Formule :C22H22N4O2Degré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :374.44Ref: TM-T9991
1mg38,00€5mg85,00€10mg111,00€25mg224,00€50mg318,00€100mg462,00€200mg627,00€1mL*10mM (DMSO)104,00€PD-149164
CAS :PD-149164 is an agonist of the CCK-A receptor.Formule :C33H38FN3O5Couleur et forme :SolidMasse moléculaire :575.67JNJ-5207787
CAS :JNJ-5207787, a blood-brain barrier-crossing Y2 receptor antagonist, is >100x selective against Y1/Y4/Y5 and inhibits human/rat Y2 with pIC50s of 7.0/7.1.Formule :C32H38N4O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :510.67CRL-42872 free base
CAS :CRL-42872 free base is a bioactive chemical.Formule :C22H26N6O6SCouleur et forme :SolidMasse moléculaire :502.54Azepexole hydrochloride
CAS :Azepexole hydrochloride (4H-Oxazolo[4,5-d]azepin-2-amine, 6-ethyl-5,6,7,8-tetrahydro-, hydrochloride (1:1)) is a potent α2-Adrenoceptor agonist with anaestheticFormule :C9H16ClN3ODegré de pureté :99.88% - 99.89%Couleur et forme :SoildMasse moléculaire :217.7GLP-1R Agonist DMB
CAS :GLP-1R Agonist DMB is an agonist of glucagon-like peptide 1 receptor (GLP-1R; KB = 26.3 nM for the recombinant human receptor).Formule :C13H15Cl2N3O2SDegré de pureté :99.52%Couleur et forme :SolidMasse moléculaire :348.25[D-Trp8]-γ-MSH
CAS :[D-Trp8]-γ-MSH is a selective melanocortin 3 (MC3) receptor agonist (IC50 values are 6.7, 340 and 600 nM for human MC3, MC5 and MC4 receptors respectively).Formule :C74H99N21O16SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :1570.79Neuropeptide Y5 receptor ligand-1
CAS :Neuropeptide Y5 receptor ligand-1 (Compound 54), a carbazole derivative, acts as a powerful antagonist to the neuropeptide Y5 (NPY-5) receptor [1].Formule :C19H17N3O2Couleur et forme :SolidMasse moléculaire :319.36GB-110 hydrochloride
GB-110 HCl: potent, nonpeptidic oral PAR2 agonist; triggers Ca2+ release in HT29 cells; EC50 0.28 μM.Formule :C33H49ClN6O5Couleur et forme :SolidMasse moléculaire :645.23Bz-Dab(nbd)-awfpp-nle-NH2
CAS :Bz-Dab(nbd)-ala-trp-phe-pro-pro-nle-NH2 is a fluorescent NK2 antagonist.Formule :C56H65N13O11Couleur et forme :SolidMasse moléculaire :1096.2HTL22562
CAS :HTL22562 is a calcitonin gene-related peptide (CGRP) receptor antagonist for acute treatment of migraine.Formule :C40H49N11O5Couleur et forme :SolidMasse moléculaire :763.904Ramelteon metabolite M-II
CAS :Ramelteon M-II binds MT1/MT2 with IC50s: 208/1470 pM; it's the main metabolite and a melatonin receptor agonist.Formule :C16H21NO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :275.34Minaprine
CAS :Minaprine is a reversible inhibitor of MAO-A, used in the treatment of various depressive states.Formule :C17H22N4ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :298.38Motapizone
CAS :Motapizone (NAT 05-239) is a selective PDE3 inhibitor that suppresses cytokine release, increases intracellular cAMP, and inhibits human platelet aggregation.Formule :C12H12N4OSDegré de pureté :95.26%Couleur et forme :SolidMasse moléculaire :260.32KB-5492 FA
KB-5492 FA is a selective sigma receptor inhibitor with antiulcerogenic effects.CAS 번호128-52-56-8Formule :C24H32N2O8Degré de pureté :98.12%Couleur et forme :SolidMasse moléculaire :476.52Substance P (1-9)
CAS :Substance P (1-9), a nonapeptide, slows its own inactivation and stimulates neurons.Formule :C52H77N15O12Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1104.26Azirkitug
Azirkitug is a humanized IgG1κ antibody targeting CCR8, with HumanIgG1kappa, Isotype Control serving as its corresponding isotype control.Couleur et forme :Odour LiquidDenrakibart
Denrakibart is a humanized IgG2κ antibody targeting CCL17, with HumanIgG2kappa, Isotype Control serving as the corresponding isotype control.Couleur et forme :Odour LiquidCCR2 antagonist 1
