
Inhibiteurs
Les inhibiteurs sont des molécules qui se lient aux enzymes, récepteurs ou autres protéines pour réduire ou bloquer leur activité biologique. Ces composés sont largement utilisés en recherche pour étudier les voies biologiques, comprendre les mécanismes des maladies et développer des médicaments thérapeutiques. Les inhibiteurs jouent un rôle crucial dans le traitement de diverses maladies, y compris le cancer, les maladies cardiovasculaires et les infections. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de haute qualité pour soutenir vos recherches en biochimie, biologie cellulaire et développement pharmaceutique.
Sous-catégories appartenant à la catégorie "Inhibiteurs"
- Angiogenèse(2.519 produits)
- Apoptose(5.786 produits)
- Cycle cellulaire/point de contrôle(4.444 produits)
- Chromatine/Épigénétique(2.235 produits)
- Signalisation du cytosquelette(1.382 produits)
- Altération de l'ADN/réparation de l'ADN(2.823 produits)
- Endocrinologie/Hormones(3.499 produits)
- Enzyme(3.639 produits)
- GPCR/G-Protéine(8.314 produits)
- Immunologie et Inflammation(3.516 produits)
- Virus de la grippe(296 produits)
- Signalisation JAK/STAT(404 produits)
- Signalisation MAPK(1.199 produits)
- Transporteur membranaire/Canal ionique(2.786 produits)
- Métabolisme(9.417 produits)
- Microbiologie/Virologie(6.967 produits)
- Neuroscience(9.920 produits)
- Autres inhibiteurs(37.931 produits)
- Oxydation-Réduction(41 produits)
- Signalisation PI3K/Akt/mTOR(1.399 produits)
- Protéases/Protéasome(1.596 produits)
- Cellules souche et Dérivés(832 produits)
- Tyrosine Kinase/Adaptateurs(2.015 produits)
- Ubiquitination(1.646 produits)
Affichez 16 plus de sous-catégories
66627 produits trouvés pour "Inhibiteurs"
Trier par
Degré de pureté (%)
0
100
|
0
|
50
|
90
|
95
|
100
Sulfo-NHS-Biotin
CAS :<p>Sulfo-NHS-Biotin: water-soluble for biotinylation, targets cell proteins, aids in protein detection with Streptavidin.</p>Formule :C14H18N3NaO8S2Degré de pureté :98.69% - 99.92%Couleur et forme :SolidMasse moléculaire :443.42Vandetanib hydrochloride
CAS :<p>Vandetanib hydrochloride is an oral VEGFR2 inhibitor with an IC50 of 40 nM, also targeting VEGFR3 (110 nM) and EGFR (500 nM).</p>Formule :C22H25BrClFN4O2Couleur et forme :SolidMasse moléculaire :511.81Amezinium methylsulfate
CAS :<p>Amezinium methylsulfate (Lu-1631) has multiple mechanisms, including stimulation of α and β-1 receptors and inhibition of noradrenaline and tyramine uptake.</p>Formule :C12H15N3O5SDegré de pureté :99.64%Couleur et forme :SolidMasse moléculaire :313.333-Methyladipic acid
CAS :<p>3-Methyladipic acid: a final metabolite in phytanic acid degradation, excreted in urine, especially in ARD patients who lack alternate pathways.</p>Formule :C7H12O4Degré de pureté :99.87%Couleur et forme :SolidMasse moléculaire :160.17Laurolitsine
CAS :<p>Laurolitsine ((+)-Norboldine), an alkaloid, is extracted from the leaves of Peumus boldus Molina.</p>Formule :C18H19NO4Degré de pureté :99.39%Couleur et forme :SolidMasse moléculaire :313.35Flupentixol dihydrochloride
