
Inhibiteurs
Les inhibiteurs sont des molécules qui se lient aux enzymes, récepteurs ou autres protéines pour réduire ou bloquer leur activité biologique. Ces composés sont largement utilisés en recherche pour étudier les voies biologiques, comprendre les mécanismes des maladies et développer des médicaments thérapeutiques. Les inhibiteurs jouent un rôle crucial dans le traitement de diverses maladies, y compris le cancer, les maladies cardiovasculaires et les infections. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de haute qualité pour soutenir vos recherches en biochimie, biologie cellulaire et développement pharmaceutique.
Sous-catégories appartenant à la catégorie "Inhibiteurs"
- Angiogenèse(2.833 produits)
- Apoptose(6.315 produits)
- Cycle cellulaire/point de contrôle(4.875 produits)
- Chromatine/Épigénétique(2.612 produits)
- Signalisation du cytosquelette(1.566 produits)
- Altération de l'ADN/réparation de l'ADN(2.872 produits)
- Endocrinologie/Hormones(3.754 produits)
- Enzyme(3.672 produits)
- GPCR/G-Protéine(9.015 produits)
- Immunologie et Inflammation(3.901 produits)
- Virus de la grippe(300 produits)
- Signalisation JAK/STAT(415 produits)
- Signalisation MAPK(1.256 produits)
- Transporteur membranaire/Canal ionique(3.153 produits)
- Métabolisme(10.140 produits)
- Microbiologie/Virologie(7.620 produits)
- Neuroscience(10.405 produits)
- Autres inhibiteurs(35.850 produits)
- Oxydation-Réduction(40 produits)
- Signalisation PI3K/Akt/mTOR(1.429 produits)
- Protéases/Protéasome(1.691 produits)
- Cellules souche et Dérivés(733 produits)
- Tyrosine Kinase/Adaptateurs(1.982 produits)
- Ubiquitination(1.726 produits)
Affichez 16 plus de sous-catégories
66518 produits trouvés pour "Inhibiteurs"
Trier par
Degré de pureté (%)
0
100
|
0
|
50
|
90
|
95
|
100
Heparin sodium salt
CAS :Heparin sodium, a sulfated glycosaminoglycan, acts as an anticoagulant and inhibits exosome-cell interactions.Formule :C9H20N3NaO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :241.267L-Norleucine
CAS :L-Norleucine ((S)-Norleucine) is an isomer of leucine, specifically affects protein synthesis in skeletal muscle, and has antivirus activity.Formule :C6H13NO2Degré de pureté :98.35%Couleur et forme :SolidMasse moléculaire :131.17Pseudouridine
CAS :Pseudouridine, prevalent in non-coding RNAs, boosts tRNA and rRNA function by RNA stabilization.Formule :C9H12N2O6Degré de pureté :99.3%Couleur et forme :SolidMasse moléculaire :244.2GsMTx4 TFA (1209500-46-8 free base)
GsMTx4 TFA is a spider venom peptide that selectively inhibits cationic permeable mechanically-sensitive channels (MSCs). Cost-effective and quality-assured.Formule :C187H279N48O48S6F3Degré de pureté :98% - 99.81%Couleur et forme :SolidMasse moléculaire :4216.935-Methylcytosine
CAS :5-Methylcytosine is a methylated nucleotide base found in eukaryotic DNA.Formule :C5H7N3ODegré de pureté :99.17%Couleur et forme :SolidMasse moléculaire :125.13OSS_128167
CAS :OSS_128167 (SIRT6-IN-1) is a specific SIRT6 inhibitor, and for SIRT6(IC50=89 μM), SIRT1(IC50=1578 μM) and SIRT2(IC50=751 μM).Formule :C19H14N2O6Degré de pureté :97.47% - 98.6%Couleur et forme :SolidMasse moléculaire :366.32NSC632839
CAS :NSC-632839 (Ubiquitin Isopeptidase Inhibitor II) is a nonselective isopeptidase inhibitor, which inhibits USP2 (EC50: 45±4 μM), USP7 (EC50: 37±1 μM), and SENP2Formule :C21H22ClNODegré de pureté :99.74% - 99.88%Couleur et forme :SolidMasse moléculaire :339.86SR9238
CAS :SR9238 is a synthetic agonist of liver X receptor inverse (IC50s: 214 nM and 43 nM for LXRα and LXRβ, respectively).Formule :C31H33NO7S2Degré de pureté :98.99% - 99.95%Couleur et forme :SolidMasse moléculaire :595.73E6446 dihydrochloride
CAS :E6446 dihydrochloride is a novel synthetic antagonist for nucleic acid-sensing TLRs; potently suppressed DNA stimulation of HEK:TLR9 cells with IC50 of 10 nM.