CAS :CCR2 antagonist 1 is a high-affinity and long-residence-time antagonist of CCR2 (Ki: 2.4 nM).Formule :C28H32BrF3N2OCouleur et forme :SolidMasse moléculaire :549.47Neuropeptide Y 13-36 (porcine)
CAS :Neuropeptide Y 13-36 (porcine) is a selective neuropeptide Y2 receptor agonist.Formule :C135H209N41O36Couleur et forme :SolidMasse moléculaire :2982.408Org 13011
CAS :Org 13011 has CNS activity and induces conditioned taste aversion by mediating 5-HT 1A receptors.Formule :C18H25F3N4ODegré de pureté :98.02%Couleur et forme :SoildMasse moléculaire :370.41Ref: TM-T28258L
1mg109,00€5mg261,00€10mg374,00€25mg583,00€50mg803,00€100mg1.063,00€200mg1.431,00€1mL*10mM (DMSO)266,00€CCR8 antagonist 1
CAS :CCR8 antagonist 1 is an antagonist of C-C Motif Chemokine Receptor 8 (CCR8) with a Ki value of 1.6 nM.Formule :C26H29N3O5SDegré de pureté :99.51%Couleur et forme :SolidMasse moléculaire :495.59[Ala11,D-Leu15]-Orexin B acetate
[Ala11,D-Leu15]-Orexin B acetate is a selective agonist of orexin-2 receptor (OX2) with an EC50 of 0.13 nM, showing 400-fold selectivity over OX1 (52 nM).Formule :C122H210N44O37SDegré de pureté :98.18%Couleur et forme :SolidMasse moléculaire :2917.31Lanepitant 2HCl
CAS :Lanepitant 2HCl is a non-peptide neurokinin-1 receptor antagonist that can be used to study painful neuropathy-like disorders such as migraine.Formule :C33H47Cl2N5O3Degré de pureté :98.67%Couleur et forme :SolidMasse moléculaire :632.66Orexin B, rat, mouse
CAS :Orexin B, rat, mouse is an endogenous agonist at Orexin receptor with Kis of 420 and 36 nM for OX1 and OX2, respectively.Formule :C126H215N45O34SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :2936.45Cafelkibart
Cafelkibart is a chimeric IgG1κ monoclonal antibody targeting CCR8, with HumanIgG1kappa, Isotype Control serving as its corresponding isotype control.Couleur et forme :Odour LiquidTagmokitug
CAS :Tagmokitug is a humanized IgG1κ monoclonal antibody inhibitor targeting CCR8. It exhibits anti-tumor activity and is applicable in cancer immunotherapy research, including studies on breast cancer, colon cancer, and lung cancer.8-iso Prostaglandin E2
CAS :"8-iso PGE2: Isoprostane from arachidonic acid, potent rat renal vasoconstrictor, reduces GFR and renal flow by 80%, no BP effect."Formule :C20H32O5Couleur et forme :SolidMasse moléculaire :352.47PSB-SB-1203
CAS :PSB-SB-1203 (Compound 25b) is a dual CB1/CB2 ligand that blocks the CB1 receptor and activates the CB2 receptor with a CB1 Ki of 0.244 μM, a CB2 Ki of 0.210 μM, and an EC50 of 0.054 μM. It shows potential for research in obesity and cancer.Formule :C25H30O4Couleur et forme :SolidMasse moléculaire :394.5CCR6 antagonist 2
CCR6 antagonist2 (Compound 20c) acts as a CCR6 antagonist with a Ki of 1.1 nM. It inhibits CCL20-induced calcium influx with an IC50 of 4.9 nM and suppresses the chemotactic migration of CCR6+ T cells with an IC50 of 190 nM.Formule :C19H24N4O4Couleur et forme :SolidMasse moléculaire :372.42BE-24566B
CAS :BE-24566B, a polyketide from S. violaceusniger, inhibits various bacteria and blocks ET receptors (ETA IC50=11 μM, ETB=3.9 μM).Formule :C27H24O7Couleur et forme :SolidMasse moléculaire :460.4825-HT6R antagonist 6
5-HT6R antagonist 6 (Compound PP15) exhibits high affinity and selectivity for the 5-HT6R receptor, with a Ki of 42 nM. It demonstrates weak antiproliferative activity on tumor cells and low toxicity toward normal cells. 5-HT6R antagonist 6 is applicable in tumor research.Formule :C24H26N4O2SCouleur et forme :SolidMasse moléculaire :434.55Tirzepatide
CAS :Tirzepatide (LY-3298176) is a dual glucose-dependent polypeptide (GIP) (EC50=0.042 nM) and glucagon-like peptide-1 (GLP-1) (EC50=0.086 nM) receptor agonist.Formule :C225H348N48O68Degré de pureté :99.52% - 99.99%Couleur et forme :SolidMasse moléculaire :4813.45PG 931 acetate
PG 931 acetate is a potent agonist of melanocortin 4 (MC4) receptors.