CAS :<p>Flupentixol dihydrochloride is used in therapy of schizophrenia as well as in anxiolytic and depressive disorders.</p>Formule :C23H27Cl2F3N2OSDegré de pureté :98.76% - >99.99%Couleur et forme :White Or Off-White SolidMasse moléculaire :507.43OJV-VI
CAS :<p>OJV-VI is a natural product found in ophiopogonis.</p>Formule :C44H70O16Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :855.02Phlorizin dihydrate
CAS :<p>1. Phlorizin dihydrate (Phloridzin dihydrate) can significantly inhibit oxidative DNA damage.</p>Formule :C21H26O11Degré de pureté :97.21%Couleur et forme :Solid CrystallineMasse moléculaire :454.42AMG-131 besylate
CAS :<p>AMG-131 besylate: Hypoglycemic, potent partial PPARγ agonist, lowers glucose in diabetic rodents with fewer side effects than TZDs.</p>Formule :C27H18Cl4N2O6S2Couleur et forme :SolidMasse moléculaire :672.37Ganoderic acid D
CAS :<p>Ganoderic acid D, a Ganoderma component, inhibits HeLa cell growth with an IC50 of 17.3µM after 48h.</p>Formule :C30H42O7Degré de pureté :98.06% - 99.98%Couleur et forme :SolidMasse moléculaire :514.65Dehydroeburicoic acid monoacetate
CAS :<p>Dehydroeburicoic acid monoacetate (3-O-Acetyldehydroeburicoic acid) is a triterpenoid of lanolin isolated from Wolfiporia cocos.</p>Formule :C33H50O4Degré de pureté :96.47%Couleur et forme :SolidMasse moléculaire :510.75Polymyxin B nonapeptide acetate
<p>Polymyxin B nonapeptide acetate, a low toxicity derivative of polymyxin B, disrupts Gram-negative bacteria membranes.</p>Formule :C45H78N14O13Degré de pureté :97.63% - 98.55%Couleur et forme :SolidMasse moléculaire :1023.19GSK-4716
CAS :<p>GSK4716 is an ERRβ/γ agonist (IC50 = 2 μM) that can activate the receptor with similar potency as the protein ligand</p>Formule :C17H18N2O2Degré de pureté :99.53%Couleur et forme :SolidMasse moléculaire :282.34Thiazole Orange
CAS :<p>Thiazole Orange is a dye that can be used for reticulocyte analysis.</p>Formule :C26H24N2O3S2Degré de pureté :99.29% - 99.93%Couleur et forme :SolidMasse moléculaire :476.61Santonin
CAS :<p>Santonin (alpha-Santonin) is a potent antiparasitic agent.</p>Formule :C15H18O3Degré de pureté :99.43% - 99.8%Couleur et forme :SolidMasse moléculaire :246.3PMEDAP
CAS :<p>PMEDAP is a potent inhibitor of Moloney murine sarcoma virus (MSV)-induced tumor formation and associated mortality and an inhibitor of human immunodeficiency</p>Formule :C8H13N6O4PDegré de pureté :99.77%Couleur et forme :SolidMasse moléculaire :288.2BDP5290
CAS :<p>BDP5290 is a potent inhibitor of both ROCK and MRCK(IC50s of 5 nM, 50 nM, 10 nM and 100 nM for ROCK1, ROCK2, MRCKα and MRCKβ, respectively.)</p>Formule :C17H18ClN7ODegré de pureté :97.22%Couleur et forme :SolidMasse moléculaire :371.825-Methoxysalicylic acid
CAS :<p>5-Methoxysalicylic acid (5-MeOSA), a natural product, serves as an effective matrix for oligonucleotide analysis in MALDI MS when used alongside spermine.</p>Formule :C8H8O4Degré de pureté :97.38%Couleur et forme :SolidMasse moléculaire :168.15BC-1258
CAS :<p>BC-1258 is a unique small molecule F-box/LRR-repeat protein 2 (FBXL2) activator.</p>Formule :C22H22N4S2Degré de pureté :97.48% - 99.64%Couleur et forme :SolidMasse moléculaire :406.57Galunisertib