Formule :C27H37Cl2N3O3Degré de pureté :98.44%Couleur et forme :SolidMasse moléculaire :522.51Ref: TM-T4068
1mg96,00€2mg127,00€5mg205,00€10mg321,00€25mg620,00€50mg895,00€100mg1.216,00€200mg1.634,00€DTT
CAS :DTT (DL-Dithiothreitol) is a strong reducing agent. DTT has anti-disulfide ptosis activity. High-Quality, Low-Cost!Formule :C4H10O2S2Degré de pureté :98.54% - ≥95%Couleur et forme :SolidMasse moléculaire :154.25Mebrofenin
CAS :Tc 99m Mebrofenin, a diagnostic radiopharmaceutical, is a DISIDA-linked Tc-99m ion available in a kit for radio-labeling.Formule :C15H19BrN2O5Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :387.23Acetyl Pentapeptide-1 acetate
Acetyl Pentapeptide-1 acetate is an histone deacetylase inhibitor.Formule :C34H55N9O12Degré de pureté :99.09%Couleur et forme :SolidMasse moléculaire :781.86NCGC00378430
CAS :NCGC00378430 is a potent SIX1/EYA2 interaction inhibitor that disrupts the SIX1/EYA2 complex, EMT, and Metastasis.Formule :C22H23N3O5SDegré de pureté :99.74%Couleur et forme :SolidMasse moléculaire :441.5Ref: TM-T9205
1mg46,00€5mg92,00€10mg137,00€25mg250,00€50mg360,00€100mg502,00€200mg682,00€1mL*10mM (DMSO)100,00€Hederacolchiside E
CAS :Hederacolchiside E: antioxidant, neuroprotective in AD, reduces oxidative stress, inhibits lipid peroxidation.Formule :C65H106O30Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :1367.52BRD7552
CAS :BRD7552 is an inducer of transcription factor PDX1, which increases insulin expression. BRD7552 increases PDX1 expression in mouse αTC cells but not βTC cells.Formule :C33H33N3O15Degré de pureté :>99.99% - ≥98%Couleur et forme :SolidMasse moléculaire :711.63Allyl Methyl Sulfide
CAS :Allyl Methyl Sulfide is a bioactive organosulfur compound found in garlic with antibacterial, antioxidant, and anticancer activities.Formule :C4H8SDegré de pureté :≥98%Couleur et forme :Clear Colorless LiquidMasse moléculaire :88.17α-Estradiol
CAS :Alpha-Estradiol (Epiestradiol) is an estrogen that inhibits 5alpha-reductase and has potential in the study of androgenetic alopecia.Formule :C18H24O2Degré de pureté :99.65% - 99.86%Couleur et forme :SolidMasse moléculaire :272.38Delafloxacin
CAS :Delafloxacin (WQ-3034, RX-3341, ABT-492) is a potent antibiotic for levofloxacin-resistant S. pneumoniae (MIC: 0.0078-0.125 μg/ml).Formule :C18H12ClF3N4O4Degré de pureté :99.76%Couleur et forme :SolidMasse moléculaire :440.76Tubeimoside III
CAS :Tubeimoside III has anti-inflammatory, anti-tumor, and anti-tumorigenic activities, stronger than those of tubeimoside II.Formule :C64H100O31Degré de pureté :99.64% - 99.86%Couleur et forme :SolidMasse moléculaire :1365.46Ref: TM-T4S1849
2mg39,00€5mg56,00€10mg93,00€25mg150,00€50mg215,00€100mg320,00€200mg477,00€1mL*10mM (DMSO)126,00€Sweroside
CAS :Sweroside: hepatoprotective, potential anti-osteoporotic for MG-63 cells and rat osteoblasts.