Formule :C61H89N15O13Degré de pureté :98.74%Couleur et forme :SolidMasse moléculaire :1240.45Ornipressin
CAS :Ornipressin is a vasoconstrictor, haemostatic and renal agent.Formule :C45H63N13O12S2Degré de pureté :98%Couleur et forme :White PowderMasse moléculaire :1042.19Apigenin 6,8-di-C-α-L-arabinopyranoside
CAS :Apigenin 6,8-di-C-alpha-L-arabinopyranoside is a useful organic compound for research related to life sciences.Formule :C25H26O13Couleur et forme :SolidMasse moléculaire :534.47CAY10597
CAS :PGD2 effects via DP1/CRTH2/DP2 receptors; CAY10597 blocks CRTH2/DP2 (Ki=37nM), R enantiomer stronger (Ki=23-22nM), inhibits eosinophil migration (IC50=40nM).
Formule :C20H14ClFN2O5Couleur et forme :SolidMasse moléculaire :416.79D-Epinephrine
CAS :D-Epinephrine: a hormone and drug, boosts heart rate, muscle blood flow, pupil size, and sugar levels in stress responses.
Formule :C9H13NO3Couleur et forme :SolidMasse moléculaire :183.2[Tyr3]Octreotate
CAS :[Tyr3]Octreotate is a long peptide compound containing 8 amino acids and is a functional DOTA chelating agent with covalent bonds.Formule :C49H64N10O12S2Degré de pureté :98.21%Couleur et forme :SoildMasse moléculaire :1049.22CRSP-1
CAS :Central CT receptor agonist, 350x stronger than CT, no CGRP or adrenomedullin action, inhibits osteoclasts, affects rat feeding, body temp, and calcium.Formule :C175H294N54O49S5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :4098.88AL 34662
CAS :AL 34662 is a selective and potent 5-HT2A receptor agonist with IC50s of 0.77 nM and 1.5 nM for rat and human 5-HT2 receptors, respectively.AL 34662 is also aFormule :C10H13N3ODegré de pureté :99.97%Couleur et forme :SolidMasse moléculaire :191.23Nemifitide diTFA
CAS :Nemifitide diTFA is a synthetic pentapeptide with antidepressant properties, resembling MIF, that crosses the blood-brain barrier.Formule :C37H45F7N10O10Degré de pureté :99.78% - 99.84%Couleur et forme :SolidMasse moléculaire :922.8Neuropeptide Y (1-24) (human)
CAS :Neuropeptide Y (1-24) inhibits rat vas deferens twitch and activates NMDA-induced neurons in rat hippocampus.Formule :C116H170N30O40SCouleur et forme :SolidMasse moléculaire :2656.835-trans Latanoprost (free acid)
CAS :Latanoprost, a prodrug eye drop, turns into active acid inside the body and treats high eye pressure. Its trans isomer also likely reduces eye pressure.Formule :C23H34O5Couleur et forme :SolidMasse moléculaire :390.52Prolactin-Releasing Peptide (12-31), rat
CAS :Prolactin-Releasing Peptide (12-31), rat, a fragment of PrRP, exhibits high affinity for GPR10 receptors and stimulates calcium mobilization in CHOK1 cellsFormule :C104H158N32O26Couleur et forme :SolidMasse moléculaire :2272.571,2,3-Trilinoelaidoyl-rac-glycerol
CAS :1,2,3-Trilinoelaidoyl-glycerol is a TAG with linoelaidic acid; reduces rat serum thromboxane B2, PGF2, and PGE.Formule :C57H98O6Couleur et forme :SolidMasse moléculaire :879.4051-Octadecyl Lysophosphatidic Acid
CAS :1-Octadecyl LPA, an LPA analog with stearic acid at sn-1, has strong platelet aggregation (EC50=9 nM) via G protein receptors.Formule :C21H45O6PCouleur et forme :SolidMasse moléculaire :424.5594-Oxo-5-phenylpentanoic aci