CAS :<p>Galunisertib (LY2157299) is a selective TGF-β receptor type I (TGF-βRI) inhibitor. Galunisertib has antitumor activity. Cost-effective and quality-assured.</p>Formule :C22H19N5ODegré de pureté :97.09% - 99.98%Couleur et forme :SolidMasse moléculaire :369.42L(+)-Leucinol
CAS :<p>L(+)-Leucinol is a potent inhibitor of leucine aminopeptidase.</p>Formule :C6H15NODegré de pureté :98%Couleur et forme :Clear Colorless To Slightly Yellow LiquidMasse moléculaire :117.19JHU37160
CAS :<p>JHU37160 is a DREADD agonist with Ki of 1.9 nM for hM3Dq, 3.6 nM for hM4Di, and EC50 of 18.5 nM (hM3Dq), 0.2 nM (hM4Di) in HEK-293 cell assays.</p>Formule :C19H20ClFN4Degré de pureté :99.87%Couleur et forme :SolidMasse moléculaire :358.84LB-60-OF61 hydrochloride
CAS :<p>LB-60-OF61 hydrochloride is a potent NAMPT enzyme inhibitor with cytotoxic effects, targeting MYC-overexpressing cell lines.</p>Formule :C29H31ClN6O2Couleur et forme :SolidMasse moléculaire :531.06Ondansetron
CAS :<p>Ondansetron (GR 38032) is a serotonin 5-HT3 receptor antagonist used mainly as an antiemetic.</p>Formule :C18H19N3ODegré de pureté :99.92%Couleur et forme :White To Yellow CrystalsMasse moléculaire :293.362"-O-Galloylhyperin
CAS :<p>2"-O-Galloylhyperin (FT-0689359) found in Pyrola. It increases ruminal fiber fermentability by formed wall-bound lignin in primary maize cell walls.</p>Formule :C28H24O16Degré de pureté :98.79% - 99.32%Couleur et forme :SolidMasse moléculaire :616.48YM976
CAS :<p>YM976 is an orally active PDE4 inhibitor (IC50:2.2 nM)</p>Formule :C17H16ClN3ODegré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :313.78MYLS22
CAS :<p>MYLS22: selective OPA1 inhibitor, halts tumor growth & angiogenesis, affects NFkB & gene expression, anti-cancer properties.</p>Formule :C24H21N5O2SDegré de pureté :98.82% - 99.77%Couleur et forme :SolidMasse moléculaire :443.52Cyclo(his-pro)
CAS :<p>Cyclo(his-pro) is a cyclic dipeptide that shields against oxidative damage by activating Nrf2.</p>Formule :C11H14N4O2Degré de pureté :99.87%Couleur et forme :SolidMasse moléculaire :234.25SR-18292
CAS :<p>SR-18292 inhibits PGC-1α, enhances acetylation, lowers gluconeogenesis, and cuts hepatic glucose production.</p>Formule :C23H30N2O2Degré de pureté :99.16% - 99.91%Couleur et forme :SolidMasse moléculaire :366.5VU0134992
CAS :<p>VU0134992 is an Kir4.1 blocker with an IC50 value of 0.97 μM</p>Formule :C20H31BrN2O2Degré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :411.38DIM-C-pPhOCH3
CAS :<p>DIM-C-pPhOCH3 (C-DIM5) is a Nerve Growth Factor-Induced Bα (NGFI-Bα, Nur77) agonist</p>Formule :C24H20N2ODegré de pureté :99.69%Couleur et forme :SolidMasse moléculaire :352.43CLP290
CAS :<p>CLP290 is an activator of the neuron-specific K+-Cl cotransporter KCC2 and displays potential for the treatment of a wide range of neurological and psychiatric</p>Formule :C19H21FN4O3SDegré de pureté :99.93% - >99.99%Couleur et forme :SolidMasse moléculaire :404.46SRS11-92
CAS :<p>SRS11-92 (AA9) is a ferroptosis inhibitor and a derivative of ferrostatin-1</p>Formule :C22H28N2O2Degré de pureté :98.58%Couleur et forme :SolidMasse moléculaire :352.47Doxycycline (hyclate)