Formule :C16H22O9Degré de pureté :98.87% - 99.89%Couleur et forme :SolidMasse moléculaire :358.34Rhamnose monohydrate
CAS :Rhamnose monohydrate (L-(+)-Rhamnose Monohydrate) is a naturally-occurring deoxy sugar that is found primarily in plants and some bacteria.Formule :C6H12O5·H2ODegré de pureté :99.71% - 99.90%Couleur et forme :White Crystalline Powder One Of The Rarer SugarsMasse moléculaire :182.17Indigo
CAS :Indigo (Indigotin) is extracted from Indigo blue.Formule :C16H10N2O2Degré de pureté :99.01%Couleur et forme :Dark Blue Solid PowderMasse moléculaire :262.26Dihydrolanosterol
CAS :Dihydrolanosterol, a sterol derived from lanosterol, undergoes demethylation by cytochrome P450 14alpha-demethylase in mammals and yeast.Formule :C30H52ODegré de pureté :98% - 99.53%Couleur et forme :SolidMasse moléculaire :428.73Dihydroergocristine mesylate
CAS :DHEC mesylate is a vasodilator and α-adrenergic antagonist used for vascular dementia and as a geroprotector.Formule :C36H45N5O8SDegré de pureté :98.9% - 99.79%Couleur et forme :SolidMasse moléculaire :707.84Etidronic acid
CAS :Etidronic acid (HEDP) is a diphosphonate which affects calcium metabolism. It inhibits ectopic calcification and slows down bone resorption and bone turnover.Formule :C2H8O7P2Degré de pureté :99.93% - ≥95%Couleur et forme :Liquid SyrupMasse moléculaire :206.03Arctiin
CAS :Arctiin (Arctigenin-4-glucoside) acts on an agonists of the adiponectin receptor 1 with anti-cancer effects.Formule :C27H34O11Degré de pureté :98.22% - 99.81%Couleur et forme :White To Off-White SolidMasse moléculaire :534.55Orantinib
CAS :Orantinib (NSC 702827) , a excellent effective against PDGFR autophosphorylation with Ki of 8 nM, also highly inhibits Flk-1 and FGFR1 trans-phosphorylation.Formule :C18H18N2O3Degré de pureté :98.92% - 99.52%Couleur et forme :SolidMasse moléculaire :310.351-Aminocyclobutanecarboxylic acid
CAS :1-Aminocyclobutanecarboxylic acid (ACBC) is a NMDA receptor partial agonist. 1-Aminocyclobutanecarboxylic acid act at the glycine site, NR1[1].Formule :C5H9NO2Degré de pureté :99.94%Couleur et forme :White To Tan Powder Crystals Crystalline Powder And/Or With ChunksMasse moléculaire :115.13N-Formyl-Met-Leu-Phe
CAS :N-Formyl-Met-Leu-Phe (N-Formyl-MLF) (fMLF) is a synthetic peptide that acts as an agonist at formyl peptide receptors (FPR; Ki = 0.8 pM).Formule :C21H31N3O5SDegré de pureté :98.69% - 98.69%Couleur et forme :SolidMasse moléculaire :437.55Acacetin
CAS :Acacetin (5,7-Dihydroxy-4'-methoxyflavone) is an O-methylated flavone found in various plants, shows antinociceptive, anti-inflammatory, and antioxidantFormule :C16H12O5Degré de pureté :96.26% - ≥95%Couleur et forme :Pale-Yellow NeedlesMasse moléculaire :284.26ILK-IN-2
CAS :ILK-IN-2 (OSU-T315) is a novel potent, orally active ILK (integrin-linked kinase) inhibitor with IC50 of 0.6 μM.Formule :C30H30F3N5ODegré de pureté :99.30%Couleur et forme :SolidMasse moléculaire :533.59Ref: TM-T5488
1mg46,00€5mg92,00€10mg122,00€25mg154,00€50mg182,00€100mg266,00€200mg386,00€1mL*10mM (DMSO)130,00€SEA0400
CAS :SEA0400 is a selective inhibitor of the Na+/Ca2+ exchanger.Formule :C21H19F2NO3Degré de pureté :98.88% - 99.55%Couleur et forme :SolidMasse moléculaire :371.38Ref: TM-T3508
1mg37,00€2mg52,00€5mg77,00€10mg124,00€25mg219,00€50mg358,00€100mg537,00€500mg1.189,00€1mL*10mM (DMSO)71,00€Tri-Salicylic Acid
CAS :Tri-Salicylic Acid, a product of the thermal decomposition of aspirin, is a compound for proteomics research.