CAS :4-Oxo-5-phenylpentanoic aci is a useful organic compound for research related to life sciences. The catalog number is T125056 and the CAS number is 3183-15-1.Formule :C11H12O3Couleur et forme :SolidMasse moléculaire :192.214LysoPalloT-NH-amide-C3-ph-m-O-C11
CAS :LysoPalloT-NH-amide-C3-ph-m-O-C11 is an agonist of the GPR174 receptor with an EC50 value of 34 nM.Formule :C27H47N2O9PCouleur et forme :SolidMasse moléculaire :574.64Neuronostatin-13 (human)
CAS :Neuronostatin-13: human-conserved, 13-amino-acid peptide with amidated C-terminus.Formule :C64H110N20O16Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1415.68Mitemcinal fumarate
CAS :Mitemcinal fumarate is a erythromycin derivative that is used to treat gastroesophageal reflux disease.Formule :C84H142N2O28Couleur et forme :SolidMasse moléculaire :1628.02CH-0076989
CAS :CH-0076989 is a chemokine receptor CCR3 agonist.Formule :C24H22Br2N2O2Couleur et forme :SolidMasse moléculaire :530.25Formoterol O-β-D-Glucuronide
CAS :Formoterol O-β-D-glucuronide is a metabolite of formoterol .Formule :C25H32N2O10Couleur et forme :SolidMasse moléculaire :520.535Mirtazapine N-oxide
CAS :Mirtazapine N-oxide, a mirtazapine metabolite, is produced by CYP1A2 and CYP3A4 in human liver.Formule :C17H19N3OCouleur et forme :SolidMasse moléculaire :281.359Nesiritide
CAS :Nesiritide, recombinant human B-type natriuretic peptide, binds NPR-A/C with Kd 7.3/13 pM.Formule :C143H244N50O42S4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :3464.04Fpl 14294
CAS :Fpl 14294 is a novel CCK-8 agonist with effective intranasal anorectic activity in the rat.Formule :C45H56N8O13S3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1013.17Velmupressin acetate
CAS :Potent, selective, short-acting peptidic V2R agonist; EC50: 0.07 nM (hV2R), 0.02 nM (rV2R).Formule :C44H64ClN11O10S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1006.6316,16-dimethyl Prostaglandin F2α
CAS :16,16-dimethyl Prostaglandin F2α can be used in related research in the field of life sciences. Its product number is T37993 and CAS number is 39746-23-1.Formule :C22H38O5Couleur et forme :SolidMasse moléculaire :382.541(+)-ORM-10921
CAS :(+)-ORM-10921 is a conformation of ORM-10921 and can be used in chemical synthesis studies.Formule :C18H23NO2Degré de pureté :99.23%Couleur et forme :SoildMasse moléculaire :285.38Ularitide
CAS :Ularitide is a 32-amino acid peptide from ANP prohormone, resistant to dog kidney cortex peptidase.Formule :C145H234N52O44S3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :3505.97Calcitonin (8-32), salmon
CAS :Calcitonin (8-32), salmon: selective amylin receptor antagonist, regulates calcium/phosphorus, thyroid origin, 32-aa peptide.Formule :C119H198N36O37Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :2725.06PSA1 (141-150)
CAS :This Prostate Specific Antigen 1 peptide was used in the immunotherapy of cancer experiments.Formule :C55H93N13O13SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :1176.47
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