CAS :<p>Doxycycline hyclate (WC2031) is a synthetic tetracycline derivative with similar antimicrobial activity. Doxycycline hyclate is also an inhibitor of MMP.</p>Formule :C22H24N2O8·HClC2H6OH2ODegré de pureté :97.48% - >99.99%Couleur et forme :Yellow Crystallien PowderMasse moléculaire :512.90MID-1
CAS :<p>MID-1 is an inhibitor of MG53-IRS-1 (Mitsugumin 53-Insulin Receptor Substrate-1) interaction.</p>Formule :C12H11N3O4SDegré de pureté :99.39%Couleur et forme :SolidMasse moléculaire :293.3Bisdemethoxycurcumin
CAS :<p>Bisdemethoxycurcumin (Curcumin III) is a natural demethoxy derivative of curcumin. Bisdemethoxycurcumin is a potent activator of macrophage phagocytosis.</p>Formule :C19H16O4Degré de pureté :99.34% - 99.75%Couleur et forme :SolidMasse moléculaire :308.33HA 155
CAS :<p>HA 155 (Autotaxin Inhibitor IV) is a boronic acid-based compound, inhibiting ATX with IC50 of 5.7 nM by selectively binding to its catalytic threonine.</p>Formule :C24H19BFNO5SDegré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :463.29Clomifene hydrochloride
CAS :<p>Clomifene hydrochloride: an oral, safe, easy-use drug to induce ovulation for infertility treatment.</p>Formule :C26H29Cl2NOCouleur et forme :SolidMasse moléculaire :442.42PQR530
CAS :<p>PQR530, a potent dual PI3K/mTORC1/2 inhibitor, blocks PKB and pS6 phosphorylation (IC50: 0.07 μM) and has antitumor properties.</p>Formule :C18H23F2N7O2Degré de pureté :99.5%Couleur et forme :SolidMasse moléculaire :407.42Pyridoxal 5'-phosphate hydrate
CAS :<p>Pyridoxal 5'-phosphate hydrate (PLP)(1:x), the active form of vitamin B6, is a cofactor for many different enzymes involved in transamination reactions,</p>Formule :C8H10NO6PDegré de pureté :97.52%Couleur et forme :SolidMasse moléculaire :247.14Daurisoline
CAS :<p>Daurisoline ((R,R)-Daurisoline) is a hERG inhibitor. Daurisoline is also an autophagy blocker.</p>Formule :C37H42N2O6Degré de pureté :98% - 99.96%Couleur et forme :Light Yellow PowderMasse moléculaire :610.74RS-25344 hydrochloride
CAS :<p>RS 25344 hydrochloride is a phosphodiesterase (PDE) 4 inhibitor</p>Formule :C19H14ClN5O4Degré de pureté :99.25%Couleur et forme :SolidMasse moléculaire :411.8α-Cyano-4-hydroxycinnamic acid
CAS :<p>α-Cyano-4-hydroxycinnamic acid (α-Cyano-4-hydroxycinnamic acid(α-CHCA)) (α-CHCA) is an inhibitor of monocarboxylate transporter 1 (MCT1) that blocks pyruvate</p>Formule :C10H7NO3Degré de pureté :99.8% - 99.86%Couleur et forme :PowderMasse moléculaire :189.17Fraxinol
CAS :<p>Fraxinol, a metabolite, is derived from 5,7-dimethoxy-2H-chromen-2-one by CYP enzymes through aromatic hydroxylation.</p>Formule :C11H10O5Degré de pureté :≥95%Couleur et forme :SolidMasse moléculaire :222.19NAI
CAS :<p>NAI (5S rRNA modificator 2) is an RNA SHAPE reagent.</p>Formule :C10H9N3ODegré de pureté :99.5%Couleur et forme :SolidMasse moléculaire :187.2BFMO (biogenic Fe-Mn oxides)
CAS :<p>BFMO reduces Fe(II), Mn(II), As(III&V) levels and removes As in high Fe(II) & Mn(II) water.</p>Formule :C12H12N2O4Degré de pureté :99.4%Couleur et forme :SolidMasse moléculaire :248.23Tiadinil