Formule :C21H14O7Degré de pureté :97.02%Couleur et forme :SolidMasse moléculaire :378.33DL-Mannitol
CAS :DL-Mannitol is a osmotic diuretic, it may play a role in reducing off-target 68Ga-PSMA renal uptakeFormule :C6H14O6Degré de pureté :99.48%Couleur et forme :Orthorhombic Needles From Alc (Ntp 1992)Masse moléculaire :182.17N-[3,5-bis(trifluoromethyl)phenyl]-N'-[(9r)-6'-methoxycinchonan-9-yl]- thiourea
CAS :N-[3,5-bis(trifluoromethyl)phenyl]-N'-[(9R)-6'-methoxycinchonan-9-yl]thiourea is a bifunctional organocatalyst derived from cinchona alkaloids.Formule :C29H28F6N4OSDegré de pureté :99.83%Couleur et forme :SolidMasse moléculaire :594.61Kansuinine A
CAS :Kansuinine A, a 95% ethanol extract from the roots of E. kansui, possesses an inhibitory effect on IL-6-induced Stat3 activation by activating ERK1/2.Formule :C37H46O15Degré de pureté :99.28% - 99.96%Couleur et forme :SolidMasse moléculaire :730.75BTR-1
CAS :5-Benzylidene-3-ethyl rhodanine(BTR-1 (5-Benzylidene-3-ethyl rhodanine)) is an active anti-cancer agent. BTR-1 activates apoptosis and induces cell death.Formule :C12H11NOS2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :249.35Ref: TM-T5822
2mg34,00€5mg50,00€10mg84,00€25mg137,00€50mg200,00€100mg304,00€200mg442,00€1mL*10mM (DMSO)56,00€Siamenoside I
CAS :Siamenoside I, a bioactive mogroside, inhibits maltase with an IC50 of 12 mM.Formule :C54H92O24Degré de pureté :99.79% - 99.81%Couleur et forme :SolidMasse moléculaire :1125.29Ref: TM-TN2208
1mg60,00€5mg116,00€10mg178,00€25mg301,00€50mg429,00€100mg593,00€1mL*10mM (DMSO)212,00€Obtusin
CAS :Obtusin is a natural product.Formule :C18H16O7Degré de pureté :99.13%Couleur et forme :SolidMasse moléculaire :344.32Dryocrassin ABBA
CAS :Dryocrassin ABBA (Dryocrassin) is a flavonoid natural product derived from Dryopteris crassirhizoma, with antiviral and antibacterial activities.Formule :C43H48O16Degré de pureté :98.43%Couleur et forme :SolidMasse moléculaire :820.83ML359
CAS :ML359 is a protein disulfide isomerase inhibitor.Formule :C23H28ClNO4Degré de pureté :99.68%Couleur et forme :SolidMasse moléculaire :417.93Ref: TM-T25821
1mg88,00€5mg187,00€10mg301,00€25mg525,00€50mg742,00€100mg1.035,00€1mL*10mM (DMSO)207,00€Benperidol Hydrochloride
CAS :Benperidol Hydrochloride is a potent D2/D4 dopamine receptor antagonist, used as antipsychotic and neuroleptic.Formule :C22H25ClFN3O2Couleur et forme :SolidMasse moléculaire :417.91Antitubercular agent-30
CAS :Antitubercular agent-30 has antitubercular activity.Formule :C12H10N2O3SDegré de pureté :99.97%Couleur et forme :SolidMasse moléculaire :262.28Bevirimat
CAS :Bevirimat (PA-457) is a first-in-class inhibitor of HIV-1 maturation, blocking the cleavage of the Gag capsid (CA) precursor, CA-SPI, to mature CA proteinFormule :C36H56O6Degré de pureté :99.4% - ≥95%Couleur et forme :SolidMasse moléculaire :584.83Mavacoxib
CAS :Mavacoxib is a selective inhibitor of cyclooxygenase-2 (COX-2) ,with Anti-Tumour activity.Formule :C16H11F4N3O2SDegré de pureté :99.90%Couleur et forme :SolidMasse moléculaire :385.34Mulberroside A
CAS :1.Formule :C26H32O14Degré de pureté :99.05% - 99.4%Couleur et forme :SolidMasse moléculaire :568.52Ref: TM-T6S1597
1mg47,00€5mg95,00€10mg137,00€25mg240,00€50mg403,00€100mg582,00€1mL*10mM (DMSO)108,00€2-Ethylbutyric Acid