CAS :<p>Tiadinil, a plant activator of systemic acquired resistance, boosts the production of herbivore-induced plant volatiles.</p>Formule :C11H10ClN3OSDegré de pureté :99.72%Couleur et forme :SolidMasse moléculaire :267.7319-Hydroxybufalin
CAS :<p>19-Hydroxybufalin is a natural product, inhibits epithelial-mesenchymal transition and attenuates the migration and invasion of PC3 cells.</p>Formule :C24H34O5Degré de pureté :98.74%Couleur et forme :SolidMasse moléculaire :402.52Inecalcitol
CAS :<p>Inecalcitol is a unique vitamin D3 analog that induces apoptosis and has anticancer activity.Cost-effective and quality-assured.</p>Formule :C26H40O3Degré de pureté :99.96%Couleur et forme :SolidMasse moléculaire :400.59AG-494
CAS :<p>AG-494 (Tyrphostin B48) is an inhibitor of epidermal growth factor receptor kinase.</p>Formule :C16H12N2O3Degré de pureté :98.69%Couleur et forme :SolidMasse moléculaire :280.28Engeletin
CAS :<p>1.</p>Formule :C21H22O10Degré de pureté :99.72% - 99.99%Couleur et forme :SolidMasse moléculaire :434.39ASP7663
CAS :<p>ASP7663 is a TRPA1 Receptor Agonist and exhibiting an abdominal analgesic effect in vivo.</p>Formule :C14H14FNO3Degré de pureté :98.61%Couleur et forme :SolidMasse moléculaire :263.26Cycloastragenol
CAS :<p>Cycloastragenol, a saponin from Astragalus, could be a new depression treatment.</p>Formule :C30H50O5Degré de pureté :99.85% - 99.92%Couleur et forme :SolidMasse moléculaire :490.71NB-598 Maleate
CAS :<p>NB-598 Maleate is a competitive squalene epoxidase (SE) inhibitor.</p>Formule :C31H35NO5S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :565.74TETRAHYDROPIPERINE
CAS :<p>Tetrahydropiperine (Cosmoperine) is a natural product derived from piperine, can be used to treat convulsion, epilepsy, relieve pain, and control insects.</p>Formule :C17H23NO3Degré de pureté :98.04% - 99.61%Couleur et forme :Off-White Low Melting Solid With Characteristic OdourMasse moléculaire :289.37Herbacetin
CAS :<p>1.</p>Formule :C15H10O7Degré de pureté :96.89% - 99.51%Couleur et forme :SolidMasse moléculaire :302.24Famotidine hydrochloride
CAS :<p>Famotidine hydrochloride is a competitive histamine H2-receptor antagonist. Its main pharmacodynamic effect is the inhibition of gastric secretion.</p>Formule :C8H15N7O2S3·xHClCouleur et forme :SolidMasse moléculaire :373.89PF-04802367
CAS :<p>PF-04802367 is a highly selective GSK-3 inhibitor with an IC50 of 2.1 nM based on a recombinant human GSK-3β enzyme assay and 1.1 nM based on ADP-Glo assay.</p>Formule :C16H16ClN5O3Degré de pureté :98.76%Couleur et forme :SolidMasse moléculaire :361.78GSK2981278
CAS :<p>GSK2981278 (ROR gama modulator 1) is a highly potent and selective inverse agonist of retinoic acid receptor-related orphan receptor gamma (ROR gamma).</p>Formule :C25H35NO5SDegré de pureté :99.31% - 99.67%Couleur et forme :SolidMasse moléculaire :461.61Oclacitinib maleate
CAS :<p>Oclacitinib maleate is a selective JAK inhibitor (IC50: 10-99 nM; JAK1 cytokines: 36-249 nM), with no effect on 38 non-JAK kinases.</p>Formule :C15H23N5O2S·C4H4O4Degré de pureté :99.17%Couleur et forme :SolidMasse moléculaire :453.51DMU-2139