CAS :2-Ethylbutyric acid is an internal standard that can be used in calibration methods for VFA analytical standards for feces.Formule :C6H12O2Degré de pureté :97.19%Couleur et forme :LiquidMasse moléculaire :116.16Pempidine tartrate
CAS :Pempidine tartrate, a nicotinic antagonist, was used for hypertension but replaced by more specific drugs.Formule :C14H27NO6Couleur et forme :SolidMasse moléculaire :305.37Quisinostat
CAS :Quisinostat (JNJ-26481585), a second-gen HDAC inhibitor, is most potent for HDAC1 (IC50 0.11 nM) and selectively affects HDACs 2, 4, 10, and 11.Formule :C21H26N6O2Degré de pureté :96.01% - ≥98%Couleur et forme :SolidMasse moléculaire :394.47Sodium taurodeoxycholate hydrate
CAS :Sodium taurodeoxycholate hydrate (Taurodeoxycholic acid sodium salt monohydrate) has been used in a study to assess the effect of submicellar concentrations ofFormule :C26H44NO6S·Na·H2ODegré de pureté :99.78%Couleur et forme :SolidMasse moléculaire :539.70L-745870 hydrochloride
CAS :L-745870 hydrochloride has excellent brain penetration. L-745870 hydrochloride is a high-affinity, selective and orally active human dopamine D4 receptorFormule :C18H20Cl2N4Degré de pureté :97.36%Couleur et forme :SolidMasse moléculaire :363.28Ref: TM-T11799
5mg38,00€10mg62,00€25mg105,00€50mg170,00€100mg245,00€200mg354,00€1mL*10mM (DMSO)33,00€2-Aminopurine
CAS :2-Aminopurine is a double-stranded RNA-dependent protein kinase, protein kinase R (PKR) inhibitor.Formule :C5H5N5Degré de pureté :99.51%Couleur et forme :White To Light Yellow Crystal PowderMasse moléculaire :135.13Seltorexant hydrochloride
CAS :Seltorexant hydrochloride is a selective, orally active and high-affinity antagonist of OX2R with pKi values of 8.0 and 8.1 for human and rat OX2R.Formule :C21H23ClFN7ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :443.91Madrasin
CAS :Madrasin (DDD00107587) is a potent and cell penetrant splicing inhibitor that interferes with the early stages of spliceosome assembly.Formule :C16H17N5O2Degré de pureté :99.06% - 99.61%Couleur et forme :SolidMasse moléculaire :311.34Tafluprost
CAS :Tafluprost, a prostaglandin analog, is the selective agonist of fluoroprostaglandin (FP) receptor PGF2α.Formule :C25H34F2O5Degré de pureté :97.7% - 99.67%Couleur et forme :LiquidMasse moléculaire :452.53BMS-779788
CAS :BMS-779788 (XL-652) is an LXRα/β partial agonist (IC50: 68/14 nM).Formule :C28H29ClN2O3SDegré de pureté :98.65% - 99.24%Couleur et forme :SolidMasse moléculaire :509.06Futibatinib
CAS :Futibatinib (TAS-120) is an orally active, potent,and irreversible FGFR inhibitor of FGFR1, FGFR2, FGFR3, and FGFR4.Cost-effective and quality-assured.Formule :C22H22N6O3Degré de pureté :97.66% - 99.44%Couleur et forme :SolidMasse moléculaire :418.45Ref: TM-T5044
1mg50,00€5mg114,00€10mg167,00€25mg313,00€50mg485,00€100mg627,00€200mg890,00€1mL*10mM (DMSO)127,00€MFCD01827729
CAS :EMTPC, a thiophene amino acid derivative, may have anti-inflammatory, analgesic, anticonvulsant, anticancer, and immune-modulating properties.Formule :C14H15NO2SDegré de pureté :99.37%Couleur et forme :SolidMasse moléculaire :261.34ABX-1431
CAS :ABX-1431 (Elcubragistat) is a selective and orally available CNS-penetrant monoacylglycerol lipase (MAGL/MGLL) inhibitor (IC50: 14 nM).Formule :C20H22F9N3O2Degré de pureté :99.8% - 99.96%Couleur et forme :SolidMasse moléculaire :507.392,4-Diaminophenoxyethanol HCl