CAS :<p>DMU2139 is a specific CYP1B1 inhibitor (CYP1B1 and CYP1A1 with IC50 of 9 nM and 795 nM, respectively).</p>Formule :C19H15NO2Degré de pureté :98.88%Couleur et forme :SolidMasse moléculaire :289.33Homocarnosine acetate
<p>Homocarnosine acetate is a dipeptide unique to brain consisting of γ-aminobutyric acid (GABA) and histidine.</p>Formule :C12H20N4O5Degré de pureté :99.52%Couleur et forme :SolidMasse moléculaire :300.31JNK-IN-8
CAS :<p>JNK-IN-8 (JNK Inhibitor XVI) is an irreversible JNK1/2/4 inhibitor (IC50: 4.7/18.7/1 nM).</p>Formule :C29H29N7O2Degré de pureté :99.24% - >99.99%Couleur et forme :SolidMasse moléculaire :507.59L-Ornithine hydrochloride
CAS :<p>L-Ornithine HCl enhances energy use, reduces fatigue, aids ammonia excretion, and is vital in the urea cycle.</p>Formule :C5H13ClN2O2Degré de pureté :99.58%Couleur et forme :SolidMasse moléculaire :168.62Indoximod
CAS :<p>Indoximod (NLG-8189) is a methylated tryptophan that inhibits IDO to boost T cell function by preventing tryptophan depletion.</p>Formule :C12H14N2O2Degré de pureté :97.82% - 99.55%Couleur et forme :SolidMasse moléculaire :218.25(+)-Magnoflorine chloride
CAS :<p>(+)-Magnoflorine chloride (Escholine chloride) has anti-inflammatory activity, it can inhibit inflammations.</p>Formule :C20H24ClNO4Degré de pureté :97.06%Couleur et forme :SolidMasse moléculaire :377.86Nanterinone mesylate
CAS :<p>Nanterinone Mesylate is the mesylate form of Nanterinone that is a novel positive inotropic and balanced vasodilator.</p>Formule :C16H19N3O4SCouleur et forme :SolidMasse moléculaire :349.4Bupranolol
CAS :<p>Bupranolol blocks β2-adrenergic receptor; treats angina, hypertension, glaucoma, arrhythmia, and prevents clots.</p>Formule :C14H22ClNO2Degré de pureté :97.63%Couleur et forme :SolidMasse moléculaire :271.78Nemifitide acetate(173240-15-8 free base)
<p>Nemifitide acetate, synthetic 5-amino acid antidepressant, has quick effect, mimics MIF.</p>Formule :C35H47FN10O8Degré de pureté :97.97%Couleur et forme :SolidMasse moléculaire :754.85Propantheline
CAS :<p>Propantheline: oral muscarinic receptor blocker for smooth muscle issues, hyperhidrosis, and bladder control.</p>Formule :C23H30NO3Couleur et forme :SolidMasse moléculaire :368.49PCI-34051
CAS :<p>PCI-34051 is an effective and selective HDAC8 inhibitor (IC50: 10 nM).</p>Formule :C17H16N2O3Degré de pureté :97.219% - 98.29%Couleur et forme :SolidMasse moléculaire :296.32NU1025
CAS :<p>NU1025 (NSC-696807) is a potent PARP inhibitor with IC50 of 400 nM.</p>Formule :C9H8N2O2Degré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :176.17Kinsenoside
CAS :<p>Kinsenoside ((+)-Kinsenoside) shows significant antihepatotoxic, and anti-inflammatory activities.</p>Formule :C10H16O8Degré de pureté :99.2% - >99.99%Couleur et forme :SolidMasse moléculaire :264.23Propyphenazone
CAS :<p>Propyphenazone: an anti-inflammatory, analgesic, antipyretic pyrazolone; prodrug; COX-2 inhibitor.</p>Formule :C14H18N2ODegré de pureté :99.64%Couleur et forme :SolidMasse moléculaire :230.31C29