CAS :Isophorone, a monoterpene with related 1,8-cineole and camphor, offers cancer protection, antimicrobial and antioxidant effects.Formule :C8H14Cl2N2O2Degré de pureté :98.11%Couleur et forme :Pale Grey To Pale Pink-Grey Solid PowderMasse moléculaire :241.12BMS-986020
CAS :BMS-986020 (AM152) is a selective antagonist of LPA1.Formule :C29H26N2O5Degré de pureté :98.82% - >99.99%Couleur et forme :SolidMasse moléculaire :482.53D159687
CAS :D159687 is a selective PDE4D inhibitor,had a procognitive profile as it improved memory in the novel object recognition test but had no antidepressant benefit.Formule :C21H19ClN2O2Degré de pureté :97.57%Couleur et forme :SolidMasse moléculaire :366.84TABERSONINE HYDROCHLORIDE
CAS :TABERSONINE HYDROCHLORIDE is a natural product extracted from the bean of Voacanga africana, is a potent inhibitor against Aβ(1 42) aggregation and toxicity.Formule :C21H25ClN2O2Degré de pureté :98.17%Couleur et forme :SolidMasse moléculaire :372.89Aminopurvalanol A
CAS :Aminopurvalanol A is a competitive, selective and cell-permeable inhibitor of cyclin-dependent kinase (CDK) that potently inhibits Cyclin A/cdk2, Cyclin B/cdk1Formule :C19H26ClN7ODegré de pureté :99.73%Couleur et forme :SolidMasse moléculaire :403.91Ref: TM-T22260
2mg39,00€5mg60,00€10mg92,00€25mg173,00€50mg269,00€100mg389,00€200mg555,00€1mL*10mM (DMSO)62,00€Trifluridine/tipiracil hydrochloride mixture
CAS :Trifluridine/tipiracil hydrochloride mixture (TAS-102) is a novel oral combination drug containing trifluridine (TFT) and Tipiracil hydrochloride (TTP) in aFormule :C29H34Cl2F6N8O12Degré de pureté :98% - 99.79%Couleur et forme :SolidMasse moléculaire :871.53Ref: TM-T3658
2mg37,00€5mg54,00€10mg93,00€25mg148,00€50mg236,00€100mg358,00€200mg538,00€500mg842,00€1mL*10mM (DMSO)73,00€Isomucronulatol 7-O-glucoside
CAS :Isomucronulatol 7-O-glucoside is a natural productFormule :C23H28O10Degré de pureté :99.33% - 99.92%Couleur et forme :SolidMasse moléculaire :464.46Ref: TM-TN1787
1mg84,00€5mg177,00€10mg295,00€25mg497,00€50mg708,00€100mg964,00€1mL*10mM (DMSO)146,00€(+)-ISOPINOCAMPHEOL
CAS :(+)-ISOPINOCAMPHEOL is a natural product.Formule :C10H18ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :154.25ML324
CAS :ML324(IC50=920 nM) is a specific inhibitor of jumonji histone demethylase (JMJD2).Formule :C21H23N3O2Degré de pureté :98.22% - 98.57%Couleur et forme :SolidMasse moléculaire :349.43Ref: TM-T6593
2mg34,00€5mg49,00€10mg74,00€25mg122,00€50mg205,00€100mg334,00€200mg494,00€1mL*10mM (DMSO)79,00€C-Reactive Protein (CRP) 174-185 acetate
CRP (174-185) acetate boosts human monocytes' and macrophages' tumor-killing action; mimics full CRP's antitumor effects.Formule :C64H97N13O18Degré de pureté :98.74% - 99.21%Couleur et forme :SolidMasse moléculaire :1336.53Afzelin
CAS :Afzelin (Kaempferol-3-O-rhamnoside) has several cellular activities such as DNA-protective, antibacterial, antioxidant, and anti-inflammatory as well as UV-Formule :C21H20O10Degré de pureté :98.92% - 99.38%Couleur et forme :SolidMasse moléculaire :432.38Ref: TM-TN1362
1mg48,00€5mg125,00€10mg180,00€25mg299,00€50mg439,00€100mg627,00€1mL*10mM (DMSO)117,00€Dioctanoylglycol
CAS :Dioctanoylglycol (ethane-1,2-diyl dioctanoate) is a diacylglycerol kinase inhibitor.Formule :C18H34O4Degré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :314.46Bepridil free base
CAS :Bepridil: Class IV anti-arrhythmic, calcium blocker, dilates coronary arteries.Formule :C24H34N2OCouleur et forme :SolidMasse moléculaire :366.54JI-101
CAS :JI-101 (CGI-1842) is an oral multi-kinase inhibitor that targets VEGFR-2, PDGFR-β, and EphB4.Formule :C22H20BrN5O2Degré de pureté :99.41% - 99.97%Couleur et forme :SolidMasse moléculaire :466.33Hamamelitannin
CAS :Hamamelitannin, from Hamamelis virginiana bark, is cytotoxic, disrupts biofilms, enhances antibiotic effectiveness, and protects cells from peroxide damage.Formule :C20H20O14Degré de pureté :99.58% - 99.99%Couleur et forme :SolidMasse moléculaire :484.366-AZATHYMINE
CAS :6-azathymine inhibits D-3-aminoisobutyrate-pyruvate aminotransferase; 6-azauracil competes with beta-alanine, uncompetitive with pyruvic acid, Ki ~8.9 mM.Formule :C4H5N3O2Degré de pureté :99.47%Couleur et forme :SolidMasse moléculaire :127.1Hypocrellin A
CAS :Hypocrellin A is a natural PKC inhibitor with light-induced antitumor, antifungal and antiviral activities.Cost-effective and quality-assured.Formule :C30H26O10Degré de pureté :98% - 99.95%Couleur et forme :SolidMasse moléculaire :546.52Dubermatinib
CAS :Dubermatinib (TP0903) is a potent and selective Axl kinase inhibitor.Formule :C24H30ClN7O2SDegré de pureté :98.65% - 99.58%Couleur et forme :SolidMasse moléculaire :516.06Importazole
CAS :Importazole is an inhibitor of the nuclear transport receptor importin-β.Formule :C20H22N4Degré de pureté :99.6% - >99.99%Couleur et forme :SolidMasse moléculaire :318.42Ref: TM-T3445
5mg49,00€10mg69,00€25mg144,00€50mg215,00€100mg356,00€200mg532,00€500mg852,00€1mL*10mM (DMSO)54,00€6''-O-xylosyl-glycitin
CAS :6''-O-xylosyl-glycitin is isolated from the flower of Pueraria thunbergiana Benth.Formule :C27H30O14Degré de pureté :99.65% - 99.68%Couleur et forme :SolidMasse moléculaire :578.52Rivanicline hemioxalate
Rivanicline hemioxalate is a selective α4β2 nicotinic receptor agonist (K i =26 nM), over 1,000x preference to α7 (K i =3.6 μM), with limited side effects.Formule :C12H16N2O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :207.23Phosalone
CAS :Phosalone is an organophosphate chemical commonly used as an insecticide and acaricide.Formule :C12H15ClNO4PS2Degré de pureté :98.45% - ≥95%Couleur et forme :Crystals SolidMasse moléculaire :367.81Maltol
CAS :Maltol (Palatone) is a naturally occurring organic compound that is flavour enhancer and flavouring agent.Formule :C6H6O3Degré de pureté :98.88% - 99.8%Couleur et forme :50% Alcohol Aqueous Solution) 5 3 (Ntp 1992)Masse moléculaire :126.11U-73343
CAS :U-73343 is an inactive analog of U-73122 and can be used as a negative control. U-73122 dose-dependently inhibits acid secretion irrespective of the stimulant.Formule :C29H42N2O3Degré de pureté :99.06%Couleur et forme :SolidMasse moléculaire :466.66BS194
CAS :BS194 is as a potent cyclin-dependent protein kinases (CDKs) inhibitor.Formule :C20H27N5O3Degré de pureté :99.85%Couleur et forme :SolidMasse moléculaire :385.46SC-58125
CAS :SC-58125 is a selective cyclooxygenase 2 (COX-2) inhibitor. SC-58125 exhibits antitumor activity, and also inhibits oedema at sites of inflammation.Formule :C17H12F4N2O2SDegré de pureté :99.57%Couleur et forme :SolidMasse moléculaire :384.35Ref: TM-T23333
5mg37,00€10mg60,00€25mg119,00€50mg178,00€100mg301,00€200mg432,00€1mL*10mM (DMSO)55,00€SRT 1720 dihydrochloride