CAS :<p>C29 inhibits TLR2/1 and TLR2/6 in human cells, but only TLR2/1 in mouse macrophages.</p>Formule :C16H15NO4Degré de pureté :96.34% - 97.37%Couleur et forme :SolidMasse moléculaire :285.29MALTOTETRAOSE
CAS :<p>Maltotetraose (Fujioligo 450) are potent inhibitors of TNF-α-induced intercellular adhesion molecule-1 (ICAM-1) expression.</p>Formule :C24H42O21Degré de pureté :99.02% - 99.87%Couleur et forme :SolidMasse moléculaire :666.58Gefarnate
CAS :<p>Gefarnate is a synthetic compound used for the treatment of gastric ulcers,and also used in the treatment of dry eye syndrome.</p>Formule :C27H44O2Degré de pureté :98.36%Couleur et forme :SolidMasse moléculaire :400.64Venetoclax
CAS :<p>Venetoclax (ABT-199) is a selective inhibitor of Bcl-2 (Ki < 0.010 nM), binding over 3 orders of magnitude less avidly to Bcl-xL, and Bcl-W (Kis = 48/245 nM).</p>Formule :C45H50ClN7O7SDegré de pureté :98.00% - 99.97%Couleur et forme :SolidMasse moléculaire :868.44Vildagliptin dihydrate
CAS :<p>Vildagliptin dihydrate: potent, selective DPP-IV inhibitor with 3.5 nM IC50, high oral bioavailability, effective against hyperglycemia.</p>Formule :C17H29N3O4Couleur et forme :SolidMasse moléculaire :339.436CRT0044876
CAS :<p>CRT0044876 (7-NO2-ICA) is a potent and selective APE1 inhibitor with IC50 of ~3 μM.</p>Formule :C9H6N2O4Degré de pureté :98.27% - 98.98%Couleur et forme :Brown PowderMasse moléculaire :206.15TMC647055 Choline Hydroxide Salt
<p>TMC647055 is a potent HCV NS5B inhibitor with low toxicity and good pharmacokinetics, under clinical evaluation.</p>Formule :C37H53N5O8SDegré de pureté :99.44%Couleur et forme :SolidMasse moléculaire :727.91PDE10-IN-1
CAS :<p>PDE10-IN-1 (SEP-0372814) is used for treating CNS and metabolic disorders.</p>Formule :C21H19N7Degré de pureté :99.65%Couleur et forme :SolidMasse moléculaire :369.42Tivozanib
CAS :<p>Tivozanib (KRN951) is an oral VEGFRs 1-3 inhibitor with potential antiangiogenic and cancer-fighting properties.</p>Formule :C22H19ClN4O5Degré de pureté :98.08% - 99.67%Couleur et forme :SolidMasse moléculaire :454.86Licarbazepine
CAS :<p>Licarbazepine (10,11-hydroxy-10,11 Dihydrocarbamezer) is the pharmacologically active metabolite of oxcarbazepine, a drug indicated for the treatment of partial</p>Formule :C15H14N2O2Degré de pureté :99.11%Couleur et forme :SolidMasse moléculaire :254.28Ciwujianoside A1
CAS :<p>Ciwujianoside A1 comes from Acanthopanax senticosus.</p>Formule :C59H96O26Degré de pureté :99.6%Couleur et forme :SolidMasse moléculaire :1221.38Skatole
CAS :<p>Skatole (3-Methyl-1H-indole), produced by bacteria, regulates intestinal epithelial cellular functions through activating aryl hydrocarbon receptors and p38.</p>Formule :C9H9NDegré de pureté :99.74%Couleur et forme :Leaves From Petroleum Ether; White-Brown Scales SolidMasse moléculaire :131.17Evolocumab
CAS :<p>Evolocumab is an inhibitor of the humanized monoclonal antibody PCSK9.Evolocumab can inhibit the binding of PCSK9 to LDLR.Cost-effective and quality-assured.</p>Degré de pureté :95% - 98.3%Couleur et forme :LiquidMasse moléculaire :144 kDaGlycochenodeoxycholic Acid
CAS :<p>Glycochenodeoxycholic Acid (Lithocholylglycine) is a glycine conjugate of lithocholic acid, a bile acid.</p>Formule :C26H43NO5Degré de pureté :97% - 99.97%Couleur et forme :SolidMasse moléculaire :449.62Potassium 1H-indol-3-yl sulfate
CAS :<p>Potassium 1H-indol-3-yl sulfate (Potassium 3-indoxyl sulfate) is an agonist for the human Aryl Hydrocarbon Receptor (AhR).</p>Formule :C8H6KNO4SDegré de pureté :99.52% - >99.99%Couleur et forme :White To Off-White Crystalline PowderMasse moléculaire :251.3Fenclozic acid
CAS :<p>[2-(4-Chlorophenyl)-1,3-thiazol-4-yl]acetic acid (2-[2-(4-CHLOROPHENYL)-1,3-THIAZOL-4-YL]ACETIC ACID) is an anti-inflammatory thiazole</p>Formule :C11H8ClNO2SDegré de pureté :98.05%Couleur et forme :SolidMasse moléculaire :253.7Chitin
CAS :<p>Chitin: a structural polysaccharide in fungi cell walls, insect exoskeletons, and aquatic creature hard parts.</p>Formule :C14H25NO9Degré de pureté :98%Couleur et forme :White Amorphous Semitransparent Mass SolidMasse moléculaire :351.352GW 284543 hydrochloride
CAS :<p>GW 284543 hydrochloride is a selective inhibitor of MEK5 .</p>Formule :C23H21ClN2O3Degré de pureté :99.73%Couleur et forme :SolidMasse moléculaire :408.87(R)-baclofen
CAS :<p>(R)-baclofen (STX209), a derivative of gamma-aminobutyric acid, is commonly utilized for the treatment of spasticity.</p>Formule :C10H12ClNO2Degré de pureté :97.20% - 98.94%Couleur et forme :SolidMasse moléculaire :213.66LMPTP INHIBITOR 1 dihydrochloride
CAS :<p>LMPTP Inhibitor 1 Dihydrochloride is a compound selectively targeting low molecular weight protein tyrosine phosphatase (LMPTP), exhibiting potent inhibitory</p>Formule :C28H38Cl2N4ODegré de pureté :99.83%Couleur et forme :SolidMasse moléculaire :517.53Triptorelin acetate(57773-63-4 free base)
CAS :<p>Triptorelin acetate is a GnRH agonist for hormone-responsive cancers, precocious puberty, and assisted reproduction.</p>Formule :C66H86N18O15Degré de pureté :99.90%Couleur et forme :White PowderMasse moléculaire :1371.533-Methyluridine
CAS :<p>3-Methyluridine is a modified RNA nucleoside of cellular RNA and commonly found in the form of RNA modifications.</p>Formule :C10H14N2O6Degré de pureté :99.79%Couleur et forme :SolidMasse moléculaire :258.23Delpazolid
CAS :<p>Delpazolid (LCB01-0371) is an oxazolidinone that's effective against Gram-positive bacteria and more active than linezolid in systemic infections.</p>Formule :C14H17FN4O3Degré de pureté :99.62% - 99.69%Couleur et forme :SolidMasse moléculaire :308.31Propiosyringone
CAS :<p>Propiosyringone is from the degradation of Eucalyptus globulus wood by wood-rotting fungi.</p>Formule :C11H14O4Degré de pureté :99.77%Couleur et forme :SolidMasse moléculaire :210.23L-Leucine
CAS :<p>L-Leucine is an essential amino acid vital for protein synthesis, metabolism, muscle and bone repair, blood sugar control, and wound healing.</p>Formule :C6H13NO2Degré de pureté :99.83%Couleur et forme :White Solid CrystallineMasse moléculaire :131.17CP 376395
CAS :<p>CP 376395 (CP-316311) is an effective and specific Corticotropin-releasing factor 1 (CRF1) receptor antagonist.</p>Formule :C21H30N2ODegré de pureté :99.86% - 99.94%Couleur et forme :SolidMasse moléculaire :326.48