CAS :SRT 1720 dihydrochloride is a selective activator of SIRT1 (EC1.5: 0.16 μM) and shows less potent activities on SIRT2 (EC1.5: 37 μM) and SIRT3 (EC1.5: 300 μM).Formule :C25H25Cl2N7OSDegré de pureté :98.58%Couleur et forme :SolidMasse moléculaire :542.48JZL195
CAS :JZL195 is a selective and efficacious dual FAAH/MAGL inhibitor.Formule :C24H23N3O5Degré de pureté :99.81%Couleur et forme :SolidMasse moléculaire :433.46Lumefantrine
CAS :Lumefantrine, an antimalarial, treats malaria with artemether, effective against Plasmodium spp. including in chloroquine-resistant areas.Formule :C30H32Cl3NODegré de pureté :98.36%Couleur et forme :Yellow SolidMasse moléculaire :528.94SHU 9119 acetate
SHU 9119 acetate: hMC3R & hMC4R antagonist, hMC5R partial agonist. IC50: MC3R 0.23nM, MC4R 0.06nM, MC5R 0.09nM.Formule :C56H75N15O11Degré de pureté :99.8%Couleur et forme :SolidMasse moléculaire :1134.29Haloperidol lactate
CAS :Haloperidol lactate: a potent antipsychotic for acute/chronic schizophrenia and polyarousal syndrome research.Formule :C24H29ClFNO5Couleur et forme :SolidMasse moléculaire :465.95Tenacissoside H
CAS :Tenacissoside H (Tenacissimoside C) has antitumor activity on esophageal cancer through arresting cell cycle and regulating PI3K/Akt-NF-κB transduction cascade.Formule :C42H66O14Degré de pureté :97.25% - 99.78%Couleur et forme :SolidMasse moléculaire :794.97Ref: TM-T6S1844
5mg43,00€10mg60,00€25mg96,00€50mg138,00€100mg198,00€200mg295,00€1mL*10mM (DMSO)52,00€Cellulase
CAS :Cellulase is an enzyme that catalyzes the hydrolysis of certain linkages in cellulose.Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :N/ATelekin
CAS :Telekin, a sesquiterpene lactone from Carpesium divaricatum, strongly inhibits cancer cell growth.Formule :C15H20O3Degré de pureté :99.86% - 99.97%Couleur et forme :SolidMasse moléculaire :248.32SKF 38393 hydrochloride
CAS :SKF 38393 hydrochloride (SKF38393 HCl) is a selective dopamine D1/D5 receptor agonist.Formule :C16H17NO2·HClDegré de pureté :99.1% - 99.51%Couleur et forme :SolidMasse moléculaire :291.77L-Cysteine hydrochloride hydrate
CAS :L-Cysteine HCl hydrate: precursor to H2S, taurine, glutathione; suppresses ghrelin, reducing appetite.Formule :C3H10ClNO3SDegré de pureté :99.86%Couleur et forme :White Solid PowderMasse moléculaire :175.643-Methylbut-2-enoic acid
CAS :3-Methylbut-2-enoic acid (Senecioic acid) appears in the urine of patients with 3-Methylcrotonic aciduria.Formule :C5H8O2Degré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :100.12Tafamidis
CAS :Tafamidis stabilizes TTR, preventing amyloid buildup; binds with negative cooperativity (Kd1: 3 nM, Kd2: 278 nM); treats familial amyloid polyneuropathy.Formule :C14H7Cl2NO3Degré de pureté :99.34% - 99.65%Couleur et forme :SolidMasse moléculaire :308.12Fevipiprant
CAS :Fevipiprant (NVP-QAW039) is a selective, potent, reversible competitive CRTh2 antagonist.Formule :C19H17F3N2O4SDegré de pureté :99.32% - 99.59%Couleur et forme :SolidMasse moléculaire :426.41Xylan
CAS :Xylan represents the main hemicellulose component in the secondary plant cell walls of flowering plants.Formule :C5H10O5Degré de pureté :85%Couleur et forme :SolidMasse moléculaire :150.13Methyl isoeugenol
CAS :Methyl isoeugenol (MIE), a natural flavor, is 93.7% of Pimenta leaf oil and used as a food additive and calming treatment.Formule :C11H14O2Degré de pureté :99.87%Couleur et forme :SolidMasse moléculaire :178.23
